Hydrochloric Acid

Hydrochloric Acid

SCHEMBL3180076

COc1c(Cl)ccnc1CCl.Cl

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Hydrochloric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA known ✓ P21397 1/20 0.36
GLA known ✓ P06280 1/20 0.32
ADRA1A known ✓ P35348 1/20 0.31
CCR5 known ✓ P51681 1/20 0.31
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
HSD17B10 Q99714 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
BLM P54132 1/20 0.32
CASP6 P55212 1/20 0.32
PMP22 Q01453 1/20 0.32
HIF1A Q16665 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30557385 0.98 ALDH1A1 (0.35) MAOARAB9AALDH1A1KDM4EHSD17B10
SCHEMBL1178052 0.98 ALDH1A1 (0.35) MAOARAB9AALDH1A1KDM4EHSD17B10
Hydrochloric Acid SCHEMBL3186456 0.88
Hydrochloric Acid SCHEMBL5268510 0.85 ALDH1A1 (0.38) MAOARAB9AALDH1A1KDM4EHSD17B10
SCHEMBL8710507 0.83 TAS1R3 (0.36) MAOARAB9AALDH1A1KDM4EHSD17B10
SCHEMBL3170691 0.83 ALDH1A1 (0.39) MAOARAB9AALDH1A1KDM4EHSD17B10
SCHEMBL25384445 0.81 LOX (0.41) MAOARAB9AALDH1A1KDM4EHSD17B10
SCHEMBL7104913 0.81 ALDH1A1 (0.34) MAOARAB9AALDH1A1KDM4EHSD17B10
Hydrochloric Acid SCHEMBL1002426 0.81 RAB9A (0.43) MAOARAB9AALDH1A1KDM4ESMN1; SMN2
SCHEMBL8840465 0.81 ALDH1A1 (0.34) MAOARAB9AALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100022779-A1 Isotopically substituted proton pump inhibitors NYCOMED GMBH (DE) 2010-01-28 US disclosed
US-20100010047-A1 Isotopically substituted proton pump inhibitors TAKEDA GMBH (DE) 2010-01-14 US disclosed
US-7601737-B2 2-Pyridinyl)methylsulfinyl]-1H-benzimidazole derivatives; substituents include methoxy and difluoromethoxy; at least one alkyl hydrogen is replaced by a deuterium atom: 5-difluoromethoxy-2-[(3-methoxy-4-monodeuteriomethoxy)-2-pyridinyl)methylsulfinyl]-1H-benzimidazole; gastrointestinal disorders NYCOMED GMBH (DE) 2009-10-13 US disclosed
US-20080146610-A1 2-Pyridinyl)methylsulfinyl]-1H-benzimidazole derivatives; substituents include methoxy and difluoromethoxy; at least one alkyl hydrogen is replaced by a deuterium atom: 5-difluoromethoxy-2-[(3-methoxy-4-monodeuteriomethoxy)-2-pyridinyl)methylsulfinyl]-1H-benzimidazole; gastrointestinal disorders NYCOMED GMBH (DE) 2008-06-19 US disclosed
EP-1912947-A1 ISOTOPICALLY SUBSTITUTED PANTOPRAZOLE Nycomed GmbH (DE) 2008-04-23 EP disclosed
EP-1910293-A1 ISOTOPICALLY SUBSTITUTED PROTON PUMP INHIBITORS Nycomed GmbH (DE) 2008-04-16 EP disclosed
WO-2007012651-A1 ISOTOPICALLY SUBSTITUTED PANTOPRAZOLE NYCOMED GMBH (DE) 2007-02-01 WO disclosed
WO-2007012650-A1 ISOTOPICALLY SUBSTITUTED PROTON PUMP INHIBITORS NYCOMED GMBH (DE) 2007-02-01 WO disclosed
US-6884810-B2 Benzimidazole derivatives ZERIA PHARMACEUTICAL CO., LTD. (JP) 2005-04-26 US disclosed
EP-1428825-A1 BENZIMIDAZOLE DERIVATIVES Zeria Pharmaceutical Co., Ltd. (JP) 2004-06-16 EP disclosed
US-20030236411-A1 Benzimidazole derivatives ZERIA PHARMACEUTICAL CO., LTD. (JP) 2003-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022779-A1 Isotopically substituted proton pump inhibitors SLC10A2, ABCB11, SLC10A1 MAOA 1435/4885GLA 2170/4885ADRA1A 1317/4885
US-20080146610-A1 2-Pyridinyl)methylsulfinyl]-1H-benzimidazole derivatives; substituents include methoxy and difluoromethoxy; at least one alkyl hydrogen is replaced by a deuterium atom: 5-difluoromethoxy-2-[(3-methoxy-4-monodeuteriomethoxy)-2-pyridinyl)methylsulfinyl]-1H-benzimidazole; gastrointestinal disorders SLC10A2, CYP2J2, CYP2D6 MAOA 1499/4885GLA 3599/4885ADRA1A 1687/4885
US-20100010047-A1 Isotopically substituted proton pump inhibitors SLC10A2, ABCB11, SLC10A1 MAOA 1435/4885GLA 2170/4885ADRA1A 1317/4885
US-20030236411-A1 Benzimidazole derivatives CYP2E1, CYP1A1, CYP1B1 MAOA 195/4885GLA 3511/4885ADRA1A 300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.