Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | HSP90AA1 | P07900 | 1/20 | 1.00 |
| ▸ | TSHR | P16473 | 6/20 | 0.67 |
| ▸ | LMNA | P02545 | 2/20 | 0.67 |
| ▸ | ALDH1A1 | P00352 | 6/20 | 0.55 |
| ▸ | ACHE | P22303 | 1/20 | 0.55 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.55 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.55 |
| ▸ | HTT | P42858 | 2/20 | 0.52 |
| ▸ | KMT2A | Q03164 | 2/20 | 0.52 |
| ▸ | GAA | P10253 | 1/20 | 0.52 |
| ▸ | CES2 | O00748 | 1/20 | 0.52 |
| ▸ | CES1 | P23141 | 1/20 | 0.52 |
| ▸ | MEN1 | O00255 | 1/20 | 0.52 |
| ▸ | DDX3X | O00571 | 1/20 | 0.52 |
| ▸ | POLB | P06746 | 1/20 | 0.52 |
| ▸ | MAPT | P10636 | 1/20 | 0.52 |
| ▸ | CTDSP1 | Q9GZU7 | 1/20 | 0.52 |
| ▸ | TP53 | P04637 | 1/20 | 0.50 |
| ▸ | NFE2L2 | Q16236 | 1/20 | 0.48 |
| ▸ | CA2 | P00918 | 1/20 | 0.48 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL31482901 | 1.00 | HSP90AA1 (1.00) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL30468119 | 1.00 | HSP90AA1 (1.00) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL4909394 | 0.88 | HSP90AA1 (0.79) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL31405188 | 0.87 | HSP90AA1 (0.77) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL11356136 | 0.87 | HSP90AA1 (0.77) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL20347051 | 0.87 | HSP90AA1 (0.77) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL1818188 | 0.85 | HSP90AA1 (0.74) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL4902082 | 0.84 | HSP90AA1 (0.71) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL4910155 | 0.84 | HSP90AA1 (0.71) | HSP90AA1TSHRLMNAALDH1A1ACHE | |
| SCHEMBL288228 | 0.83 | HSP90AA1 (0.71) | HSP90AA1TSHRLMNAALDH1A1ACHE |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 258 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-2931703-B1 | METHOD FOR PRODUCING BIS (3-AMINOPHENYL) DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2018-11-28 | — | — | EP | claimed |
| US-20150329485-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2015-11-19 | — | — | US | claimed |
| EP-2931703-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | Bayer CropScience AG (DE) | 2015-10-21 | — | — | EP | claimed |
| WO-2014090913-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2014-06-19 | — | — | WO | claimed |
| US-7732534-B2 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION (JP) | 2010-06-08 | — | — | US | claimed |
| US-20080051552-A1 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION | 2008-02-28 | — | — | US | claimed |
| US-20080051519-A1 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION (JP) | 2008-02-28 | — | — | US | claimed |
| US-6989263-B1 | Method for identifying and using compounds that inactivate HIV-1 and other retroviruses by attacking highly conserved zinc fingers in the viral nucleocapsid protein | THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 2006-01-24 | — | — | US | claimed |
| EP-1435930-A2 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2004-07-14 | — | — | EP | claimed |
| US-20030198648-A1 | Methods for identifying compounds which inhibit binding of nucleocapsid 7 protein to HIV-1 RNA | ACHILION PHARMACEUTICALS | 2003-10-23 | — | — | US | claimed |
| WO-2003060098-A2 | METHODS FOR IDENTIFYING COMPOUNDS WHICH INHIBIT BINDING OF NUCLEOCAPSID 7 PROTEIN TO HIV-1 RNA | ACHILLION PHARMACEUTICALS, INC. (US) | 2003-07-24 | — | — | WO | claimed |
| WO-2003032969-A2 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2003-04-24 | — | — | WO | claimed |
| EP-0782632-B1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | US GOV HEALTH & HUMAN SERV (US) | 2003-04-16 | — | — | EP | claimed |
| US-6001555-A | DISSOCIATING A ZINC FINGER BY CONTACTING THE PROTEIN WITH A DISULFIDE, A MALEIMIDE, AN ALPHA-HALOGENATED KETONE, A HYDRAZIDE, A NITRIC OXIDE OR DERIVATIVES, CUPRIC IONS, FERRIC IONS OR THEIR COMPLEXES; SYNERGISTIC EFFECTS WITH VIRICIDES | THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1999-12-14 | — | — | US | claimed |
| EP-0782632-A1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the Secretary of the Department of Health and Human Services (US) | 1997-07-09 | — | — | EP | claimed |
| WO-1996009406-A9 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | — | 1996-05-23 | — | — | WO | claimed |
| WO-1996009406-A1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1996-03-28 | — | — | WO | claimed |
| EP-0693056-A1 | PROCESS FOR THE PREPARATION OF ARYL- AND HETEROARYLSULPHURPENTAFLUORIDES | ZENECA LIMITED (GB) | 1996-01-24 | — | — | EP | claimed |
| WO-1994022817-A1 | PROCESS FOR THE PREPARATION OF ARYL- AND HETEROARYLSULPHURPENTAFLUORIDES | ZENECA LIMITED (GB) | 1994-10-13 | — | — | WO | claimed |
| JP-56043338-A | — | — | None | — | — | JP | disclosed |
| JP-1165586-A | — | — | None | — | — | JP | disclosed |
| CN-116283684-B | Green preparation method of diphenyl sulfide and derivative thereof | 常州大学 | 2025-04-08 | — | — | CN | disclosed |
| US-20230278965-A1 | NOVEL CARBONOHYDRAZONOYL DICYANIDE COMPOUNDS COMPRISING 2 OR MORE ARYL OR HETEROARYL CONNECTED VIA LINKER AND USE THEREOF | KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) | 2023-09-07 | — | — | US | disclosed |
| CN-116283684-A | Green preparation method of diphenyl sulfide and derivative thereof | 常州大学 | 2023-06-23 | — | — | CN | disclosed |
| CN-110845287-B | Method for selective vulcanization of aliphatic amine | 陕西师范大学 | 2023-02-14 | — | — | CN | disclosed |
| WO-2023001999-A1 | C2-THIOETHER TRYPTOPHAN TRIMERS AND TETRAMERS FOR THE TREATMENT OF BETACORONOAVIRUS INFECTIONS | 1. CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (CSIC) (ES) | 2023-01-26 | — | — | WO | disclosed |
| EP-4122917-A1 | C2-THIOETHER TRYPTOPHAN TRIMERS AND TETRAMERS AND USE THEREOF | Consejo Superior de Investigaciones Científicas (CSIC) (ES) | 2023-01-25 | — | — | EP | disclosed |
| CN-113956521-B | Preparation method of super-hydrophobic antifouling anti-drag material | 中国船舶重工集团公司第七二五研究所 | 2022-12-13 | — | — | CN | disclosed |
| US-11500247-B2 | Liquid crystal sensor | PLATYPUS TECHNOLOGIES, LLC (US) | 2022-11-15 | — | — | US | disclosed |
| CN-113956521-A | Preparation method of super-hydrophobic antifouling anti-drag material | 中国船舶重工集团公司第七二五研究所 | 2022-01-21 | — | — | CN | disclosed |
| CN-111116461-B | Palladium-catalyzed o-toluidine amide gamma-C- (sp)3) Synthesis method of H sulfur/selenium ether compound | 浙江工业大学 | 2021-07-27 | — | — | CN | disclosed |
| US-20200409221-A1 | LIQUID CRYSTAL SENSOR | PLATYPUS TECHNOLOGIES, LLC | 2020-12-31 | — | — | US | disclosed |
| CN-111373077-A | Sn or Sn alloy plating solution and method for producing Sn or Sn alloy plating | 上村工业株式会社 | 2020-07-03 | — | — | CN | disclosed |
| US-20200208285-A1 | ELECTROLYTIC SN OR SN ALLOY PLATING SOLUTION AND METHOD FOR PRODUCING SN OR SN ALLOY PLATED ARTICLE | UEMURA KOGYO KK (JP) | 2020-07-02 | — | — | US | disclosed |
| CN-111116461-A | Palladium-catalyzed o-toluidine amide gamma-C- (sp)3) Synthesis method of H sulfur/selenium ether compound | 浙江工业大学 | 2020-05-08 | — | — | CN | disclosed |
| CN-110845287-A | Method for selective vulcanization of aliphatic amine | 陕西师范大学 | 2020-02-28 | — | — | CN | disclosed |
| US-10239831-B2 | Method for producing bis(3-aminophenyl)disulfides and 3-aminothiols | BAYER CROPSCIENCE AG (DE) | 2019-03-26 | — | — | US | disclosed |
| EP-2931703-B1 | METHOD FOR PRODUCING BIS (3-AMINOPHENYL) DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2018-11-28 | — | — | EP | disclosed |
| US-20180258036-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2018-09-13 | — | — | US | disclosed |
| US-10053421-B2 | Method for producing bis(3-aminophenyl)disulfides and 3-aminothiols | BAYER CROPSCIENCE AG (DE) | 2018-08-21 | — | — | US | disclosed |
| US-9949480-B2 | N-alkylthio beta-lactams, alkyl-coenzyme A asymmetric disulfides, and aryl-alkyl disulfides as anti-bacterial agents | UNIVERSITY OF SOUTH FLORIDA (US) | 2018-04-24 | — | — | US | disclosed |
| US-20170212088-A1 | DETECTION OF GAS-PHASE ANALYTES USING LIQUID CRYSTALS | PLATYPUS TECHNOLOGIES, LLC | 2017-07-27 | — | — | US | disclosed |
| US-9575037-B2 | Detection of gas-phase analytes using liquid crystals | PLATYPUS TECHNOLOGIES, LLC (US) | 2017-02-21 | — | — | US | disclosed |
| EP-2805940-B1 | PYRAZINE CARBOXAMIDE COMPOUND | ASTELLAS PHARMA INC (JP) | 2016-11-23 | — | — | EP | disclosed |
| US-20160274084-A1 | DETECTION OF VAPOR PHASE COMPOUNDS BY CHANGES IN PHYSICAL PROPERTIES OF A LIQUID CRYSTAL | PLATYPUS TECHNOLOGIES, LLC | 2016-09-22 | — | — | US | disclosed |
| US-20160160178-A1 | IMMUNOTHERAPY USING STEM CELLS | WHITE OAK IND INC (US) | 2016-06-09 | — | — | US | disclosed |
| US-9341576-B2 | Detection of vapor phase compounds by changes in physical properties of a liquid crystal | PLATYPUS TECHNOLOGIES, LLC (US) | 2016-05-17 | — | — | US | disclosed |
| US-20160018371-A1 | DETECTION OF GAS-PHASE ANALYTES USING LIQUID CRYSTALS | PLATYPUS TECHNOLOGIES, LLC | 2016-01-21 | — | — | US | disclosed |
| US-20150327547-A1 | N-ALKYLTHIO BETA-LACTAMS, ALKYL-COENZYME A ASYMMETRIC DISULFIDES, AND ARYL-ALKYL DISULFIDES AS ANTI-BACTERIAL AGENTS | UNIVERSITY OF SOUTH FLORIDA (US) | 2015-11-19 | — | — | US | disclosed |
| US-20150329485-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2015-11-19 | — | — | US | disclosed |
| US-20150329485-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2015-11-19 | — | — | US | disclosed |
| EP-2931703-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | Bayer CropScience AG (DE) | 2015-10-21 | — | — | EP | disclosed |
| US-9096635-B2 | N-alkylthio beta-lactams, alkyl-coenzyme A asymmetric disulfides, and aryl-alkyl disulfides as anti-bacterial agents | UNIVERSITY OF SOUTH FLORIDA (US) | 2015-08-04 | — | — | US | disclosed |
| US-9085540-B2 | Pyrazinecarboxamide compound | ASTELLAS PHARMA INC. (JP) | 2015-07-21 | — | — | US | disclosed |
| US-20150125489-A1 | METHOD FOR THE PREPARATION OF DENDRITIC CELL VACCINES | LABORATORIOS DEL DR. ESTEVE S.A. (ES) | 2015-05-07 | — | — | US | disclosed |
| CN-104530007-A | Preparation method of mono-substituted carbazolyl sulfide compound | UNIV HUNAN | 2015-04-22 | — | — | CN | disclosed |
| EP-2819696-A1 | METHOD FOR THE PREPARATION OF DENDRITIC CELL VACCINES | Laboratorios Del. Dr. Esteve, S.A. (ES) | 2015-01-07 | — | — | EP | disclosed |
| EP-2805940-A1 | PYRAZINE CARBOXAMIDE COMPOUND | Astellas Pharma Inc. (JP) | 2014-11-26 | — | — | EP | disclosed |
| US-20140323463-A1 | PYRAZINECARBOXAMIDE COMPOUND | ASTELLAS PHARMA INC. (JP) | 2014-10-30 | — | — | US | disclosed |
| WO-2014165196-A1 | DETECTION OF GAS-PHASE ANALYTES USING LIQUID CRYSTALS | PLATYPUS TECHNOLOGIES, LLC (US) | 2014-10-09 | — | — | WO | disclosed |
| CN-104080774-A | Pyrazine carboxamide compound | ASTELLAS PHARMA INC | 2014-10-01 | — | — | CN | disclosed |
| US-20140235565-A1 | N-ALKYLTHIO BETA-LACTAMS, ALKYL-COENZYME A ASYMMETRIC DISULFIDES, AND ARYL-ALKYL DISULFIDES AS ANTI-BACTERIAL AGENTS | UNIVERSITY OF SOUTH FLORIDA (US) | 2014-08-21 | — | — | US | disclosed |
| WO-2014090913-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | BAYER CROPSCIENCE AG (DE) | 2014-06-19 | — | — | WO | disclosed |
| US-8722937-B2 | Asymmetric disulfides and aryl-alkyl disulfides as anti-bacterial agents | UNIVERSITY OF SOUTH FLORIDA (US) | 2014-05-13 | — | — | US | disclosed |
| WO-2013127976-A1 | METHOD FOR THE PREPARATION OF DENDRITIC CELL VACCINES | LABORATORIOS DEL DR. ESTEVE, S.A. (ES) | 2013-09-06 | — | — | WO | disclosed |
| US-20120288951-A1 | DETECTION OF VAPOR PHASE COMPOUNDS BY CHANGES IN PHYSICAL PROPERTIES OF A LIQUID CRYSTAL | PLATYPUS TECHNOLOGIES, LLC (US) | 2012-11-15 | — | — | US | disclosed |
| US-20120122860-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | PLEXXIKON, INC. | 2012-05-17 | — | — | US | disclosed |
| US-20120122860-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | PLEXXIKON, INC. | 2012-05-17 | — | — | US | disclosed |
| US-20120122860-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | PLEXXIKON, INC. | 2012-05-17 | — | — | US | disclosed |
| US-8178355-B2 | Detection of vapor phase compounds by changes in physical properties of a liquid crystal | PLATYPUS TECHNOLOGIES, LLC. (US) | 2012-05-15 | — | — | US | disclosed |
| EP-2427433-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | Plexxikon, Inc. (US) | 2012-03-14 | — | — | EP | disclosed |
| EP-2344879-A2 | DETECTION OF VAPOR PHASE COMPOUNDS BY CHANGES IN PHYSICAL PROPERTIES OF A LIQUID CRYSTAL | Platypus Technologies, LLC (US) | 2011-07-20 | — | — | EP | disclosed |
| US-7871982-B2 | Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient | MEIJI SEIKA KAISHA, LTD. (JP) | 2011-01-18 | — | — | US | disclosed |
| US-7833331-B2 | Non-toxic corrosion-protection pigments based on cobalt | UNIVERSITY OF DAYTON (US) | 2010-11-16 | — | — | US | disclosed |
| WO-2010129570-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | PLEXXIKON, INC. (US) | 2010-11-11 | — | — | WO | disclosed |
| WO-2010129570-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | PLEXXIKON, INC. (US) | 2010-11-11 | — | — | WO | disclosed |
| EP-1225205-B1 | Carbon black reacted with diazonium salts and products | CABOT CORP (US) | 2010-10-06 | — | — | EP | disclosed |
| US-7789958-B2 | Non-toxic corrosion-protection pigments based on manganese | UNIVERSITY OF DAYTON (US) | 2010-09-07 | — | — | US | disclosed |
| US-20100144698-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2010-06-10 | — | — | US | disclosed |
| US-20100144698-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2010-06-10 | — | — | US | disclosed |
| US-20100144698-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2010-06-10 | — | — | US | disclosed |
| US-7732534-B2 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION (JP) | 2010-06-08 | — | — | US | disclosed |
| US-20100093096-A1 | DETECTION OF VAPOR PHASE COMPOUNDS BY CHANGES IN PHYSICAL PROPERTIES OF A LIQUID CRYSTAL | PLATYPUS TECHNOLOGIES, LLC (US) | 2010-04-15 | — | — | US | disclosed |
| EP-1942156-B1 | Carbon black reacted with diazonium salts and products | CABOT CORP (US) | 2010-04-14 | — | — | EP | disclosed |
| WO-2010031047-A2 | DETECTION OF VAPOR PHASE COMPOUNDS BY CHANGES IN PHYSICAL PROPERTIES OF A LIQUID CRYSTAL | PLATYPUS TECHNOLOGIES, LLC (US) | 2010-03-18 | — | — | WO | disclosed |
| US-7626027-B2 | Substituted 1H-pyrrolo[2,3-c]pyridine-2-carboxamides and related analogs as inhibitors of casein kinase Iε | AVENTIS PHARMACEUTICALS INC (US) | 2009-12-01 | — | — | US | disclosed |
| US-20090163628-A1 | NON-TOXIC CORROSION-PROTECTION PIGMENTS BASED ON COBALT | STURGILL JEFFREY ALLEN | 2009-06-25 | — | — | US | disclosed |
| US-20090156512-A1 | potent activity against resistant pneumococci | MEIJI SEIKA KAISHA, LTD. (JP) | 2009-06-18 | — | — | US | disclosed |
| US-20090143351-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2009-06-04 | — | — | US | disclosed |
| US-20090143351-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2009-06-04 | — | — | US | disclosed |
| US-20090143351-A1 | SUBSTITUTED AZETIDINONES | DAIAMED (US) | 2009-06-04 | — | — | US | disclosed |
| US-7541008-B2 | Fluid reactor | UNIVERSITY OF DURHAM OF UNIVERSITY OFFICE (GB) | 2009-06-02 | — | — | US | disclosed |
| US-7541008-B2 | Fluid reactor | UNIVERSITY OF DURHAM OF UNIVERSITY OFFICE (GB) | 2009-06-02 | — | — | US | disclosed |
| US-7541008-B2 | Fluid reactor | UNIVERSITY OF DURHAM OF UNIVERSITY OFFICE (GB) | 2009-06-02 | — | — | US | disclosed |
| EP-1747220-B1 | SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON | AVENTIS PHARMA INC (US) | 2009-04-15 | — | — | EP | disclosed |
| US-7501404-B2 | Substituted azetidinones | DAIMED (US) | 2009-03-10 | — | — | US | disclosed |
| US-7501404-B2 | Substituted azetidinones | DAIMED (US) | 2009-03-10 | — | — | US | disclosed |
| US-7501404-B2 | Substituted azetidinones | DAIMED (US) | 2009-03-10 | — | — | US | disclosed |
| EP-1809602-B1 | INDOLE DERIVATIVES USEFUL AS PROGESTERONE RECEPTOR MODULATORS | JANSSEN PHARMACEUTICA NV (BE) | 2008-10-29 | — | — | EP | disclosed |
| EP-1970377-A1 | LINCOMYCIN DERIVATIVE AND ANTIBACTERIAL AGENT CONTAINING THE SAME AS ACTIVE INGREDIENT | MEIJI SEIKA KAISHA LTD. (JP) | 2008-09-17 | — | — | EP | disclosed |
| US-7422793-B2 | Non-toxic corrosion-protection rinses and seals based on rare earth elements | UNIVERSITY OF DAYTON (US) | 2008-09-09 | — | — | US | disclosed |
| US-20080200496-A1 | SUBSTITUTED 1H-PYRROLO[3,2-b, 3,2-c, and 2,3-c]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE Ie | AVENTIS PHARMACEUTICALS INC. (US) | 2008-08-21 | — | — | US | disclosed |
| US-7407711-B2 | Non-toxic corrosion-protection conversion coats based on rare earth elements | UNIVERSITY OF DAYTON (US) | 2008-08-05 | — | — | US | disclosed |
| US-20080182815-A1 | Act against several infective agents, and most notably Bacillus spp. and Staphylococcus spp., including infection caused by methicillin-resistant Staphylococcus aureus (MRSA) | UNIVERSITY OF SOUTH FLORIDA | 2008-07-31 | — | — | US | disclosed |
| US-7402672-B2 | Substituted 1H-pyrrolo[3,2-b, 3,2-c, and 2,3-c]pyridine-2-carboxamides and related analogs as inhibitors of casein kinase lepsilon | AVENTIS PHARMACEUTICALS INC. (US) | 2008-07-22 | — | — | US | disclosed |
| EP-1942156-A1 | Carbon black reacted with diazonium salts and products | Cabot Corporation (US) | 2008-07-09 | — | — | EP | disclosed |
| US-20080139664-A1 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2008-06-12 | — | — | US | disclosed |
| US-20080099112-A1 | Reduced sensitivity melt-pourable Tritonal replacements | ALLIANT TECHSYSTEMS INC. | 2008-05-01 | — | — | US | disclosed |
| US-7345084-B2 | Indole derivatives useful as progesterone receptor modulators | JANSSEN PHARMACEUTICA N.V. (BE) | 2008-03-18 | — | — | US | disclosed |
| US-20080051552-A1 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION | 2008-02-28 | — | — | US | disclosed |
| US-20080051519-A1 | Polymers functionalized with nitro compounds | BRIDGESTONE CORPORATION (JP) | 2008-02-28 | — | — | US | disclosed |
| EP-1879900-A2 | SULFOXIMINE-PYRIMIDINE MACROCYCLES AND THE SALTS THEREOF, A PROCESS FOR MAKING THEM, AND THEIR PHARMACEUTICAL USE AGAINST CANCER | Bayer Schering Pharma Aktiengesellschaft (DE) | 2008-01-23 | — | — | EP | disclosed |
| EP-1011729-B1 | OLIGONUCLEOTIDES WHICH SPECIFICALLY BIND RETROVIRAL NUCLEOCAPSID PROTEINS | US GOV HEALTH & HUMAN SERV (US) | 2008-01-09 | — | — | EP | disclosed |
| EP-1871741-A2 | SUBSTITUTED AZETIDINONES | Daiamed, Inc. (US) | 2008-01-02 | — | — | EP | disclosed |
| US-7294211-B2 | Non-toxic corrosion-protection conversion coats based on cobalt | UNIVERSITY OF DAYTON (US) | 2007-11-13 | — | — | US | disclosed |
| US-7294185-B2 | In absence of exterior applies electrical current; wear resistance | CABOT CORPORATION (US) | 2007-11-13 | — | — | US | disclosed |
| US-7291217-B2 | Non-toxic corrosion-protection pigments based on rare earth elements | UNIVERSITY OF DAYTON (US) | 2007-11-06 | — | — | US | disclosed |
| EP-1809602-A1 | INDOLE DERIVATIVES USEFUL AS PROGESTERONE RECEPTOR MODULATORS | JANSSEN PHARMACEUTICA N.V. (BE) | 2007-07-25 | — | — | EP | disclosed |
| US-20070149673-A1 | NON-TOXIC CORROSION-PROTECTION PIGMENTS BASED ON MANGANESE | STURGILL JEFFREY A | 2007-06-28 | — | — | US | disclosed |
| US-7235142-B2 | Non-toxic corrosion-protection rinses and seals based on cobalt | UNIVERSITY OF DAYTON (US) | 2007-06-26 | — | — | US | disclosed |
| US-20070135511-A1 | INDOLE DERIVATIVES USEFUL AS PROGESTERONE RECEPTOR MODULATORS | JIANG WEIQIN | 2007-06-14 | — | — | US | disclosed |
| US-20070105832-A1 | Substituted azetidinones | Cadrenal Therapeutics, Inc. | 2007-05-10 | — | — | US | disclosed |
| US-20070105832-A1 | Substituted azetidinones | Cadrenal Therapeutics, Inc. | 2007-05-10 | — | — | US | disclosed |
| US-20070105832-A1 | Substituted azetidinones | Cadrenal Therapeutics, Inc. | 2007-05-10 | — | — | US | disclosed |
| US-7183309-B2 | Indole derivatives useful as progesterone receptor modulators | JANSSEN PHARMACEUTICA N.V. (BE) | 2007-02-27 | — | — | US | disclosed |
| EP-1747220-A1 | SUBSTITUTED 1H-PYRROLO 3,2-B, 3,2-C, AND 2,3-C¨PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON | Aventis Pharmaceuticals Inc. (US) | 2007-01-31 | — | — | EP | disclosed |
| US-20060252782-A1 | Sulfoximine-macrocycle compounds and salts thereof, pharmaceutical compositions comprising said compounds, methods of preparing same and uses of same | SCHERING AKTIENGESELLSCHAFT (DE) | 2006-11-09 | — | — | US | disclosed |
| WO-2006108695-A2 | SULFOXIMINE-PYRIMIDINE MACROCYCLES AND THE SALTS THEREOF , A PROCESS FOR MAKING THEM, AND THEIR PHARMACEUTICAL USE AGAINST CANCER | BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) | 2006-10-19 | — | — | WO | disclosed |
| WO-2006108039-A2 | SUBSTITUTED AZETIDINONES | DAIAMED, INC. (US) | 2006-10-12 | — | — | WO | disclosed |
| EP-1710246-A1 | Sulfoximine-pyrimidine Macrocycles and the salts thereof, a process for making them, and their pharmaceutical use against cancer | Schering Aktiengesellschaft (DE) | 2006-10-11 | — | — | EP | disclosed |
| US-7101676-B2 | Methods for identifying compounds which inhibit binding of nucleocapsid 7 protein to HIV-1 RNA | ACHILION PHARMACEUTICALS | 2006-09-05 | — | — | US | disclosed |
| US-7067024-B2 | Reduced sensitivity, melt-pourable TNT replacements | ALLIANT TECHSYSTEMS INC. (US) | 2006-06-27 | — | — | US | disclosed |
| US-20060111427-A1 | Indole derivatives useful as progesterone receptor modulators | JANSSEN PHARMACEUTICA N.V. (BE) | 2006-05-25 | — | — | US | disclosed |
| WO-2006049889-A1 | INDOLE DERIVATIVES USEFUL AS PROGESTERONE RECEPTOR MODULATORS | JANSSEN PHARMACEUTICA N.V. (BE) | 2006-05-11 | — | — | WO | disclosed |
| EP-0799281-B2 | CARBON BLACK REACTED WITH DIAZONIUM SALTS AND PRODUCTS | CABOT CORP (US) | 2006-03-29 | — | — | EP | disclosed |
| US-6989263-B1 | Method for identifying and using compounds that inactivate HIV-1 and other retroviruses by attacking highly conserved zinc fingers in the viral nucleocapsid protein | THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 2006-01-24 | — | — | US | disclosed |
| US-6984644-B2 | Treatment of skin disorders using thieno[2,3-D]pyrimidinediones | ASTRAZENECA AB (SE) | 2006-01-10 | — | — | US | disclosed |
| US-6964714-B2 | Reduced sensitivity, melt-pourable tritonal replacements | ALLIANT TECHSYSTEMS INC. (US) | 2005-11-15 | — | — | US | disclosed |
| US-6960688-B2 | Use of compounds for the elevation of pyruvate dehydrogenase activity | ASTRAZENECA AB (SE) | 2005-11-01 | — | — | US | disclosed |
| US-20050214184-A1 | Fluid reactor | UNIVERSITY OF DURHAM OF UNIVERSITY OFFICE (GB) | 2005-09-29 | — | — | US | disclosed |
| US-6943268-B2 | Method for induction of L-selectin shedding | SCIENCE & TECHNOLOGY CORPORATION @ UNM (US) | 2005-09-13 | — | — | US | disclosed |
| WO-2005061498-A1 | SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON | AVENTIS PHARMACEUTICALS INC. (US) | 2005-07-07 | — | — | WO | disclosed |
| US-20050131012-A1 | Substituted 1H-pyrrolo[3,2-b, 3,2-c, and 2,3-c]pyridine-2-carboxamides and related analogs as inhibitors of casein kinase lepsilon | AVENTIS PHARMACEUTICALS INC. (US) | 2005-06-16 | — | — | US | disclosed |
| US-20050043408-A1 | Anti-glycation agents for preventing age- diabetes- and smoking-related complications | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2005-02-24 | — | — | US | disclosed |
| US-20050034629-A1 | In absence of exterior applies electrical current; wear resistance | BELMONT JAMES A (US) | 2005-02-17 | — | — | US | disclosed |
| EP-1472319-A1 | NON-TOXIC CORROSION PROTECTION PIGMENTS BASED ON COBALT | UNIVERSITY OF DAYTON (US) | 2004-11-03 | — | — | EP | disclosed |
| WO-2004065305-A1 | NON-TOXIC CORROSION-PROTECTION PIGMENTS BASED ON MANGANESE | UNIVERSITY OF DAYTON (US) | 2004-08-05 | — | — | WO | disclosed |
| EP-1435930-A2 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2004-07-14 | — | — | EP | disclosed |
| US-20040104377-A1 | Non-toxic corrosion-protection pigments based on rare earth elements | UNIVERSITY OF DAYTON | 2004-06-03 | — | — | US | disclosed |
| US-6740151-B2 | IN THE ABSENCE OF AN EXTERNALLY APPLIED ELECTRIC CURRENT SUFFICIENT TO REDUCE THE DIAZONIUM SALT AND ATTACH AN ORGANIC GROUP; IMPROVED ABRASION RESISTANCE. | CABOT CORPORATION | 2004-05-25 | — | — | US | disclosed |
| EP-1399400-A1 | REDUCED SENSITIVITY, MELT-POURABLE TNT REPLACEMENTS | ALLIANT TECHSYSTEMS INC. (US) | 2004-03-24 | — | — | EP | disclosed |
| EP-1399399-A1 | REDUCED SENSITIVITY, MELT-POURABLE TRITONAL REPLACEMENTS | ALLIANT TECHSYSTEMS INC. (US) | 2004-03-24 | — | — | EP | disclosed |
| EP-1082110-B1 | USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY | ASTRAZENECA AB (SE) | 2004-03-24 | — | — | EP | disclosed |
| US-20040020568-A1 | Non-toxic corrosion-protection conversion coats based on rare earth elements | DAYTON, UNIVERSITY OF | 2004-02-05 | — | — | US | disclosed |
| WO-2004009114-A1 | METHOD FOR DISCOVERING SUBSTANCES FOR INHIBITING ENZYMES | PHARMACIA & UPJOHN COMPANY (US) | 2004-01-29 | — | — | WO | disclosed |
| US-20040016910-A1 | Non-toxic corrosion-protection rinses and seals based on rare earth elements | DAYTON, UNIVERSITY OF | 2004-01-29 | — | — | US | disclosed |
| US-20040018581-A1 | Method for discovering substances for inhibiting enzymes | PHARMACIA AND UPJOHN COMPANY | 2004-01-29 | — | — | US | disclosed |
| US-20040011252-A1 | Non-toxic corrosion-protection pigments based on manganese | UNIVERSITY OF DAYTON | 2004-01-22 | — | — | US | disclosed |
| US-20040009979-A1 | Use of compounds for the elevation of pyruvate dehydrogenase activity | ZENECA LIMITED | 2004-01-15 | — | — | US | disclosed |
| US-20030234063-A1 | Non-toxic corrosion-protection conversion coats based on cobalt | DAYTON, UNIVERSITY OF | 2003-12-25 | — | — | US | disclosed |
| US-20030230363-A1 | Non-toxic corrosion-protection rinses and seals based on cobalt | UNIVERSITY OF DAYTON | 2003-12-18 | — | — | US | disclosed |
| WO-2003095086-A2 | FLUID REACTOR | THE UNIVERSITY OF DURHAM (GB) | 2003-11-20 | — | — | WO | disclosed |
| US-20030198648-A1 | Methods for identifying compounds which inhibit binding of nucleocapsid 7 protein to HIV-1 RNA | ACHILION PHARMACEUTICALS | 2003-10-23 | — | — | US | disclosed |
| US-20030191142-A1 | Thieno[2,3-d]pyrimidinediones, their preparation and use in therapy | ASTRAZENECA AB | 2003-10-09 | — | — | US | disclosed |
| US-20030140993-A1 | Reduced sensitivity, melt-pourable tritonal replacements | NORTHROP GRUMMAN SYSTEMS CORPORATION | 2003-07-31 | — | — | US | disclosed |
| WO-2003060191-A2 | NON-TOXIC CORROSION-PROTECTION CONVERSION COATINGES ABSED ON COBALT | UNIVERSITY OF DAYTON (US) | 2003-07-24 | — | — | WO | disclosed |
| WO-2003060192-A1 | NON-TOXIC CORROSION-PROTECTION RINSES AND SEALS BASED ON COBALT | UNIVERSITY OF DAYTON (US) | 2003-07-24 | — | — | WO | disclosed |
| WO-2003060098-A2 | METHODS FOR IDENTIFYING COMPOUNDS WHICH INHIBIT BINDING OF NUCLEOCAPSID 7 PROTEIN TO HIV-1 RNA | ACHILLION PHARMACEUTICALS, INC. (US) | 2003-07-24 | — | — | WO | disclosed |
| WO-2003060019-A1 | NON-TOXIC CORROSION PROTECTION PIGMENTS BASED ON COBALT | UNIVERSITY OF DAYTON (US) | 2003-07-24 | — | — | WO | disclosed |
| US-20030095914-A1 | In the absence of an externally applied electric current sufficient to reduce the diazonium salt and attach an organic group; improved abrasion resistance. | BELMONT JAMES A (US) | 2003-05-22 | — | — | US | disclosed |
| US-20030092763-A1 | Method for induction of L-selectin shedding | SCIENCE & TECHNOLOGY CORPORATION @UNM | 2003-05-15 | — | — | US | disclosed |
| WO-2003032969-A2 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | NATIONAL RESEARCH COUNCIL OF CANADA (CA) | 2003-04-24 | — | — | WO | disclosed |
| EP-0782632-B1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | US GOV HEALTH & HUMAN SERV (US) | 2003-04-16 | — | — | EP | disclosed |
| WO-2003002486-A1 | REDUCED SENSITIVITY, MELT-POURABLE TNT REPLACEMENTS | ALLIANT TECHSYSTEMS INC. (US) | 2003-01-09 | — | — | WO | disclosed |
| WO-2003002485-A1 | REDUCED SENSITIVITY, MELT-POURABLE TRITONAL REPLACEMENTS | ALLIANT TECHSYSTEMS INC. (US) | 2003-01-09 | — | — | WO | disclosed |
| US-20030005988-A1 | Reduced sensitivity, melt-pourable TNT replacements | NORTHROP GRUMMAN SYSTEMS CORPORATION | 2003-01-09 | — | — | US | disclosed |
| US-6498275-B1 | Use of compounds for the elevation of pyruvate dehydrogenase activity | ASTRAZENECA AB (SE) | 2002-12-24 | — | — | US | disclosed |
| US-6498189-B1 | SUPPRESSION OF INFLAMMATION AND OF LYMPH NODE ENTRY BY CALMODULIN ANTAGONISTS; CELL ASSOCIATED PROTEIN DISULFIDE ISOMERASE INHIBITORS; P-AMINOPHENYLARSINE OXIDES | UNIVERSITY OF NEW MEXICO | 2002-12-24 | — | — | US | disclosed |
| US-6494946-B1 | PROCESSES FOR PREPARING A CARBON BLACK PRODUCT HAVING AN ORGANIC GROUP ATTACHED TO THE CARBON BLACK. IN ONE PROCESS AT LEAST ONE DIAZONIUM SALT REACTS WITH A CARBON BLACK IN THE ABSENCE OF AN EXTERNALLY APPLIED ELECTRIC CURRENT SUFFICIENT | CABOT CORPORATION | 2002-12-17 | — | — | US | disclosed |
| US-20020183337-A1 | For use in immunosuppression; for reducing the risk of, a reversible obstructive airways disease | ASTRAZENECA AB. | 2002-12-05 | — | — | US | disclosed |
| US-6469014-B1 | IMMUNOSUPPRESSIVE ACTIVITY | ASTRAZENECA AB (SE) | 2002-10-22 | — | — | US | disclosed |
| EP-0991653-B1 | NOVEL COMPOUNDS | ASTRAZENECA AB (SE) | 2002-10-16 | — | — | EP | disclosed |
| US-6432294-B1 | ELECTROCHEMICAL OXIDATION OF DISULFIDES IN ARENE SOLUTIONS FOR SYNTHESIS OF ORGANOTHIATED PRODUCT | THE UNIVERSITY OF ARIZONA | 2002-08-13 | — | — | US | disclosed |
| EP-0799281-B1 | CARBON BLACK REACTED WITH DIAZONIUM SALTS AND PRODUCTS | CABOT CORP (US) | 2002-07-24 | — | — | EP | disclosed |
| EP-1225205-A2 | Carbon black reacted with diazonium salts and products | CABOT CORPORATION (US) | 2002-07-24 | — | — | EP | disclosed |
| US-6342502-B1 | ANTIASTHMATICS | ASTRAZENECA AB (GB) | 2002-01-29 | — | — | US | disclosed |
| US-6316190-B1 | FOR DETECTING OR PURIFYING HUMAN IMMUNODEFICIENCY VIRUS(HIV) FROM BLOOD SAMPLE | THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES | 2001-11-13 | — | — | US | disclosed |
| CN-1303281-A | Application of compound in enhancing activity of pyruvate dehydrogenase | ASTRA ZENECA LTD (SE) | 2001-07-11 | — | — | CN | disclosed |
| US-6207838-B1 | ELECTROLYSIS IN LIQUID SULFUR DIOXIDE | THE UNIVERSITY OF ARIZONA | 2001-03-27 | — | — | US | disclosed |
| EP-1082110-A1 | USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY | AstraZeneca AB (SE) | 2001-03-14 | — | — | EP | disclosed |
| US-6180635-B1 | NOVEL THIENO(2,3-D)PYRIMIDINEDIONES WHICH EXHIBIT PHARMACOLOGICAL ACTIVITY, IN PARTICULAR IMMUNOSUPPRESSIVE ACTIVITY; TREATING ALLOGRAFT REJECTION | ASTRAZENECA UK LIMITED (GB) | 2001-01-30 | — | — | US | disclosed |
| EP-1048752-A2 | Electrochemically generated organothiating reagents and their use | ALBEMARLE CORPORATION (US) | 2000-11-02 | — | — | EP | disclosed |
| EP-1011729-A2 | OLIGONUCLEOTIDES WHICH SPECIFICALLY BIND RETROVIRAL NUCLEOCAPSID PROTEINS | THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 2000-06-28 | — | — | EP | disclosed |
| EP-0991653-A1 | NOVEL COMPOUNDS | Astra Pharmaceuticals Limited (GB) | 2000-04-12 | — | — | EP | disclosed |
| US-6042643-A | AS PIGMENT TO COLOR PLASTICS, PAPER, TEXTILE, RUBBER, AQUEOUS INKS | CABOT CORPORATION (US) | 2000-03-28 | — | — | US | disclosed |
| EP-0590885-B1 | Antibiotic carbapenem compounds | ZENECA LTD (GB) | 2000-03-15 | — | — | EP | disclosed |
| US-6001555-A | DISSOCIATING A ZINC FINGER BY CONTACTING THE PROTEIN WITH A DISULFIDE, A MALEIMIDE, AN ALPHA-HALOGENATED KETONE, A HYDRAZIDE, A NITRIC OXIDE OR DERIVATIVES, CUPRIC IONS, FERRIC IONS OR THEIR COMPLEXES; SYNERGISTIC EFFECTS WITH VIRICIDES | THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1999-12-14 | — | — | US | disclosed |
| WO-1999062506-A1 | USE OF COMPOUNDS FOR THE ELEVATION OF PYRUVATE DEHYDROGENASE ACTIVITY | ASTRAZENECA AB (SE) | 1999-12-09 | — | — | WO | disclosed |
| EP-0784614-B1 | THE PREPARATION OF FLUORINATED ORGANIC COMPOUNDS | F2 CHEMICALS LIMITED (GB) | 1999-10-06 | — | — | EP | disclosed |
| US-5900029-A | COLORING FIBER OR TEXTILE | CABOT CORPORATION (US) | 1999-05-04 | — | — | US | disclosed |
| US-5851280-A | Reaction of carbon black with diazonium salts, resultant carbon black products and their uses | CABOT CORPORATION (US) | 1998-12-22 | — | — | US | disclosed |
| WO-1998054190-A1 | NOVEL COMPOUNDS | ASTRA PHARMACEUTICALS LTD. (GB) | 1998-12-03 | — | — | WO | disclosed |
| US-5821263-A | ANTICARCINOGENIC AGENT; CHARACTERIZED BY C3' NITROGEN BEARING ONE OR TWO SULFUR SUBSTITUENTS | BRISTOL-MYERS SQUIBB COMPANY (US) | 1998-10-13 | — | — | US | disclosed |
| US-5741935-A | Preparation of organic pentafluorosulphur compounds | BRITISH NUCLEAR FUELS PLC (GB) | 1998-04-21 | — | — | US | disclosed |
| WO-1998008833-A1 | SULFENAMIDE TAXANE DERIVATIVES | BRISTOL-MYERS SQUIBB COMPANY (US) | 1998-03-05 | — | — | WO | disclosed |
| WO-1997044064-A2 | OLIGONUCLEOTIDES WHICH SPECIFICALLY BIND RETROVIRAL NUCLEOCAPSID PROTEINS | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1997-11-27 | — | — | WO | disclosed |
| EP-0799281-A1 | CARBON BLACK REACTED WITH DIAZONIUM SALTS AND PRODUCTS | CABOT CORPORATION (US) | 1997-10-08 | — | — | EP | disclosed |
| US-5663164-A | CEPHALOSPORIN ANTIBIOTICS AS BACTERICIDES | ROUSSEL UCLAF (FR) | 1997-09-02 | — | — | US | disclosed |
| EP-0784614-A1 | THE PREPARATION OF FLUORINATED ORGANIC COMPOUNDS | British Nuclear Fuels PLC (GB) | 1997-07-23 | — | — | EP | disclosed |
| EP-0782632-A1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the Secretary of the Department of Health and Human Services (US) | 1997-07-09 | — | — | EP | disclosed |
| WO-1997005106-A1 | THE PREPARATION OF FLUORINATED ORGANIC COMPOUNDS | BRITISH NUCLEAR FUELS PLC (GB) | 1997-02-13 | — | — | WO | disclosed |
| WO-1996018688-A1 | CARBON BLACK REACTED WITH DIAZONIUM SALTS AND PRODUCTS | CABOT CORPORATION (US) | 1996-06-20 | — | — | WO | disclosed |
| US-5527791-A | Carbapenem antibiotic compounds | ZENECA LIMITED (GB) | 1996-06-18 | — | — | US | disclosed |
| WO-1996009406-A9 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | — | 1996-05-23 | — | — | WO | disclosed |
| WO-1996009406-A1 | A METHOD FOR IDENTIFYING AND USING COMPOUNDS THAT INACTIVATE HIV-1 AND OTHER RETROVIRUSES BY ATTACKING HIGHLY CONSERVED ZINC FINGERS IN THE VIRAL NUCLEOCAPSID PROTEIN | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) | 1996-03-28 | — | — | WO | disclosed |
| EP-0693056-A1 | PROCESS FOR THE PREPARATION OF ARYL- AND HETEROARYLSULPHURPENTAFLUORIDES | ZENECA LIMITED (GB) | 1996-01-24 | — | — | EP | disclosed |
| EP-0489360-B1 | Water-soluble azocompounds, process for their preparation and their use as dyes | HOECHST AG (DE) | 1995-09-20 | — | — | EP | disclosed |
| WO-1994022817-A1 | PROCESS FOR THE PREPARATION OF ARYL- AND HETEROARYLSULPHURPENTAFLUORIDES | ZENECA LIMITED (GB) | 1994-10-13 | — | — | WO | disclosed |
| EP-0590885-A1 | Antibiotic carbapenem compounds | ZENECA LIMITED (GB) | 1994-04-06 | — | — | EP | disclosed |
| US-5300633-A | Lightfast, washfast | HOECHST AKTIENGESELLSCHAFT (DE) | 1994-04-05 | — | — | US | disclosed |
| US-5216138-A | With vinyl sulfonyl group | HOECHST AKTIENGESELLSCHAFT (DE) | 1993-06-01 | — | — | US | disclosed |
| EP-0513657-A2 | Water-soluble azo compounds, process for their preparation and their use as dyes | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-11-19 | — | — | EP | disclosed |
| EP-0489360-A1 | Water-soluble azocompounds, process for their preparation and their use as dyes | HOECHST AKTIENGESELLSCHAFT (DE) | 1992-06-10 | — | — | EP | disclosed |
| CN-1034012-A | A kind of synthesis method of reactive blue dye | DALIAN POLYTECHNICAL COLLEGE (CN) | 1989-07-19 | — | — | CN | disclosed |
| JP-H01165586-A | ANTI TUMOR PRODRUG | BRISTOL MYERS CO | 1989-06-29 | — | — | JP | disclosed |
| EP-0317956-A2 | Anti-tumor prodrugs | Bristol-Myers Squibb Company (US) | 1989-05-31 | — | — | EP | disclosed |
| US-4826851-A | 2-substituted ergoline urea and thio-urea derivatives having neurolyptic/dopaminergic activity | SCHERING AKTIENGESELLSCHAFT (DE) | 1989-05-02 | — | — | US | disclosed |
| EP-0217735-A2 | 2-Substituted ergoline derivatives | SCHERING AKTIENGESELLSCHAFT (DE) | 1987-04-08 | — | — | EP | disclosed |
| US-4656290-A | Process for preparing thio, dithio or carbonyl compounds | CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) | 1987-04-07 | — | — | US | disclosed |
| EP-0150026-A2 | Chemical process | CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) | 1985-07-31 | — | — | EP | disclosed |
| US-4504568-A | Sensitive silver halide photothermographic materials for producing dye images | EASTMAN KODAK COMPANY (US) | 1985-03-12 | — | — | US | disclosed |
| EP-0025339-B1 | MICROBICIDAL SULFONES, COMPOSITIONS THEREOF AND METHODS OF PREPARING THEM | UNIROYAL, INC. (US) | 1984-05-30 | — | — | EP | disclosed |
| EP-0093363-A1 | Process for the preparation of disulphides | CASSELLA Aktiengesellschaft (DE) | 1983-11-09 | — | — | EP | disclosed |
| EP-0086774-A1 | TREATMENT OF COCCIDIAL INFECTIONS WITH AMIDINOUREA OR AMIDINOTHIOUREA DERIVATIVES | RORER INTERNATIONAL (OVERSEAS) INC. (US) | 1983-08-31 | — | — | EP | disclosed |
| WO-1983000625-A1 | TREATMENT OF COCCIDIAL INFECTIONS WITH AMIDINOUREA OR AMIDINOTHIOUREA DERIVATIVES | STUDT, WILLIAM, LYON | 1983-03-03 | — | — | WO | disclosed |
| US-4335142-A | MICROBIOCIDES | UNIROYAL, INC. (US) | 1982-06-15 | — | — | US | disclosed |
| EP-0035393-A1 | Poultry feeds containing and methods of using anovulatory compounds, and novel anovulatory imidazolines | MERCK & CO. INC. (US) | 1981-09-09 | — | — | EP | disclosed |
| US-4287201-A | CONTAINING A 2-(SUBSTITUTED PHENYLIMINO)IMIDAZOLIDINE COMPOUND | MERCK & CO., INC. (US) | 1981-09-01 | — | — | US | disclosed |
| US-4286964-A | Polyfunctional epoxides and halohydrins used as bridging groups to bind aromatic amine group-containing alcohols and thiols to hydroxyl bearing substrates | SEED BRIAN S | 1981-09-01 | — | — | US | disclosed |
| JP-S5643338-A | SCORCH RETARDER FOR HALOGEN-CONTAINING POLYMER RUBBER AND PREVENTION OF SCORCH OF SAID RUBBER | SANSHIN KAGAKU KOGYO KK | 1981-04-22 | — | — | JP | disclosed |
| EP-0027377-A1 | Derivatives of hydroxyl-bearing substrates, process for their preparation and a method of application | Seed, Brian Sarsfield (US) | 1981-04-22 | — | — | EP | disclosed |
| EP-0025339-A1 | Microbicidal sulfones, compositions thereof and methods of preparing them | UNIROYAL, INC. (US) | 1981-03-18 | — | — | EP | disclosed |
| US-4130661-A | ANTICOCCIDIAL | MERCK & CO., INC. (US) | 1978-12-19 | — | — | US | disclosed |
| US-4098893-A | PYRIDINE DERIVATIVES AND THEIR USE AS ANTICOCCIDIAL AGENTS | SANKYO COMPANY LIMITED (JP) | 1978-07-04 | — | — | US | disclosed |
| US-4094982-A | PYRIDINE SULFONAMIDES AND THEIR USE AS ANTICOCCIDIAL AGENTS | SANKYO COMPANY LIMITED (JA) | 1978-06-13 | — | — | US | disclosed |
| US-4083984-A | 1-Substituted phenyl-4(1H)-pyridinone hydrazones and composition therewith for treatment of coccidiosis | MERCK & CO., INC. (US) | 1978-04-11 | — | — | US | disclosed |
| US-4079069-A | ANTIPROTOZOAL, ANTIPARASITIC | MERCK & CO., INC. (US) | 1978-03-14 | — | — | US | disclosed |
| US-4073791-A | ANTICOCCIDIAL | MERCK & CO., INC. (US) | 1978-02-14 | — | — | US | disclosed |
| US-4054663-A | POULTRY FEEDS | SANKYO COMPANY LIMITED (JA) | 1977-10-18 | — | — | US | disclosed |
| US-4053608-A | 3-NITROPYRIDINE CARBOXAMIDES, POULTRY FEED | SANKYO COMPANY LIMITED (JA) | 1977-10-11 | — | — | US | disclosed |
| US-4053602-A | POULTRY FEED; ANTIPROTOZOAL, ANTIPARASITIC | MERCK & CO., INC. (US) | 1977-10-11 | — | — | US | disclosed |
| US-4044133-A | FEED SUPPLEMENT, POULTRY, THIENO-PYRIDINE, OR FURO-PYRIDINE BASE N | MERCK & CO., INC. (US) | 1977-08-23 | — | — | US | disclosed |
| US-4006143-A | COCCIDIOSTATS | MERCK & CO., INC. (US) | 1977-02-01 | — | — | US | disclosed |
| US-3994724-A | SUBSTITUTED ANILINE PHOTOCONDUCTOR | SCOTT PAPER COMPANY (US) | 1976-11-30 | — | — | US | disclosed |
| US-3991185-A | Methods for treating coccidiosis with emimycin and its derivatives | MERCK & CO., INC. (US) | 1976-11-09 | — | — | US | disclosed |
| US-3983238-A | Substituted pyridinol-containing compositions and methods for the treatment of coccidiosis | SANKYO COMPANY LIMITED (JA) | 1976-09-28 | — | — | US | disclosed |
| US-3957997-A | Anticoccidial complexes of 4,4'-dinitrocarbanilides | MERCK & CO., INC. (US) | 1976-05-18 | — | — | US | disclosed |
| US-3935311-A | Substitute pyridinol-containing compositions and methods for the treatment of coccidiosis | SANKYO COMPANY LIMITED (JA) | 1976-01-27 | — | — | US | disclosed |
| US-3935311-A | Substitute pyridinol-containing compositions and methods for the treatment of coccidiosis | SANKYO COMPANY LIMITED (JA) | 1976-01-27 | — | — | US | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (28 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-20070105832-A1 | Substituted azetidinones | F2R, CPA3, CFD | HSP90AA1 4432/4885TSHR 414/4885LMNA 1127/4885 |
| US-20080182815-A1 | Act against several infective agents, and most notably Bacillus spp. and Staphylococcus spp., including infection caused by methicillin-resistant Staphylococcus aureus (MRSA) | SQOR, TST, COASY | HSP90AA1 427/4885TSHR 4113/4885LMNA 2815/4885 |
| US-20050043408-A1 | Anti-glycation agents for preventing age- diabetes- and smoking-related complications | AGER, GID4, GALE | HSP90AA1 1444/4885TSHR 4241/4885LMNA 509/4885 |
| US-20120122860-A1 | SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS | BRAF, RAF1, ARAF | HSP90AA1 550/4885TSHR 2679/4885LMNA 3902/4885 |
| US-20080139664-A1 | ANTI-GLYCATION AGENTS FOR PREVENTING AGE-, DIABETES-, AND SMOKING-RELATED COMPLICATIONS | AGER, GID4, GALE | HSP90AA1 1439/4885TSHR 4320/4885LMNA 479/4885 |
| US-20160160178-A1 | IMMUNOTHERAPY USING STEM CELLS | CD14, ICOS, BMP4 | HSP90AA1 1615/4885TSHR 1550/4885LMNA 2622/4885 |
| US-20230278965-A1 | NOVEL CARBONOHYDRAZONOYL DICYANIDE COMPOUNDS COMPRISING 2 OR MORE ARYL OR HETEROARYL CONNECTED VIA LINKER AND USE THEREOF | AADAC, CBR3, MTCL3 | HSP90AA1 3895/4885TSHR 4231/4885LMNA 2555/4885 |
| US-20040009979-A1 | Use of compounds for the elevation of pyruvate dehydrogenase activity | PDHA1, PDK1, PDHB | HSP90AA1 483/4885TSHR 3602/4885LMNA 1594/4885 |
| US-20080200496-A1 | SUBSTITUTED 1H-PYRROLO[3,2-b, 3,2-c, and 2,3-c]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE Ie | CSNK1E, CSNK1G3, CSNK2A3 | HSP90AA1 4163/4885TSHR 3252/4885LMNA 589/4885 |
| US-20140323463-A1 | PYRAZINECARBOXAMIDE COMPOUND | EGFR, ERBB2, ALK | HSP90AA1 3176/4885TSHR 2449/4885LMNA 4103/4885 |
| US-20150125489-A1 | METHOD FOR THE PREPARATION OF DENDRITIC CELL VACCINES | CCR7, CD69, CD14 | HSP90AA1 622/4885TSHR 4841/4885LMNA 1497/4885 |
| US-20150327547-A1 | N-ALKYLTHIO BETA-LACTAMS, ALKYL-COENZYME A ASYMMETRIC DISULFIDES, AND ARYL-ALKYL DISULFIDES AS ANTI-BACTERIAL AGENTS | COASY, SQOR, TST | HSP90AA1 959/4885TSHR 4071/4885LMNA 2590/4885 |
| US-20100144698-A1 | SUBSTITUTED AZETIDINONES | F2R, CPA3, CFD | HSP90AA1 4432/4885TSHR 414/4885LMNA 1127/4885 |
| US-20090156512-A1 | potent activity against resistant pneumococci | H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, NAT1, NPM1 | HSP90AA1 1581/4885TSHR 1003/4885LMNA 48/4885 |
| US-20020183337-A1 | For use in immunosuppression; for reducing the risk of, a reversible obstructive airways disease | TPMT, TSLP, TYMP | HSP90AA1 3318/4885TSHR 3760/4885LMNA 4754/4885 |
| US-20050131012-A1 | Substituted 1H-pyrrolo[3,2-b, 3,2-c, and 2,3-c]pyridine-2-carboxamides and related analogs as inhibitors of casein kinase lepsilon | CSNK2A3, PACSIN2, CSNK1G3 | HSP90AA1 4403/4885TSHR 2103/4885LMNA 342/4885 |
| US-20180258036-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | GSS, QSOX1, SQOR | HSP90AA1 947/4885TSHR 3827/4885LMNA 3832/4885 |
| US-20070135511-A1 | INDOLE DERIVATIVES USEFUL AS PROGESTERONE RECEPTOR MODULATORS | PRLHR, GNRHR, ADCYAP1R1 | HSP90AA1 2502/4885TSHR 230/4885LMNA 1228/4885 |
| US-20060252782-A1 | Sulfoximine-macrocycle compounds and salts thereof, pharmaceutical compositions comprising said compounds, methods of preparing same and uses of same | TEK, FLT1, TIE1 | HSP90AA1 4752/4885TSHR 1194/4885LMNA 4670/4885 |
| US-10239831-B2 | Method for producing bis(3-aminophenyl)disulfides and 3-aminothiols | GSS, QSOX1, SQOR | HSP90AA1 947/4885TSHR 3827/4885LMNA 3832/4885 |
| US-20140235565-A1 | N-ALKYLTHIO BETA-LACTAMS, ALKYL-COENZYME A ASYMMETRIC DISULFIDES, AND ARYL-ALKYL DISULFIDES AS ANTI-BACTERIAL AGENTS | COASY, SQOR, TST | HSP90AA1 959/4885TSHR 4071/4885LMNA 2590/4885 |
| US-20090143351-A1 | SUBSTITUTED AZETIDINONES | F2R, CPA3, CFD | HSP90AA1 4432/4885TSHR 414/4885LMNA 1127/4885 |
| US-20060111427-A1 | Indole derivatives useful as progesterone receptor modulators | PRLHR, GNRHR, ADCYAP1R1 | HSP90AA1 2502/4885TSHR 230/4885LMNA 1228/4885 |
| US-20150329485-A1 | METHOD FOR PRODUCING BIS(3-AMINOPHENYL)DISULFIDES AND 3-AMINOTHIOLS | GSS, QSOX1, SQOR | HSP90AA1 947/4885TSHR 3827/4885LMNA 3832/4885 |
| US-20030191142-A1 | Thieno[2,3-d]pyrimidinediones, their preparation and use in therapy | TYMP, DPYD, TYMS | HSP90AA1 2700/4885TSHR 1938/4885LMNA 4234/4885 |
| US-20030198648-A1 | Methods for identifying compounds which inhibit binding of nucleocapsid 7 protein to HIV-1 RNA | MRPS27, SNRPE, NSUN2 | HSP90AA1 2171/4885TSHR 4796/4885LMNA 2733/4885 |
| US-10053421-B2 | Method for producing bis(3-aminophenyl)disulfides and 3-aminothiols | GSS, QSOX1, SQOR | HSP90AA1 947/4885TSHR 3827/4885LMNA 3832/4885 |
| US-20030092763-A1 | Method for induction of L-selectin shedding | PDIA5, PDIA4, PDIA6 | HSP90AA1 1036/4885TSHR 4422/4885LMNA 4121/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.