SCHEMBL312084

SCHEMBL312084

O=C(SSSSC(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 5/20 0.50
CES2 O00748 5/20 0.50
TSHR P16473 3/20 0.50
ALDH1A1 P00352 3/20 0.50
DAO P14920 1/20 0.50
NAPRT Q6XQN6 1/20 0.50
TDP1 Q9NUW8 4/20 0.46
CYP3A4 P08684 2/20 0.46
MAPT P10636 2/20 0.46
CA2 P00918 2/20 0.46
CA4 P22748 2/20 0.46
HSD17B10 Q99714 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA9 Q16790 2/20 0.46
POLB P06746 1/20 0.46
PARP1 P09874 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL168007 0.89 CES1 (0.55) CES1CES2TSHRALDH1A1DAO
Hydrochloric Acid SCHEMBL28496848 0.86 CES1 (0.52) CES1CES2TSHRALDH1A1DAO
Hydrogen Sulfide SCHEMBL28111724 0.86 CES1 (0.52) CES1CES2TSHRALDH1A1DAO
Water SCHEMBL27612226 0.86 CES1 (0.52) CES1CES2TSHRALDH1A1DAO
SCHEMBL8932412 0.81 CES1 (0.43) CES1CES2TSHRALDH1A1DAO
SCHEMBL5031044 0.80 KMT2A (0.47) CES1CES2TSHRALDH1A1DAO
SCHEMBL11742945 0.80 CES1 (0.46) CES1CES2TSHRALDH1A1DAO
SCHEMBL8494639 0.80 CA2 (0.48) CES1CES2TSHRALDH1A1DAO
SCHEMBL11621561 0.78 HPGD (0.48) CES1CES2TSHRALDH1A1DAO
SCHEMBL11623306 0.78 CES1 (0.48) CES1CES2TSHRALDH1A1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 409 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12492220-B2 Method for the preparation of oligonucleotides THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2025-12-09 US claimed
US-20230192751-A1 METHOD FOR THE PREPARATION OF OLIGONUCLEOTIDES THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIV (CA) 2023-06-22 US claimed
US-8304532-B2 Method for preparing oligonucleotides GIRINDUS AG (DE) 2012-11-06 US claimed
EP-1525212-B1 METHOD FOR PREPARING OLIGONUCLEOTIDES GIRINDUS AG (DE) 2012-09-12 EP claimed
US-20110224424-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2011-09-15 US claimed
US-20100069623-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2010-03-18 US claimed
US-20060089494-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2006-04-27 US claimed
EP-1525212-A1 METHOD FOR PREPARING OLIGONUCLEOTIDES Girindus AG (DE) 2005-04-27 EP claimed
EP-0948512-B1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2004-10-06 EP claimed
WO-2004013154-A1 METHOD FOR PREPARING OLIGONUCLEOTIDES GIRINDUS AG (DE) 2004-02-12 WO claimed
EP-1386925-A1 Method for preparing oligonucleotides Girindus AG (DE) 2004-02-04 EP claimed
US-20030114662-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2003-06-19 US claimed
US-20020128466-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2002-09-12 US claimed
US-6403781-B2 REACTING A PHOSPHORDIAMIDITE WITH A SUPPORT-BOUND SYNTHON TO FORM A SUPPORT BOUND PHOSPHORAMIDITE, PROTECTING TO FORM A SUPPORT BOUND PHOSHITE, SULFURIZING THE PHOSPHITE TO FORM A PROTECTED PHOSPHORTHIOATE AND DEPROTECTING ISIS PHARMACEUTICALS, INC. 2002-06-11 US claimed
EP-0948512-A4 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2001-10-24 EP claimed
US-20010003132-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2001-06-07 US claimed
US-6172217-B1 SULFURIZATION OF PHOSPORDIAMIDITE; DEBLOCKING ISIS PHARMACEUTICALS INC. 2001-01-09 US claimed
EP-0948512-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1999-10-13 EP claimed
WO-1998029427-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO claimed
US-12590115-B2 Technologies useful for oligonucleotide preparation WAVE LIFE SCIENCES LTD. (SG) 2026-03-31 US disclosed
US-20260008806-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD (SG) 2026-01-08 US disclosed
US-12492220-B2 Method for the preparation of oligonucleotides THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2025-12-09 US disclosed
US-12435105-B2 Technologies for oligonucleotide preparation WAVE LIFE SCIENCES LTD. (SG) 2025-10-07 US disclosed
US-20240327448-A1 LITHIUM REAGENTS AND THEIR USES IN SOLID PHASE SYNTHESIS OLIX US, INC. 2024-10-03 US disclosed
WO-2024173777-A1 LITHIUM REAGENTS AND THEIR USES IN SOLID PHASE SYNTHESIS OLIX US, INC. (US) 2024-08-22 WO disclosed
US-20240158432-A1 COMPOSITIONS COMPRISING DICHLOROACETIC ACID, PROCESSES FOR PREPARING SAME AND USES THEREOF SHANGHAI STA PHARMACEUTICAL R&D CO., LTD. (CN) 2024-05-16 US disclosed
US-11873318-B2 Compositions comprising dichloroacetic acid, processes for preparing same and uses thereof CHANGZHOU SYNTHEALL PHARMACEUTICALS CO., LTD. (CN) 2024-01-16 US disclosed
US-20230348524-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD. (SG) 2023-11-02 US disclosed
US-20230192751-A1 METHOD FOR THE PREPARATION OF OLIGONUCLEOTIDES THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIV (CA) 2023-06-22 US disclosed
US-20230123981-A1 4'-O-METHYLENE PHOSPHONATE NUCLEIC ACIDS AND ANALOGUES THEREOF NOVO NORDISK A/S (DK) 2023-04-20 US disclosed
EP-4153605-A1 COMPOSITIONS COMPRISING DICHLOROACETIC ACID, PROCESSES FOR PREPARING SAME AND USES THEREOF Changzhou Syntheall Pharmaceuticals Co., Ltd. (CN) 2023-03-29 EP disclosed
US-20230089442-A1 TECHNOLOGIES USEFUL FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD. (SG) 2023-03-23 US disclosed
US-11608355-B2 Technologies for oligonucleotide preparation WAVE LIFE SCIENCES LTD. (SG) 2023-03-21 US disclosed
CN-115836080-A Composition comprising dichloroacetic acid, process for its preparation and its use 常州合全药业有限公司 2023-03-21 CN disclosed
US-20230002438-A1 COMPOSITIONS COMPRISING DICHLOROACETIC ACID, PROCESSES FOR PREPARING SAME AND USES THEREOF SHANGHAI STA PHARMACEUTICAL R&D CO., LTD. (CN) 2023-01-05 US disclosed
CN-115298192-A 4' -O-methylene phosphonate nucleic acids and analogs thereof 迪克纳制药公司 2022-11-04 CN disclosed
EP-3941924-A1 TECHNOLOGIES USEFUL FOR OLIGONUCLEOTIDE PREPARATION Wave Life Sciences Ltd. (SG) 2022-01-26 EP disclosed
CN-113748116-A Techniques useful for oligonucleotide preparation 波涛生命科学有限公司 2021-12-03 CN disclosed
WO-2021233406-A1 COMPOSITIONS COMPRISING DICHLOROACETIC ACID, PROCESSES FOR PREPARING SAME AND USES THEREOF CHANGZHOU SYNTHEALL PHARMACEUTICALS CO., LTD. (CN) 2021-11-25 WO disclosed
US-20210309690-A1 OLIGONUCLEOTIDE SYNTHESIS ROCHE INNOVATION CT COPENHAGEN AS (DK) 2021-10-07 US disclosed
WO-2021146488-A1 4'-O-METHYLENE PHOSPHONATE NUCLEIC ACIDS AND ANALOGUES THEREOF DICERNA PHARMACEUTICALS, INC. (US) 2021-07-22 WO disclosed
US-20200392491-A1 Method of Preparing Oligonucleotide Compounds NOGRA PHARMA LIMITED (IE) 2020-12-17 US disclosed
WO-2020191252-A1 TECHNOLOGIES USEFUL FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD. (SG) 2020-09-24 WO disclosed
CN-111479818-A Method and system for synthesizing oligonucleotides 深圳华大生命科学研究院 2020-07-31 CN disclosed
EP-3684755-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION Wave Life Sciences Ltd. (SG) 2020-07-29 EP disclosed
US-20200231620-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD. (SG) 2020-07-23 US disclosed
EP-3658155-A1 METHOD OF PREPARING OLIGONUCLEOTIDE COMPOUNDS Celgene Corporation (US) 2020-06-03 EP disclosed
CN-111148519-A Method for preparing oligonucleotide compound 细胞基因公司 2020-05-12 CN disclosed
CN-111108096-A Oligonucleotide preparation technology 波涛生命科学有限公司 2020-05-05 CN disclosed
US-10597421-B2 Protected monomer and method of final deprotection for RNA synthesis AGILENT TECHNOLOGIES, INC. (US) 2020-03-24 US disclosed
EP-3491002-A2 SYNTHESIS OF OLIGONUCLEOTIDES COMPRISING ACHIRAL 3'-S- OR 5'-S-PHOSPHOROTHIOLATE INTERNUCLEOSIDE LINKAGE Roche Innovation Center Copenhagen A/S (DK) 2019-06-05 EP disclosed
CN-109641932-A Oligonucleotide synthesis comprising connector between achirality 3 '-S- or 5 '-S phosphorothioic acid ester nucleosides 罗氏创新中心哥本哈根有限公司 2019-04-16 CN disclosed
WO-2019055951-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION WAVE LIFE SCIENCES LTD. (SG) 2019-03-21 WO disclosed
WO-2019023439-A1 METHOD OF PREPARING OLIGONUCLEOTIDE COMPOUNDS CELGENE CORPORATION (US) 2019-01-31 WO disclosed
EP-2331558-B1 PROTECTED MONOMERS AND METHODS OF DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES INC (US) 2018-09-12 EP disclosed
US-20180186826-A1 PROTECTED MONOMER AND METHOD OF FINAL DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES, INC. 2018-07-05 US disclosed
US-9896472-B2 Protected monomer and method of final deprotection for RNA synthesis AGILENT TECHNOLOGIES, INC. (US) 2018-02-20 US disclosed
US-20170130029-A1 POLYSULFIDE ADDITIVE, METHOD FOR PRODUCTION THEREOF AND USE THEREOF IN RUBBER MIXTURES LANXESS DEUTSCHLAND GMBH (DE) 2017-05-11 US disclosed
EP-2540734-B1 Process and reagents for oligonucleotide synthesis and purification ALNYLAM PHARMACEUTICALS INC (US) 2016-03-30 EP disclosed
US-9273086-B2 Protected monomer and method of final deprotection for RNA synthesis AGILENT TECHNOLOGIES, INC. (US) 2016-03-01 US disclosed
EP-1028124-B2 Improved deprotection method for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS INC (US) 2016-01-27 EP disclosed
US-20160002282-A1 Protected Monomer and Method of Final Deprotection for RNA Synthesis AGILENT TECHNOLOGIES, INC. 2016-01-07 US disclosed
US-20150240053-A1 POLYSULFIDE ADDITIVE, METHOD FOR PRODUCTION THEREOF AND USE THEREOF IN RUBBER MIXTURES LANXESS DEUTSCHLAND GMBH (DE) 2015-08-27 US disclosed
CN-104661832-A Polysulphide additive, method for production thereof, and use thereof in rubber mixtures LANXESS DEUTSCHLAND GMBH 2015-05-27 CN disclosed
US-20140179875-A1 SULFURIZATION REAGENTS ON SOLID SUPPORTS GIRINDUS AMERICA, INC. (US) 2014-06-26 US disclosed
EP-1023310-B2 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2014-05-21 EP disclosed
US-8552175-B2 Sulfur transfer reagents for oligonucleotide synthesis A.M. Chemicals, Inc. (US) 2013-10-08 US disclosed
US-8541599-B2 Supports for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2013-09-24 US disclosed
US-8431693-B2 Process for desilylation of oligonucleotides ALNYLAM PHARMACEUTICALS, INC. (US) 2013-04-30 US disclosed
EP-1501851-B1 PROCESS FOR PREPARING OLIGONUCLEOTIDES NITTO DENKO AVECIA INC (US) 2013-02-13 EP disclosed
WO-2013017469-A1 SULFURIZATION REAGENTS ON SOLID SUPPORTS GIRINDUS AMERICA, INC. (US) 2013-02-07 WO disclosed
EP-1789460-B1 POLYMERIC BEADS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS INC (US) 2013-01-09 EP disclosed
EP-2540734-A2 Process and reagents for oligonucleotide synthesis and purification Alnylam Pharmaceuticals, Inc. (US) 2013-01-02 EP disclosed
US-20120289691-A1 PROTECTED MONOMER AND METHOD OF FINAL DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES, INC. (US) 2012-11-15 US disclosed
US-8304532-B2 Method for preparing oligonucleotides GIRINDUS AG (DE) 2012-11-06 US disclosed
EP-1525212-B1 METHOD FOR PREPARING OLIGONUCLEOTIDES GIRINDUS AG (DE) 2012-09-12 EP disclosed
US-20120184724-A1 PROTECTED MONOMERS AND METHODS OF DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES, INC. (US) 2012-07-19 US disclosed
US-20120165547-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2012-06-28 US disclosed
US-8193337-B2 Oxidation process AVECIA BIOTECHNOLOGY, INC. (US) 2012-06-05 US disclosed
WO-2012059510-A1 BACK PRESSURE CONTROL DURING SOLID-PHASE SYNTHESIS ON POLYMERIC SUPPORTS GIRINDUS AMERICA, INC. (US) 2012-05-10 WO disclosed
US-8153725-B2 Supports for oligomer synthesis ISIS PHARMACEUTICALS, INC (US) 2012-04-10 US disclosed
US-20120071640-A1 Sulfurizing reagents and their use for oligonucleotides synthesis GIRINDUS AMERICA, INC. (US) 2012-03-22 US disclosed
US-8093397-B2 Activators for oligonucleotide synthesis AVECIA BIOTECHNOLOGY, INC. (US) 2012-01-10 US disclosed
CN-102307889-A Sulfurizing reagents and their use for oligonucleotides synthesis GIRINDUS AMERICA INC 2012-01-04 CN disclosed
US-8063198-B2 Processes and reagents for desilylation of oligonucleotides ALNYLAM PHARMACEUTICALS, INC. (US) 2011-11-22 US disclosed
US-8058448-B2 Processes and reagents for sulfurization of oligonucleotides ALNYLAM PHARMACEUTICALS, INC. (US) 2011-11-15 US disclosed
EP-2382227-A1 SULFURIZING REAGENTS AND THEIR USE FOR OLIGONUCLEOTIDES SYNTHESIS Girindus America, Inc. (US) 2011-11-02 EP disclosed
CN-101076546-B Polymeric beads for oligomer synthesis ISIS PHARMACEUTICALS INC 2011-10-26 CN disclosed
US-20110224424-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2011-09-15 US disclosed
US-20110196145-A1 PROCESS FOR DESILYLATION OF OLIGONUCLEOTIDES ALNYLAM PHARMACEUTICALS, INC. (US) 2011-08-11 US disclosed
US-20110160082-A1 Mobility-Modified Nucleobase Polymers and Methods of Using Same Life Technologies Corporation (US) 2011-06-30 US disclosed
EP-2331558-A2 PROTECTED MONOMERS AND METHODS OF DEPROTECTION FOR RNA SYNTHESIS Agilent Technologies, Inc. (US) 2011-06-15 EP disclosed
US-20110137021-A1 SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS A.M. Chemicals, Inc. 2011-06-09 US disclosed
US-7897338-B2 Mobility-modified nucleobase polymers and methods of using same APPLIED BIOSYSTEMS, LLC (US) 2011-03-01 US disclosed
EP-1575975-B1 PROCESS FOR THE PREPARATION OF OLIGONUCLEOTIDES AVECIA BIOTECHNOLOGY INC (US) 2010-10-27 EP disclosed
US-20100234528-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2010-09-16 US disclosed
US-7759480-B2 Chloral-free DCA in oligonucleotide synthesis ISIS PHARMACEUTICALS, INC. (US) 2010-07-20 US disclosed
WO-2010072831-A1 SULFURIZING REAGENTS AND THEIR USE FOR OLIGONUCLEOTIDES SYNTHESIS GIRINDUS AMERICA, INC (US) 2010-07-01 WO disclosed
US-20100137572-A1 OXIDATION PROCESS NITTO DENKO AVECIA, INC. 2010-06-03 US disclosed
US-7723511-B2 Synthesis of sulfurized oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2010-05-25 US disclosed
US-7723528-B2 Sulfur transfer reagents for oligonucleotide synthesis AM CHEMICALS LLC (US) 2010-05-25 US disclosed
US-7718810-B2 Supports such as glass and styrene polymers functionalized with tricyclic hetercyclic anhydrides and imides, used in the preparation of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2010-05-18 US disclosed
US-7700706-B2 Polymeric beads for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2010-04-20 US disclosed
US-20100076183-A1 PROTECTED MONOMER AND METHOD OF FINAL DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES, INC. 2010-03-25 US disclosed
WO-2010034024-A2 PROTECTED MONOMERS AND METHODS OF DEPROTECTION FOR RNA SYNTHESIS AGILENT TECHNOLOGIES, INC. (US) 2010-03-25 WO disclosed
US-20100069623-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2010-03-18 US disclosed
US-7635772-B2 Process for the preparation of oligonucleotides AVECIA BIOTECHNOLOGY INC. (US) 2009-12-22 US disclosed
US-20090306358-A1 SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS AM CHEMICALS LLC 2009-12-10 US disclosed
US-20090286085-A1 POLYMERIC BEADS FOR OLIGOMER SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2009-11-19 US disclosed
EP-1379698-B1 MOBILITY-MODIFIED NUCLEOBASE POLYMERS AND METHODS OF USING SAME APPLIED BIOSYSTEMS LLC (US) 2009-08-26 EP disclosed
US-7576119-B2 Supports for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2009-08-18 US disclosed
US-20090187027-A1 PROCESSES AND REAGENTS FOR SULFURIZATION OF OLIGONUCLEOTIDES ALNYLAM PHARMACEUTICALS, INC. (US) 2009-07-23 US disclosed
US-20090131682-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2009-05-21 US disclosed
US-20090085006-A1 Activators for oligonucleotide synthesis AVECIA BIOTECHNOLOGY, INC. (US) 2009-04-02 US disclosed
US-7511125-B2 Pyrimidine derivatives for labeled binding partners CARLSBAD (US) 2009-03-31 US disclosed
US-7501505-B2 Activators for oligonucleotide synthesis AVECIA BIOTECHNOLOGY, INC. (US) 2009-03-10 US disclosed
WO-2009007736-A1 OXIDATION PROCESS AVECIA BIOTECHNOLOGY INC. (US) 2009-01-15 WO disclosed
US-7476709-B2 Process for preparing oligonucleotides AVECIA BIOTECHNOLOGY INC. (US) 2009-01-13 US disclosed
US-20090005549-A1 Processes and Reagents for Desilylation of Oligonucleotides ALNYLAM PHARMACEUTICALS, INC. (US) 2009-01-01 US disclosed
EP-1212339-B1 2'-O-ACETAMIDO MODIFIED MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS INC (US) 2008-12-31 EP disclosed
US-20080293929-A1 SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2008-11-27 US disclosed
CN-100430411-C Activators for oligonucleotide synthesis AVECIA LTD (US) 2008-11-05 CN disclosed
US-7446193-B2 Methods for detection of chloral hydrate in dichloroacetic acid ISIS PHARMACEUTICALS, INC. (US) 2008-11-04 US disclosed
US-7427675-B2 Compounds and methods for the characterization of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2008-09-23 US disclosed
US-7378516-B2 Synthesis of sulfurized oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2008-05-27 US disclosed
US-20080119645-A1 Immobilization; solid phase synthesis ISIS PHARMACEUTICALS, INC. (US) 2008-05-22 US disclosed
CN-100384864-C Process for the preparation of oligonucleotides AVECIA LTD (US) 2008-04-30 CN disclosed
US-20080097028-A1 POLYMERIC BEADS FOR OLIGOMER SYNTHESIS LSIS PHARMACEUTICALS, INC. (US) 2008-04-24 US disclosed
US-7348391-B2 Polymeric beads for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2008-03-25 US disclosed
US-20080021224-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2008-01-24 US disclosed
CN-101076546-A Polymeric beads for oligomer synthesis ISIS PHARMACEUTICALS INC (US) 2007-11-21 CN disclosed
US-20070265435-A1 PROCESS FOR THE SYNTHESIS OF OLIGOMERIC COMPOUNDS RAVIKUMAR VASULINGA T 2007-11-15 US disclosed
EP-1028124-B1 Improved deprotection method for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS INC (US) 2007-10-31 EP disclosed
US-7276599-B2 Oligonucleotide synthesis with alternative solvents ISIS PHARMACEUTICALS, INC. (US) 2007-10-02 US disclosed
US-7273933-B1 Methods for synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2007-09-25 US disclosed
US-20070196847-A1 METHODS FOR DETECTION OF CHLORAL HYDRATE IN DICHLOROACETIC ACID ISIS PHARMACEUTICALS, INC. (US) 2007-08-23 US disclosed
EP-1490515-A4 CHLORAL-FREE DCA IN OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS INC (US) 2007-07-11 EP disclosed
US-7227016-B2 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2007-06-05 US disclosed
US-7227015-B2 Synthesis of sulfurized oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2007-06-05 US disclosed
US-20070123703-A1 CHLORAL-FREE DCA IN OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2007-05-31 US disclosed
EP-1789460-A2 POLYMERIC BEADS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2007-05-30 EP disclosed
EP-1379698-A4 MOBILITY-MODIFIED NUCLEOBASE POLYMERS AND METHODS OF USING SAME APPLERA CORP (US) 2007-04-25 EP disclosed
US-7202264-B2 Supports such as glass and styrene polymers functionalized with tricyclic hetercyclic anhydrides and imides, used in the preparation of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2007-04-10 US disclosed
US-7199236-B2 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2007-04-03 US disclosed
US-7186822-B2 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2007-03-06 US disclosed
US-7173123-B2 Methods for detection of chloral hydrate in dichloroacetic acid ISIS PHARMACEUTICALS, INC. (US) 2007-02-06 US disclosed
US-20070026434-A1 Mobility-Modified Nucleobase Polymers and Methods of Using Same APPLERA CORPORATION (US) 2007-02-01 US disclosed
US-7169916-B2 Chloral-free DCA in oligonucleotide synthesis ISIS PHARMACEUTICALS, INC. (US) 2007-01-30 US disclosed
US-RE39464-E1 Oligonucleolotides having site specific chiral phosphorothioate internucleoside linkages ISIS PHARMACEUTICALS INC. (US) 2007-01-09 US disclosed
US-20070004911-A1 Silylated oligonucleotide compounds AVECIA LIMITED (GB) 2007-01-04 US disclosed
EP-1737878-A2 PROCESS AND REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS AND PURIFICATION Alnylam Pharmaceuticals Inc. (US) 2007-01-03 EP disclosed
EP-1356115-B1 METHODS FOR DETECTION OF CHLORAL HYDRATE IN DICHLOROACETIC ACID ISIS PHARMACEUTICALS INC (US) 2006-11-29 EP disclosed
US-RE39324-E1 Pyrimidine derivatives and oligonucleotides containing same ISIS PHARMACEUTICALS, INC. (US) 2006-10-03 US disclosed
US-20060149052-A1 Process for the preparation of oligonucleotides AVECIA LIMITED (GB) 2006-07-06 US disclosed
US-7057027-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2006-06-06 US disclosed
EP-1660512-A2 OLIGONUCLEOTIDE SYNTHESIS WITH ALTERNATIVE SOLVENTS ISIS PHARMACEUTICALS, INC. (US) 2006-05-31 EP disclosed
EP-0904275-B1 PREPARATION OF PHOSPHOROTHIOATE OLIGOMERS UNIV MCGILL (CA) 2006-05-17 EP disclosed
US-7041816-B2 solid phase deprotection of cyanoethyl groups on the phosphorothioate backbone of an oligonucleotide with an amine deprotecting agent (triethylamine); cleaving the oligonucleotide from the support; minimal acrylonitrile nucleobase adduct formation; by-product inhibition ISIS PHARMACEUTICALS, INC. (US) 2006-05-09 US disclosed
US-20060089494-A1 Method for preparing oligonucleotides GIRINDUS AG (DE) 2006-04-27 US disclosed
WO-2006029023-A2 POLYMERIC BEADS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2006-03-16 WO disclosed
CN-1747963-A Process for preparing oligonucleotides AVECIA LTD (GB) 2006-03-15 CN disclosed
US-20060051800-A1 Polymeric beads for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2006-03-09 US disclosed
US-20060041114-A1 Activators for oligonucleotide synthesis NITTO DENKO AVECIA, INC. 2006-02-23 US disclosed
US-20060040308-A1 Compounds and methods for the characterization of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2006-02-23 US disclosed
US-7002006-B2 Protection of nucleosides ISIS PHARMACEUTICALS, INC. (US) 2006-02-21 US disclosed
US-20060036028-A1 Process for preparing oligonucleotides NITTO DENKO AVECIA, INC. 2006-02-16 US disclosed
EP-1404696-B1 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS AVECIA BIOTECHNOLOGY INC (US) 2006-02-08 EP disclosed
EP-1097162-B1 OLIGONUCLEOTIDES HAVING SITE SPECIFIC CHIRAL PHOSPHOROTHIOATE INTERNUCLEOSIDE LINKAGES ISIS PHARMACEUTICALS INC (US) 2006-01-18 EP disclosed
US-20060003952-A1 Oligomeric compounds having modified phosphate groups ISIS PHARMACEUTICALS, INC. (US) 2006-01-05 US disclosed
EP-1608669-A1 SILYLATED OLIGONUCLEOTIDE COMPOUNDS Avecia Limited (GB) 2005-12-28 EP disclosed
US-20050267300-A1 Processes and reagents for oligonucleotide synthesis and purification ALNYLAM PHARMACEUTICALS 2005-12-01 US disclosed
US-6967079-B2 Pyrimidine derivatives for labeled binding partners ISIS PHARMACEUTICALS, INC. (US) 2005-11-22 US disclosed
WO-2005108411-A2 SUBSTITUTED PIXYL PROTECTING GROUPS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2005-11-17 WO disclosed
US-6962783-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2005-11-08 US disclosed
WO-2005097817-A2 PROCESS AND REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS AND PURIFICATION ALNYLAM PHARMACEUTICALS, INC. (US) 2005-10-20 WO disclosed
US-6951931-B2 Pyrimidine derivatives for labeled binding partners ISIS PHARMACEUTICALS, INC. (US) 2005-10-04 US disclosed
US-20050208588-A1 Supports for oligomer synthesis ISIS PHARMACEUTICALS, INC. (US) 2005-09-22 US disclosed
EP-1575975-A1 PROCESS FOR THE PREPARATION OF OLIGONUCLEOTIDES Avecia Limited (GB) 2005-09-21 EP disclosed
US-20050182251-A1 Process for the synthesis of oligomeric compounds IONIS PHARMACEUTICALS, INC. 2005-08-18 US disclosed
CN-1649889-A Process for preparing oligonucleotides AVECIA LTD (GB) 2005-08-03 CN disclosed
US-20050165226-A1 Synthesis of sulfurized oligonucleotides ISIS PHARMACEUTICALS INC. 2005-07-28 US disclosed
US-20050137390-A1 Process for the synthesis of oligomeric compounds IONIS PHARMACEUTICALS, INC. 2005-06-23 US disclosed
US-20050137391-A1 Process for the synthesis of oligomeric compounds IONIS PHARMACEUTICALS, INC. 2005-06-23 US disclosed
US-20050113569-A1 Methods for detection of chloral hydrate in dichloroacetic acid ISIS PHARMACEUTICALS, INC. 2005-05-26 US disclosed
EP-1525212-A1 METHOD FOR PREPARING OLIGONUCLEOTIDES Girindus AG (DE) 2005-04-27 EP disclosed
US-20050075490-A1 Chloral-free DCA in oligonucleotide synthesis IONIS PHARMACEUTICALS, INC. 2005-04-07 US disclosed
US-6875593-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2005-04-05 US disclosed
US-6870039-B2 Synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 2005-03-22 US disclosed
WO-2005020885-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF SEVERE ACUTE RESPIRATORY SYNDROME (SARS) ISIS PHARMACEUTICALS, INC. (US) 2005-03-10 WO disclosed
US-6861518-B2 Hybrid oligonucleotide MCGILL UNIVERSITY (CA) 2005-03-01 US disclosed
US-20050042644-A1 Mobility-modified nucleobase polymers and methods of using same APPLERA CORPORATION (US) 2005-02-24 US disclosed
EP-1317466-B1 SYNTHONS FOR OLIGONUCLEOTIDE SYNTHESIS AVECIA BIOTECHNOLOGY INC (US) 2005-02-23 EP disclosed
US-6858722-B2 Oligomer phosphoramidite compositions and processes for synthesizing the same ISIS PHARMACEUTICALS, INC. (US) 2005-02-22 US disclosed
US-6858715-B2 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2005-02-22 US disclosed
US-20050026192-A1 Oligonucleotide synthesis with alternative solvents ISIS PHARMACEUTICALS, INC. (US) 2005-02-03 US disclosed
EP-1501851-A1 PROCESS FOR PREPARING OLIGONUCLEOTIDES Avecia Limited (GB) 2005-02-02 EP disclosed
US-20050020826-A1 Pyrimidine derivatives for labeled binding partners LIN KUEI-YING (US) 2005-01-27 US disclosed
US-6846922-B1 Reacting phosphoramidite with hydroxyl group of nucleoside or oligonucleotide linked to solid support in presence of activating reagent comprising at least one pyridinium salt and at least one substituted imidazole ISIS PHARMACEUTICALS, INC. (US) 2005-01-25 US disclosed
US-20040265802-A9 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES FROEHLER BRIAN (US) 2004-12-30 US disclosed
WO-2004113553-A2 METHOD OF PRODUCING PURE AMIDITES AND OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2004-12-29 WO disclosed
EP-1490515-A1 CHLORAL-FREE DCA IN OLIGONUCLEOTIDE SYNTHESIS ISIS Pharmaceuticals, Inc. (US) 2004-12-29 EP disclosed
WO-2004108081-A2 OLIGONUCLEOTIDE SYNTHESIS WITH ALTERNATIVE SOLVENTS ISIS PHARMACEUTICALS, INC. (US) 2004-12-16 WO disclosed
EP-1023310-B1 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2004-12-08 EP disclosed
EP-1027364-B1 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS INC (US) 2004-12-08 EP disclosed
US-20040242897-A1 Universal support media for synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. 2004-12-02 US disclosed
US-6825338-B2 SELECTIVE FUNCTIONALIZATION OF OLIGONUCLEOTIDES WITH CONJUGATE GROUPS WITHOUT THE NEED FOR POST-SYNTHETIC LABELING; SOLID PHASE SYNTHESIS; DEBLOCKING AN ACID LABILE HYDROXYL GROUP AND REACTING WITH A PHOSPHORAMIDITE ISIS PHARMACEUTICALS, INC. 2004-11-30 US disclosed
CN-1549820-A Activators for oligonucleotide synthesis ƽ 2004-11-24 CN disclosed
US-20040220395-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. 2004-11-04 US disclosed
US-20040219577-A1 Process for the synthesis of oligomeric compounds IONIS PHARMACEUTICALS, INC. 2004-11-04 US disclosed
US-6809195-B1 COMPRISES A MODIFIED PHOSPHORAMIDITE PROTOCOL IN WHICH OXIDATION AND CAPPING STEPS ARE COMBINED INTO A SINGLE STEP; INCREASED EFFICIENCY; SOLID PHASE SYNTHESIS ISIS PHARMACEUTICALS, INC. 2004-10-26 US disclosed
WO-2004085454-A1 SILYLATED OLIGONUCLEOTIDE COMPOUNDS AVECIA LIMITED (GB) 2004-10-07 WO disclosed
US-20040198972-A1 Processes for the preparation of oligonucleotides ISIS PHARMACEUTICALS, INC. 2004-10-07 US disclosed
EP-0948512-B1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2004-10-06 EP disclosed
US-6800743-B2 FOR USE AS LABELS IN DIAGNOSTIC ASSAYS AND IN ENHANCING BINDING TO COMPLEMENTARY BASES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-20040185491-A1 Methods for synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2004-09-23 US disclosed
WO-2004072234-A2 PROTECTION OF NUCLEOSIDES ISIS PHARMACEUTICALS, INC. (US) 2004-08-26 WO disclosed
US-6780989-B2 HYBRID OLIGONUCLEOTIDE ISIS PHARMACEUTICALS, INC. 2004-08-24 US disclosed
US-20040158055-A1 Protection of nucleosides IONIS PHARMACEUTICALS, INC. 2004-08-12 US disclosed
US-20040152905-A1 Universal building blocks and support media for synthesis of oligonucleotides and their analogs ISIS PHARMACEUTICALS, INC. 2004-08-05 US disclosed
EP-0986571-B1 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS AVECIA BIOTECHNOLOGY INC (US) 2004-07-14 EP disclosed
US-6762281-B2 GENERATING PREFERENTIAL OLIGOMERS; GENERATE OLIGOMER, DEPROTECT, EXPOSE TO PHOSPHOROUS, OXIDIZE, EXPOSE TO SULFUR, CLEAVE, RECOVER PRODUCT ISIS PHARMACEUTICALS, INC. 2004-07-13 US disclosed
WO-2004055036-A1 PROCESS FOR THE PREPARATION OF OLIGONUCLEOTIDES AVECIA LIMITED (GB) 2004-07-01 WO disclosed
EP-1356115-A4 METHODS FOR DETECTION OF CHLORAL HYDRATE IN DICHLOROACETIC ACID ISIS PHARMACEUTICALS INC (US) 2004-06-23 EP disclosed
EP-1119578-B1 IMPROVED PROCESS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS INC (US) 2004-06-16 EP disclosed
US-6743905-B2 BIOPOLYMER FOR USE IN THE DETECTION OF PREERENTIAL SEQUENCES IN SAMPLE APPLERA CORPORATION 2004-06-01 US disclosed
EP-1084134-A4 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS INC (US) 2004-05-26 EP disclosed
US-20040097722-A9 Preparation of phosphorothioate oligomers MCGILL UNIVERSITY 2004-05-20 US disclosed
US-20040082774-A1 Novel phosphate and thiophosphate protecting groups ISIS PHARMACEUTICALS, INC. 2004-04-29 US disclosed
CN-1489633-A Method for detecting chloral hydrate in dichloroacetic acid ISISҩ�﹫˾ 2004-04-14 CN disclosed
EP-1404696-A1 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS Avecia Biotechnology, Inc. (US) 2004-04-07 EP disclosed
US-20040063925-A1 Synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2004-04-01 US disclosed
WO-2004013154-A1 METHOD FOR PREPARING OLIGONUCLEOTIDES GIRINDUS AG (DE) 2004-02-12 WO disclosed
WO-2004011474-A1 UNIVERSAL SUPPORT MEDIA FOR SYNTHESIS OF OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2004-02-05 WO disclosed
EP-1386925-A1 Method for preparing oligonucleotides Girindus AG (DE) 2004-02-04 EP disclosed
EP-1379541-A1 LABELED OLIGONUCLEOTIDES, METHODS FOR MAKING SAME, AND COMPOUNDS USEFUL THEREFOR ISIS Pharmaceuticals, Inc. (US) 2004-01-14 EP disclosed
EP-1379698-A1 MOBILITY-MODIFIED NUCLEOBASE POLYMERS AND METHODS OF USING SAME Applera Corporation (US) 2004-01-14 EP disclosed
US-6677471-B2 USED FOR PREPARATION OF OLIGOMERIC COMPOUNDS HAVING PHOSPHITE, PHOSPHODIESTER, PHOSPHOROTHIOATE, PHOSPHORODITHIOATE OR OTHER LINKAGES ISIS PHARMACEUTICALS, INC. 2004-01-13 US disclosed
US-20030229218-A1 Synthons for oligonucleotide synthesis AVECIA BIOTECHNOLOGY INC. 2003-12-11 US disclosed
US-20030229220-A1 Oligomer phosphoramidite compositions and processes for synthesizing the same RAVIKUMAR VASULINGA T (US) 2003-12-11 US disclosed
US-20030229219-A1 Preparation of phosphorothioate oligomers ISIS PHARMACEUTICALS, INC. 2003-12-11 US disclosed
US-6653468-B1 Bicyclic heptane derivatives linked to controlled pore glass or copolymers of polystyrene; can be cleaved and used for subsequent reactions ISIS PHARMACEUTICALS, INC. 2003-11-25 US disclosed
US-6649750-B1 Nucleoside linked to a support through heterocyclic base and amide bond; deblocking/deprotecting; capping/oxidizing; purity; reduced levels of byproducts containing abasic sites ISIS PHARMACEUTICALS, INC. 2003-11-18 US disclosed
US-20030212267-A1 Synthesis of sulfurized oligonucleotides IONIS PHARMACEUTICALS, INC. 2003-11-13 US disclosed
US-6645716-B2 Detecting nuclear magnetic resonance spectrum of chloral hydrate in sample; obtain sample of dichloroacetic acid, monitor resonance spectrum for presence of chloral hydrate ISIS PHARMACEUTICALS, INC. 2003-11-11 US disclosed
US-6646114-B2 Especially phosphorothioate oligonucleotides, and to intermediates used in that process; solution phase synthesis having improved efficiencies and enhanced convenience and cost ISIS PHARMACEUTICALS, INC. 2003-11-11 US disclosed
US-20030208061-A1 Labeled oligonucleotides, methods for making same, and compounds useful therefor ISIS PHARMACEUTICALS, INC. 2003-11-06 US disclosed
WO-2003091267-A1 PROCESS FOR PREPARING OLIGONUCLEOTIDES AVECIA LIMITED (GB) 2003-11-06 WO disclosed
US-20030207824-A1 Pyrimidine derivatives for labeled binding partners MATTEUCCI MARK D (US) 2003-11-06 US disclosed
US-6642373-B2 Phosphitylating using pyridinium salt activators; forming phosphorate or phosphorothioate intersugar linkages ISIS PHARMACEUTICALS, INC. 2003-11-04 US disclosed
EP-1356115-A1 METHODS FOR DETECTION OF CHLORAL HYDRATE IN DICHLOROACETIC ACID ISIS PHARMACEUTICALS, INC. (US) 2003-10-29 EP disclosed
WO-2003085136-A1 CHLORAL-FREE DCA IN OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2003-10-16 WO disclosed
US-20030191304-A1 Activators for oligonucleotide synthesis IONIS PHARMACEUTICALS, INC. 2003-10-09 US disclosed
US-20030190626-A1 Phosphorothioate monoester modified oligomers ISIS PHARMACEUTICALS, INC. 2003-10-09 US disclosed
US-20030176677-A1 Pyrimidine derivatives for labeled binding partners IONIS PHARMACEUTICALS, INC. 2003-09-18 US disclosed
US-20030170680-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines FROEHLER BRIAN (US) 2003-09-11 US disclosed
US-6617437-B1 Modified oligonucleotide of given formula; useful in diagnostics and therapeutics ISIS PHARMACEUTICALS, INC. 2003-09-09 US disclosed
US-6610842-B1 Removing hydroxyl protecting group from compound of given formula and treating with another compound; wide range of diagnostic and therapeutic uses ISIS PHARMACEUTICALS, INC. 2003-08-26 US disclosed
US-6610837-B1 Preparation of an oligonucleotide compound of given formula by reacting with given compounds, followed by oxidation or sulfurization ISIS PHARMACEUTICALS, INC. 2003-08-26 US disclosed
US-20030153743-A1 Processes for the synthesis of oligomeric compounds MANOHARAN MUTHIAH (US) 2003-08-14 US disclosed
US-20030149260-A1 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. 2003-08-07 US disclosed
US-6596857-B1 Oligomer for use as tool in human diagnostics and therapeutics MCGILL UNIVERSITY (CA) 2003-07-22 US disclosed
EP-1066308-A4 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2003-07-02 EP disclosed
US-20030114662-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2003-06-19 US disclosed
US-20030114660-A1 Preparation of phosphorothioate oligomers JUST GEORGE (CA) 2003-06-19 US disclosed
EP-1317466-A2 SYNTHONS FOR OLIGONUCLEOTIDE SYNTHESIS Avecia Biotechnology, Inc. (US) 2003-06-11 EP disclosed
WO-2003045969-A1 COUPLING REAGENT FOR H-PHOSPHONATE CHEMISTRY AVECIA BIOTECHNOLOGY INC. (US) 2003-06-05 WO disclosed
US-20030096980-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. 2003-05-22 US disclosed
EP-1311526-A1 PROCESSES FOR THE PREPARATION OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2003-05-21 EP disclosed
US-20030088088-A1 Process for the synthesis of oligomeric compounds IONIS PHARMACEUTICALS, INC. 2003-05-08 US disclosed
EP-0719272-B1 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS INC (US) 2003-05-07 EP disclosed
US-6559279-B1 Generation of peptide linked oligomers; generate solid support, expose to deprotecting agent, incubate with nucleoside, cap, cleave and recover peptide derivative ISIS PHARMACEUTICALS, INC. 2003-05-06 US disclosed
US-20030072712-A1 Pyrimidine derivatives for labeled binding partners LIN KUEI-YING (US) 2003-04-17 US disclosed
US-20030069412-A1 Synthesis of oligonucleotides RAVIKUMAR VASULINGA (US) 2003-04-10 US disclosed
EP-1246833-A4 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2003-04-09 EP disclosed
US-6531590-B1 Having bioreversible phosphate blocking groups, using a phosphoramite reactant carrying the phosphate blocking group; designed for cleavage by carboxyesterases to yield unprotected oligonucleotides ISIS PHARMACEUTICALS, INC. 2003-03-11 US disclosed
US-20030045698-A1 Compounds, processes and intermediates for synthesis of mixed backbone oligomeric compounds ISIS PHARMACEUTICALS, INC. 2003-03-06 US disclosed
US-6521775-B2 Genetically engineered oligonucleotides for use as diagnostic and therapeutic tools in gene therapy ISIS PHARMACEUTICALS, INC. 2003-02-18 US disclosed
EP-1244682-A4 PROCESS FOR THE PREPARATION OF OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS INC (US) 2003-02-05 EP disclosed
WO-2003004512-A1 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS AVECIA BIOTECHNOLOGY INC. (US) 2003-01-16 WO disclosed
US-6500944-B2 FOR SOLID PHASE BIOSYNTHESIS AVECIA BIOTECHNOLOGY, INC. 2002-12-31 US disclosed
US-20020182602-A1 Mobility-modified nucleobase polymers and methods of using same APPLIED BIOSYSTEMS, INC. 2002-12-05 US disclosed
US-6486312-B2 LIQUID PHASE BIOSYNTHESIS ISIS PHARMACEUTICALS, INC. 2002-11-26 US disclosed
EP-1256589-A2 Oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2002-11-13 EP disclosed
US-6476216-B1 Preparation of phosphorothioate oligomers MCGILL UNIVERSITY (CA) 2002-11-05 US disclosed
US-20020156235-A1 Process for preparing peptide derivatized oligomeric compounds IONIS PHARMACEUTICALS, INC. 2002-10-24 US disclosed
WO-2002083954-A1 MOBILITY-MODIFIED NUCLEOBASE POLYMERS AND METHODS OF USING SAME APPLERA CORPORATION (US) 2002-10-24 WO disclosed
EP-0637965-B1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES ISIS PHARMACEUTICALS INC (US) 2002-10-16 EP disclosed
US-6465628-B1 METHOD OF SYNTHESIS WITH DEPROTECTION OF OLIGOMERS ISIS PHARMACEUTICALS, INC. 2002-10-15 US disclosed
US-20020147331-A1 Methods for synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2002-10-10 US disclosed
WO-2002079216-A1 LABELED OLIGONUCLEOTIDES, METHODS FOR MAKING SAME, AND COMPOUNDS USEFUL THEREFOR ISIS PHARMACEUTICALS, INC. (US) 2002-10-10 WO disclosed
EP-1246833-A1 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2002-10-09 EP disclosed
US-6462184-B2 PROVIDING A PURINE OR PYRIMIDINE BASE CONTAINING NUCLEOSIDE WITH ACID LABILE HYDROXYL PROTECTING GROUP AND A BASE LABILE HYDROXY PROTECTING GROUP SUBSTITUTIONS, DEBLOCKING HYDROXY GROUP, TREATING WITH PHOSPHONATE COMPOUND, CONDENSING AGENT ISIS PHARMACEUTICALS, INC. 2002-10-08 US disclosed
EP-1244682-A1 PROCESS FOR THE PREPARATION OF OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2002-10-02 EP disclosed
EP-1175432-A4 PROCESSES FOR THE SYNTHESIS OF OLIGOMERS USING PHOSPHORAMIDITE COMPOSITIONS ISIS PHARMACEUTICALS INC (US) 2002-09-25 EP disclosed
EP-1212339-A4 2'-O-ACETAMIDO MODIFIED MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS INC (US) 2002-09-18 EP disclosed
US-20020128466-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2002-09-12 US disclosed
US-20020119483-A1 Methods for detection of chloral hydrate in dichloroacetic acid IONIS PHARMACEUTICALS, INC. 2002-08-29 US disclosed
EP-1159282-A4 COMPOUNDS, PROCESSES AND INTERMEDIATES FOR SYNTHESIS OF MIXED BACKBONE OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS INC (US) 2002-08-28 EP disclosed
US-6440943-B1 MIMIC AND/OR MODULATE THE ACTIVITY OF WILD-TYPE NUCLEIC ACIDS; THE 5' AND THE 3'-TERMINAL INTERNUCLEOSIDE LINKAGES ARE CHIRALLY SP AND INTERNAL INTERNUCLEOSIDE LINKAGES ARE CHIRALLY RP; RESISTANT TO NUCLEASE DEGRADATION; PSORIASIS ISIS PHARMACEUTICALS, INC. 2002-08-27 US disclosed
WO-2002062811-A2 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2002-08-15 WO disclosed
WO-2002061138-A1 METHODS FOR DETECTION OF CHLORAL HYDRATE IN DICHLOROACETIC ACID ISIS PHARMACEUTICALS, INC. (US) 2002-08-08 WO disclosed
US-6414127-B1 INCREASED AFFINITY TO COMPLEMENTARY OLIGONUCLEOTIDES; DNA SEQUENCING; MEDICAL DIAGNOSIS; NUCLEASE RESISTANCE ISIS PHARMACEUTICALS, INC. 2002-07-02 US disclosed
EP-1112279-A4 METHODS FOR THE PREPARATION OF CONJUGATED OLIGOMERS ISIS PHARMACEUTICALS INC (US) 2002-06-19 EP disclosed
EP-1212339-A1 2'-O-ACETAMIDO MODIFIED MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 2002-06-12 EP disclosed
US-6403781-B2 REACTING A PHOSPHORDIAMIDITE WITH A SUPPORT-BOUND SYNTHON TO FORM A SUPPORT BOUND PHOSPHORAMIDITE, PROTECTING TO FORM A SUPPORT BOUND PHOSHITE, SULFURIZING THE PHOSPHITE TO FORM A PROTECTED PHOSPHORTHIOATE AND DEPROTECTING ISIS PHARMACEUTICALS, INC. 2002-06-11 US disclosed
US-6399756-B1 OLIGONUCLEOTIDE ISIS PHARMACEUTICALS, INC. 2002-06-04 US disclosed
US-20020055623-A1 Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS. INC. 2002-05-09 US disclosed
US-6384209-B1 HIGHLY EFFIENT PROCESS BY CONTACTING OLIGONUCLEOTIDE HAVING INTERNUCLEOSIDE LINKAGE OF A PHOSPHOROUS III ATOM WITH A REAGENT OF DEFINED STRUCTURE; REAGENTS ARE INEXPENSIVE TO MAKE AND STABLE IN STORAGE AVECIA BIOTECHNOLOGY, INC. (GB) 2002-05-07 US disclosed
US-6380368-B1 GENETIC ENGINEERING ISIS PHARMACEUTICALS, INC. 2002-04-30 US disclosed
EP-1119578-A4 IMPROVED PROCESS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS INC (US) 2002-04-17 EP disclosed
WO-2002020543-A2 SYNTHONS FOR OLIGONUCLEOTIDE SYNTHESIS AVECIA BIOTECHNOLOGY INC. (US) 2002-03-14 WO disclosed
WO-2002020544-A1 PROCESS FOR PREPARING PEPTIDE DERIVATIZED OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2002-03-14 WO disclosed
EP-1097162-A4 OLIGONUCLEOTIDES HAVING SITE SPECIFIC CHIRAL PHOSPHOROTHIOATE INTERNUCLEOSIDE LINKAGES ISIS PHARMACEUTICALS INC (US) 2002-03-06 EP disclosed
WO-2002014340-A1 PROCESSES FOR THE PREPARATION OF OLIGONUCLEOTIDES_______________ ISIS PHARMACEUTICALS, INC. (US) 2002-02-21 WO disclosed
EP-1175432-A1 PROCESSES FOR THE SYNTHESIS OF OLIGOMERS USING PHUSPHORAMIDITE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 2002-01-30 EP disclosed
US-20020010326-A1 NOVEL SULFURIZING REAGENT 3-PHENYL-1,2,4-DITHIAZOLINE-5-ONE NITTO DENKO AVECIA, INC. 2002-01-24 US disclosed
US-6335437-B1 REACTING NUCLEOSIDE OR OLIGONUCLEOTIDE WITH ELECTROPHILIC HALOACETYL LINKER ISIS PHARMACEUTICALS, INC. 2002-01-01 US disclosed
EP-1159282-A1 COMPOUNDS, PROCESSES AND INTERMEDIATES FOR SYNTHESIS OF MIXED BACKBONE OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
US-6326478-B1 OLIGONUCLEOTIDES AND MEDICAL DIAGNOSIS, METABOLISM ISIS PHARMACEUTICALS, INC. 2001-12-04 US disclosed
EP-0948512-A4 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2001-10-24 EP disclosed
US-6294664-B1 PREPARING OLIGONUCLEOTIDE BLOCKS HAVING COMMON SUBSEQUENCES, PHOSPITYLATING, AND PERFORMING SOLID PHASE SYNTHESIS (SPS) TO FORM TARGET OLIGONUCLEOTIDES WHEREIN THE SYNTHONS USED IN SPS COMPRISE PHOSPHITYLATED OLIGONUCLEOTIDE BLOCKS ISIS PHARMACEUTICALS, INC. 2001-09-25 US disclosed
US-20010018510-A1 Synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2001-08-30 US disclosed
US-20010016652-A1 Compounds, processes and intermediates for synthesis of mixed backbone oligomeric compounds ISIS PHARMACEUTICALS, INC. 2001-08-23 US disclosed
US-6274725-B1 PROVIDING COMPOUND HAVING A HYDROXYL GROUP; REACTING WITH PHOSPHITYLATING REAGENT IN THE PRESENCE OF A PYRIDINUM SALT IN A SOLVENT UNDER CONDITIONS OF TIME, TEMPERATURE AND PRESSURE TO YIELD PHOSPHITYLATED COMPOUND ISIS PHARMACEUTICALS, INC. 2001-08-14 US disclosed
EP-1119578-A1 IMPROVED PROCESS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2001-08-01 EP disclosed
WO-2001051502-A1 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2001-07-19 WO disclosed
WO-2001049701-A1 PROCESS FOR THE PREPARATION OF OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2001-07-12 WO disclosed
EP-1112279-A1 METHODS FOR THE PREPARATION OF CONJUGATED OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 2001-07-04 EP disclosed
US-20010003132-A1 Method of synthesizing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. 2001-06-07 US disclosed
US-6242591-B1 Synthesis of sulfurized 2'-substituted oligonucleotides ISIS PHARMACEUTICALS, INC. 2001-06-05 US disclosed
EP-1023310-A4 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 2001-05-16 EP disclosed
EP-1097162-A2 OLIGONUCLEOTIDES HAVING SITE SPECIFIC CHIRAL PHOSPHOROTHIOATE INTERNUCLEOSIDE LINKAGES ISIS PHARMACEUTICALS, INC. (US) 2001-05-09 EP disclosed
US-6211350-B1 REACTING SYNTHON WITH TWO NUCLEOSIDE UNITS AND WITH SYNTHON HAVING ONE NUCLEOSIDE UNIT TO OBTAIN OLIGONUCLEOTIDE CONTAINING PHOSPHOROTHIOATE GROUPS ISIS PHARMACEUTICALS, INC. 2001-04-03 US disclosed
US-6207819-B1 SYNTHESIZING OLIGONUCLEOTIDE BY DEBLOCKING AND COUPLING NUCLEOTIDES TOGETHER, THEN TREATING WITH OXIDIZING SOLUTION TO CONVERT H-PHOSPHONATE LINKAGES TO PHOSPHODIESTER, PHOSPHOROTHIOATE, PHOSPHORAMIDATE OR BORANOPHOSPHATE ISIS PHARMACEUTICALS, INC. 2001-03-27 US disclosed
EP-1084134-A1 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2001-03-21 EP disclosed
WO-2001014400-A1 2'-O-ACETAMIDO MODIFIED MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 2001-03-01 WO disclosed
EP-1066308-A1 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2001-01-10 EP disclosed
US-6172217-B1 SULFURIZATION OF PHOSPORDIAMIDITE; DEBLOCKING ISIS PHARMACEUTICALS INC. 2001-01-09 US disclosed
US-6169177-B1 EFFICIENT REMOVAL OF ALLYL PROTECTING GROUPS DURING OLIGONUCLEOTIDE SYNTHESIS BY TREATING WITH SOLUTION OF CONCENTRATED AMMONIUM HYDROXIDE CONTAINING A MERCAPTO COMPOUND ISIS PHARMACEUTICALS, INC. 2001-01-02 US disclosed
US-6160152-A Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2000-12-12 US disclosed
US-6160109-A Preparation of phosphorothioate and boranophosphate oligomers ISIS PHARMACEUTICALS, INC. (US) 2000-12-12 US disclosed
WO-2000068241-A1 PROCESSES FOR THE SYNTHESIS OF OLIGOMERS USING PHUSPHORAMIDITE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 2000-11-16 WO disclosed
US-6147200-A NUCLEOSIDES FOR SOLID PHASE SYNTHESIS OF OLIGONUCLEOTIDES HAVING INCREASED NUCLEASE RESISTANCE AND BETTER BINDING AFFINITY; DIAGNOSIS; ANTISENSE THERAPY ISIS PHARMACEUTICALS, INC. (US) 2000-11-14 US disclosed
US-6124450-A Processes and intermediates for phosphorous-containing covalent linkages ISIS PHARMACEUTICALS, INC. (US) 2000-09-26 US disclosed
WO-2000055179-A1 NOVEL PHOSPHATE AND THIOPHOSPHATE PROTECTING GROUPS ISIS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed
US-6121437-A SYNTHESIS OF OLIGONUCLEOTIDES USING OLIGONUCLEOTIDES OR NUCLEOTIDES WITH PROTECTED INTERNUCLEOSIDIC PHOSPHORUS FUNCTIONALITIES WHICH CAN BE REMOVED UNDER MILD CONDITIONS AND PRODUCE NONTOXIC BY-PRODUCTS ISIS PHARMACEUTICALS, INC. (US) 2000-09-19 US disclosed
US-6114519-A PHOSPHITYLATION; OXIDATION ACYL DISULFIDE ISIS PHARMACEUTICALS, INC. (US) 2000-09-05 US disclosed
WO-2000047593-A1 COMPOUNDS, PROCESSES AND INTERMEDIATES FOR SYNTHESIS OF MIXED BACKBONE OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed
EP-1027364-A2 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS, INC. (US) 2000-08-16 EP disclosed
EP-1028124-A2 Improved process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2000-08-16 EP disclosed
EP-1023310-A1 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2000-08-02 EP disclosed
US-6096881-A Sulfur transfer reagents for oligonucleotide synthesis HYBRIDON, INC. (US) 2000-08-01 US disclosed
US-6084082-A SOLID PHASE SYNTHESIS BY ATTACHING BETA-LACTAM HAVING NUCLEOBASE TO SOLID SUPPORT, DEPROTECTING HYDROXY GROUP, REACTING FREE HYDROXYL GROUP WITH BETA-LACTAMTIDE HAVING ACTIVATED PHOSPHITE GROUP, AND OXIDIZING ISIS PHARMACEUTICALS, INC. (US) 2000-07-04 US disclosed
US-6069243-A USING ACETONITRILE HAVING WATER CONTENT BETWEEN 30 AND 1250 PPM AS WASHING AGENT BEFORE OR AFTER COUPLING OR OXIDATION STEPS OR AS OXIDIZING AGENT IN SOLID PHASE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2000-05-30 US disclosed
WO-2000027859-A1 IMPROVED PROCESSES FOR THE SYNTHESIS OF OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2000-05-18 WO disclosed
US-6051699-A Process for the synthesis of oligomeric compounds ISIS PHARMACEUTICALS, INC. (US) 2000-04-18 US disclosed
WO-2000020431-A1 IMPROVED PROCESS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 2000-04-13 WO disclosed
EP-0986571-A1 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS HYBRIDON, INC. (US) 2000-03-22 EP disclosed
WO-2000014098-A1 METHODS FOR THE PREPARATION OF CONJUGATED OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 2000-03-16 WO disclosed
US-6031092-A Preparation of phosphorothioate oligomers MC GILL UNIVERSITY (CA) 2000-02-29 US disclosed
US-6028183-A Pyrimidine derivatives and oligonucleotides containing same GILEAD SCIENCES, INC. (US) 2000-02-22 US disclosed
US-6020475-A Process for the synthesis of oligomeric compounds ISIS PHARMEUTICALS, INC. (US) 2000-02-01 US disclosed
WO-2000004034-A2 OLIGONUCLEOTIDES HAVING SITE SPECIFIC CHIRAL PHOSPHOROTHIOATE INTERNUCLEOSIDE LINKAGES ISIS PHARMACEUTICALS, INC. (US) 2000-01-27 WO disclosed
US-6007992-A MIXING DERIVATIVE WITH A SAMPLE CONTAINING TARGET NUCLEIC ACIDS, AND INCUBATING FORMING A COMPLEX; FOR DIAGNOSTIC ASSAYS AND TO ENHANCE BINDING TO COMPLEMENTARY BASES GILEAD SCIENCES, INC. (US) 1999-12-28 US disclosed
US-6005096-A FOR OLIGONUCLEOTIDES THAT ARE MODIFIED TO ENHANCE THE BINDING AFFINITY AND TO BEAR DETECTABLE LABELS; FOR DIAGNOSTIC USE GILEAD SCIENCES, INC. (US) 1999-12-21 US disclosed
US-6001982-A Synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 1999-12-14 US disclosed
WO-1999062922-A1 ACTIVATORS FOR OLIGONUCLEOTIDE SYNTHESIS ISIS PHARMACEUTICALS, INC. (US) 1999-12-09 WO disclosed
EP-0948512-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1999-10-13 EP disclosed
WO-1999043694-A1 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1999-09-02 WO disclosed
US-5945521-A Preparation of phosphorothioate oligomers MCGILL UNIVERSITY (CA) 1999-08-31 US disclosed
WO-1999024452-A9 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS INC (US) 1999-08-12 WO disclosed
WO-1999024452-A2 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS, INC. (US) 1999-05-20 WO disclosed
WO-1999019340-A1 IMPROVED SYNTHESIS OF SULFURIZED OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1999-04-22 WO disclosed
WO-1998054198-A9 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS HYBRIDON INC (US) 1999-04-01 WO disclosed
EP-0904275-A1 PREPARATION OF PHOSPHOROTHIOATE OLIGOMERS McGILL UNIVERSITY (CA) 1999-03-31 EP disclosed
US-5866691-A Lactam nucleic acids ISIS PHARMACEUTICALS, INC. (US) 1999-02-02 US disclosed
WO-1999003873-A2 NOVEL SULFURIZING REAGENT 3-PHENYL-1,2,4-DITHIAZOLINE-5-ONE HYBRIDON, INC. (US) 1999-01-28 WO disclosed
US-5859232-A Process for the synthesis of oligomeric phosphite, phosphodiester, phosphorothioate and phosphorodithioate compounds ISIS PHARMACEUTICALS, INC. (US) 1999-01-12 US disclosed
EP-0766688-A4 SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS INC (US) 1998-12-30 EP disclosed
US-5852168-A Sulfurization of phosphorus-containing compounds REGENTS OF THE UNIVERSITY OF MINESOTA (US) 1998-12-22 US disclosed
US-5847106-A Monomeric and dimeric nucleosides with silyl-containing diamino phosphorous linkages ISIS PHARMACEUTICALS INC. (US) 1998-12-08 US disclosed
WO-1998054198-A1 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS HYBRIDON, INC. (US) 1998-12-03 WO disclosed
WO-1998049181-A1 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS HYBRIDON, INC. (US) 1998-11-05 WO disclosed
US-5830653-A ABILITY TO INHIBIT GENE EXPRESSION GILEAD SCIENCES, INC. (US) 1998-11-03 US disclosed
WO-1998029427-A1 METHOD OF SYNTHESIZING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO disclosed
US-5763588-A Pyrimidine derivatives for labeled binding partners GILEAD SCIENCES, INC. (US) 1998-06-09 US disclosed
US-5734041-A Preparation of chiral phosphorothioate oligomers MCGILL UNIVERSITY (CA) 1998-03-31 US disclosed
WO-1998008809-A1 NOVEL SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS HYBRIDON, INC. (US) 1998-03-05 WO disclosed
US-5705621-A Oligomeric phosphite, phosphodiester, Phosphorothioate and phosphorodithioate compounds and intermediates for preparing same ISIS PHARMACEUTICALS, INC. (US) 1998-01-06 US disclosed
WO-1997041130-A2 SULFURIZATION OF PHOSPHORUS-CONTAINING COMPOUNDS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1997-11-06 WO disclosed
US-5645985-A USED FOR DIAGNOSIS TO DETECT VIRUSES OR DISEASED CONDITIONS GILEAD SCIENCES, INC. (US) 1997-07-08 US disclosed
WO-1997014710-A1 PREPARATION OF PHOSPHOROTHIOATE OLIGOMERS MCGILL UNIVERSITY (US) 1997-04-24 WO disclosed
EP-0766688-A1 SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1997-04-09 EP disclosed
US-5614621-A Process for preparing oligonucleotides using silyl-containing diamino phosphorous reagents ISIS PHARMACEUTICALS, INC. (US) 1997-03-25 US disclosed
US-5594121-A DETECT VIRUSES, DISEASES GILEAD SCIENCES, INC. (US) 1997-01-14 US disclosed
US-5571902-A OLIGOMERIZATION IN THE PRESENCE OF TETRAZOLE COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 1996-11-05 US disclosed
US-5554746-A Lactam nucleic acids ISIS PHARMACEUTICALS, INC. (US) 1996-09-10 US disclosed
EP-0719272-A1 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS GILEAD SCIENCES, INC. (US) 1996-07-03 EP disclosed
US-5502177-A POLYCYCLIC STRUCTURE BOUND TO OLIGONUCLEOTIDE, FLUORESCENT LABEL, IMMUNOASSAY GILEAD SCIENCES, INC. (US) 1996-03-26 US disclosed
EP-0695306-A1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PURINES GILEAD SCIENCES, INC. (US) 1996-02-07 EP disclosed
EP-0637965-A4 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES. GILEAD SCIENCES INC (US) 1996-01-24 EP disclosed
WO-1995032980-A1 SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1995-12-07 WO disclosed
EP-0653438-A2 Oligonucleotide compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-17 EP disclosed
WO-1995007918-A2 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS GILEAD SCIENCES, INC. (US) 1995-03-23 WO disclosed
EP-0637965-A1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES GILEAD SCIENCES, INC. (US) 1995-02-15 EP disclosed
WO-1994024144-A2 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PURINES GILEAD SCIENCES, INC. (US) 1994-10-27 WO disclosed
WO-1993013118-A1 SYNTHESIS OF PHOSPHOROTHIOATE ANALOGUES OF OLIGO- AND POLYNUCLEOTIDES KING'S COLLEGE LONDON (GB) 1993-07-08 WO disclosed
WO-1993010820-A1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES GILEAD SCIENCES, INC. (US) 1993-06-10 WO disclosed
US-4399075-A Process for producing chlorinated phenoxytoluene derivatives ASAHI CHEMICAL COMPANY, LIMITED (JP) 1983-08-16 US disclosed
US-4399075-A Process for producing chlorinated phenoxytoluene derivatives ASAHI CHEMICAL COMPANY, LIMITED (JP) 1983-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030190626-A1 Phosphorothioate monoester modified oligomers DCLRE1B, SNRPE, POLRMT CES1 3375/4885CES2 4338/4885TSHR 2653/4885
US-20210309690-A1 OLIGONUCLEOTIDE SYNTHESIS RNGTT, RTCB, TYMS CES1 2428/4885CES2 3597/4885TSHR 2070/4885
US-20020128466-A1 Method of synthesizing phosphorothioate oligonucleotides RNGTT, TYMP, MTAP CES1 3379/4885CES2 4411/4885TSHR 1934/4885
US-20030114662-A1 Method of synthesizing phosphorothioate oligonucleotides RNGTT, TYMP, MTAP CES1 3379/4885CES2 4411/4885TSHR 1934/4885
US-20070026434-A1 Mobility-Modified Nucleobase Polymers and Methods of Using Same PCNA, PNKP, SAMHD1 CES1 4015/4885CES2 3182/4885TSHR 3939/4885
US-20020182602-A1 Mobility-modified nucleobase polymers and methods of using same PCNA, PNKP, SAMHD1 CES1 4015/4885CES2 3182/4885TSHR 3939/4885
US-20120071640-A1 Sulfurizing reagents and their use for oligonucleotides synthesis RRM1, SRRT, NSUN2 CES1 2337/4885CES2 3785/4885TSHR 1504/4885
US-20020156235-A1 Process for preparing peptide derivatized oligomeric compounds IAPP, PTMS, NGLY1 CES1 4792/4885CES2 4881/4885TSHR 3062/4885
US-20090286085-A1 POLYMERIC BEADS FOR OLIGOMER SYNTHESIS NEFM, NOD2, MACF1 CES1 4712/4885CES2 4601/4885TSHR 4838/4885
US-20050137391-A1 Process for the synthesis of oligomeric compounds PFAS, DIS3, EXOSC4 CES1 3984/4885CES2 2639/4885TSHR 3941/4885
US-20060036028-A1 Process for preparing oligonucleotides RTCB, POLRMT, POLM CES1 2004/4885CES2 3168/4885TSHR 3722/4885
US-20030208061-A1 Labeled oligonucleotides, methods for making same, and compounds useful therefor METTL16, BCDIN3D, GARS1 CES1 1444/4885CES2 1668/4885TSHR 3410/4885
US-20040185491-A1 Methods for synthesis of oligonucleotides RNGTT, POLL, TYMP CES1 3140/4885CES2 2529/4885TSHR 970/4885
US-20040063925-A1 Synthesis of oligonucleotides RNGTT, POLRMT, POLI CES1 3229/4885CES2 4046/4885TSHR 2331/4885
US-20100069623-A1 Method for preparing oligonucleotides RNGTT, NSUN2, RNMT CES1 2452/4885CES2 2762/4885TSHR 2547/4885
US-11608355-B2 Technologies for oligonucleotide preparation POLRMT, DCLRE1B, RNGTT CES1 2271/4885CES2 4249/4885TSHR 2860/4885
US-20010003132-A1 Method of synthesizing phosphorothioate oligonucleotides RNGTT, TYMP, MTAP CES1 3379/4885CES2 4411/4885TSHR 1934/4885
US-20030072712-A1 Pyrimidine derivatives for labeled binding partners DDB1, RRBP1, PRPF31 CES1 2896/4885CES2 3970/4885TSHR 2809/4885
US-20120289691-A1 PROTECTED MONOMER AND METHOD OF FINAL DEPROTECTION FOR RNA SYNTHESIS NSUN2, SNRPB2, RNGTT CES1 4258/4885CES2 3112/4885TSHR 1669/4885
US-20020010326-A1 NOVEL SULFURIZING REAGENT 3-PHENYL-1,2,4-DITHIAZOLINE-5-ONE BPNT1, DNTT, TST CES1 3159/4885CES2 3454/4885TSHR 3174/4885
US-20030170680-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines NUDT1, DHX15, DDX5 CES1 3840/4885CES2 4627/4885TSHR 3775/4885
US-20110196145-A1 PROCESS FOR DESILYLATION OF OLIGONUCLEOTIDES ALKBH1, DIMT1, RNGTT CES1 1507/4885CES2 964/4885TSHR 3087/4885
US-20060040308-A1 Compounds and methods for the characterization of oligonucleotides POLRMT, DCLRE1B, RNGTT CES1 1142/4885CES2 1054/4885TSHR 2682/4885
US-20260008806-A1 TECHNOLOGIES FOR OLIGONUCLEOTIDE PREPARATION RNGTT, RNMT, NSUN2 CES1 1538/4885CES2 1633/4885TSHR 1346/4885
US-20030229220-A1 Oligomer phosphoramidite compositions and processes for synthesizing the same PHOSPHO1, OSGEP, DTYMK CES1 4262/4885CES2 4548/4885TSHR 3963/4885
US-20230002438-A1 COMPOSITIONS COMPRISING DICHLOROACETIC ACID, PROCESSES FOR PREPARING SAME AND USES THEREOF AGXT, DDC, GRHPR CES1 921/4885CES2 516/4885TSHR 4683/4885
US-20090306358-A1 SULFUR TRANSFER REAGENTS FOR OLIGONUCLEOTIDE SYNTHESIS POLRMT, TST, DNTT CES1 3968/4885CES2 3824/4885TSHR 2699/4885
US-20060051800-A1 Polymeric beads for oligomer synthesis NEFM, NOD2, MACF1 CES1 4712/4885CES2 4601/4885TSHR 4838/4885
US-20100137572-A1 OXIDATION PROCESS POLRMT, POLN, POLB CES1 4341/4885CES2 4333/4885TSHR 1981/4885
US-20090131682-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ILK, NOP2, PFAS CES1 4288/4885CES2 2416/4885TSHR 4585/4885
US-20080097028-A1 POLYMERIC BEADS FOR OLIGOMER SYNTHESIS NEFM, NOD2, MACF1 CES1 4712/4885CES2 4601/4885TSHR 4838/4885
US-20040198972-A1 Processes for the preparation of oligonucleotides RNGTT, RNMT, NUDT1 CES1 3662/4885CES2 3982/4885TSHR 3203/4885
US-20030088088-A1 Process for the synthesis of oligomeric compounds PFAS, DIS3, EXOSC4 CES1 3984/4885CES2 2639/4885TSHR 3941/4885
US-20060041114-A1 Activators for oligonucleotide synthesis MED12, RBM12, RPS12 CES1 1315/4885CES2 2838/4885TSHR 1293/4885
US-20050182251-A1 Process for the synthesis of oligomeric compounds PFAS, DIS3, EXOSC4 CES1 3984/4885CES2 2639/4885TSHR 3941/4885
US-12435105-B2 Technologies for oligonucleotide preparation POLRMT, DCLRE1B, RNGTT CES1 2271/4885CES2 4249/4885TSHR 2860/4885
US-20050075490-A1 Chloral-free DCA in oligonucleotide synthesis DCLRE1B, DCTD, DDT CES1 422/4885CES2 235/4885TSHR 678/4885
US-20070265435-A1 PROCESS FOR THE SYNTHESIS OF OLIGOMERIC COMPOUNDS PFAS, DIS3, EXOSC4 CES1 3984/4885CES2 2639/4885TSHR 3941/4885
US-20040265802-A9 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES NUDT1, DHX15, DDX5 CES1 3840/4885CES2 4627/4885TSHR 3775/4885
US-20090005549-A1 Processes and Reagents for Desilylation of Oligonucleotides ALKBH1, DIMT1, RNGTT CES1 1520/4885CES2 990/4885TSHR 2468/4885
US-20120165547-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ILK, NOP2, PFAS CES1 4288/4885CES2 2416/4885TSHR 4585/4885
US-20010016652-A1 Compounds, processes and intermediates for synthesis of mixed backbone oligomeric compounds PPIP5K2, NUDT1, ITPA CES1 4236/4885CES2 3951/4885TSHR 4500/4885
US-20030153743-A1 Processes for the synthesis of oligomeric compounds PPIP5K2, NUDT21, NUDT1 CES1 4073/4885CES2 4735/4885TSHR 3095/4885
US-20080021224-A1 SUPPORTS FOR OLIGOMER SYNTHESIS ILK, NOP2, PFAS CES1 4288/4885CES2 2416/4885TSHR 4585/4885
US-20030229218-A1 Synthons for oligonucleotide synthesis POLI, TYMP, POLRMT CES1 2738/4885CES2 4053/4885TSHR 1349/4885
US-20040219577-A1 Process for the synthesis of oligomeric compounds PFAS, DIS3, EXOSC4 CES1 3984/4885CES2 2639/4885TSHR 3941/4885
US-20060149052-A1 Process for the preparation of oligonucleotides CPSF7, CPSF1, CPSF6 CES1 3456/4885CES2 3594/4885TSHR 2641/4885
US-20040152905-A1 Universal building blocks and support media for synthesis of oligonucleotides and their analogs POLM, POLRMT, POLB CES1 3785/4885CES2 4432/4885TSHR 3397/4885
US-20150240053-A1 POLYSULFIDE ADDITIVE, METHOD FOR PRODUCTION THEREOF AND USE THEREOF IN RUBBER MIXTURES PUF60, RPS21, RPS4Y1 CES1 3782/4885CES2 2001/4885TSHR 4724/4885
US-20030176677-A1 Pyrimidine derivatives for labeled binding partners DDB1, RRBP1, PRPF31 CES1 2896/4885CES2 3970/4885TSHR 2809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.