SCHEMBL366066

SCHEMBL366066

Cc1ccc([C@@H](O)C(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.62
MAPK1 P28482 1/20 0.62
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
BLM P54132 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ACHE P22303 1/20 0.42
ALOX5 P09917 1/20 0.42
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
POLB P06746 1/20 0.42
SRD5A2 P31213 1/20 0.41
HPGD P15428 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
PSMB5 P28074 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245404 1.00 LMNA (0.62) LMNAMAPK1KEAP1NFE2L2BLM
SCHEMBL245405 1.00 LMNA (0.62) LMNAMAPK1KEAP1NFE2L2BLM
SCHEMBL11835765 0.94 LMNA (0.56) LMNAMAPK1KEAP1NFE2L2BLM
D-Alanine SCHEMBL11208357 0.90 LMNA (0.52) LMNAMAPK1KEAP1NFE2L2BLM
D-Alanine SCHEMBL11207612 0.90 LMNA (0.52) LMNAMAPK1KEAP1NFE2L2BLM
Alanine SCHEMBL11209772 0.90 LMNA (0.52) LMNAMAPK1KEAP1NFE2L2BLM
Alanine SCHEMBL11204313 0.90 LMNA (0.52) LMNAMAPK1KEAP1NFE2L2BLM
D-Alanine SCHEMBL11496478 0.88 LMNA (0.50) LMNAMAPK1KEAP1NFE2L2BLM
SCHEMBL275597 0.87 LMNA (0.79) LMNAMAPK1BLMNPSR1TSHR
SCHEMBL9000789 0.81 LMNA (0.62) LMNAMAPK1BLMNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 186 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113355367-B Application of ketoacid reductase in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2024-03-26 CN claimed
US-20220281839-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2022-09-08 US claimed
CN-113355299-B Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2022-05-24 CN claimed
US-11306069-B2 Benzimidazole derivatives as dual histamine H1 and histamine H4 receptor ligands BIOPROJET (FR) 2022-04-19 US claimed
CN-113355299-A Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-09-07 CN claimed
CN-113355367-A Application of ketoacid reductase in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-09-07 CN claimed
CN-108410831-B Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-07-27 CN claimed
EP-3486243-B1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2020-04-15 EP claimed
EP-3486243-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS Bioprojet (FR) 2019-05-22 EP claimed
US-20190144421-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET (FR) 2019-05-16 US claimed
CN-108410831-A Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2018-08-17 CN claimed
CN-102660471-B Production of chiral alpha-hydroxy acid and its strain by using biological catalysis method UNIV ZHEJIANG TECHNOLOGY 2014-11-05 CN claimed
CN-102660470-B Sinorhizobium fredii and its application in producing chiral alpha-hydroxy acid by biologically splitting alpha-hydroxy acid raceme UNIV ZHEJIANG TECHNOLOGY 2013-07-31 CN claimed
CN-102660471-A Production of chiral alpha-hydroxy acid and its strain by using biological catalysis method UNIV ZHEJIANG TECHNOLOGY 2012-09-12 CN claimed
CN-102660470-A Sinorhizobium fredii and its application in producing chiral alpha-hydroxy acid by biologically splitting alpha-hydroxy acid raceme UNIV ZHEJIANG TECHNOLOGY 2012-09-12 CN claimed
US-7985572-B2 Modified nitrilases and their use in methods for the production of carboxylic acids BASF SE (DE) 2011-07-26 US claimed
EP-1599584-B1 MODIFIED NITRILASES AND THEIR USE IN METHODS FOR THE PRODUCTION OF CARBOXYLIC ACIDS BASF SE (DE) 2009-07-01 EP claimed
US-20070112216-A1 Method for producing chiral mercapto amino acids DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO KG (AT) 2007-05-17 US claimed
US-20060259999-A1 Modified nitrilases and their use in methods for the production of carboxylic acids BASF AKTIENGESELLSCHAFT (DE) 2006-11-16 US claimed
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2026-05-07 US disclosed
US-20260125390-A1 SOLID FORMS OF MACROCYCLIC COMPOUNDS, SALTS AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE SAME KURA ONCOLOGY INC (US) 2026-05-07 US disclosed
EP-4720073-A1 SOLID FORMS OF A MACROCYCLIC FARNESYLTRANSFERASE INHIBITOR AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE MACROCYCLIC COMPOUND AND ITS SOLID FORMS Kura Oncology, Inc. (US) 2026-04-08 EP disclosed
US-12466835-B1 Solid forms of macrocyclic compounds, salts and formulations thereof, and methods of preparing and using the same KURA ONCOLOGY, INC. (US) 2025-11-11 US disclosed
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-09-16 US disclosed
US-12384757-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds ACLARIS THERAPEUTICS, INC. (US) 2025-08-12 US disclosed
WO-2024245364-A1 SOLID FORMS OF A MACROCYCLIC FARNESYLTRANSFERASE INHIBITOR AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE MACROCYCLIC COMPOUND AND ITS SOLID FORMS KURA ONCOLOGY, INC. (US) 2024-12-05 WO disclosed
US-12134608-B2 Benzimidazole derivatives as dual histamine H1 and histamine H4 receptor ligands BIOPROJET (FR) 2024-11-05 US disclosed
CN-113355367-B Application of ketoacid reductase in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2024-03-26 CN disclosed
CN-111757874-B Methods for preparing modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2024-03-08 CN disclosed
US-20240043398-A1 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS, INC. 2024-02-08 US disclosed
US-20240025877-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED 2024-01-25 US disclosed
CN-111051280-B Process for preparing pyrrolidine compounds 弗特克斯药品有限公司 2023-12-22 CN disclosed
CN-108047033-B Reaction device and method for preparing mandelic acid compound 江西科苑生物药业有限公司 2023-12-01 CN disclosed
US-20230339934-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2023-10-26 US disclosed
US-20230339934-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2023-10-26 US disclosed
US-11767309-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds ACLARIS THERAPEUTICS, INC. (US) 2023-09-26 US disclosed
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS, INC. 2023-06-29 US disclosed
CN-110317212-B Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-10-21 CN disclosed
US-11465985-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-10-11 US disclosed
US-20220281839-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2022-09-08 US disclosed
US-11434201-B2 Processes for preparing pyrrolidine compounds VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-09-06 US disclosed
US-20220235025-A1 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS ACLARIS THERAPEUTICS INC (US) 2022-07-28 US disclosed
CN-109689667-B Porous chiral material and use thereof 南开大学 2022-07-12 CN disclosed
EP-3527573-B9 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES INC (US) 2022-07-06 EP disclosed
CN-113355299-B Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2022-05-24 CN disclosed
CN-108997253-B Mandelic acid derivatives containing 1,3, 4-oxadiazole thioether and application thereof 贵州大学 2022-05-24 CN disclosed
CN-114394983-A Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-04-26 CN disclosed
US-11306069-B2 Benzimidazole derivatives as dual histamine H1 and histamine H4 receptor ligands BIOPROJET (FR) 2022-04-19 US disclosed
EP-3661915-B1 PROCESSES FOR PREPARING PYRROLIDINE COMPOUNDS VERTEX PHARMA (US) 2022-03-09 EP disclosed
CN-113355299-A Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-09-07 CN disclosed
CN-113355367-A Application of ketoacid reductase in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-09-07 CN disclosed
US-20210246117-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS (SAN DIEGO) LLC 2021-08-12 US disclosed
EP-3500582-B1 POROUS CHIRAL MATERIALS AND USES THEREOF UNIV NANKAI (CN) 2021-08-11 EP disclosed
CN-108410831-B Ketoacid reductase, gene, engineering bacterium and application in synthesis of chiral aromatic 2-hydroxy acid 浙江工业大学 2021-07-27 CN disclosed
EP-3419974-B1 PROCESS FOR THE SEPARATION OF ENANTIOMERS OF PIPERAZINE DERIVATIVES ASCENEURON SA (CH) 2021-05-05 EP disclosed
US-10975096-B2 Synthesis of polycyclic-carbamoylpyridone compounds GILEAD SCIENCES, INC. (US) 2021-04-13 US disclosed
EP-3783001-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2021-02-24 EP disclosed
US-10857517-B2 Porous chiral materials and uses thereof NANKAI UNIVERSITY (CN) 2020-12-08 US disclosed
US-20200369608-A1 PROCESSES FOR PREPARING PYRROLIDINE COMPOUNDS VERTEX PHARMACEUTICALS (SAN DIEGO) LLC 2020-11-26 US disclosed
EP-3720849-A2 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR Vertex Pharmaceuticals Incorporated (US) 2020-10-14 EP disclosed
CN-111757874-A Method for producing modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2020-10-09 CN disclosed
EP-3527573-B1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES INC (US) 2020-08-12 EP disclosed
US-20200223866-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2020-07-16 US disclosed
EP-3661915-A1 PROCESSES FOR PREPARING PYRROLIDINE COMPOUNDS Vertex Pharmaceuticals Incorporated (US) 2020-06-10 EP disclosed
CN-111051280-A Process for producing pyrrolidine compound 弗特克斯药品有限公司 2020-04-21 CN disclosed
EP-3486243-B1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2020-04-15 EP disclosed
CN-110317212-A The synthesis of polycyclic carbamoylpyridone compound 吉利德科学公司 2019-10-11 CN disclosed
EP-3527573-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2019-08-21 EP disclosed
US-10344021-B2 Process for the separation of enantiomers of piperazine derivatives ASCENEURON S A (CH) 2019-07-09 US disclosed
EP-3500582-A1 POROUS CHIRAL MATERIALS AND USES THEREOF Nankai University (CN) 2019-06-26 EP disclosed
WO-2019113476-A2 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-06-13 WO disclosed
EP-3486243-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS Bioprojet (FR) 2019-05-22 EP disclosed
US-20190144421-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS BIOPROJET (FR) 2019-05-16 US disclosed
CN-106470975-B Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2019-04-26 CN disclosed
CN-109689667-A Porous chiral material and use thereof 南开大学 2019-04-26 CN disclosed
WO-2019028228-A1 PROCESSES FOR PREPARING PYRROLIDINE COMPOUNDS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-02-07 WO disclosed
EP-3419974-A1 PROCESS FOR THE SEPARATION OF ENANTIOMERS OF PIPERAZINE DERIVATIVES Asceneuron SA (CH) 2019-01-02 EP disclosed
CN-108997253-A Mandelic acid derivatives and its application of the one kind containing \" 1,3,4- oxadiazoles thioether \ 贵州大学 2018-12-14 CN disclosed
CN-108884081-A The method for separating the enantiomer of bridged piperazine derivatives 阿森纽荣股份公司 2018-11-23 CN disclosed
US-10113025-B2 Functionalized ketone-aldehyde condensation resins EVONIK DEGUSSA GMBH (DE) 2018-10-30 US disclosed
WO-2018035660-A1 POROUS CHIRAL MATERIALS AND USES THEREOF NANKAI UNIVERSITY (CN) 2018-03-01 WO disclosed
US-20180022757-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2018-01-25 US disclosed
WO-2017144635-A1 PROCESS FOR THE SEPARATION OF ENANTIOMERS OF PIPERAZINE DERIVATIVES ASCENEURON S. A. (CH) 2017-08-31 WO disclosed
EP-3157933-A2 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2017-04-26 EP disclosed
CN-106470975-A Synthesis of Polycyclic Carbamoylpyridone Compounds 吉利德科学公司 2017-03-01 CN disclosed
CN-106046281-A FUNCTIONALIZED KETONE-ALDEHYDE CONDENSATION RESINS 赢创德固赛有限公司 2016-10-26 CN disclosed
US-20160289366-A1 FUNCTIONALIZED KETONE-ALDEHYDE CONDENSATION RESINS EVONIK DEGUSSA GMBH (DE) 2016-10-06 US disclosed
US-9315792-B2 Nitrilases, nucleic acids encoding them and methods for making and using them BASF ENZYMES LLC (US) 2016-04-19 US disclosed
US-20150368264-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2015-12-24 US disclosed
WO-2015195656-A2 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES ,INC. (US) 2015-12-23 WO disclosed
US-9217164-B2 Nitrilases, nucleic acids encoding them and methods for making and using them BASF ENZYMES LLC (US) 2015-12-22 US disclosed
EP-2327766-B1 Nitrilases BASF ENZYMES LLC (US) 2015-12-02 EP disclosed
EP-2319919-B1 Nitrilases BASF ENZYMES LLC (US) 2015-08-12 EP disclosed
EP-1576108-B1 NITRILASES, NUCLEIC ACIDS ENCODING THEM AND METHODS FOR MAKING AND USING THEM BASF ENZYMES LLC (US) 2015-07-08 EP disclosed
US-20150125928-A1 NITRILASES, NUCLEIC ACIDS ENCODING THEM AND METHODS FOR MAKING AND USING THEM BASF ENZYMES LLC 2015-05-07 US disclosed
EP-2327767-B1 Nitrilases BASF ENZYMES LLC (US) 2015-04-29 EP disclosed
EP-2327765-B1 Nitrilases BASF ENZYMES LLC (US) 2015-04-01 EP disclosed
CN-102170864-B Treatment of Respiratory Diseases PULMAGEN THERAPUTICS INFLAMMATION LTD 2015-04-01 CN disclosed
US-8906663-B2 Nitrilases VERENIUM CORPORATION (US) 2014-12-09 US disclosed
US-8906663-B2 Nitrilases VERENIUM CORPORATION (US) 2014-12-09 US disclosed
CN-102660471-B Production of chiral alpha-hydroxy acid and its strain by using biological catalysis method UNIV ZHEJIANG TECHNOLOGY 2014-11-05 CN disclosed
US-8815569-B2 Methods for preserving and/or storing cells having a nitrilase or nitrile hydratase activity BASF SE (DE) 2014-08-26 US disclosed
US-8778651-B2 Nitrilases, nucleic acids encoding them and methods for making and using them VERENIUM CORPORATION (US) 2014-07-15 US disclosed
EP-2423211-B1 PROCESSES FOR PRODUCING (1S,6S)- OR (1R,6R)-CIS-2,8-DIAZABICYCLO[4.3.0]NONANE AND INTERMEDIATE THEREOF KANEKA CORP (JP) 2014-04-16 EP disclosed
CN-102660624-B Alpha-hydroxy acid deracemisation method and strain UNIV ZHEJIANG TECHNOLOGY 2013-10-16 CN disclosed
CN-102660470-B Sinorhizobium fredii and its application in producing chiral alpha-hydroxy acid by biologically splitting alpha-hydroxy acid raceme UNIV ZHEJIANG TECHNOLOGY 2013-07-31 CN disclosed
US-20130177949-A1 NITRILASES VERENIUM CORPORATION (US) 2013-07-11 US disclosed
US-20130177949-A1 NITRILASES VERENIUM CORPORATION (US) 2013-07-11 US disclosed
US-8334125-B2 Nucleic acids encoding nitrilases VERENIUM CORPORATION (US) 2012-12-18 US disclosed
US-8334125-B2 Nucleic acids encoding nitrilases VERENIUM CORPORATION (US) 2012-12-18 US disclosed
EP-2222272-B1 Respiratory disease treatment PULMAGEN THERAPEUTICS INFLAMMATION LTD (GB) 2012-11-07 EP disclosed
CN-102660471-A Production of chiral alpha-hydroxy acid and its strain by using biological catalysis method UNIV ZHEJIANG TECHNOLOGY 2012-09-12 CN disclosed
CN-102660624-A Alpha-hydroxy acid deracemisation method and strain UNIV ZHEJIANG TECHNOLOGY 2012-09-12 CN disclosed
CN-102660470-A Sinorhizobium fredii and its application in producing chiral alpha-hydroxy acid by biologically splitting alpha-hydroxy acid raceme UNIV ZHEJIANG TECHNOLOGY 2012-09-12 CN disclosed
EP-2423211-A1 PROCESSES FOR PRODUCING (1S,6S)- OR (1R,6R)-CIS-2,8-DIAZABICYCLO[4.3.0]NONANE AND INTERMEDIATE THEREOF Kaneka Corporation (JP) 2012-02-29 EP disclosed
WO-2012007814-A2 THREE COMPONENT CO-CRYSTAL FORMATION BETWEEN DIASTEREOMERIC MIXTURES OF 3-ALKYL-4-((S)-1'PHENYLETHYLAMINO) BUTANOIC ACID AND OPTICALLY PURE 1, 1'-BI-2-NAPHTHOL LUPIN LIMITED (IN) 2012-01-19 WO disclosed
US-20120009637-A1 Nitrilases, Nucleic Acids Encoding Them and Methods For Making and Using Them VERENIUM CORPORATION (US) 2012-01-12 US disclosed
US-20110263839-A1 Nucleic Acids Encoding Nitrilases VERENIUM CORPORATION (US) 2011-10-27 US disclosed
US-20110263839-A1 Nucleic Acids Encoding Nitrilases VERENIUM CORPORATION (US) 2011-10-27 US disclosed
CN-102170864-A Treatment of Respiratory Diseases ARGENTA DISCOVERY LTD 2011-08-31 CN disclosed
US-7993901-B2 Nitrilases and methods for making and using them VERENIUM CORPORATION (US) 2011-08-09 US disclosed
US-7993901-B2 Nitrilases and methods for making and using them VERENIUM CORPORATION (US) 2011-08-09 US disclosed
US-7985572-B2 Modified nitrilases and their use in methods for the production of carboxylic acids BASF SE (DE) 2011-07-26 US disclosed
EP-2327767-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP disclosed
EP-2327766-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP disclosed
EP-2327765-A1 Nitrilases Verenium Corporation (US) 2011-06-01 EP disclosed
EP-2319919-A1 Nitrilases Verenium Corporation (US) 2011-05-11 EP disclosed
EP-2222272-A1 RESPIRATORY DISEASE TREATMENT Pulmagen Therapeutics (Inflammation) Limited (GB) 2010-09-01 EP disclosed
US-20100086986-A1 Increased activity and stability at increased pH and temperature; making a chiral alpha -hydroxy acid molecule, a chiral amino acid molecule, a chiral beta -hydroxy acid molecule, or a chiral gamma-hydroxy acid molecule, from a molecule with a cyanohydrin moiety or an aminonitrile moiety VERENIUM CORPORATION (US) 2010-04-08 US disclosed
US-20100086986-A1 Increased activity and stability at increased pH and temperature; making a chiral alpha -hydroxy acid molecule, a chiral amino acid molecule, a chiral beta -hydroxy acid molecule, or a chiral gamma-hydroxy acid molecule, from a molecule with a cyanohydrin moiety or an aminonitrile moiety VERENIUM CORPORATION (US) 2010-04-08 US disclosed
WO-2010015818-A1 RESPIRATORY DISEASE TREATMENT ARGENTA DISCOVERY LIMITED (GB) 2010-02-11 WO disclosed
US-7651849-B2 Increased activity and stability at increased pH and temperature VERENIUM CORPORATION 2010-01-26 US disclosed
US-7651849-B2 Increased activity and stability at increased pH and temperature VERENIUM CORPORATION 2010-01-26 US disclosed
US-20100009426-A1 synthetic or recombinant polypeptide having a nitrilase activity; have increased activity and stability at increased pH and temperature VERENIUM CORPORATION (US) 2010-01-14 US disclosed
US-7608445-B1 Nitrilases, nucleic acids encoding them and methods for making and using them VERENIUM CORPORATION (US) 2009-10-27 US disclosed
US-20090176976-A1 Increased activity and stability at increased pH and temperature VERENIUM CORPORATION 2009-07-09 US disclosed
US-20090176976-A1 Increased activity and stability at increased pH and temperature VERENIUM CORPORATION 2009-07-09 US disclosed
EP-1599584-B1 MODIFIED NITRILASES AND THEIR USE IN METHODS FOR THE PRODUCTION OF CARBOXYLIC ACIDS BASF SE (DE) 2009-07-01 EP disclosed
US-7521216-B2 Nitrilases and methods for making and using them VERENIUM CORPORATION (US) 2009-04-21 US disclosed
US-7521216-B2 Nitrilases and methods for making and using them VERENIUM CORPORATION (US) 2009-04-21 US disclosed
EP-2039762-A2 Nitralases Verenium Corporation (US) 2009-03-25 EP disclosed
EP-1578910-A4 NITRILASES VERENIUM CORP (US) 2008-06-04 EP disclosed
US-20070149599-A1 Polymorphs of bicifadine hydrochloride DOV PHARMACEUTICAL, INC. 2007-06-28 US disclosed
US-20070112216-A1 Method for producing chiral mercapto amino acids DSM FINE CHEMICALS AUSTRIA NFG GMBH & CO KG (AT) 2007-05-17 US disclosed
US-20070082938-A1 Polymorphs of bicifadine hydrochloride DOV PHARMACEUTICAL, INC. 2007-04-12 US disclosed
EP-1236714-B1 ACETALSULFONATE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING STYRENE OXIDE DERIVATIVE MITSUBISHI RAYON CO (JP) 2007-01-17 EP disclosed
US-20060259999-A1 Modified nitrilases and their use in methods for the production of carboxylic acids BASF AKTIENGESELLSCHAFT (DE) 2006-11-16 US disclosed
US-7094799-B2 A single, thermodynamical stable crystal structure, is crystallized from a cooled and agitated solvent solution, analgesic drug for reducing pain DOV PHARMACEUTICAL, INC. (US) 2006-08-22 US disclosed
EP-1562900-A4 POLYMORPHS OF BICIFADINE HYDROCHLORIDE DOV PHARMACEUTICAL INC (US) 2006-07-12 EP disclosed
US-20060110808-A1 Methods for preserving and/or storing cellshaving a nitrilase or nitrile hydratase avtivity BASF AKTIENGESELLSCHAFT 2006-05-25 US disclosed
CN-1735594-A Polymorphs of bicifadine hydrochloride DOV PHARMACEUTICALS INC (US) 2006-02-15 CN disclosed
CN-1235875-C Substituted alpha-hydroxy acid caspase inhibitors and uses thereof CYTOVIA INC (US) 2006-01-11 CN disclosed
EP-1599584-A1 MODIFIED NITRILASES AND THEIR USE IN METHODS FOR THE PRODUCTION OF CARBOXYLIC ACIDS BASF AKTIENGESELLSCHAFT (DE) 2005-11-30 EP disclosed
EP-1578910-A2 NITRILASES DIVERSA CORPORATION (US) 2005-09-28 EP disclosed
EP-1562900-A1 POLYMORPHS OF BICIFADINE HYDROCHLORIDE DOV Pharmaceutical Inc. (US) 2005-08-17 EP disclosed
WO-2004076655-A1 MODIFIED NITRILASES AND THEIR USE IN METHODS FOR THE PRODUCTION OF CARBOXYLIC ACIDS BASF AKTIENGESELLSCHAFT (DE) 2004-09-10 WO disclosed
US-6743944-B1 FORMING DIASTEREOMERIC SALT OF RACEMIC 4-AMINO-2-METHYL-BUTANE-1-OL AND OPTICALLY ACTIVE ORGANIC ACID; CRYSTALLI-ZATION; ALKALI SOLUTION DECOMPOSITION MITSUBISHI RAYON CO., LTD. (JP) 2004-06-01 US disclosed
WO-2004043920-A1 POLYMORPHS OF BICIFADINE HYDROCHLORIDE DOV PHARMACEUTICALS, INC. (US) 2004-05-27 WO disclosed
US-20040102638-A1 Polymorphs of bicifadine hydrochloride EUTHYMICS BIOSCIENCE, INC. 2004-05-27 US disclosed
EP-0838448-B1 Process for the separation of a mixture of enantiomers DSM IP ASSETS BV (NL) 2004-04-21 EP disclosed
US-6642395-B1 Esterifying mandelic acid derivative; protecting hydroxyl group and reducing ester; sulfonating and epoxidizing MITSUBISHI RAYON CO., LTD. (JP) 2003-11-04 US disclosed
EP-0915080-B1 Process for preparing optically active amines and optically active carboxylic acids, and intermediates for preparation YAMAKAWA CHEMICAL IND (JP) 2003-03-26 EP disclosed
WO-2003000840-A2 NITRILASES DIVERSA CORPORATION (US) 2003-01-03 WO disclosed
US-6495522-B1 PREVENTING APOPTOTIC CELL DEATH IN WHICH THE LOSS OF CELLS, TISSUES OR ENTIRE ORGANS OCCURS CYTOVIA, INC. 2002-12-17 US disclosed
CN-1382119-A Substituted alpha-hydroxy acid caspase inhibitors and uses thereof CYTOVIA INC (US) 2002-11-27 CN disclosed
US-6465684-B2 DIASTEREOMER COMPLEX OF AT LEAST THREE COMPOUNDS, AT LEAST ONE IS A RESOLVING AGENT IN OPTICALLY ACTIVE FORM, AND AT LEAST ONE IS AN ENANTIOMER IN OPTICALLY ACTIVE FORM; RAPID SEPARATION DSM N.V. (NL) 2002-10-15 US disclosed
EP-1236714-A1 ACETALSULFONATE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING STYRENE OXIDE DERIVATIVE Mitsubishi Rayon Co., Ltd. (JP) 2002-09-04 EP disclosed
EP-1219593-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE AMINOALCOHOL Mitsubishi Rayon Co., Ltd. (JP) 2002-07-03 EP disclosed
EP-1212295-A1 SUBSTITUTED $g(a)-HYDROXY ACID CASPASE INHIBITORS AND THE USE THEREOF Cytovia, Inc. (US) 2002-06-12 EP disclosed
US-6342636-B1 REACTION OF ARYLALKYLAMINE WITH NAPHTHYLGLYCOLIC ACID AND DECOMPOSITION A DIASTEROMER SALT TO OBTAIN AN ENANTIOMORPH YAMAKAWA CHEMICAL INDUSTRY CO., LTD. (JP) 2002-01-29 US disclosed
US-20010051747-A1 Process for the separation of a mixture of enantiomers DSM N.V. 2001-12-13 US disclosed
US-6235927-B1 OPTICAL RESOLUTION OF ENANTIOMORPHS OF COMPLEXES DSM N.V. (NL) 2001-05-22 US disclosed
WO-2001016093-A1 SUBSTITUTED α-HYDROXY ACID CASPASE INHIBITORS AND THE USE THEREOF CYTOVIA, INC. (US) 2001-03-08 WO disclosed
EP-0915080-A1 Process for preparing optically active amines and optically active carboxylic acids, and intermediates for preparation YAMAKAWA CHEMICAL INDUSTRY CO., LTD. (JP) 1999-05-12 EP disclosed
EP-0838448-A1 Process for the separation of a mixture of enantiomers DSM N.V. (NL) 1998-04-29 EP disclosed
EP-0816316-A1 PROCESS FOR PRODUCING 1,2-ETHANEDIOL DERIVATIVES NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-01-07 EP disclosed
EP-0146269-B1 HETERO-POLYCYCLIC AROMATIC COMPOUND IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-01-03 EP disclosed
US-4650882-A Dyes having two 5-membered lactone rings fused to a central cyclohexa-1.4-diene nucleus IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-03-17 US disclosed
EP-0146269-A2 Hetero-polycyclic aromatic compound IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-06-26 EP disclosed
EP-0033583-B1 DYESTUFFS COMPRISING TWO 5-MEMBERED HETEROCYCLIC NUCLEI FUSED TO A CENTRAL CYCLOHEXADIENE NUCLEUS, PROCESSES FOR THEIR PREPARATION AND THEIR USE FOR COLOURING SYNTHETIC TEXTILE MATERIALS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-10-12 EP disclosed
EP-0023080-B1 SUBSTITUTED 2,7-DIOXO-2,7-DIHYDROBENZO(1:2-B; 5,6-B1)DIFURAN OR DIPYRROLE DYESTUFFS, PROCESSES FOR THEIR PREPARATION AND THEIR USE FOR THE COLOURATION OF AROMATIC POLYESTER TEXTILE MATERIALS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-07-27 EP disclosed
US-4333877-A Substituted 2,7-dioxo-2,7-dihydrobenzo[1:2-b; 5:6-b1 ]difuran or -dipyrrole dyestuffs, their preparation and their use IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-06-08 US disclosed
EP-0033583-A1 Dyestuffs comprising two 5-membered heterocyclic nuclei fused to a central cyclohexadiene nucleus, processes for their preparation and their use for colouring synthetic textile materials IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-08-12 EP disclosed
EP-0023080-A1 Substituted 2,7-dioxo-2,7-dihydrobenzo(1:2-b; 5,6-b1)difuran or dipyrrole dyestuffs, processes for their preparation and their use for the colouration of aromatic polyester textile materials IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-01-28 EP disclosed
US-4218380-A OXIDATION OF THE A-HYDROXY-ARYLACETIC ACID BAYER AKTIENGESELLSCHAFT (DE) 1980-08-19 US disclosed
US-4091214-A ALPHA-HYDROXY CARBOXYLIC ACID ELI LILLY AND COMPANY (US) 1978-05-23 US disclosed
US-4091214-A ALPHA-HYDROXY CARBOXYLIC ACID ELI LILLY AND COMPANY (US) 1978-05-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (33 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150368264-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS CPS1, SDHA, DHPS LMNA 2030/4885MAPK1 4044/4885KEAP1 2541/4885
US-20070149599-A1 Polymorphs of bicifadine hydrochloride SF3B5, SFPQ, BBC3 LMNA 1689/4885MAPK1 4459/4885KEAP1 1264/4885
US-20260125390-A1 SOLID FORMS OF MACROCYCLIC COMPOUNDS, SALTS AND FORMULATIONS THEREOF, AND METHODS OF PREPARING AND USING THE SAME FDPS, PCTP, MTTP LMNA 3952/4885MAPK1 2771/4885KEAP1 3724/4885
US-12466835-B1 Solid forms of macrocyclic compounds, salts and formulations thereof, and methods of preparing and using the same FNTA, SF3B1, SF3A1 LMNA 1318/4885MAPK1 2101/4885KEAP1 473/4885
US-20200223866-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS CPS1, SDHA, DHPS LMNA 2030/4885MAPK1 4044/4885KEAP1 2541/4885
US-10344021-B2 Process for the separation of enantiomers of piperazine derivatives CYP3A5, CYP4Z1, HTR5A LMNA 1321/4885MAPK1 1627/4885KEAP1 273/4885
US-11767309-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds PIR, PUM1, ZRANB2 LMNA 780/4885MAPK1 924/4885KEAP1 483/4885
US-12384757-B2 Methods of synthesizing substituted pyridinone-pyridinyl compounds PIR, PUM1, ZRANB2 LMNA 780/4885MAPK1 924/4885KEAP1 483/4885
US-20210246117-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1B, SCNN1G LMNA 3683/4885MAPK1 1948/4885KEAP1 817/4885
US-20190144421-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS HRH4, HRH3, HRH1 LMNA 4746/4885MAPK1 3692/4885KEAP1 1280/4885
US-20200369608-A1 PROCESSES FOR PREPARING PYRROLIDINE COMPOUNDS MTAP, PRMT5, TET3 LMNA 1837/4885MAPK1 1217/4885KEAP1 4489/4885
US-20220235025-A1 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS PIR, PUM1, ZRANB2 LMNA 780/4885MAPK1 924/4885KEAP1 483/4885
US-20110263839-A1 Nucleic Acids Encoding Nitrilases RNGTT, NSUN2, DNTT LMNA 1303/4885MAPK1 4328/4885KEAP1 3317/4885
US-20240043398-A1 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS PIR, PUM1, ZRANB2 LMNA 780/4885MAPK1 924/4885KEAP1 483/4885
US-20260125363-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SLC26A4, SLC26A3 LMNA 1827/4885MAPK1 366/4885KEAP1 1258/4885
US-20180022757-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS CPS1, SDHA, DHPS LMNA 2030/4885MAPK1 4044/4885KEAP1 2541/4885
US-20070082938-A1 Polymorphs of bicifadine hydrochloride SF3B5, SFPQ, BBC3 LMNA 1689/4885MAPK1 4459/4885KEAP1 1264/4885
US-20100086986-A1 Increased activity and stability at increased pH and temperature; making a chiral alpha -hydroxy acid molecule, a chiral amino acid molecule, a chiral beta -hydroxy acid molecule, or a chiral gamma-hydroxy acid molecule, from a molecule with a cyanohydrin moiety or an aminonitrile moiety ASPH, AHSA1, DNPH1 LMNA 697/4885MAPK1 2286/4885KEAP1 2503/4885
US-20040102638-A1 Polymorphs of bicifadine hydrochloride SF3B5, SFPQ, BBC3 LMNA 1689/4885MAPK1 4459/4885KEAP1 1264/4885
US-20240025877-A1 PROCESSES FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1B, SCNN1G LMNA 3445/4885MAPK1 2625/4885KEAP1 842/4885
US-20010051747-A1 Process for the separation of a mixture of enantiomers EPHX2, VKORC1, ALDH1A2 LMNA 270/4885MAPK1 4593/4885KEAP1 401/4885
US-20230339934-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS TRPV4, TRPV1, TRPV2 LMNA 4199/4885MAPK1 1813/4885KEAP1 1024/4885
US-11434201-B2 Processes for preparing pyrrolidine compounds MTAP, PRMT5, TET3 LMNA 1837/4885MAPK1 1217/4885KEAP1 4489/4885
US-20230202999-A9 METHODS OF SYNTHESIZING SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS PIR, PUM1, ZRANB2 LMNA 780/4885MAPK1 924/4885KEAP1 483/4885
US-11465985-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SCNN1G LMNA 3683/4885MAPK1 1948/4885KEAP1 817/4885
US-12415798-B2 Processes for making modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SCNN1G LMNA 3445/4885MAPK1 2625/4885KEAP1 842/4885
US-20120009637-A1 Nitrilases, Nucleic Acids Encoding Them and Methods For Making and Using Them RNGTT, NSUN2, NSUN3 LMNA 1395/4885MAPK1 4287/4885KEAP1 2794/4885
US-10857517-B2 Porous chiral materials and uses thereof ANXA7, XDH, OPRM1 LMNA 219/4885MAPK1 1200/4885KEAP1 3938/4885
US-20070112216-A1 Method for producing chiral mercapto amino acids CPN1, AKR1C3, AHCY LMNA 1994/4885MAPK1 2896/4885KEAP1 1368/4885
US-20220281839-A1 BENZIMIDAZOLE DERIVATIVES AS DUAL HISTAMINE H1 AND HISTAMINE H4 RECEPTOR LIGANDS HRH4, HRH3, HRH1 LMNA 4626/4885MAPK1 3796/4885KEAP1 1128/4885
US-12134608-B2 Benzimidazole derivatives as dual histamine H1 and histamine H4 receptor ligands HRH4, HRH3, HRH1 LMNA 4626/4885MAPK1 3796/4885KEAP1 1128/4885
US-10975096-B2 Synthesis of polycyclic-carbamoylpyridone compounds CPS1, SDHA, DHPS LMNA 2030/4885MAPK1 4044/4885KEAP1 2541/4885
US-11306069-B2 Benzimidazole derivatives as dual histamine H1 and histamine H4 receptor ligands HRH4, HRH3, HRH1 LMNA 4746/4885MAPK1 3692/4885KEAP1 1280/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.