SCHEMBL414754

SCHEMBL414754

O=C(Nc1ccccc1C(=O)O)c1ccccc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.83
KMT2A Q03164 3/20 0.83
PKM P14618 2/20 0.83
DHODH Q02127 1/20 0.80
MAPT P10636 1/20 0.70
GRIK1 P39086 1/20 0.70
TDP1 Q9NUW8 1/20 0.70
KCNK2 O95069 1/20 0.67
KCNK10 P57789 1/20 0.67
NPC1 O15118 1/20 0.65
RAB9A P51151 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
KDM4D Q6B0I6 1/20 0.65
KDM4C Q9H3R0 1/20 0.65
LTC4S Q16873 1/20 0.63
SUCNR1 Q9BXA5 1/20 0.61
POLB P06746 2/20 0.61
MDM4 O15151 1/20 0.61
TP53 P04637 1/20 0.61
HDAC3 O15379 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31053873 1.00 MEN1 (0.83) MEN1KMT2APKMDHODHMAPT
SCHEMBL8439303 0.98 MEN1 (0.80) MEN1KMT2APKMDHODHMAPT
SCHEMBL15183709 0.96 KMT2A (0.77) MEN1KMT2APKMDHODHMAPT
SCHEMBL14855554 0.96 KMT2A (0.77) MEN1KMT2APKMDHODHMAPT
SCHEMBL2028671 0.96 DHODH (0.86) MEN1KMT2APKMDHODHMAPT
SCHEMBL12700422 0.92 DHODH (0.81) MEN1KMT2APKMDHODHMAPT
SCHEMBL14855907 0.91 DHODH (0.73) MEN1KMT2APKMDHODHMAPT
SCHEMBL4670044 0.91 DHODH (0.78) MEN1KMT2APKMDHODHMAPT
SCHEMBL16404480 0.91 DHODH (0.78) MEN1KMT2APKMDHODHMAPT
SCHEMBL2029098 0.91 MEN1 (1.00) MEN1KMT2APKMDHODHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 306 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115626879-A Preparation method of 2-phenylalanyl-benzoic acid derivative 广州同隽医药科技有限公司 2023-01-20 CN claimed
CN-109232275-B Preparation method of 4-nitrodiphenylamine and 4-nitrosodiphenylamine 科迈化工股份有限公司 2021-06-11 CN claimed
CN-106102477-B Compositions with reduced bitter taste perception 宝洁公司 2020-03-17 CN claimed
EP-2621462-B1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR PROCTER & GAMBLE (US) 2020-02-12 EP claimed
EP-3160592-B1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION PROCTER & GAMBLE (US) 2018-10-31 EP claimed
US-9827320-B2 Compositions with reduced bitter taste perception THE PROCTER & GAMBLE COMPANY (US) 2017-11-28 US claimed
EP-3160592-A1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION The Procter & Gamble Company (US) 2017-05-03 EP claimed
CN-102993203-B The preparations and applicatio of 8-phenyl yanthine analog derivative WENZHOU MEDICAL COLLEGE (CN) 2015-11-25 CN claimed
WO-2015131001-A1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION THE PROCTER & GAMBLE COMPANY (US) 2015-09-03 WO claimed
US-20150238613-A1 Compositions With Reduced Bitter Taste Perception THE PROCTER & GAMBLE COMPANY 2015-08-27 US claimed
EP-2621462-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR The Procter and Gamble Company (US) 2013-08-07 EP claimed
CN-102993203-A Preparation of 8-benzyl xanthine derivative and application WENZHOU MEDICAL COLLEGE 2013-03-27 CN claimed
WO-2012055170-A1 USE OF CYTOPLASMIC C-MYC FOR REGULATING IMMUNE RESPONSES THE UNIVERSITY OF HONG KONG (CN) 2012-05-03 WO claimed
US-20120107317-A1 USE OF CYTOPLASMIC C-MYC FOR REGULATING IMMUNE RESPONSES THE UNIVERSITY OF HONG KONG (CN) 2012-05-03 US claimed
WO-2012044728-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR THE PROCTER & GAMBLE COMPANY (US) 2012-04-05 WO claimed
US-20120082628-A1 Oral Care Compositions With Improved Flavor THE PROCTER & GAMBLE COMPANY 2012-04-05 US claimed
EP-0199276-A2 Process for preparaing substituted 2-phenyl-4H-3,1-benzoxazin-4-ones BASF Aktiengesellschaft (DE) 1986-10-29 EP claimed
EP-0024669-B1 SUBSTITUTED N-BENZOYLANTHRANILIC ACID DERIVATIVES AND THEIR ANHYDRO DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS HERBICIDES AND COMPOSITIONS THEREFOR BASF Aktiengesellschaft (DE) 1983-04-06 EP claimed
US-4235925-A N-Benzoylanthranilate derivatives as phytopathogenic fungicidal agents SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-11-25 US claimed
JP-54002322-A None JP disclosed
WO-2026087024-A1 ORAL BIOFILM MODULATION SYMRISE AG (DE) 2026-04-30 WO disclosed
EP-4719062-A2 METHODS FOR IMPROVING PLANT RESPONSE TO PESTS AND PATHOGENS Newleaf Symbiotics, Inc. (US) 2026-04-08 EP disclosed
WO-2025122372-A1 METHODS FOR AFFECTING PLANT PESTS AND PATHOGENS NEWLEAF SYMBIOTICS, INC. (US) 2025-06-12 WO disclosed
US-20250099539-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS MASSACHUSETTS EYE AND EAR INFIRMARY 2025-03-27 US disclosed
EP-3383502-B1 ORAL CARE PRODUCT AND METHODS OF USE AND MANUFACTURE THEREOF COLGATE PALMOLIVE CO (US) 2025-03-05 EP disclosed
US-12239651-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2025-03-04 US disclosed
US-20250064762-A1 A SUBSTITUTED AROMATIC DICARBONIC ACID AMIDE AS AN INHIBITOR OF THE FERROPTOSIS SUPPRESSOR PROTEIN-1 (FSP1) UNIV WUERZBURG J MAXIMILIANS (DE) 2025-02-27 US disclosed
US-20240409939-A1 COMBINATION OF OLIGONUCLEOTIDES FOR MODULATING RTEL1 AND FUBP1 HOFFMANN-LA ROCHE INC. 2024-12-12 US disclosed
CN-119095603-A Combinations of oligonucleotides for modulating RTEL1 and FUBP1 豪夫迈·罗氏有限公司 2024-12-06 CN disclosed
US-12156899-B2 Methods and compositions for regenerating hair cells and/or supporting cells MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-12-03 US disclosed
WO-2024243521-A2 METHODS FOR IMPROVING PLANT RESPONSE TO PESTS AND PATHOGENS NEWLEAF SYMBIOTICS, INC. (US) 2024-11-28 WO disclosed
EP-4456888-A1 A SUBSTITUTED AROMATIC DICARBONIC ACID AMIDE AS AN INHIBITOR OF THE FERROPTOSIS SUPPRESSOR PROTEIN-1 (FSP1) Julius-Maximilians-Universität Würzburg (DE) 2024-11-06 EP disclosed
EP-4448106-A1 COMBINATION OF OLIGONUCLEOTIDES FOR MODULATING RTEL1 AND FUBP1 Hoffmann-La Roche Inc. (US) 2024-10-23 EP disclosed
US-20240299432-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY 2024-09-12 US disclosed
US-12043653-B2 Efficient delivery of therapeutic molecules to cells of the inner ear MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-07-23 US disclosed
US-20240150758-A1 USE OF FUBP1 INHIBITORS FOR TREATING HEPATITIS B VIRUS INFECTION HOFFMANN LA ROCHE (US) 2024-05-09 US disclosed
US-11963968-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-04-23 US disclosed
US-20240108040-A1 HIGH INTENSITY SWEETENERS FIRMENICH INCORPORATED (US) 2024-04-04 US disclosed
US-11852631-B2 Biomarkers predictive of anti-immune checkpoint response DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-12-26 US disclosed
EP-2775839-B1 METHODS FOR ASSESSING REPELLANT QUALITY OF ORGANIC MATERIALS AND METHODS AND COMPOSITIONS FOR REPELLING ARTHROPODS UNIV CALIFORNIA (US) 2023-12-06 EP disclosed
US-11834392-B2 KDM4B inhibitors for the treatment of inflammatory diseases and disorders MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2023-12-05 US disclosed
US-11834392-B2 KDM4B inhibitors for the treatment of inflammatory diseases and disorders MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2023-12-05 US disclosed
US-11758933-B2 High intensity sweeteners FIRMENICH INCORPORATED (US) 2023-09-19 US disclosed
US-20230277574-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY 2023-09-07 US disclosed
US-11732262-B2 Use of FUBP1 inhibitors for treating hepatitis B virus infection UNIVERSITE CLAUDE BERNARD LYON I (FR) 2023-08-22 US disclosed
WO-2023126338-A1 A SUBSTITUTED AROMATIC DICARBONIC ACID AMIDE AS AN INHIBITOR OF THE FERROPTOSIS SUPPRESSOR PROTEIN-1 (FSP1) JULIUS-MAXIMILIANS-UNIVERSITÄT WÜRZBURG (DE) 2023-07-06 WO disclosed
WO-2023111210-A1 COMBINATION OF OLIGONUCLEOTIDES FOR MODULATING RTEL1 AND FUBP1 F. HOFFMANN-LA ROCHE AG (CH) 2023-06-22 WO disclosed
US-20230131993-A1 COMPOSITION COMPRISING AN AVENANTHRAMIDE OR AN ANALOGUE THEREOF WITH IMPROVED STABILITY SYMRISE AG (DE) 2023-04-27 US disclosed
US-20230129036-A1 AVENANTHRAMIDE COMPOSITIONS WITH IMPROVED SOLUBILITY COMPRISING 4-HYDROXYPHENONE SYMRISE AG (DE) 2023-04-27 US disclosed
US-20230129036-A1 AVENANTHRAMIDE COMPOSITIONS WITH IMPROVED SOLUBILITY COMPRISING 4-HYDROXYPHENONE SYMRISE AG (DE) 2023-04-27 US disclosed
US-20230131993-A1 COMPOSITION COMPRISING AN AVENANTHRAMIDE OR AN ANALOGUE THEREOF WITH IMPROVED STABILITY SYMRISE AG (DE) 2023-04-27 US disclosed
US-20230118467-A1 COSMETIC OR PHARMACEUTICAL USE OF AVENANTHRAMIDE L SYMRISE AG (DE) 2023-04-20 US disclosed
CN-115943307-A MR1 ligands and pharmaceutical compositions for immunomodulation 巴塞尔大学 2023-04-07 CN disclosed
US-20230099822-A1 MR1 LIGANDS AND PHARMACEUTICAL COMPOSITIONS FOR IMMUNOMODULATION UNIVERSITÄT BASEL (CH) 2023-03-30 US disclosed
US-11590152-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2023-02-28 US disclosed
CN-115626879-A Preparation method of 2-phenylalanyl-benzoic acid derivative 广州同隽医药科技有限公司 2023-01-20 CN disclosed
EP-4090969-A1 MR1 LIGANDS AND PHARMACEUTICAL COMPOSITIONS FOR IMMUNOMODULATION Universität Basel (CH) 2022-11-23 EP disclosed
CN-115103840-A Substituted thiophenecarboxamides, thiophenecarboxylic acids and derivatives thereof 拜耳公司 2022-09-23 CN disclosed
US-20220288051-A1 METHODS FOR TREATING CANCER USING SERIAL ADMINISTRATION OF E3 UBIQUITIN LIGASE DEGRADERS DANA-FARBER CANCER INSTITUTE, INC. 2022-09-15 US disclosed
US-20220281941-A1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2022-09-08 US disclosed
US-11370823-B2 Efficient delivery of therapeutic molecules to cells of the inner ear MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2022-06-28 US disclosed
EP-3368542-B1 HIGH INTENSITY SWEETENERS FIRMENICH INCORPORATED (US) 2022-06-22 EP disclosed
US-11357246-B2 High intensity sweeteners FIRMENICH INCORPORATED (US) 2022-06-14 US disclosed
US-20220119344-A1 KDM4B INHIBITORS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DISORDERS MUSC FOUNDATION FOR RESEARCH DEVELOPMENT D/B/A ZUCKER INSTITUTE FOR INNOVATION COMMERCIALIZATION 2022-04-21 US disclosed
US-20220031590-A1 ORAL CARE COMPOSITION SYMRISE AG (DE) 2022-02-03 US disclosed
CN-113683615-A Evodiamine derivative and preparation and application thereof 南华大学 2021-11-23 CN disclosed
EP-3212773-B1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR MASSACHUSETTS EYE & EAR INFIRMARY (US) 2021-09-15 EP disclosed
US-20210227863-A1 HIGH INTENSITY SWEETENERS SENOMYX, INC. 2021-07-29 US disclosed
WO-2021144475-A1 MR1 LIGANDS AND PHARMACEUTICAL COMPOSITIONS FOR IMMUNOMODULATION UNIVERSITÄT BASEL (CH) 2021-07-22 WO disclosed
CN-105218386-B Salts or co-crystals of 3- (3-dimethylamino-1-ethyl-2-methyl-propyl) -phenol 格吕伦塔尔有限公司 2021-07-06 CN disclosed
CN-108473484-B Compounds useful as TRPM8 modulators 弗门尼舍公司 2021-06-29 CN disclosed
CN-109232275-B Preparation method of 4-nitrodiphenylamine and 4-nitrosodiphenylamine 科迈化工股份有限公司 2021-06-11 CN disclosed
EP-3356356-B1 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 FIRMENICH INCORPORATED (US) 2021-05-26 EP disclosed
EP-3800179-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2021-04-07 EP disclosed
CN-108135802-B Oral care compositions and methods of using the same 高露洁-棕榄公司 2021-04-06 CN disclosed
WO-2021050832-A2 METHODS FOR TREATING CANCER USING SERIAL ADMINISTRATION OF E3 UBIQUITIN LIGASE DEGRADERS DANA-FARBER CANCER INSTITUTE, INC. (US) 2021-03-18 WO disclosed
US-20210072248-A1 BIOMARKERS PREDICTIVE OF ANTI-IMMUNE CHECKPOINT RESPONSE DANA-FARBER CANCER INSTITUTE, INC. 2021-03-11 US disclosed
EP-3355849-B1 ORAL CARE COMPOSITIONS AND METHODS OF USING THE COMPOSITIONS COLGATE PALMOLIVE CO (US) 2021-03-10 EP disclosed
EP-3775208-A1 USE OF FUBP1 INHIBITORS FOR TREATING HEPATITIS B VIRUS INFECTION F. Hoffmann-La Roche AG (CH) 2021-02-17 EP disclosed
CN-112359018-A Methods and compositions for regenerating hair cells and/or supporting cells 麻省眼耳医院 2021-02-12 CN disclosed
US-20210030775-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY 2021-02-04 US disclosed
US-20210024934-A1 USE OF FUBP1 INHIBITORS FOR TREATING HEPATITIS B VIRUS INFECTION UNIVERSITE CLAUDE BERNARD LYON I (FR) 2021-01-28 US disclosed
EP-3533436-B1 COMPOSITIONS COMPRISING MENTHOL, ISOBORNYL BUTYRATE AND APRITONE PROCTER & GAMBLE (US) 2020-12-23 EP disclosed
CN-112055749-A Use of FUBP1 inhibitors for the treatment of hepatitis B virus infection 豪夫迈·罗氏有限公司 2020-12-08 CN disclosed
EP-3743057-A1 TREATMENT OF HEARING LOSS Massachusetts Eye & Ear Infirmary (US) 2020-12-02 EP disclosed
US-20200338160-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2020-10-29 US disclosed
CN-111836802-A Fungicidal acibenzoates 拜耳公司 2020-10-27 CN disclosed
CN-108517022-B Solid catalyst component for olefin polymerization, catalyst and application thereof 北京利和知信科技有限公司 2020-10-27 CN disclosed
CN-104869987-B Methods and compositions for regenerating hair cells and/or supporting cells 麻省眼耳医院 2020-10-16 CN disclosed
EP-2998001-B1 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS PROCTER & GAMBLE (US) 2020-07-22 EP disclosed
EP-3656765-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2020-05-27 EP disclosed
EP-3653600-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2020-05-20 EP disclosed
EP-3650439-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2020-05-13 EP disclosed
EP-3636629-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2020-04-15 EP disclosed
CN-106102477-B Compositions with reduced bitter taste perception 宝洁公司 2020-03-17 CN disclosed
EP-2621462-B1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR PROCTER & GAMBLE (US) 2020-02-12 EP disclosed
CN-110603253-A Heteroaryl phenylamino quinolines and analogs 拜耳公司 2019-12-20 CN disclosed
WO-2019193165-A1 USE OF FUBP1 INHIBITORS FOR TREATING HEPATITIS B VIRUS INFECTION F. HOFFMANN-LA ROCHE AG (CH) 2019-10-10 WO disclosed
EP-2854750-B1 TRPA1 ANTAGONISTS FOR REDUCING NEGATIVE SENSATIONS CAUSED BY HYDROGEN PEROXIDE PROCTER & GAMBLE (US) 2019-10-02 EP disclosed
EP-3533436-A1 COMPOSITIONS COMPRISING MENTHOL, ISOBORNYL BUTYRATE AND APRITONE The Procter & Gamble Company (US) 2019-09-04 EP disclosed
US-10392371-B2 Compounds useful as modulators of TRPM8 SENOMYX, INC. (US) 2019-08-27 US disclosed
WO-2019148067-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2019-08-01 WO disclosed
WO-2019143880-A1 BIOMARKERS PREDICTIVE OF ANTI-IMMUNE CHECKPOINT RESPONSE DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-07-25 WO disclosed
US-20190177308-A9 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 SENOMYX, INC. 2019-06-13 US disclosed
EP-2892523-B1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS MASSACHUSETTS EYE & EAR INFIRMARY (US) 2019-05-01 EP disclosed
EP-3160592-B1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION PROCTER & GAMBLE (US) 2018-10-31 EP disclosed
US-20180280263-A1 Oral Care Compositions and Methods of Using the Compositions COLGATE-PALMOLIVE COMPANY (US) 2018-10-04 US disclosed
US-20180273517-A1 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 SENOMYX INC (US) 2018-09-27 US disclosed
EP-3368542-A2 HIGH INTENSITY SWEETENERS Senomyx, Inc. (US) 2018-09-05 EP disclosed
EP-3356356-A1 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 Senomyx, Inc. (US) 2018-08-08 EP disclosed
EP-3355849-A1 ORAL CARE COMPOSITIONS AND METHODS OF USING THE COMPOSITIONS Colgate-Palmolive Company (US) 2018-08-08 EP disclosed
CN-108135802-A Oral care composition and the method using the composition 高露洁-棕榄公司 2018-06-08 CN disclosed
US-9937115-B2 Oral care compositions with improved flavor THE PROCTER & GAMBLE COMPANY (US) 2018-04-10 US disclosed
US-9937115-B2 Oral care compositions with improved flavor THE PROCTER & GAMBLE COMPANY (US) 2018-04-10 US disclosed
US-9937115-B2 Oral care compositions with improved flavor THE PROCTER & GAMBLE COMPANY (US) 2018-04-10 US disclosed
US-9937115-B2 Oral care compositions with improved flavor THE PROCTER & GAMBLE COMPANY (US) 2018-04-10 US disclosed
US-9932340-B2 Substituted indoles ABBVIE INC. (US) 2018-04-03 US disclosed
EP-3287447-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2018-02-28 EP disclosed
US-20180052161-A1 BIOMARKERS FOR MALARIA DIAGNOSIS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2018-02-22 US disclosed
US-20180049960-A1 Methods And Compositions For Modifying Sensorial Perception PROCTER & GAMBLE (US) 2018-02-22 US disclosed
US-20170349589-A9 Substituted Indoles ABBVIE INC. (US) 2017-12-07 US disclosed
US-9827320-B2 Compositions with reduced bitter taste perception THE PROCTER & GAMBLE COMPANY (US) 2017-11-28 US disclosed
US-20170327557-A1 Efficient delivery of therapeutic molecules to cells of the inner ear PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-11-16 US disclosed
US-9790469-B2 Established human brown adipocyte line and method for differentiation from an hMADS cell line CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2017-10-17 US disclosed
EP-3212773-A1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR Massachusetts Eye & Ear Infirmary (US) 2017-09-06 EP disclosed
US-9732071-B2 Compounds useful as modulators of TRPM8 SENOMYX, INC. (US) 2017-08-15 US disclosed
CN-106999973-A System and method for discharging edible material 阿甘芳香和精细化工有限公司 2017-08-01 CN disclosed
US-20170174688-A1 Substituted Indoles ABBVIE INC. (US) 2017-06-22 US disclosed
US-20170143022-A1 Compositions Incorporating an Umami Flavor Agent SENOMYX INC (US) 2017-05-25 US disclosed
US-20170119032-A1 HIGH INTENSITY SWEETENERS FIRMENICH INCORPORATED 2017-05-04 US disclosed
WO-2017075257-A2 HIGH INTENSITY SWEETENERS SENOMYX, INC. (US) 2017-05-04 WO disclosed
EP-3160592-A1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION The Procter & Gamble Company (US) 2017-05-03 EP disclosed
WO-2017062019-A1 ORAL CARE COMPOSITIONS AND METHODS OF USING THE COMPOSITIONS COLGATE-PALMOLIVE COMPANY (US) 2017-04-13 WO disclosed
US-20170096418-A1 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 FIRMENICH INCORPORATED 2017-04-06 US disclosed
US-20170087199-A1 COMPOSITIONS FOR DELIVERING A COOLING SENSATION SENOMYX INC (US) 2017-03-30 US disclosed
EP-3126831-A1 METHOD FOR SCREENING TRP CHANNELS The Procter & Gamble Company (US) 2017-02-08 EP disclosed
US-20160376263-A1 BITTER TASTE MODIFIERS INCLUDING SUBSTITUTED 1-BENZYL-3-(1-(ISOXAZOL-4-YLMETHYL)-1H-PYRAZOL-4-YL)IMIDAZOLIDINE-2,4-DIONES AND COMPOSITIONS THEREOF SENOMYX INC (US) 2016-12-29 US disclosed
US-20160331659-A1 Methods And Compositions For Modifying Sensorial Perception PROCTER & GAMBLE (US) 2016-11-17 US disclosed
US-9491942-B2 Methods for assessing repellant quality of organic materials and methods and compositions for repelling arthropods THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-11-15 US disclosed
US-9491942-B2 Methods for assessing repellant quality of organic materials and methods and compositions for repelling arthropods THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-11-15 US disclosed
WO-2016149386-A1 BIOMARKERS FOR MALARIA DIAGNOSIS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2016-09-22 WO disclosed
US-9427415-B2 Methods and compositions for modifying sensorial perception THE PROCTER & GAMBLE COMPANY (US) 2016-08-30 US disclosed
US-20160158136-A1 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS PROCTER & GAMBLE (US) 2016-06-09 US disclosed
WO-2016069906-A1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2016-05-06 WO disclosed
CN-105473554-A Fused piperidine amides as modulators of ion channels VERTEX PHARMA 2016-04-06 CN disclosed
EP-2998001-A1 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS The Procter and Gamble Company (US) 2016-03-23 EP disclosed
CN-102993203-B The preparations and applicatio of 8-phenyl yanthine analog derivative WENZHOU MEDICAL COLLEGE (CN) 2015-11-25 CN disclosed
WO-2015153184-A1 METHOD FOR SCREENING TRP CHANNELS THE PROCTER & GAMBLE COMPANY (US) 2015-10-08 WO disclosed
US-20150272907-A1 Methods And Compositions For Modifying Sensorial Perception THE PROCTER & GAMBLE COMPANY 2015-10-01 US disclosed
US-9133142-B2 Salts or co-crystals of 3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol GRUENENTHAL GMBH (DE) 2015-09-15 US disclosed
WO-2015131001-A1 COMPOSITIONS WITH REDUCED BITTER TASTE PERCEPTION THE PROCTER & GAMBLE COMPANY (US) 2015-09-03 WO disclosed
US-20150238613-A1 Compositions With Reduced Bitter Taste Perception THE PROCTER & GAMBLE COMPANY 2015-08-27 US disclosed
US-20150209406-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2015-07-30 US disclosed
EP-2892523-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS Massachusetts Eye & Ear Infirmary (US) 2015-07-15 EP disclosed
EP-1959915-B1 MIXTURES COMPRISING ANTHRANILIC ACID AMIDES AND ANTIDANDRUFF AGENTS AS COSMETIC AND PHARMACEUTICAL COMPOSITIONS FOR ALLEVIATING ITCHING SYMRISE AG (DE) 2015-05-13 EP disclosed
EP-2854750-A2 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS The Procter & Gamble Company (US) 2015-04-08 EP disclosed
US-8993622-B2 Antiviral compounds EIRIUM AB (SE) 2015-03-31 US disclosed
US-8993622-B2 Antiviral compounds EIRIUM AB (SE) 2015-03-31 US disclosed
US-8911795-B2 Compositions comprising dihydroavenanthramide D and climbazole as cosmetic and pharmaceutical compositions for alleviating itching SYMRISE AG (DE) 2014-12-16 US disclosed
US-8911795-B2 Compositions comprising dihydroavenanthramide D and climbazole as cosmetic and pharmaceutical compositions for alleviating itching SYMRISE AG (DE) 2014-12-16 US disclosed
US-20140128352-A1 COMPOUNDS AND METHODS FOR MODULATING MITOCHONDRIAL METABOLISM AND REACTIVE OXYGEN SPECIES PRODUCTION BUCK INSTITUTE FOR RESEARCH ON AGING (US) 2014-05-08 US disclosed
US-20140128352-A1 COMPOUNDS AND METHODS FOR MODULATING MITOCHONDRIAL METABOLISM AND REACTIVE OXYGEN SPECIES PRODUCTION BUCK INSTITUTE FOR RESEARCH ON AGING (US) 2014-05-08 US disclosed
WO-2014039908-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2014-03-13 WO disclosed
WO-2013176897-A2 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS THE PROCTER & GAMBLE COMPANY (US) 2013-11-28 WO disclosed
US-20130315843-A1 COMPOSITION FOR REDUCTION OF TRPA1 AND TRPV1 SENSATIONS THE PROCTER & GAMBLE COMPANY (US) 2013-11-28 US disclosed
US-20130225644-A1 MODIFIED LYSINE-MIMETIC COMPOUNDS ZEALAND PHARMA A/S (DK) 2013-08-29 US disclosed
US-20130210915-A1 ANTIVIRAL COMPOUNDS EIRIUM AB (SE) 2013-08-15 US disclosed
US-20130210915-A1 ANTIVIRAL COMPOUNDS EIRIUM AB (SE) 2013-08-15 US disclosed
EP-1567143-B1 ANTHRANILIC ACID AMIDES AND THE DERIVATIVES THEREOF AS COSMETIC AND PHARMACEUTICAL AGENTS SYMRISE AG (DE) 2013-08-14 EP disclosed
EP-1567143-B1 ANTHRANILIC ACID AMIDES AND THE DERIVATIVES THEREOF AS COSMETIC AND PHARMACEUTICAL AGENTS SYMRISE AG (DE) 2013-08-14 EP disclosed
EP-2621462-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR The Procter and Gamble Company (US) 2013-08-07 EP disclosed
EP-2621462-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR The Procter and Gamble Company (US) 2013-08-07 EP disclosed
CN-103140209-A Oral care compositions with improved flavor PROCTER & GAMBLE 2013-06-05 CN disclosed
EP-2595971-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2013-05-29 EP disclosed
US-8431540-B2 Modified lysine-mimetic compounds ZEALAND PHARMA A/S (DK) 2013-04-30 US disclosed
US-8409552-B2 Anthranillic acid amides and derivatives thereof as cosmetic and pharmaceutical active compounds SYMRISE AG (DE) 2013-04-02 US disclosed
US-8409552-B2 Anthranillic acid amides and derivatives thereof as cosmetic and pharmaceutical active compounds SYMRISE AG (DE) 2013-04-02 US disclosed
US-8409552-B2 Anthranillic acid amides and derivatives thereof as cosmetic and pharmaceutical active compounds SYMRISE AG (DE) 2013-04-02 US disclosed
CN-102993203-A Preparation of 8-benzyl xanthine derivative and application WENZHOU MEDICAL COLLEGE 2013-03-27 CN disclosed
US-20120315233-A1 ANTHRANILLIC ACID AMIDES AND DERIVATIVES THEREOF AS COSMETIC AND PHARMACEUTICAL ACTIVE COMPOUNDS SYMRISE AG (DE) 2012-12-13 US disclosed
US-20120315233-A1 ANTHRANILLIC ACID AMIDES AND DERIVATIVES THEREOF AS COSMETIC AND PHARMACEUTICAL ACTIVE COMPOUNDS SYMRISE AG (DE) 2012-12-13 US disclosed
US-20120315233-A1 ANTHRANILLIC ACID AMIDES AND DERIVATIVES THEREOF AS COSMETIC AND PHARMACEUTICAL ACTIVE COMPOUNDS SYMRISE AG (DE) 2012-12-13 US disclosed
US-20120245106-A1 MODIFIED LYSINE-MIMETIC COMPOUNDS ZEALAND PHARMA A/S (DK) 2012-09-27 US disclosed
US-8203016-B2 Anthranilic acid amides and derivatives thereof as cosmetic and pharmaceutical agents SYMRISE AG (DE) 2012-06-19 US disclosed
US-8203016-B2 Anthranilic acid amides and derivatives thereof as cosmetic and pharmaceutical agents SYMRISE AG (DE) 2012-06-19 US disclosed
US-8203016-B2 Anthranilic acid amides and derivatives thereof as cosmetic and pharmaceutical agents SYMRISE AG (DE) 2012-06-19 US disclosed
WO-2012055170-A1 USE OF CYTOPLASMIC C-MYC FOR REGULATING IMMUNE RESPONSES THE UNIVERSITY OF HONG KONG (CN) 2012-05-03 WO disclosed
US-20120107317-A1 USE OF CYTOPLASMIC C-MYC FOR REGULATING IMMUNE RESPONSES THE UNIVERSITY OF HONG KONG (CN) 2012-05-03 US disclosed
WO-2012044728-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR THE PROCTER & GAMBLE COMPANY (US) 2012-04-05 WO disclosed
WO-2012044728-A1 ORAL CARE COMPOSITIONS WITH IMPROVED FLAVOR THE PROCTER & GAMBLE COMPANY (US) 2012-04-05 WO disclosed
US-20120082628-A1 Oral Care Compositions With Improved Flavor THE PROCTER & GAMBLE COMPANY 2012-04-05 US disclosed
US-20120082628-A1 Oral Care Compositions With Improved Flavor THE PROCTER & GAMBLE COMPANY 2012-04-05 US disclosed
US-20120082628-A1 Oral Care Compositions With Improved Flavor THE PROCTER & GAMBLE COMPANY 2012-04-05 US disclosed
US-20120082628-A1 Oral Care Compositions With Improved Flavor THE PROCTER & GAMBLE COMPANY 2012-04-05 US disclosed
US-20120022117-A1 Salts or Co-Crystals of 3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol GRUENENTHAL GMBH (DE) 2012-01-26 US disclosed
WO-2012010316-A1 SALTS OR CO-CRYSTALS OF 3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2012-01-26 WO disclosed
EP-2405914-A1 COMPOSITIONS AND METHODS FOR PROPHYLAXIS AND TREATMENT OF ADDICTIONS Omeros Corporation (US) 2012-01-18 EP disclosed
WO-2011155898-A1 NEW ANTIVIRAL COMPOUNDS WADELL GOERAN (SE) 2011-12-15 WO disclosed
US-8026272-B2 Modified lysine-mimetic compounds ZEALAND PHARMA A/S (DK) 2011-09-27 US disclosed
EP-2356242-A2 METHODS FOR USING POSITIVELY AND NEGATIVELY SELECTABLE GENES IN A FILAMENTOUS FUNGAL CELL Novozymes Inc. (US) 2011-08-17 EP disclosed
EP-2352831-A1 METHODS FOR PRODUCING POLYPEPTIDES IN ENZYME-DEFICIENT MUTANTS OF FUSARIUM VENENATUM Novozymes Inc. (US) 2011-08-10 EP disclosed
US-7973163-B2 Fused quinoline derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LTD. (JP) 2011-07-05 US disclosed
US-20110117066-A1 ESTABLISHED HUMAN BROWN ADIPOCYTE LINE AND METHOD FOR DIFFERENTIATION FROM AN HMADS CELL LINE UNIVERSITE DE NICE SOPHIA ANTIPOLIS (FR) 2011-05-19 US disclosed
US-7943770-B2 Fused quinoline derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-05-17 US disclosed
US-20110071197-A1 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS BIOLIPOX AB (LV) 2011-03-24 US disclosed
US-20110039808-A1 Multitarget Compounds Active at a PPAR and Cannabinoid Receptor NOGRA PHARMA LIMITED (IE) 2011-02-17 US disclosed
US-20100261103-A1 ORGANIC PIGMENT FINE PARTICLES AND METHOD OF PRODUCING THE SAME, PIGMENT-DISPERSION COMPOSITION, PHOTOCURABLE COMPOSITION AND INK-JET INK CONTAINING THE SAME, AND COLOR FILTER USING THE SAME AND METHOD OF PRODUCING THE SAME FUJIFILM CORPORATION (JP) 2010-10-14 US disclosed
US-20100249206-A1 MODIFIED LYSINE-MIMETIC COMPOUNDS Zealand Pharma A/S and Wyeth 2010-09-30 US disclosed
US-20100248390-A1 COMPOSITIONS AND METHODS FOR IDENTIFYING LIGANDS OF ODORANT RECEPTORS DUKE UNIVERSITY (US) 2010-09-30 US disclosed
EP-2230312-A1 Probe compound for detecting and isolating enzymes and means and methods using the same Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2010-09-22 EP disclosed
CN-101842362-A Benzothiazole compounds INST MEDICAL W & E HALL 2010-09-22 CN disclosed
WO-2010105103-A1 COMPOSITIONS AND METHODS FOR PROPHYLAXIS AND TREATMENT OF ADDICTIONS OMEROS CORPORATION (US) 2010-09-16 WO disclosed
EP-2222287-A2 MULTITARGET COMPOUNDS ACTIVE AT A PPAR AND CANNABINOID RECEPTOR Giuliani International Limited (IE) 2010-09-01 EP disclosed
US-20100189648-A1 INHIBITORS FOR DISRUPTING THE INTERACTION OF UBIQUITINATION RELATED ENZYMES AND USES THEREOF HUANG LAN 2010-07-29 US disclosed
US-20100189648-A1 INHIBITORS FOR DISRUPTING THE INTERACTION OF UBIQUITINATION RELATED ENZYMES AND USES THEREOF HUANG LAN 2010-07-29 US disclosed
EP-1740584-B9 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2010-06-09 EP disclosed
WO-2010039840-A1 METHODS FOR PRODUCING POLYPEPTIDES IN ENZYME-DEFICIENT MUTANTS OF FUSARIUM VENENATUM NOVOZYMES, INC. (US) 2010-04-08 WO disclosed
WO-2010039889-A2 METHODS FOR USING POSITIVELY AND NEGATIVELY SELECTABLE GENES IN A FILAMENTOUS FUNGAL CELL NOVOZYMES, INC. (US) 2010-04-08 WO disclosed
WO-2010009091-A2 ANTI-INFLAMMATORY AND ANTI-ALLERGY EXTRACTS FROM NETTLE HERBALSCIENCE GROUP, LLC (US) 2010-01-21 WO disclosed
US-20100009927-A1 Anti-Inflammatory and Anti-Allergy Extracts from Nettle HERBALSCIENCE GROUP LLC (US) 2010-01-14 US disclosed
US-20090297468-A1 Mixtures Comprising Anthranilic Acid Amides and Cooling Agents as Cosmetic and Pharmaceutical Compositions for Alleviating Itching SYMRISE GMBH & CO. KG (DE) 2009-12-03 US disclosed
US-20090297468-A1 Mixtures Comprising Anthranilic Acid Amides and Cooling Agents as Cosmetic and Pharmaceutical Compositions for Alleviating Itching SYMRISE GMBH & CO. KG (DE) 2009-12-03 US disclosed
US-7622496-B2 antiarrhythmia agents; 1-(2-Amino-acetyl)-4-(benzoylamino)-pyrrolidine-2-carboxylic acid; desirable bioavailability properties ZEALAND PHARMA A/S (DK) 2009-11-24 US disclosed
US-20090275568-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 US disclosed
US-20090270625-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMTED (JP) 2009-10-29 US disclosed
US-20090264342-A1 COMPOSITIONS AND METHODS FOR ANTIBIOTIC POTENTIATION AND DRUG DISCOVERY TRUSTEES OF BOSTON UNIVERSITY (US) 2009-10-22 US disclosed
US-20090258893-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-15 US disclosed
US-7592453-B2 Fused quinoline derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-22 US disclosed
US-20090226537-A1 MIXTURES COMPRISING ANTHRANILIC ACID AMIDES AND ANTIDANDRUFF AGENTS AS COSMETIC AND PHARMACEUTICAL COMPOSITIONS FOR ALLEVIATING ITCHING SYMRISE GMBH & CO. KG (DE) 2009-09-10 US disclosed
US-20090226537-A1 MIXTURES COMPRISING ANTHRANILIC ACID AMIDES AND ANTIDANDRUFF AGENTS AS COSMETIC AND PHARMACEUTICAL COMPOSITIONS FOR ALLEVIATING ITCHING SYMRISE GMBH & CO. KG (DE) 2009-09-10 US disclosed
US-20090209536-A1 AMINOQUINAZOLINE CANNABINOID RECEPTOR MODULATORS FOR TREATMENT OF DISEASE KALYPSYS, INC. (US) 2009-08-20 US disclosed
EP-2080760-A1 Fused quinoline derivative and use thereof Takeda Pharmaceutical Company Limited (JP) 2009-07-22 EP disclosed
WO-2009080821-A2 RECEPTOR TARGETING LIGANDS GIULIANI INTERNATIONAL LIMITED (IE) 2009-07-02 WO disclosed
JP-2009107972-A AMINOBENZALDEHYDE COMPOUND, METHOD FOR PRODUCING THE SAME, AND METHOD FOR PRODUCING AMINOBENZOIC ACID COMPOUND FUJI CHEM IND CO LTD 2009-05-21 JP disclosed
US-20090118135-A1 METHODS AND COMPOUNDS FOR REGULATING APOPTOSIS THE BURNHAM INSTITUTE (US) 2009-05-07 US disclosed
US-20090118135-A1 METHODS AND COMPOUNDS FOR REGULATING APOPTOSIS THE BURNHAM INSTITUTE (US) 2009-05-07 US disclosed
EP-2028936-A2 COMPOSITIONS AND METHODS FOR ANTIBIOTIC POTENTIATION AND DRUG DISCOVERS TRUSTEES OF BOSTON UNIVERSITY (US) 2009-03-04 EP disclosed
EP-2021331-A1 2-PHENYL-5-AMINO-1,3,4-OXADIAZOLES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS GLAXO GROUP LIMITED (GB) 2009-02-11 EP disclosed
US-20090035306-A1 QUINAZOLINONE MODULATORS OF TGR5 KALYPSYS, INC. (US) 2009-02-05 US disclosed
WO-2008147826-A1 MALARIA LIVER STAGE DRUGS SEATTLE BIOMEDICAL RESEARCH INSTITUTE (US) 2008-12-04 WO disclosed
EP-1740584-B1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2008-12-03 EP disclosed
US-20080039452-A1 Fused Quinoline Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-02-14 US disclosed
EP-1886662-A1 Anti-microbial compounds for treating bad breath Symrise GmbH & Co. KG (DE) 2008-02-13 EP disclosed
EP-1886662-A1 Anti-microbial compounds for treating bad breath Symrise GmbH & Co. KG (DE) 2008-02-13 EP disclosed
US-20080008660-A1 Antimicrobially active compounds for treating bad breath SYMRISE GMBH & CO. KG (DE) 2008-01-10 US disclosed
US-20080008660-A1 Antimicrobially active compounds for treating bad breath SYMRISE GMBH & CO. KG (DE) 2008-01-10 US disclosed
US-20080008660-A1 Antimicrobially active compounds for treating bad breath SYMRISE GMBH & CO. KG (DE) 2008-01-10 US disclosed
WO-2007138033-A1 2-PHENYL-5-AMINO-1,3,4-OXADIAZOLES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS GLAXO GROUP LIMITED (GB) 2007-12-06 WO disclosed
WO-2007095187-A2 COMPOSITIONS AND METHODS FOR ANTIBIOTIC POTENTIATION AND DRUG DISCOVERY TRUSTEES OF BOSTON UNIVERSITY (US) 2007-08-23 WO disclosed
US-20070149460-A1 Modified lysine-mimetic compounds ZEALAND PHARMA A/S (DK) 2007-06-28 US disclosed
WO-2007062957-A1 MIXTURES COMPRISING ANTHRANILIC ACID AMIDES AND ANTIDANDRUFF AGENTS AS COSMETIC AND PHARMACEUTICAL COMPOSITIONS FOR ALLEVIATING ITCHING SYMRISE GMBH & CO. KG (DE) 2007-06-07 WO disclosed
US-7186739-B2 Stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas IMMUPHARMA (FRANCE) SA (FR) 2007-03-06 US disclosed
EP-1740584-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
US-7060845-B2 Stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas NEOMPS (FR) 2006-06-13 US disclosed
US-20060089413-A1 Anthranilic acid amides and derivatives thereof as cosmetic and pharmaceutical agents SYMRISE GMBH & CO. KG (DE) 2006-04-27 US disclosed
WO-2005105802-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed
US-20050159584-A1 Novel stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2005-07-21 US disclosed
US-20050159585-A1 Novel stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2005-07-21 US disclosed
EP-1165494-B1 HSV PRIMASE INHIBITORS BOEHRINGER INGELHEIM CA LTD (CA) 2003-11-05 EP disclosed
US-20030073862-A1 Compounds BIOVITRUM AB (SE) 2003-04-17 US disclosed
US-20030073862-A1 Compounds BIOVITRUM AB (SE) 2003-04-17 US disclosed
WO-2003004458-A1 NEW COMPOUNDS BIOVITRUM AB (SE) 2003-01-16 WO disclosed
WO-2003004458-A1 NEW COMPOUNDS BIOVITRUM AB (SE) 2003-01-16 WO disclosed
US-20020143191-A1 Novel stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas UREKA SARL (FR) 2002-10-03 US disclosed
EP-1165494-A2 HSV PRIMASE INHIBITORS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2002-01-02 EP disclosed
US-6323202-B1 BENZAMIDE SUBSTITUTES WITH KETONE COMPOUNDS AS ENZYME INHIBITORS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2001-11-27 US disclosed
WO-2000058270-A2 HSV PRIMASE INHIBITORS BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2000-10-05 WO disclosed
EP-0983226-A1 NEW NITROMETHYL KETONES, PROCESS FOR PREPARING THEM AND COMPOSITIONS CONTAINING THEM MERCK PATENT GmbH (DE) 2000-03-08 EP disclosed
US-5847155-A Aromatic pyrrolidine amide prolyl endopeptidase inhibitors PFIZER INC (US) 1998-12-08 US disclosed
WO-1998052906-A1 NEW NITROMETHYL KETONES, PROCESS FOR PREPARING THEM AND COMPOSITIONS CONTAINING THEM MERCK PATENT GMBH (DE) 1998-11-26 WO disclosed
EP-0750611-B1 ANILIDE DERIVATIVES AS FUNGICIDES AGREVO UK LTD (GB) 1998-07-08 EP disclosed
US-5756524-A APPLYING TO COMBAT CYTOPATHOGENIC FUNGI AGREVO UK LIMITED (GB) 1998-05-26 US disclosed
EP-0280367-B1 Glycine compounds SHELL INT RESEARCH (NL) 1993-11-03 EP disclosed
EP-0536163-A1 AROMATIC PYRROLIDINE AND THIAZOLIDINE AMIDES PFIZER INC. (US) 1993-04-14 EP disclosed
US-5164277-A Oxyalkylated derivative of ditrimethylolpropane FUJI PHOTO FILM CO., LTD. (JP) 1992-11-17 US disclosed
CN-1017799-B GLYCINE COMPOUNDS AND PROCESS FOR PREPARING THEM SHELL INT RESEARCH (NL) 1992-08-12 CN disclosed
US-5110348-A Pre-and postemergence SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1992-05-05 US disclosed
WO-1991018891-A1 AROMATIC PYRROLIDINE AND THIAZOLIDINE AMIDES PFIZER INC. (US) 1991-12-12 WO disclosed
EP-0246570-B1 ZINC AND/OR LEAD SALTS OF CARBOXYLIC ACIDS AND THEIR USE AS ANTICORROSIVES BASF Lacke + Farben AG (DE) 1989-09-13 EP disclosed
US-4837228-A HYPOTERMIC AGENTS THE UNIVERSITY OF MISSISSIPPI (US) 1989-06-06 US disclosed
US-4830775-A FOR AQUEOUS COATING SYSTEMS BASF Lacke ± Farben Aktiengesellschaft (DE) 1989-05-16 US disclosed
CN-88100995-A glycine compound and preparation method thereof 1988-09-07 CN disclosed
EP-0280367-A2 Glycine compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1988-08-31 EP disclosed
EP-0246570-A1 Zinc and/or lead salts of carboxylic acids and their use as anticorrosives BASF Lacke + Farben AG (DE) 1987-11-25 EP disclosed
US-4673740-A Preparation of substituted 2-phenyl-4H-3,1-benzoxazin-4-ones BASF AKTIENGESELLSCHAFT (DE) 1987-06-16 US disclosed
EP-0199276-A2 Process for preparaing substituted 2-phenyl-4H-3,1-benzoxazin-4-ones BASF Aktiengesellschaft (DE) 1986-10-29 EP disclosed
EP-0024669-B1 SUBSTITUTED N-BENZOYLANTHRANILIC ACID DERIVATIVES AND THEIR ANHYDRO DERIVATIVES, PROCESS FOR THEIR PREPARATION, THEIR USE AS HERBICIDES AND COMPOSITIONS THEREFOR BASF Aktiengesellschaft (DE) 1983-04-06 EP disclosed
US-4347188-A FUNGICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1982-08-31 US disclosed
US-4347188-A FUNGICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1982-08-31 US disclosed
US-4347188-A FUNGICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1982-08-31 US disclosed
US-4344862-A Reaction products of sulfonamido-carboxylic acids or carboxamido-carboxylic acids with alkanolamines, and their use as low-foaming corrosion inhibitors BASF AKTIENGESELLSCHAFT (DE) 1982-08-17 US disclosed
US-4321371-A Substituted N-benzoylanthranilic acid derivatives and their anhydro compounds BASF AKTIENGESELLSCHAFT (DE) 1982-03-23 US disclosed
US-4321371-A Substituted N-benzoylanthranilic acid derivatives and their anhydro compounds BASF AKTIENGESELLSCHAFT (DE) 1982-03-23 US disclosed
US-4321371-A Substituted N-benzoylanthranilic acid derivatives and their anhydro compounds BASF AKTIENGESELLSCHAFT (DE) 1982-03-23 US disclosed
US-4315862-A FROM CITRAL AND A RESORCINOL PERIVATIVE THE UNIVERSITY OF MISSISSIPPI (US) 1982-02-16 US disclosed
US-4303548-A Process for coating dispersed minute droplets with membrane MITSUBISHI PAPER MILLS, LTD. (JP) 1981-12-01 US disclosed
EP-0029529-A1 Reaction products of sulfone or carboxamido carboxylic acids with alkanol amines, and their use as corrosion inhibitors with low foam formation BASF Aktiengesellschaft (DE) 1981-06-03 EP disclosed
EP-0024669-A1 Substituted N-benzoylanthranilic acid derivatives and their anhydro derivatives, process for their preparation, their use as herbicides and compositions therefor BASF Aktiengesellschaft (DE) 1981-03-11 EP disclosed
EP-0024669-A1 Substituted N-benzoylanthranilic acid derivatives and their anhydro derivatives, process for their preparation, their use as herbicides and compositions therefor BASF Aktiengesellschaft (DE) 1981-03-11 EP disclosed
US-4254208-A DISPERSION, LIQUEFYING, SOLIDS FUJI PHOTO FILM CO., LTD. (JP) 1981-03-03 US disclosed
US-4235925-A N-Benzoylanthranilate derivatives as phytopathogenic fungicidal agents SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-11-25 US disclosed
US-4235925-A N-Benzoylanthranilate derivatives as phytopathogenic fungicidal agents SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-11-25 US disclosed
US-4235925-A N-Benzoylanthranilate derivatives as phytopathogenic fungicidal agents SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1980-11-25 US disclosed
US-4230727-A N-BENZYLIDENEANILINE AND DERIVATIVES WILLIAM H. RORER, INC. (US) 1980-10-28 US disclosed
US-4187317-A Sunscreen and erythema treating with N-benzylidene anilenes WILLIAM H. RORER, INC. (US) 1980-02-05 US disclosed
JP-S542322-A ALKYL N-ACYLANTHRANYLATE DERIVATIVES, THEIR PREPARATION, AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE CONTAINING THE SAME SUMITOMO CHEM CO LTD 1979-01-09 JP disclosed
JP-S542322-A ALKYL N-ACYLANTHRANYLATE DERIVATIVES, THEIR PREPARATION, AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE CONTAINING THE SAME SUMITOMO CHEM CO LTD 1979-01-09 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11370823-B2 Efficient delivery of therapeutic molecules to cells of the inner ear HES1, NOTCH1, NOTCH2 MEN1 254/4885KMT2A 2721/4885PKM 4849/4885
US-20110071197-A1 BIS-ARYL COMPOUNDS FOR USE AS MEDICAMENTS LTC4S, LTB4R2, LTB4R MEN1 2758/4885KMT2A 3849/4885PKM 2760/4885
US-20090209536-A1 AMINOQUINAZOLINE CANNABINOID RECEPTOR MODULATORS FOR TREATMENT OF DISEASE CNR2, CNR1, GPR18 MEN1 718/4885KMT2A 1424/4885PKM 1716/4885
US-20240108040-A1 HIGH INTENSITY SWEETENERS TAS2R40, TAS2R60, TAS1R1 MEN1 2644/4885KMT2A 2697/4885PKM 3251/4885
US-20120245106-A1 MODIFIED LYSINE-MIMETIC COMPOUNDS MYLK2, KCNN2, KCNN1 MEN1 1114/4885KMT2A 89/4885PKM 145/4885
US-20090035306-A1 QUINAZOLINONE MODULATORS OF TGR5 GRK5, PLAAT5, GPBAR1 MEN1 4781/4885KMT2A 4183/4885PKM 1804/4885
US-20170119032-A1 HIGH INTENSITY SWEETENERS TAS2R40, TAS2R60, TAS1R1 MEN1 2644/4885KMT2A 2697/4885PKM 3251/4885
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“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.