B-D-Galactose

B-D-Galactose

SCHEMBL79549

OC[C@H]1OC(O)[C@@H](O)[C@H](O)[C@@H]1O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LGALS3 P17931 3/20 0.58
LGALS1 P09382 2/20 0.58
LGALS9 O00182 1/20 0.58
LGALS8 O00214 1/20 0.58
CA12 O43570 3/20 0.45
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CA9 Q16790 3/20 0.45
PYGB P11216 6/20 0.44
GAA P10253 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
LMNA P02545 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
B-D-Galactose SCHEMBL9880688 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL10050866 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL2441804 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL13220216 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL18649521 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL8527882 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL23758905 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL17112445 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL21123450 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12
B-D-Galactose SCHEMBL9820102 1.00 LGALS3 (0.58) LGALS3LGALS1LGALS9LGALS8CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1113 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO claimed
US-10960570-B2 Additives for lignocellulosic composites HEXION INC. (US) 2021-03-30 US claimed
EP-3198072-B1 NON-FLUORINATED URETHANE BASED COATINGS CHEMOURS CO FC LLC (US) 2020-10-28 EP claimed
US-20190270219-A1 ADDITIVES FOR LIGNOCELLULOSIC COMPOSITES HEXION INC. 2019-09-05 US claimed
US-10011617-B2 Isocyanate derived organosilanes THE CHEMOURS COMPANY FC, LLC (US) 2018-07-03 US claimed
US-8212013-B2 Phenyl 3,4,6-tri-O-benzyl-2-O-(1,1,2,2-tetramethyl-dimethylene phosphonoyl)- beta -D-thioglucopyranoside; inhibits formation of o-ester by-product resulting from the conventional glycosilation reaction of pyranose compounds of 1,2-trans form, affording 1,2-transglycoside compounds with high selectivity OTSUKA CHEMICAL CO., LTD. (JP) 2012-07-03 US claimed
US-20080177049-A1 Process for Producing 1,2-Trans-Glycoside Compound GLYTECH, INC. (JP) 2008-07-24 US claimed
EP-1849794-A1 PROCESS FOR PRODUCING 1,2-TRANS-GLYCOSIDE COMPOUND Otsuka Chemical Co., Ltd. (JP) 2007-10-31 EP claimed
WO-2007088559-A1 PROCESS FOR PRODUCING SUBSTITUTED SULPHOXIDES JUBILANT ORGANOSYS LIMITED (IN) 2007-08-09 WO claimed
EP-1186688-B1 Hollow fibrous organic nanotube and method for producing the same NAT INST OF ADVANCED IND SCIEN (JP) 2005-06-15 EP claimed
US-6693178-B2 HALOGENATED BENZYL ETHER GALACTOPYRANOSIDE, GLUCOPYRANOSIDE, RIBOFURANOSIDE OR XYLOFURANOSIDE DERIVATIVES; STABLE, EASILY REMOVED MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2004-02-17 US claimed
US-20020045199-A1 Treatment or prophylaxis of diseases caused by pilus-forming bacteria HULTGREN SCOTT (US) 2002-04-18 US claimed
WO-1998024792-A1 ANTICOAGULANT GLYCOSIDES AND PHARMACEUTICAL COMPOSITIONS THEREOF Richter Gedeon Vegyészeti Gyár Rt. (HU) 1998-06-11 WO claimed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP claimed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP claimed
EP-0485517-A1 SYNTHESIS OF GLYCOSIDES HAVING PREDETERMINED STEREOCHEMISTRY YALE UNIVERSITY (US) 1992-05-20 EP claimed
US-5041541-A 5-C-Hydroxymethylhexose Compounds THE PROCTER & GAMBLE COMPANY (US) 1991-08-20 US claimed
WO-1991002739-A1 SYNTHESIS OF GLYCOSIDES HAVING PREDETERMINED STEREOCHEMISTRY YALE UNIVERSITY (US) 1991-03-07 WO claimed
EP-0341062-A2 Functional sugar substitutes with reduced calories THE PROCTER & GAMBLE COMPANY (US) 1989-11-08 EP claimed
US-20260137677-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 TOCRIS COOKSON LTD (GB) 2026-05-21 US disclosed
US-20260109721-A1 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON: SYNTHESIS AND LNP FORMULATION ALDEXCHEM KFT (HU) 2026-04-23 US disclosed
EP-4727929-A2 5'-MODIFIED MONOMERS, OLIGONUCLEOTIDES AND DOUBLE-STRANDED RNAS Alnylam Pharmaceuticals, Inc. (US) 2026-04-22 EP disclosed
EP-4726101-A1 WATER REPELLENT COMPOSITION AND METHOD FOR PRODUCING SAME Daikin Industries, Ltd. (JP) 2026-04-15 EP disclosed
US-20260098377-A1 FIBER STRUCTURE DAIKIN INDUSTRIES, LTD. (JP) 2026-04-09 US disclosed
US-20260062633-A1 EMULSION QUADRISE INTERNATIONAL LTD (GB) 2026-03-05 US disclosed
EP-4688653-A2 MANUFACTURING OF HYBRID ORGANIC-INORGANIC SILICA AEROGELS AEROBEL BV (BE) 2026-02-11 EP disclosed
US-20260008793-A1 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON ALDEXCHEM KFT (HU) 2026-01-08 US disclosed
EP-4673438-A1 PROTEOLYSIS-TARGETING CHIMERAS Tocris Cookson Limited (GB) 2026-01-07 EP disclosed
EP-4663716-A1 WATER REPELLENT COMPOSITION Daikin Industries, Ltd. (JP) 2025-12-17 EP disclosed
US-12497613-B2 Modified oligonucleotides ALNYLAM PHARMACEUTICALS, INC. (US) 2025-12-16 US disclosed
US-20250346778-A1 FLUORINE-CONTAINING COMPOUND DAIKIN INDUSTRIES, LTD. (JP) 2025-11-13 US disclosed
EP-4646422-A1 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON: SYNTHESIS AND LNP FORMULATION AldexChem Kft. (HU) 2025-11-12 EP disclosed
US-20250340519-A1 RADIOLABELLED COMPOUND OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2025-11-06 US disclosed
EP-4633738-A1 CYTOTOXIC COMPOUNDS Pheon Therapeutics Ltd (GB) 2025-10-22 EP disclosed
EP-4624459-A2 RADIOLABELLED COMPOUND Oxford University Innovation Limited (GB) 2025-10-01 EP disclosed
EP-4617341-A1 WATER REPELLENT COMPOSITION Daikin Industries, Ltd. (JP) 2025-09-17 EP disclosed
US-20250283066-A1 METHODS AND COMPOSITIONS UNITED KINGDOM RESEARCH AND INNOVATION (GB) 2025-09-11 US disclosed
EP-4163350-B1 WATER REPELLENT COMPOSITION, KIT, WATER REPELLENT FIBER PRODUCT AND METHOD FOR MANUFACTURING SAME MEISEI CHEMICAL WORKS LTD (JP) 2025-09-10 EP disclosed
EP-3630779-B1 ANTIBIOTIC RESISTANCE BREAKERS KING S COLLEGE LONDON (GB) 2025-09-03 EP disclosed
US-12398162-B2 Guanine analogs as telomerase substrates and telomere length affectors GERON CORPORATION (US) 2025-08-26 US disclosed
EP-4603635-A1 FIBER STRUCTURE DAIKIN INDUSTRIES, LTD. (JP) 2025-08-20 EP disclosed
EP-4598914-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 Tocris Cookson Limited (GB) 2025-08-13 EP disclosed
EP-4598582-A1 PROTEOLYSIS-TARGETING CHIMERAS AGAINST THE PAPAIN-LIKE PROTEASE OF SARS-COV-2 Tocris Cookson Limited (GB) 2025-08-13 EP disclosed
US-20250224411-A1 MOLECULAR HOPPER OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2025-07-10 US disclosed
EP-4581107-A1 EMULSION Quadrise International Ltd (GB) 2025-07-09 EP disclosed
EP-4574872-A1 FLUORINE-CONTAINING COMPOUND DAIKIN INDUSTRIES, LTD. (JP) 2025-06-25 EP disclosed
EP-4562021-A2 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON AldexChem Kft. (HU) 2025-06-04 EP disclosed
WO-2025104452-A1 COMPOUNDS FOR USE IN TREATMENT MITORX THERAPEUTICS LTD (GB) 2025-05-22 WO disclosed
US-20250163159-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2025-05-22 US disclosed
WO-2025090191-A1 TEXTILE TREATMENT FOR IMPARTING OIL REPELLENCY INCLUDES USE OF A NON-CRYSTALLINE SILICONE – (METH)ACRYLATE COPOLYMER, A CRYSTALLINE POLYMER, AND A BLOCKED ISOCYANATE DOW GLOBAL TECHNOLOGIES LLC (US) 2025-05-01 WO disclosed
WO-2025090190-A1 TEXTILE TREATMENT FOR IMPARTING OIL REPELLENCY INCLUDES USE OF A SILICONE – (METH)ACRYLATE COPOLYMER AND A URETHANE DOW SILICONES CORPORATION (US) 2025-05-01 WO disclosed
US-12286657-B2 Methods and compositions UNITED KINGDOM RESEARCH AND INNOVATION (GB) 2025-04-29 US disclosed
US-20250123276-A1 HIGHLY SENSITIVE IMMUNOASSAY REAGENT AND MEASUREMENT METHOD PCH Corporation (JP) 2025-04-17 US disclosed
WO-2025052296-A1 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON: SYNTHESIS AND LNP FORMULATION ALDEXCHEM KFT. (HU) 2025-03-13 WO disclosed
EP-4520765-A1 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON AldexChem Kft. (HU) 2025-03-12 EP disclosed
US-12247990-B2 Molecular hopper OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2025-03-11 US disclosed
WO-2025047963-A1 WATER REPELLENT COMPOSITION ダイキン工業株式会社 2025-03-06 WO disclosed
WO-2025047961-A1 WATER REPELLENT COMPOSITION ダイキン工業株式会社 2025-03-06 WO disclosed
CN-113631560-B Azetidine benzodiazepine dimers and conjugates comprising the same for the treatment of cancer 麦迪穆有限责任公司 2025-02-18 CN disclosed
WO-2025023238-A1 FIBER STRUCTURE ダイキン工業株式会社 2025-01-30 WO disclosed
US-12209099-B2 Azetidobenzodiazepine dimers and conjugates comprising them for use in the treatment of cancer MEDIMMUNE LIMITED (GB) 2025-01-28 US disclosed
EP-4488285-A2 MOLECULAR HOPPER Oxford University Innovation Limited (GB) 2025-01-08 EP disclosed
WO-2024259190-A2 5'-MODIFIED MONOMERS, OLIGONUCLEOTIDES AND DOUBLE-STRANDED RNAS ALNYLAM PHARMACEUTICALS, INC. (US) 2024-12-19 WO disclosed
EP-3824285-B1 MOLECULAR HOPPER UNIV OXFORD INNOVATION LTD (GB) 2024-12-11 EP disclosed
US-20240400536-A1 IDEBENONE DERIVATIVES AND THEIR USE IN TREATING PLANTS MITORX THERAPEUTICS LTD (GB) 2024-12-05 US disclosed
US-20240383827-A1 DIFLUOROCARBENE RADIOSYNTHESIS OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2024-11-21 US disclosed
WO-2024219501-A1 GLYCOLIPID DERIVATIVE AS MINCLE LIGAND 国立大学法人大阪大学 2024-10-24 WO disclosed
WO-2024200821-A2 MANUFACTURING OF HYBRID ORGANIC-INORGANIC SILICA AEROGELS AEROBEL BV (BE) 2024-10-03 WO disclosed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO disclosed
WO-2024185707-A1 FLUORINE-CONTAINING COMPOUND ダイキン工業株式会社 2024-09-12 WO disclosed
WO-2024180157-A1 PROTEOLYSIS-TARGETING CHIMERAS TOCRIS COOKSON LIMITED (GB) 2024-09-06 WO disclosed
CN-118414150-A Pharmaceutical composition with enhanced stability characteristics 阿奎斯蒂弗医疗股份有限公司 2024-07-30 CN disclosed
US-20240246905-A1 VINYL ISOCYANIDE COMPOUNDS AS ANTIBACTERIAL AGENTS UNIVERSITY OF LEICESTER (GB) 2024-07-25 US disclosed
EP-4396174-A1 IDEBENONE DERIVATIVES AND THEIR USE IN TREATING PLANTS Mitorx Therapeutics Limited (GB) 2024-07-10 EP disclosed
WO-2024127333-A1 CYTOTOXIC COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2024-06-20 WO disclosed
WO-2024127332-A1 CYTOTOXIC COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2024-06-20 WO disclosed
EP-4364754-A2 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2024-05-08 EP disclosed
WO-2024074849-A1 PROTEOLYSIS-TARGETING CHIMERAS AGAINST THE PAPAIN-LIKE PROTEASE OF SARS-COV-2 TOCRIS COOKSON LIMITED (GB) 2024-04-11 WO disclosed
WO-2024074848-A1 PROTACS USEFUL AGAINST THE MAIN PROTEASE SARS-COV-2 TOCRIS COOKSON LIMITED (GB) 2024-04-11 WO disclosed
US-20240109916-A1 CYTOTOXIC AGENTS PHEON THERAPEUTICS LTD (GB) 2024-04-04 US disclosed
EP-4337635-A1 VINYL ISOCYANIDE COMPOUNDS AS ANTIBACTERIAL AGENTS University of Leicester (GB) 2024-03-20 EP disclosed
EP-3612234-B1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE ADC THERAPEUTICS SA (CH) 2024-03-13 EP disclosed
WO-2024047354-A1 EMULSION QUADRISE INTERNATIONAL LIMITED (GB) 2024-03-07 WO disclosed
EP-4317991-A1 HIGHLY SENSITIVE IMMUNOASSAY REAGENT AND MEASUREMENT METHOD LSI Medience Corporation (JP) 2024-02-07 EP disclosed
WO-2024023174-A2 IONIZABLE CATIONIC LIPIDS INCORPORATING SILICON ALDEXCHEM KFT. (HU) 2024-02-01 WO disclosed
US-20240002379-A1 ASYMMETRIC CONJUGATE COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2024-01-04 US disclosed
US-20230372528-A1 GLYCOCONJUGATES UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2023-11-23 US disclosed
US-11813335-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2023-11-14 US disclosed
EP-3938372-B1 AZETIDOBENZODIAZEPINE DIMERS AND CONJUGATES COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER MEDIMMUNE LTD (GB) 2023-10-25 EP disclosed
US-20230332348-A1 SILICONE POLYETHER POLYMER TREATMENTS FOR FIBROUS SUBSTRATES THE CHEMOURS COMPANY FC, LLC (US) 2023-10-19 US disclosed
US-11779650-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2023-10-10 US disclosed
US-11771775-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2023-10-03 US disclosed
US-20230302142-A1 Cytotoxic Agents Pheon Therapeutics Ltd. (GB) 2023-09-28 US disclosed
EP-4247828-A1 PROTECTED DISACCHARIDES, THEIR PROCESS OF PREPARATION AND THEIR USE IN THE SYNTHESIS OF ZWITTERIONIC OLIGOSACCHARIDES, AND CONJUGATES THEREOF Institut Pasteur (FR) 2023-09-27 EP disclosed
US-11746116-B2 Antibiotic resistance breakers KING'S COLLEGE LONDON (GB) 2023-09-05 US disclosed
EP-4219638-A1 MODIFIED NATURAL MATERIAL AND USE THEREOF Daikin Industries, Ltd. (JP) 2023-08-02 EP disclosed
EP-4218929-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2023-08-02 EP disclosed
EP-4211192-A1 SILICONE POLYETHER POLYMER TREATMENTS FOR FIBROUS SUBSTRATES The Chemours Company FC, LLC (US) 2023-07-19 EP disclosed
US-11702473-B2 Site-specific antibody-drug conjugates MEDIMMUNE LIMITED (GB) 2023-07-18 US disclosed
US-20230220217-A1 MODIFIED NATURAL MATERIAL AND USE THEREOF DAIKIN INDUSTRIES, LTD. (JP) 2023-07-13 US disclosed
US-11690918-B2 Pyrrolobenzodiazepine-anti-CD22 antibody conjugates MEDIMMUNE LIMITED (GB) 2023-07-04 US disclosed
EP-4188927-A1 CYTOTOXIC AGENTS Pheon Therapeutics Ltd (GB) 2023-06-07 EP disclosed
WO-2023092188-A1 \"COMPOUNDS AND METHODS\ DemAgtech Pty Ltd (AU) 2023-06-01 WO disclosed
US-11649250-B2 Pyrrolobenzodiazepine conjugates MEDIMMUNE LIMITED (GB) 2023-05-16 US disclosed
US-20230135723-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2023-05-04 US disclosed
US-20230120736-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2023-04-20 US disclosed
EP-4163350-A1 WATER REPELLENT COMPOSITION, KIT, WATER REPELLENT FIBER PRODUCT AND METHOD FOR MANUFACTURING SAME MEISEI CHEMICAL WORKS, LTD. (JP) 2023-04-12 EP disclosed
WO-2023047104-A1 DIFLUOROCARBENE RADIOSYNTHESIS OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2023-03-30 WO disclosed
US-11612665-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2023-03-28 US disclosed
WO-2023041906-A1 IDEBENONE DERIVATIVES AND THEIR USE IN TREATING PLANTS MITORX THERAPEUTICS LIMITED (GB) 2023-03-23 WO disclosed
US-20230053603-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2023-02-23 US disclosed
US-20230015617-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2023-01-19 US disclosed
EP-4103727-A2 PRODUCTION OF GLYCOSYLATED PRODUCT IN HOST CELLS Inbiose N.V. (BE) 2022-12-21 EP disclosed
EP-4103726-A1 KDO-FREE PRODUCTION HOSTS FOR OLIGOSACCHARIDE SYNTHESIS Inbiose N.V. (BE) 2022-12-21 EP disclosed
US-11524969-B2 Pyrrolobenzodiazepines and conjugates thereof as antitumour agents MEDIMMUNE LIMITED (GB) 2022-12-13 US disclosed
US-20220389419-A1 MODIFIED OLIGONUCLEOTIDES ALNYLAM PHARMACEUTICALS, INC. (US) 2022-12-08 US disclosed
WO-2022238694-A1 VINYL ISOCYANIDE COMPOUNDS AS ANTIBACTERIAL AGENTS THE UNIVERSITY OF BATH (GB) 2022-11-17 WO disclosed
EP-3356477-B1 HYDROPHOBIC EXTENDERS IN FLUORINATED SURFACE EFFECT COATINGS CHEMOURS CO FC LLC (US) 2022-11-09 EP disclosed
US-11484606-B2 Pyrrolobenzodiazepine-antibody conjugates OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2022-11-01 US disclosed
US-11466032-B2 Cytotoxic agents FEMTOGENIX LIMITED 2022-10-11 US disclosed
WO-2022211009-A1 HIGHLY SENSITIVE IMMUNOASSAY REAGENT AND MEASUREMENT METHOD 株式会社LSIメディエンス 2022-10-06 WO disclosed
US-11459485-B2 Non-fluorinated coating and finish agents THE CHEMOURS COMPANY FC, LLC (US) 2022-10-04 US disclosed
US-20220306660-A1 Guanine Analogs as Telomerase Substrates and Telomere Length Affectors BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2022-09-29 US disclosed
US-20220298161-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SARL (CH) 2022-09-22 US disclosed
US-20220288221-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2022-09-15 US disclosed
EP-2771696-B1 METHODS MAKING USE OF PANELS OF METABOLITES FOR THE DIAGNOSIS AND DIFFERENTIATION OF NEONATAL ENCEPHALOPATHY INFANDX AG (DE) 2022-09-14 EP disclosed
EP-4045180-A1 DEVICE FOR AUTOMATED SYNTHESIS OF OLIGO- AND POLYSACCHARIDES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2022-08-24 EP disclosed
EP-4045182-A1 MICROWAVE-ASSISTED METHOD FOR SYNTHESIS OF OLIGO- AND POLYSACCHARIDES ON SOLID PHASE Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2022-08-24 EP disclosed
EP-4041248-A1 MODIFIED OLIGONUCLEOTIDES Alnylam Pharmaceuticals Inc. (US) 2022-08-17 EP disclosed
EP-4039280-A1 TARGETED PYRROLOBENZODIAZEPINE CONJUGATES Seagen Inc. (US) 2022-08-10 EP disclosed
EP-3612537-B1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LTD (GB) 2022-07-13 EP disclosed
US-11384098-B2 Pyrrolobenzodiazepine-antibody conjugates ADC THERAPEUTICS SA (CH) 2022-07-12 US disclosed
US-11370801-B2 Pyrrolobenzodiazepine conjugates MEDIMMUNE LIMITED (GB) 2022-06-28 US disclosed
US-11359099-B2 Hydrophobic extenders in fluorinated surface effect coatings THE CHEMOURS COMPANY FC, LLC (US) 2022-06-14 US disclosed
EP-3710066-B1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LTD (GB) 2022-06-08 EP disclosed
WO-2022106703-A1 PROTECTED DISACCHARIDES, THEIR PROCESS OF PREPARATION AND THEIR USE IN THE SYNTHESIS OF ZWITTERIONIC OLIGOSACCHARIDES, AND CONJUGATES THEREOF INSTITUT PASTEUR (FR) 2022-05-27 WO disclosed
US-20220160905-A1 FLUORINATION METHOD OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2022-05-26 US disclosed
US-20220160881-A1 AZETIDOBENZODIAZEPINE DIMERS AND CONJUGATES COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER MEDIMMUNE LIMITED (GB) 2022-05-26 US disclosed
WO-2022079211-A1 GLYCOCONJUGATES ADC THERAPEUTICS SA (CH) 2022-04-21 WO disclosed
WO-2022065382-A1 MODIFIED NATURAL MATERIAL AND USE THEREOF ダイキン工業株式会社 2022-03-31 WO disclosed
US-20220098191-A1 G-A CROSSLINKING CYTOTOXIC AGENTS Pheon Therapeutics Ltd. (GB) 2022-03-31 US disclosed
WO-2022055884-A1 SILICONE POLYETHER POLYMER TREATMENTS THE CHEMOURS COMPANY FC, LLC (US) 2022-03-17 WO disclosed
WO-2022055874-A1 SILICONE POLYETHER POLYMER TREATMENTS FOR FIBROUS SUBSTRATES THE CHEMOURS COMPANY FC, LLC (US) 2022-03-17 WO disclosed
US-11274220-B2 Hydrophobic extenders in non-fluorinated surface effect coatings THE CHEMOURS COMPANY FC, LLC (US) 2022-03-15 US disclosed
WO-2022023735-A1 CYTOTOXIC AGENTS FEMTOGENIX LIMITED (GB) 2022-02-03 WO disclosed
US-20220016261-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2022-01-20 US disclosed
EP-2558127-B1 TARGETED PYRROLOBENZODIAZEPINE CONJUGATES SEAGEN INC (US) 2022-01-19 EP disclosed
EP-3938372-A1 AZETIDOBENZODIAZEPINE DIMERS AND CONJUGATES COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER MedImmune Limited (GB) 2022-01-19 EP disclosed
EP-3939616-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics SA (CH) 2022-01-19 EP disclosed
US-20220008552-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES BLUE OWL OPPORTUNISTIC MASTER FUND I, L.P. (FORMERLY KNOWN AS OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P.) 2022-01-13 US disclosed
US-20220010296-A1 METHODS AND COMPOSITIONS UNITED KINGDOM RESEARCH AND INNOVATION (GB) 2022-01-13 US disclosed
EP-3668874-B1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LTD (GB) 2021-12-22 EP disclosed
US-20210380605-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2021-12-09 US disclosed
EP-3917924-A1 G-A CROSSLINKING CYTOTOXIC AGENTS Femtogenix Limited (GB) 2021-12-08 EP disclosed
US-20210371413-A1 POLYCYCLIC AMIDES AS CYTOTOXIC AGENTS Pheon Therapeutics Ltd. (GB) 2021-12-02 US disclosed
US-11160803-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2021-11-02 US disclosed
US-11160872-B2 Pyrrolobenzodiazepine-antibody conjugates ADC THERAPEUTICS SA (CH) 2021-11-02 US disclosed
US-20210316006-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2021-10-14 US disclosed
US-20210318340-A1 MOLECULAR HOPPER OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2021-10-14 US disclosed
US-11135303-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2021-10-05 US disclosed
EP-3356476-B1 HYDROPHOBIC EXTENDERS IN NON-FLUORINATED SURFACE EFFECT COATINGS CHEMOURS CO FC LLC (US) 2021-09-22 EP disclosed
US-20210284613-A1 RADIOLABELLED COMPOUND OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2021-09-16 US disclosed
US-20210283141-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2021-09-16 US disclosed
WO-2021160828-A1 KDO-FREE PRODUCTION HOSTS FOR OLIGOSACCHARIDE SYNTHESIS INBIOSE N.V. (BE) 2021-08-19 WO disclosed
WO-2021160827-A2 PRODUCTION OF GLYCOSYLATED PRODUCT IN HOST CELLS INBIOSE N.V. (BE) 2021-08-19 WO disclosed
EP-3579883-B1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2021-08-11 EP disclosed
EP-3535336-B1 COATINGS INCORPORATING NON-FLUORINATED CLEANABILITY ADDITIVES CHEMOURS CO FC LLC (US) 2021-08-11 EP disclosed
US-20210230395-A1 SOLID POLYMERIC ARTICLES HAVING HYDROPHOBIC COMPOUNDS INTERMIXED THEREIN THE CHEMOURS COMPANY FC, LLC (US) 2021-07-29 US disclosed
EP-3849956-A1 FLUORINATION METHOD Oxford University Innovation Limited (GB) 2021-07-21 EP disclosed
EP-3847166-A1 POLYCYCLIC AMIDES AS CYTOTOXIC AGENTS Femtogenix Limited (GB) 2021-07-14 EP disclosed
EP-3197931-B1 USE OF NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES IN COATINGS CHEMOURS CO FC LLC (US) 2021-07-14 EP disclosed
EP-3835322-A2 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2021-06-16 EP disclosed
US-20210171637-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2021-06-10 US disclosed
EP-3824285-A1 MOLECULAR HOPPER Oxford University Innovation Limited (GB) 2021-05-26 EP disclosed
US-11008439-B2 Solid polymeric articles having hydrophobic compounds intermixed therein THE CHEMOURS COMPANY FC, LLC (US) 2021-05-18 US disclosed
US-20210137940-A1 PYRROLOBENZODIAZEPINE-ANTI-PSMA ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2021-05-13 US disclosed
EP-3313453-B1 METHOD FOR IMAGING ARTHRITIS GUYS AND ST THOMAS HOSPITAL NHS FOUND TRUST (GB) 2021-04-28 EP disclosed
WO-2021074182-A1 PRODUCTION OF BIOPRODUCT IN A HOST CELL INBIOSE N.V. (BE) 2021-04-22 WO disclosed
US-20210113587-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2021-04-22 US disclosed
US-20210107923-A1 CYTOTOXIC AGENTS PHEON THERAPEUTICS LTD (GB) 2021-04-15 US disclosed
EP-3578563-B1 GUANINE ANALOGS AS TELOMERASE SUBSTRATES AND TELOMERE LENGTH AFFECTORS GERON CORP (US) 2021-04-14 EP disclosed
EP-3801630-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2021-04-14 EP disclosed
US-20210093731-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2021-04-01 US disclosed
EP-3544636-B1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2021-03-31 EP disclosed
US-10960570-B2 Additives for lignocellulosic composites HEXION INC. (US) 2021-03-30 US disclosed
US-20210079023-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF AS ANTITUMOUR AGENTS MEDIMMUNE LIMITED (GB) 2021-03-18 US disclosed
US-20210079020-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2021-03-18 US disclosed
EP-3525830-B1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LTD (GB) 2021-03-10 EP disclosed
CN-112391092-A Acrylic resin coating 上海婉静纺织科技有限公司 2021-02-23 CN disclosed
EP-2935268-B2 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LTD (GB) 2021-02-17 EP disclosed
EP-3774699-A1 RADIOLABELLED COMPOUND Oxford University Innovation Limited (GB) 2021-02-17 EP disclosed
EP-3774820-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF AS ANTITUMOUR AGENTS MedImmune Limited (GB) 2021-02-17 EP disclosed
CN-112239523-A Acrylic resin and preparation method thereof 宁波高新区巴艺新材料科技有限公司 2021-01-19 CN disclosed
US-20200405873-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2020-12-31 US disclosed
US-20200405880-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES BLUE OWL OPPORTUNISTIC MASTER FUND I, L.P. (FORMERLY KNOWN AS OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P.) 2020-12-31 US disclosed
US-20200405878-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2020-12-31 US disclosed
US-20200399365-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2020-12-24 US disclosed
WO-2020245283-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2020-12-10 WO disclosed
US-20200345861-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES BLUE OWL OPPORTUNISTIC MASTER FUND I, L.P. (FORMERLY KNOWN AS OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P.) 2020-11-05 US disclosed
US-20200338209-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2020-10-29 US disclosed
EP-3198072-B1 NON-FLUORINATED URETHANE BASED COATINGS CHEMOURS CO FC LLC (US) 2020-10-28 EP disclosed
US-10799596-B2 Pyrrolobenzodiazepine-antibody conjugates ADC THERAPEUTICS S.A. (CH) 2020-10-13 US disclosed
US-10799595-B2 Pyrrolobenzodiazepine conjugates MEDIMMUNE LIMITED (GB) 2020-10-13 US disclosed
US-20200306385-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2020-10-01 US disclosed
EP-3356474-B1 COATINGS INCORPORATING HYDROPHOBIC COMPOUNDS CHEMOURS CO FC LLC (US) 2020-09-30 EP disclosed
WO-2020187721-A1 AZETIDOBENZODIAZEPINE DIMERS AND CONJUGATES COMPRISING THEM FOR USE IN THE TREATMENT OF CANCER MEDIMMUNE LIMITED (GB) 2020-09-24 WO disclosed
EP-3710066-A1 PYRROLOBENZODIAZEPINE CONJUGATES Medimmune Limited (GB) 2020-09-23 EP disclosed
US-10780181-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2020-09-22 US disclosed
US-10780096-B2 Pyrrolobenzodiazepine-antibody conjugates ADC THERAPEUTICS SA (CH) 2020-09-22 US disclosed
US-20200289660-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2020-09-17 US disclosed
US-20200283461-A1 Guanine Analogs as Telomerase Substrates and Telomere Length Affectors BIOPHARMA CREDIT PLC [COLLATERAL AGENT] (GB) 2020-09-10 US disclosed
US-10751346-B2 Pyrrolobenzodiazepine—anti-PSMA antibody conjugates MEDIMMUNE LIMITED (GB) 2020-08-25 US disclosed
US-10736903-B2 Pyrrolobenzodiazepine-anti-PSMA antibody conjugates MEDIMMUNE LIMITED (GB) 2020-08-11 US disclosed
WO-2020157491-A1 G-A CROSSLINKING CYTOTOXIC AGENTS FEMTOGENIX LIMITED (GB) 2020-08-06 WO disclosed
US-20200247823-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2020-08-06 US disclosed
US-10729793-B2 Method for imaging arthritis GUY'S AND ST. THOMAS' HOSPITAL NHS FOUNDATION TRUST (GB) 2020-08-04 US disclosed
US-10722594-B2 Pyrrolobenzodiazepine-anti-CD22 antibody conjugates ADC THERAPEUTICS S.A. (CH) 2020-07-28 US disclosed
EP-3679045-A1 CYTOTOXIC AGENTS Femtogenix Limited (GB) 2020-07-15 EP disclosed
US-10695433-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2020-06-30 US disclosed
EP-3668874-A1 PYRROLOBENZODIAZEPINE CONJUGATES Medimmune Limited (GB) 2020-06-24 EP disclosed
US-20200147235-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2020-05-14 US disclosed
US-10640563-B2 Anti-B7-H3 antibodies and antibody drug conjugates ABBVIE INC. (US) 2020-05-05 US disclosed
US-20200129637-A1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2020-04-30 US disclosed
US-20200121803-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2020-04-23 US disclosed
WO-2020079229-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2020-04-23 WO disclosed
WO-2020079239-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2020-04-23 WO disclosed
US-20200115390-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2020-04-16 US disclosed
EP-3630779-A1 ANTIBIOTIC RESISTANCE BREAKERS Kings College London (GB) 2020-04-08 EP disclosed
EP-2182936-B1 SUBSTRATE REDUCTION THERAPY THE CHANCELLOR MASTERS AND SCHOLARS OF THE UNIV OF OXFORD (GB) 2020-04-01 EP disclosed
WO-2020053596-A1 FLUORINATION METHOD OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2020-03-19 WO disclosed
US-10576164-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2020-03-03 US disclosed
EP-3612537-A1 PYRROLOBENZODIAZEPINE CONJUGATES Medimmune Limited (GB) 2020-02-26 EP disclosed
EP-3612234-A1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE ADC Therapeutics SA (CH) 2020-02-26 EP disclosed
US-20200054761-A1 METHODS AND COMPOSITION FOR INHIBITING TUMOR GROWTH AND ENHANCING IMMUNE RESPONSES TO TUMORS THOMAS JEFFERSON UNIVERSITY (US) 2020-02-20 US disclosed
US-10561739-B2 Targeted pyrrolobenzodiazapine conjugates SEATTLE GENETICS INC. (US) 2020-02-18 US disclosed
US-10562926-B2 Guanine analogs as telomerase substrates and telomere length affectors GERON CORPORATION (US) 2020-02-18 US disclosed
US-10544223-B2 Combination therapy with an anti-axl antibody-drug conjugate ADC THERAPEUTICS SA (CH) 2020-01-28 US disclosed
WO-2020016573-A1 MOLECULAR HOPPER OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2020-01-23 WO disclosed
US-10514383-B2 Diagnosis and treatment of neonatal encephalopathy INFANDX AG (DE) 2019-12-24 US disclosed
WO-2019224340-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2019-11-28 WO disclosed
CN-110461366-A Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LTD 2019-11-15 CN disclosed
US-20190336614-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES SEAGEN INC. 2019-11-07 US disclosed
US-10449192-B2 Phthalazinone derivatives KUDO PHARMACEUTICALS LIMITED (GB) 2019-10-22 US disclosed
WO-2019197602-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF AS ANTITUMOUR AGENTS MEDIMMUNE LIMITED (GB) 2019-10-17 WO disclosed
WO-2019186135-A1 RADIOLABELLED COMPOUND OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2019-10-03 WO disclosed
EP-3544636-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics SA (CH) 2019-10-02 EP disclosed
CN-110300601-A Pyrrolobenzodiazepines *-antibody conjugates ADC治疗有限公司 2019-10-01 CN disclosed
US-10420777-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2019-09-24 US disclosed
CN-110267686-A Pyrrolobenzodiazepines *-antibody conjugates ADC治疗有限公司 2019-09-20 CN disclosed
US-20190282705-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2019-09-19 US disclosed
EP-3535336-A1 COATINGS INCORPORATING NON-FLUORINATED CLEANABILITY ADDITIVES The Chemours Company FC, LLC (US) 2019-09-11 EP disclosed
EP-3535331-A1 NON-FLUORINATED COATING AND FINISH AGENTS The Chemours Company FC, LLC (US) 2019-09-11 EP disclosed
US-20190270219-A1 ADDITIVES FOR LIGNOCELLULOSIC COMPOSITES HEXION INC. 2019-09-05 US disclosed
US-10399970-B2 Pyrridinobenzodiazepine and benzopyrridodiazecine compounds FEMTOGENIX LIMITED (GB) 2019-09-03 US disclosed
US-10392393-B2 Pyrrolobenzodiazepines MEDIMMUNE LIMITED (GB) 2019-08-27 US disclosed
US-20190256739-A1 NON-FLUORINATED COATING AND FINISH AGENTS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2019-08-22 US disclosed
US-20190256729-A1 COATINGS INCORPORATING NON-FLUORINATED CLEANABILITY ADDITIVES JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2019-08-22 US disclosed
EP-3525830-A1 PYRROLOBENZODIAZEPINE CONJUGATES Medimmune Limited (GB) 2019-08-21 EP disclosed
EP-3191490-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LTD (GB) 2019-08-07 EP disclosed
US-20190218291-A1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2019-07-18 US disclosed
US-10328084-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2019-06-25 US disclosed
US-10329352-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2019-06-25 US disclosed
CN-105209077-B Pyrrolobenzodiazepines and conjugates thereof 麦迪穆有限责任公司 2019-06-11 CN disclosed
US-10308898-B2 Method of imparting water repellency with non-fluorinated laundry treatment compositions THE CHEMOURS COMPANY FC, LLC (US) 2019-06-04 US disclosed
CN-109843335-A Pyrrolobenzodiazepines Zhuo conjugate 麦迪穆有限责任公司 2019-06-04 CN disclosed
US-20190144443-A1 ASYMMETRIC CONJUGATE COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2019-05-16 US disclosed
EP-2794624-B1 GUANINE ANALOGS AS TELOMERASE SUBSTRATES AND TELOMERE LENGTH AFFECTORS GERON CORP (US) 2019-05-15 EP disclosed
US-10287220-B2 Fluorination method OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2019-05-14 US disclosed
US-20190134216-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2019-05-09 US disclosed
EP-3197963-B1 NON-FLUORINATED MONOMERS AND POLYMERS FOR SURFACE EFFECT COMPOSITIONS CHEMOURS CO FC LLC (US) 2019-05-01 EP disclosed
US-20190119433-A1 SULFONATED FLUORINATED, NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2019-04-25 US disclosed
EP-2968594-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LTD (GB) 2019-04-24 EP disclosed
EP-3468599-A2 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-04-17 EP disclosed
EP-3469000-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-04-17 EP disclosed
EP-3468598-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-04-17 EP disclosed
EP-3468596-A2 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-04-17 EP disclosed
EP-3468993-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-04-17 EP disclosed
US-20190106447-A1 Guanine Analogs as Telomerase Substrates and Telomere Length Affectors BIOPHARMA CREDIT PLC [COLLATERAL AGENT] (GB) 2019-04-11 US disclosed
CN-109562169-A anti-CD 98 antibodies and antibody drug conjugates 艾伯维公司 2019-04-02 CN disclosed
CN-109562168-A anti-CD 98 antibodies and antibody drug conjugates 艾伯维公司 2019-04-02 CN disclosed
CN-109562170-A anti-CD 98 antibodies and antibody drug conjugates 艾伯维公司 2019-04-02 CN disclosed
US-10246608-B2 Non-fluorinated urethane based coatings THE CHEMOURS COMPANY FC, LLC (US) 2019-04-02 US disclosed
EP-3458479-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2019-03-27 EP disclosed
US-20190085017-A1 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY CLINIGEN GROUP PLC (GB) 2019-03-21 US disclosed
EP-3455225-A1 ASYMMETRIC CONJUGATE COMPOUNDS Femtogenix Limited (GB) 2019-03-20 EP disclosed
EP-2902402-B1 WATER-SOLUBLE PHOTOCHROMIC MOLECULE RIKKYO EDUCATIONAL CORP (JP) 2019-03-13 EP disclosed
WO-2019043417-A1 CYTOTOXIC AGENTS FEMTOGENIX LIMITED (GB) 2019-03-07 WO disclosed
US-20190070305-A1 BENZODIAZEPINES AND CONJUGATES THEREOF IMMUNOGEN, INC. 2019-03-07 US disclosed
WO-2019034764-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2019-02-21 WO disclosed
US-20190055254-A1 PYRROLOBENZODIAZEPINES MEDIMMUNE LIMITED (GB) 2019-02-21 US disclosed
US-10208155-B2 Sulfonated fluorinated, non-fluorinated or partially fluorinated urethanes THE CHEMOURS COMPANY FC, LLC (US) 2019-02-19 US disclosed
US-20190040270-A1 COATINGS INCORPORATING HYDROPHOBIC COMPOUNDS THE CHEMOURS COMPANY FC, LLC (US) 2019-02-07 US disclosed
US-10188746-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2019-01-29 US disclosed
US-20190015524-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2019-01-17 US disclosed
CN-106687472-B Pyrrolobenzodiazepines Zhuo and its conjugate 麦迪穆有限责任公司 2019-01-08 CN disclosed
CN-109071502-A Pyrrolobenzodiazepines * 麦迪穆有限责任公司 2018-12-21 CN disclosed
US-20180362644-A1 PYRROLOBENZODIAZEPINES AND ANTIBODY DISULFIDE CONJUGATES THEREOF GENENTECH INC (US) 2018-12-20 US disclosed
WO-2018220365-A1 ANTIBIOTIC RESISTANCE BREAKERS KING'S COLLEGE LONDON (GB) 2018-12-06 WO disclosed
EP-3408267-A1 PYRROLOBENZODIAZEPINES Medimmune Limited (GB) 2018-12-05 EP disclosed
US-10138594-B2 Partially fluorinated urethane based coatings THE CHEMOURS COMPANY FC, LLC (US) 2018-11-27 US disclosed
US-20180320309-A1 CARPET WITH HYDROPHOBIC SURFACE FINISH JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2018-11-08 US disclosed
US-20180320005-A1 HYDROPHOBIC EXTENDERS IN NON-FLUORINATED SURFACE EFFECT COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2018-11-08 US disclosed
WO-2018192944-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2018-10-25 WO disclosed
WO-2018193102-A1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE ADC THERAPEUTICS SA (CH) 2018-10-25 WO disclosed
US-20180303953-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC THERAPEUTICS S.A. (CH) 2018-10-25 US disclosed
EP-3388435-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES Seattle Genetics, Inc. (US) 2018-10-17 EP disclosed
US-10098968-B2 Anti-EGFR antibodies and antibody drug conjugates ABBVIE INC. (US) 2018-10-16 US disclosed
US-20180282514-A1 SOLID POLYMERIC ARTICLES HAVING HYDROPHOBIC COMPOUNDS INTERMIXED THEREIN JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2018-10-04 US disclosed
US-20180282571-A1 HYDROPHOBIC COMPOUND EXTENDERS IN SURFACE EFFECT COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2018-10-04 US disclosed
US-20180273774-A1 HYDROPHOBIC EXTENDERS IN FLUORINATED SURFACE EFFECT COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2018-09-27 US disclosed
US-20180250417-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2018-09-06 US disclosed
WO-2018156725-A1 METHODS AND COMPOSITIONS FOR INHIBITING TUMOR GROWTH AND ENHANCING IMMUNE RESPONSES TO TUMORS THOMAS JEFFERSON UNIVERSITY (US) 2018-08-30 WO disclosed
EP-2751120-B1 PYRROLOBENZODIAZEPINES AS UNSYMMETRICAL DIMERIC PBD COMPOUNDS FOR INCLUSION IN TARGETED CONJUGATES MEDIMMUNE LTD (GB) 2018-08-22 EP disclosed
WO-2018146199-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2018-08-16 WO disclosed
WO-2018146189-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2018-08-16 WO disclosed
WO-2018146188-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2018-08-16 WO disclosed
EP-3356474-A1 COATINGS INCORPORATING HYDROPHOBIC COMPOUNDS The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
EP-3356475-A1 HYDROPHOBIC COMPOUND EXTENDERS IN SURFACE EFFECT COATINGS The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
EP-3356477-A1 HYDROPHOBIC EXTENDERS IN FLUORINATED SURFACE EFFECT COATINGS The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
EP-3356460-A1 SOLID POLYMERIC ARTICLES HAVING HYDROPHOBIC COMPOUNDS INTERMIXED THEREIN The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
EP-3356476-A1 HYDROPHOBIC EXTENDERS IN NON-FLUORINATED SURFACE EFFECT COATINGS The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
EP-3356594-A1 CARPET WITH HYDROPHOBIC SURFACE FINISH The Chemours Company FC, LLC (US) 2018-08-08 EP disclosed
US-10035814-B2 Guanine analogs as telomerase substrates and telomere length affectors GERON CORPORATION (US) 2018-07-31 US disclosed
US-10034884-B2 Pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2018-07-31 US disclosed
EP-2755642-B1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEATTLE GENETICS INC (US) 2018-07-18 EP disclosed
EP-2968585-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LTD (GB) 2018-07-18 EP disclosed
US-20180193480-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2018-07-12 US disclosed
US-10017580-B2 Humanized anti-Tn-MUC1 antibodies and their conjugates ADC Therpeutics S.A. (CH) 2018-07-10 US disclosed
US-20180185522-A1 CONTRAST AGENT FOR IMAGING HYPOXIA OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2018-07-05 US disclosed
US-20180185523-A1 METHOD FOR IMAGING ARTHRITIS GUY'S AND ST. THOMAS' HOSPITAL NHS FOUNDATION TRUST (GB) 2018-07-05 US disclosed
US-20180185363-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2018-07-05 US disclosed
US-10011617-B2 Isocyanate derived organosilanes THE CHEMOURS COMPANY FC, LLC (US) 2018-07-03 US disclosed
EP-2906249-B1 SYNTHESIS AND INTERMEDIATES OF PYRROLOBENZODIAZEPINE DERIVATIVES FOR CONJUGATION MEDIMMUNE LTD (GB) 2018-06-27 EP disclosed
US-20180169259-A1 ANTI-CD79B ANTIBODIES AND IMMUNOCONJUGATES GENENTECH INC. (US) 2018-06-21 US disclosed
US-20180169258-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2018-06-21 US disclosed
US-9999625-B2 Pyrrolobenzodiazepine compounds FEMTOGENIX LIMITED (GB) 2018-06-19 US disclosed
US-20180162855-A1 PDD AND BPD COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2018-06-14 US disclosed
EP-3328497-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics SA (CH) 2018-06-06 EP disclosed
US-20180134717-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN LIMITED (GB) 2018-05-17 US disclosed
US-20180125796-A1 TREATMENT OF MYCOBACTERIAL INFECTION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-05-10 US disclosed
US-20180127505-A1 HUMANIZED ANTI-AXL ANTIBODIES AND THEIR CONJUGATES ADC THERAPEUTICS SA (CH) 2018-05-10 US disclosed
US-20180125997-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2018-05-10 US disclosed
US-20180125999-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2018-05-10 US disclosed
US-20180125994-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES MEDIMMUNE LIMITED (GB) 2018-05-10 US disclosed
US-20180117172-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2018-05-03 US disclosed
EP-3313453-A1 METHOD FOR IMAGING ARTHRITIS Guy's And St Thomas' Nhs Foundation Trust (GB) 2018-05-02 EP disclosed
US-9957661-B2 Polyurethanes derived from non-fluorinated or partially fluorinated polymers THE CHEMOURS COMPANY FC, LLC (US) 2018-05-01 US disclosed
EP-2751076-B1 SYNTHESIS METHOD AND INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2018-04-25 EP disclosed
WO-2018069490-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2018-04-19 WO disclosed
EP-3309162-A1 TARGETED CONJUGATES OF PYRROLOBENZODIAZEPINES Seattle Genetics, Inc. (US) 2018-04-18 EP disclosed
EP-3307743-A1 PDD AND BPD COMPOUNDS Femtogenix Limited (GB) 2018-04-18 EP disclosed
US-20180099055-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES MEDIMMUNE LIMITED (GB) 2018-04-12 US disclosed
US-9938431-B2 Use of non-fluorinated or partially fluorinated urethanes in coatings THE CHEMOURS COMPANY FC, LLC (US) 2018-04-10 US disclosed
US-20180092986-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES MEDIMMUNE LIMITED (GB) 2018-04-05 US disclosed
US-20180092985-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES MEDIMMUNE LIMITED (GB) 2018-04-05 US disclosed
US-9931414-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2018-04-03 US disclosed
US-9931415-B2 Pyrrolobenzodiazepine-antibody conjugates MEDIMMUNE LIMITED (GB) 2018-04-03 US disclosed
US-20180086828-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES MEDIMMUNE LIMITED (GB) 2018-03-29 US disclosed
EP-2422183-B1 OXIDATION STATE SENSORS AND METHODS FOR TRANSITION METAL ALLOYS ROLLS ROYCE PLC (GB) 2018-03-21 EP disclosed
US-9919056-B2 Pyrrolobenzodiazepine-anti-CD22 antibody conjugates ADC THERAPEUTICS S.A. (CH) 2018-03-20 US disclosed
US-9915025-B2 Non-fluorinated monomers and polymers for surface effect compositions THE CHEMOURS COMPANY FC, LLC (US) 2018-03-13 US disclosed
EP-3283116-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283119-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283121-A1 HUMANIZED ANTI-AXL ANTIBODIES AND THEIR CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283117-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283123-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283120-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES Medimmune Limited (GB) 2018-02-21 EP disclosed
EP-3283118-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
EP-3283122-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES ADC Therapeutics SA (CH) 2018-02-21 EP disclosed
CN-104684914-B Pyrrolobenzodiazepines are tall and erect 麦迪穆有限责任公司 2017-12-15 CN disclosed
US-20170355769-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2017-12-14 US disclosed
WO-2017214462-A2 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2017-12-14 WO disclosed
WO-2017214456-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2017-12-14 WO disclosed
WO-2017214335-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2017-12-14 WO disclosed
WO-2017214458-A2 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2017-12-14 WO disclosed
US-20170340752-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2017-11-30 US disclosed
US-9827330-B2 Anti-EGFR antibodies and antibody drug conjugates ABBVIE INC. (US) 2017-11-28 US disclosed
EP-2935268-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LTD (GB) 2017-11-22 EP disclosed
US-9821074-B2 Pyrrolobenzodiazepines and conjugates thereof GENENTECH, INC. (US) 2017-11-21 US disclosed
WO-2017194960-A1 ASYMMETRIC CONJUGATE COMPOUNDS FEMTOGENIX LIMITED (GB) 2017-11-16 WO disclosed
EP-3235820-A1 PYRROLOBENZODIAZEPINES AND ANTIBODY DISULFIDE CONJUGATES THEREOF Genentech, Inc. (US) 2017-10-25 EP disclosed
US-20170298137-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2017-10-19 US disclosed
US-20170290924-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2017-10-12 US disclosed
US-20170290920-A1 ANTI-CD22 ANTIBODIES AND IMMUNOCONJUGATES MEDIMMUNE LIMITED (GB) 2017-10-12 US disclosed
US-20170281637-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2017-10-05 US disclosed
EP-3223854-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics SA (CH) 2017-10-04 EP disclosed
US-20170274091-A1 BENZODIAZEPINES AND CONJUGATES THEREOF IMMUNOGEN, INC. 2017-09-28 US disclosed
US-20170267778-A1 HUMANIZED ANTI-TN-MUC1 ANTIBODIES AND THEIR CONJUGATES MEDIMMUNE LIMITED (GB) 2017-09-21 US disclosed
US-20170268165-A1 POLYURETHANES DERIVED FROM NON-FLUORINATED OR PARTIALLY FLUORINATED POLYMERS THE CHEMOURS COMPANY FC, LLC 2017-09-21 US disclosed
US-20170258934-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2017-09-14 US disclosed
CN-107148285-A Pyrrolobenzodiazepines * antibody conjugates ADC治疗股份有限公司 2017-09-08 CN disclosed
US-9745303-B2 Synthesis and intermediates of pyrrolobenzodiazepine derivatives for conjugation MEDIMMUNE LIMITED (GB) 2017-08-29 US disclosed
US-20170239365-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2017-08-24 US disclosed
EP-2869850-B1 IMMUNOCONJUGATES COMPRISING ANTI-CD79B ANTIBODIES GENENTECH INC (US) 2017-08-23 EP disclosed
US-9738675-B2 Water-soluble photochromic compound RIKKYO EDUCATIONAL CORPORATION (JP) 2017-08-22 US disclosed
CN-107073136-A Pyrrolobenzodiazepines Zhuo and its antibody disulphide conjugate 健泰科生物技术公司 2017-08-18 CN disclosed
US-20170233419-A1 Guanine Analogs as Telomerase Substrates and Telomere Length Affectors BIOPHARMA CREDIT PLC [COLLATERAL AGENT] (GB) 2017-08-17 US disclosed
US-9732084-B2 Pyrrolobenzodiazepines used to treat proliferative diseases MEDIMMUNE LIMITED (GB) 2017-08-15 US disclosed
US-20170226124-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2017-08-10 US disclosed
CN-107019804-A Target the tall and erect conjugate of Pyrrolobenzodiazepines 西雅图基因公司 2017-08-08 CN disclosed
WO-2017129652-A1 PYRROLOBENZODIAZEPINES MEDIMMUNE LIMITED (GB) 2017-08-03 WO disclosed
EP-3198072-A1 NON-FLUORINATED URETHANE BASED COATINGS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197932-A1 NON-FLUORINATED AND PARTIALLY FLUORINATED POLYMERS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197866-A1 PARTIALLY FLUORINATED URETHANE BASED COATINGS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197931-A1 USE OF NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES IN COATINGS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197865-A1 SULFONATED FLUORINATED, NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197903-A1 ISOCYANATE DERIVED ORGANOSILANES The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197963-A1 NON-FLUORINATED MONOMERS AND POLYMERS FOR SURFACE EFFECT COMPOSITIONS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
EP-3197927-A1 POLYURETHANES DERIVED FROM NON-FLUORINATED OR PARTIALLY FLUORINATED POLYMERS The Chemours Company FC, LLC (US) 2017-08-02 EP disclosed
US-9717736-B2 Pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2017-08-01 US disclosed
EP-3194400-A1 PYRROLOBENZODIAZEPINES AND ANTIBODY DISULFIDE CONJUGATES THEREOF Genentech, Inc. (US) 2017-07-26 EP disclosed
EP-3193940-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF Medimmune Limited (GB) 2017-07-26 EP disclosed
US-9713647-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2017-07-25 US disclosed
EP-3191490-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF Medimmune Limited (GB) 2017-07-19 EP disclosed
EP-1789430-B1 DERIVATES OF AVERMECTIN,AVERMECTIN MONOSACCHARIDE AND AVERMECTIN AGLYCONE MERIAL LTD (US) 2017-07-19 EP disclosed
US-9709571-B2 Method of drug design VAST BIOSCIENCE PTY LIMITED (AU) 2017-07-18 US disclosed
US-9707301-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2017-07-18 US disclosed
US-9702081-B2 Polyurethanes derived from non-fluorinated or partially fluorinated polymers THE CHEMOURS COMPANY FC, LLC (US) 2017-07-11 US disclosed
US-20170143846-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES SPIROGEN LIMITED (GB) 2017-05-25 US disclosed
US-20170145046-A1 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY CLINIGEN GROUP PLC (GB) 2017-05-25 US disclosed
US-20170137341-A1 FLUORINATION METHOD OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2017-05-18 US disclosed
CN-106687472-A Pyrrolobenzodiazepines and conjugates thereof 麦迪穆有限责任公司 2017-05-17 CN disclosed
CN-106687141-A Pyrrolobenzodiazepines and conjugates thereof 麦迪穆有限责任公司 2017-05-17 CN disclosed
US-9649390-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2017-05-16 US disclosed
EP-3164418-A1 HUMANIZED ANTI-TN-MUC1 ANTIBODIES AND THEIR CONJUGATES Cancer Research Technology Ltd (GB) 2017-05-10 EP disclosed
EP-2751111-B1 Asymmetrical bis-(5H-Pyrrolo[2,1-c][1,4]benzodiazepin-5-one) derivatives for the treatment of proliferative or autoimmune diseases MEDIMMUNE LTD (GB) 2017-04-26 EP disclosed
US-20170107235-A1 PYRROLOBENZODIAZEPINE COMPOUNDS FOR TREATING LYMPHOMA ADC PRODUCTS (UK) LIMITED (GB) 2017-04-20 US disclosed
EP-2751110-B1 Asymmetrical bis-(5H-Pyrrolo[2,1-c][1,4]benzodiazepin-5-one) derivatives for the treatment of proliferative and autoimmune diseases MEDIMMUNE LTD (GB) 2017-04-19 EP disclosed
US-9624227-B2 Unsymmetrical pyrrolobenzodiazepine-dimers for treatment of proliferative diseases MEDIMMUNE LIMITED (GB) 2017-04-18 US disclosed
EP-3148548-A1 PYRROLOBENZODIAZEPINE COMPOUNDS FOR TREATING LYMPHOMA ADC Products (UK) Limited (GB) 2017-04-05 EP disclosed
EP-2558445-B1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2017-03-22 EP disclosed
US-20170072065-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. 2017-03-16 US disclosed
US-9592240-B2 Targeted pyrrolobenzodiazapine conjugates SEATTLE GENETICS INC. (US) 2017-03-14 US disclosed
US-9593137-B2 Guanine analogs as telomerase substrates and telomere length affectors GERON CORPORATION (US) 2017-03-14 US disclosed
EP-2855482-B1 PYRROLOBENZODIAZEPINES MEDIMMUNE LTD (GB) 2017-03-01 EP disclosed
EP-2789622-B1 Pyrrolobenzodiazepines used to treat proliferative diseases MEDIMMUNE LTD (GB) 2017-03-01 EP disclosed
US-20170050971-A1 PYRROLOBENZODIAZEPINE COMPOUNDS PHEON THERAPEUTICS LTD (GB) 2017-02-23 US disclosed
US-9566276-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2017-02-14 US disclosed
US-9567340-B2 Unsymmetrical pyrrolobenzodiazepines-dimers for use in the treatment of proliferative and autoimmune diseases MEDIMMUNE LIMITED (GB) 2017-02-14 US disclosed
WO-2017020972-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES VAN BERKEL, Patricius Hendrikus Cornelis (CH) 2017-02-09 WO disclosed
EP-3126006-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES AbbVie Inc. (US) 2017-02-08 EP disclosed
US-9562049-B2 Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LIMITED (GB) 2017-02-07 US disclosed
EP-2057156-B1 2-METHYLMORPHOLINE PYRIDO-,PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS KUDOS PHARM LTD (GB) 2017-02-01 EP disclosed
US-9555125-B2 Benzodiazepines and conjugates thereof IMMUNOGEN, INC. (US) 2017-01-31 US disclosed
EP-3119737-A1 FLUORINATION METHOD Oxford University Innovation Limited (GB) 2017-01-25 EP disclosed
WO-2016207636-A1 METHOD FOR IMAGING ARTHRITIS GUY'S AND ST THOMAS' HOSPITAL NHS FOUNDATION TRUST (GB) 2016-12-29 WO disclosed
US-9526798-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2016-12-27 US disclosed
WO-2016198869-A1 PDD AND BPD COMPOUNDS FEMTOGENIX LIMITED (GB) 2016-12-15 WO disclosed
US-9493568-B2 Anti-EGFR antibodies and antibody drug conjugates ABBVIE INC. (US) 2016-11-15 US disclosed
WO-2016166300-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166302-A1 HUMANIZED ANTI-AXL ANTIBODIES AND THEIR CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166341-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166305-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-10-20 WO disclosed
WO-2016166304-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166297-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166301-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166298-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166307-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
WO-2016166299-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES VAN BERKEL PATRICIUS HENDRIKUS CORNELIS (CH) 2016-10-20 WO disclosed
US-9464141-B2 Anti-ETBR antibodies and immunoconjugates GENENTECH, INC. (US) 2016-10-11 US disclosed
US-20160289239-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2016-10-06 US disclosed
US-20160287721-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2016-10-06 US disclosed
WO-2016151295-A1 FLUORINATION PROCESS OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2016-09-29 WO disclosed
US-9428541-B2 Substrate reduction therapy THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2016-08-30 US disclosed
US-9399641-B2 Pyrrolobenzodiazepines as unsymmetrical dimeric PBD compounds for inclusion in targeted conjugates MEDIMMUNE LIMITED (GB) 2016-07-26 US disclosed
US-9399073-B2 Pyrrolobenzodiazepines SEATTLE GENETICS, INC. (US) 2016-07-26 US disclosed
WO-2016110702-A1 TREATMENT OF MYCOBACTERIAL INFECTION ISIS INNOVATION LIMITED (GB) 2016-07-14 WO disclosed
US-9388187-B2 Pyrrolobenzodiazepines MEDIMMUNE LIMITED (GB) 2016-07-12 US disclosed
US-9387259-B2 Pyrrolobenzodiazepines and targeted conjugates SEATTLE GENETICS, INC. (US) 2016-07-12 US disclosed
US-9387258-B2 2016-07-12 US disclosed
CN-102971329-B Pyrrolobenzodiazepines for the treatment of proliferative diseases 麦迪穆有限责任公司 2016-06-29 CN disclosed
US-9376440-B2 Pyrrolobenzodiazepines as antiproliferative agents MEDIMMUNE LIMITED (GB) 2016-06-28 US disclosed
WO-2016092325-A1 CONTRAST AGENT FOR IMAGING HYPOXIA ISIS INNOVATION LIMITED (GB) 2016-06-16 WO disclosed
WO-2016083468-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC THERAPEUTICS SA (CH) 2016-06-02 WO disclosed
US-9356318-B2 Gel polymer electrolyte composition KURARAY CO., LTD. (JP) 2016-05-31 US disclosed
US-20160144052-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN LIMITED (GB) 2016-05-26 US disclosed
US-20160129013-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES SEAGEN INC. 2016-05-12 US disclosed
US-9321774-B2 Pyrrolobenzodiazepines MEDIMMUNE LIMITED (GB) 2016-04-26 US disclosed
US-20160090392-A1 ISOCYANATE DERIVED ORGANOSILANES JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
WO-2016048643-A1 ISOCYANATE DERIVED ORGANOSILANES THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016049293-A1 USE OF NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES IN COATINGS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016048695-A1 PARTIALLY FLUORINATED URETHANE BASED COATINGS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
US-20160090688-A1 PARTIALLY FLUORINATED URETHANE BASED COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
WO-2016049278-A1 NON-FLUORINATED URETHANE BASED COATINGS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016048642-A1 NON-FLUORINATED MONOMERS AND POLYMERS FOR SURFACE EFFECT COMPOSITIONS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016048696-A1 POLYURETHANES DERIVED FROM NON-FLUORINATED OR PARTIALLY FLUORINATED POLYMERS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016049107-A1 NON-FLUORINATED AND PARTIALLY FLUORINATED POLYMERS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
US-20160090438-A1 SULFONATED FLUORINATED, NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
US-20160090687-A1 POLYURETHANES DERIVED FROM NON-FLUORINATED OR PARTIALLY FLUORINATED POLYMERS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
WO-2016048684-A1 METHOD OF IMPARTING WATER REPELLENCY WITH NON-FLUORINATED LAUNDRY TREATMENT COMPOSITIONS THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
WO-2016049282-A1 SULFONATED FLUORINATED, NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES THE CHEMOURS COMPANY FC, LLC (US) 2016-03-31 WO disclosed
US-20160090508-A1 NON-FLUORINATED URETHANE BASED COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
US-20160090686-A1 NON-FLUORINATED MONOMERS AND POLYMERS FOR SURFACE EFFECT COMPOSITIONS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
US-20160090509-A1 USE OF NON-FLUORINATED OR PARTIALLY FLUORINATED URETHANES IN COATINGS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
US-20160090505-A1 NON-FLUORINATED AND PARTIALLY FLUORINATED POLYMERS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
US-20160090560-A1 METHOD OF IMPARTING WATER REPELLENCY WITH NON-FLUORINATED LAUNDRY TREATMENT COMPOSITIONS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-03-31 US disclosed
WO-2016044560-A1 PYRROLOBENZODIAZEPINES AND ANTIBODY DISULFIDE CONJUGATES THEREOF GENENTECH, INC. (US) 2016-03-24 WO disclosed
WO-2016038383-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2016-03-17 WO disclosed
WO-2016037644-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2016-03-17 WO disclosed
US-20160074527-A1 PYRROLOBENZODIAZEPINES AND ANTIBODY DISULFIDE CONJUGATES THEREOF GENENTECH, INC. 2016-03-17 US disclosed
US-20160067258-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARM LTD (GB) 2016-03-10 US disclosed
US-9273024-B2 Synthesis of cyclic carbonates UNIVERSITY OF YORK (GB) 2016-03-01 US disclosed
US-20160056054-A1 ETCHING METHOD, ETCHING LIQUID AND ETCHING LIQUID KIT TO BE USED IN SAID METHOD, AND SEMICONDUCTOR SUBSTRATE PRODUCT MANUFACTURING METHOD FUJIFILM CORPORATION (JP) 2016-02-25 US disclosed
US-9266894-B2 2016-02-23 US disclosed
EP-2675278-B1 METHODS FOR SYNTHESIZING MOLYBDOPTERIN PRECURSOR Z DERIVATIVES ALEXION PHARMA INTERNAT SÀRL (CH) 2016-02-17 EP disclosed
US-9260382-B2 Methods of reducing virulence in bacteria UWM RESEARCH FOUNDATION (US) 2016-02-16 US disclosed
US-20160031887-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN LIMITED (GB) 2016-02-04 US disclosed
US-9242955-B2 Synthesis of cyclic carbonates UNIVERSITY OF YORK (GB) 2016-01-26 US disclosed
US-9242013-B2 Targeted pyrrolobenzodiazapine conjugates SEATTLE GENETICS INC. (US) 2016-01-26 US disclosed
EP-2968596-A2 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2016-01-20 EP disclosed
EP-2968585-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2016-01-20 EP disclosed
US-20160002144-A1 HIGH REFRACTIVE INDEX POLYMER COMPOSITION FOR OPTHALMIC APPLICATIONS CONTAMAC LTD (GB) 2016-01-07 US disclosed
US-20160000781-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2016-01-07 US disclosed
CN-105209077-A Pyrrolobenzodiazepines and conjugates thereof MEDIMMUNE LTD 2015-12-30 CN disclosed
US-9212245-B2 High performance acrylamide adhesives EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2015-12-15 US disclosed
US-9212245-B2 High performance acrylamide adhesives EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2015-12-15 US disclosed
WO-2015181559-A1 PYRROLOBENZODIAZEPINE COMPOUNDS FOR TREATING LYMPHOMA ADC PRODUCTS (UK) LIMITED (GB) 2015-12-03 WO disclosed
US-20150344482-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2015-12-03 US disclosed
US-20150337042-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2015-11-26 US disclosed
EP-2524932-B1 GEL POLYMER ELECTROLYTE COMPOSITION KURARAY CO (JP) 2015-11-25 EP disclosed
WO-2015170119-A1 OXYGEN SENSOR COMPOUNDS ISIS INNOVATION LIMITED (GB) 2015-11-12 WO disclosed
US-20150315196-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINES-DIMERS FOR USE IN THE TREATMENT OF PROLIFERATIVE AND AUTOIMMUNE DISEASES MEDIMMUNE LIMITED (GB) 2015-11-05 US disclosed
WO-2015166289-A1 PYRROLOBENZODIAZEPINE COMPOUNDS FEMTOGENIX LIMITED (GB) 2015-11-05 WO disclosed
US-20150307541-A1 WATER-SOLUBLE PHOTOCHROMIC MOLECULES RIKKYO EDUCATIONAL CORPORATION (JP) 2015-10-29 US disclosed
EP-2935268-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MedImmune Limited (GB) 2015-10-28 EP disclosed
EP-2935273-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINES-DIMERS FOR USE IN THE TREATMENT OF PROLIFERATIVE AND AUTOIMMUNE DISEASES MedImmune Limited (GB) 2015-10-28 EP disclosed
US-9169235-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2015-10-27 US disclosed
US-20150297746-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2015-10-22 US disclosed
WO-2015159076-A1 HUMANIZED ANTI-TN-MUC1 ANTIBODIES AND THEIR CONJUGATES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2015-10-22 WO disclosed
US-20150299232-A1 GUANINE ANALOGS AS TELOMERASE SUBSTRATES AND TELOMERE LENGTH AFFECTORS BIOPHARMA CREDIT PLC [COLLATERAL AGENT] (GB) 2015-10-22 US disclosed
EP-2350080-B1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN SARL (CH) 2015-10-14 EP disclosed
US-20150283258-A1 PYRROLOBENZODIAZEPINE - ANTI-PSMA ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2015-10-08 US disclosed
US-20150283263-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2015-10-08 US disclosed
US-20150283262-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2015-10-08 US disclosed
US-20150274737-A1 SYNTHESIS AND INTERMEDIATES OF PYRROLOBENZODIAZEPINE DERIVATIVES FOR CONJUGATION MEDIMMUNE LIMITED (GB) 2015-10-01 US disclosed
US-20150273078-A1 PYRROLOBENZODIAZEPINE-ANTI-PSMA ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2015-10-01 US disclosed
US-20150273077-A1 PYRROLOBENZODIAZEPINE-ANTI-HER2 ANTIBODY CONJUGATES MEDIMMUNE LIMITED (GB) 2015-10-01 US disclosed
US-20150265722-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES OWL ROCK OPPORTUNISTIC MASTER FUND I, L.P. 2015-09-24 US disclosed
WO-2015140572-A1 FLUORINATION METHOD ISIS INNOVATION LIMITED (GB) 2015-09-24 WO disclosed
WO-2015143382-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC. (US) 2015-09-24 WO disclosed
EP-2750713-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SARL (CH) 2015-09-16 EP disclosed
CN-101754769-B Use of type B lantibiotics based on antimicrobial activity NOVACTA BIOSYSTEMS LTD. (GB) 2015-09-09 CN disclosed
EP-2912043-A1 NEW ANTIBACTERIAL COMPOUNDS AND BIOLOGICAL APPLICATIONS THEREOF LABORATOIRE BIODIM (FR) 2015-09-02 EP disclosed
CN-103087841-B The method of liquid detergent compositions, its purposes, preparation method, test kit and washing articles BEIJING CONFLE TECHNOLOGY CO., LTD. (CN) 2015-09-02 CN disclosed
CN-103087847-B A kind of method of germicidal detergent composition, its purposes, preparation method and washing object BEIJING CONFLE TECHNOLOGY CO., LTD. (CN) 2015-09-02 CN disclosed
EP-2906251-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906252-A1 PYRROLOBENZODIAZEPINE-ANTI-HER2 ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906253-A1 PYRROLOBENZODIAZEPINE - ANTI-PSMA ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906249-A1 SYNTHESIS AND INTERMEDIATES OF PYRROLOBENZODIAZEPINE DERIVATIVES FOR CONJUGATION Spirogen Sàrl (CH) 2015-08-19 EP disclosed
EP-2906250-A1 PYRROLOBENZODIAZEPINE-ANTI-PSMA ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906298-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906296-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
EP-2906297-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES ADC Therapeutics S.a.r.l. (CH) 2015-08-19 EP disclosed
US-9102704-B2 Synthesis method and intermediates useful in the preparation of pyrrolobenzodiazepines SPIROGEN SARL (CH) 2015-08-11 US disclosed
US-9102670-B2 Pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2015-08-11 US disclosed
EP-2902402-A1 WATER-SOLUBLE PHOTOCHROMIC MOLECULE Rikkyo Educational Corporation (JP) 2015-08-05 EP disclosed
US-20150209444-A1 BENZODIAZEPINES AND CONJUGATES THEREOF IMMUNOGEN, INC. (US) 2015-07-30 US disclosed
EP-1812433-B1 IMIDAZO[4,5-B]PYRIDIN-2-ONE AND OXAZOLO[4,5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC COMPOUNDS CANCER REC TECH LTD (GB) 2015-07-22 EP disclosed
CN-103087842-B Germicidal detergent composition, application thereof, preparation method thereof, kit thereof and method thereof for cleaning object BEIJING CONFLE TECHNOLOGY CO LTD 2015-07-22 CN disclosed
US-20150183883-A1 ANTI-ETBR ANTIBODIES AND IMMUNOCONJUGATES GENENTECH INC (US) 2015-07-02 US disclosed
CN-104717979-A Anti-ETBR antibodies and immunoconjugates GENENTECH INC 2015-06-17 CN disclosed
US-20150158869-A1 PYRROLOBENZODIAZEPINES AS UNSYMMETRICAL DIMERIC PBD COMPOUNDS FOR INCLUSION IN TARGETED CONJUGATES MEDIMMUNE LIMITED (GB) 2015-06-11 US disclosed
EP-2879708-A2 ANTI-ETBR ANTIBODIES AND IMMUNOCONJUGATES Genentech, Inc. (US) 2015-06-10 EP disclosed
CN-104684914-A Pyrrolobenzodiazepines SPIROGEN LTD 2015-06-03 CN disclosed
US-20150133435-A1 PYRROLOBENZODIAZEPINES MEDIMMUNE LIMITED (GB) 2015-05-14 US disclosed
EP-2869849-A1 IMMUNOCONJUGATES COMPRISING ANTI-CD22 ANTIBODIES Genentech, Inc. (US) 2015-05-13 EP disclosed
EP-2869850-A1 IMMUNOCONJUGATES COMPRISING ANTI-CD79B ANTIBODIES Genentech, Inc. (US) 2015-05-13 EP disclosed
US-20150126495-A1 PYRROLOBENZODIAZEPINES MEDIMMUNE LIMITED (GB) 2015-05-07 US disclosed
US-20150111880-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES MEDIMMUNE LIMITED (GB) 2015-04-23 US disclosed
CN-104540526-A Immunoconjugates comprising anti-CD 79B antibodies GENENTECH INC 2015-04-22 CN disclosed
US-9006425-B2 Aluminum complexes and their use in the synthesis of cyclic carbonates UNIVERSITY OF YORK (GB) 2015-04-14 US disclosed
EP-2855481-A1 PYRROLOBENZODIAZEPINES UCL Business PLC (GB) 2015-04-08 EP disclosed
EP-2855482-A1 PYRROLOBENZODIAZEPINES Spirogen Sàrl (CH) 2015-04-08 EP disclosed
US-8980639-B2 Oxidation state sensors and methods for transition metal alloys ROLLS-ROYCE PLC (GB) 2015-03-17 US disclosed
WO-2015018855-A1 PENTAFLUOROETHYLATING COMPOSITIONS FUNDACIÓ INSTITUT CATALÀ D'INVESTIGACIÓ QUÍMICA (ES) 2015-02-12 WO disclosed
EP-1723152-B1 Pyrrolobenzodiazepines SPIROGEN SARL (CH) 2015-02-11 EP disclosed
EP-2835374-A1 Pentafluoroethylating compositions Fundació Institut Català d'Investigació Química (ES) 2015-02-11 EP disclosed
US-8940733-B2 Unsymmetrical pyrrolobenzodiazepine-dimers for treatment of proliferative diseases SPIROGEN SARL (CH) 2015-01-27 US disclosed
US-20140378442-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2014-12-25 US disclosed
US-8912187-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2014-12-16 US disclosed
CN-102356086-B Aluminum complexes and their use in the synthesis of cyclic carbonates UNIV NEWCASTLE 2014-11-05 CN disclosed
US-20140323726-A1 Methods for synthesizing molybdopterin precursor Z derivatives ALEXION PHARMA INTERNATIONAL SÀRL (CH) 2014-10-30 US disclosed
US-20140323726-A1 Methods for synthesizing molybdopterin precursor Z derivatives ALEXION PHARMA INTERNATIONAL SÀRL (CH) 2014-10-30 US disclosed
EP-2794624-A1 GUANINE ANALOGS AS TELOMERASE SUBSTRATES AND TELOMERE LENGTH AFFECTORS Geron Corporation (US) 2014-10-29 EP disclosed
US-20140308687-A1 Method and Use of Metabolites for the Diagnosis and Differentiation of Neonatal Encephalopathy INFANDX AG (DE) 2014-10-16 US disclosed
EP-2789622-A1 Pyrrolobenzodiazepines used to treat proliferative diseases Spirogen Sàrl (CH) 2014-10-15 EP disclosed
EP-2257559-B1 SYNTHESIS OF CYCLIC CARBONATES UNIV YORK (GB) 2014-10-15 EP disclosed
US-20140302066-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2014-10-09 US disclosed
US-20140303367-A1 Methods for Synthesizing Molybdopterin Precursor Z Derivatives ALEXION PHARMA INTERNATIONAL SÀRL (CH) 2014-10-09 US disclosed
US-20140303367-A1 Methods for Synthesizing Molybdopterin Precursor Z Derivatives ALEXION PHARMA INTERNATIONAL SÀRL (CH) 2014-10-09 US disclosed
WO-2014159981-A2 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SARL (CH) 2014-10-02 WO disclosed
US-20140294868-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2014-10-02 US disclosed
US-20140286970-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEAGEN INC. 2014-09-25 US disclosed
US-8841099-B2 Cell-based production of nonulosonates NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2014-09-23 US disclosed
WO-2014140174-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SÀRL (CH) 2014-09-18 WO disclosed
US-20140274907-A1 PYRROLOBENZODIAZEPINES SPIROGEN SARL (CH) 2014-09-18 US disclosed
US-20140275522-A1 SYNTHESIS METHOD AND INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLOBENZODIAZEPINES SPIROGEN SÁRL (CH) 2014-09-18 US disclosed
US-8829184-B2 Intermediates useful for the synthesis of pyrrolobenzodiazepines SPIROGEN SARL (CH) 2014-09-09 US disclosed
EP-2408784-B1 ALUMINUM COMPLEXES AND THEIR USE IN THE SYNTHESIS OF CYCLIC CARBONATES UNIV YORK (GB) 2014-08-27 EP disclosed
US-20140234346-A1 PYRROLOBENZODIAZEPINES SPIROGEN SÀRL (CH) 2014-08-21 US disclosed
EP-2755642-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES Seattle Genetics, Inc. (US) 2014-07-23 EP disclosed
EP-2751120-A1 PYRROLOBENZODIAZEPINES AS UNSYMMETRICAL DIMERIC PBD COMPOUNDS FOR INCLUSION IN TARGETED CONJUGATES Spirogen Sàrl (CH) 2014-07-09 EP disclosed
EP-2751076-A1 SYNTHESIS METHOD AND INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLOBENZODIAZEPINES Spirogen Sàrl (CH) 2014-07-09 EP disclosed
EP-2751111-A1 PYRROLOBENZODIAZEPINES Spirogen Sàrl (CH) 2014-07-09 EP disclosed
EP-2751110-A1 PYRROLOBENZODIAZEPINES Spirogen Sàrl (CH) 2014-07-09 EP disclosed
EP-2750713-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF Spirogen Sàrl (CH) 2014-07-09 EP disclosed
US-20140178344-A1 ACRYLAMIDE HYDROGELS FOR TISSUE ENGINEERING EMPIRE TECHNOLOGY DEVELOPMENT LLC 2014-06-26 US disclosed
WO-2014096368-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SÀRL (CH) 2014-06-26 WO disclosed
US-20140178344-A1 ACRYLAMIDE HYDROGELS FOR TISSUE ENGINEERING EMPIRE TECHNOLOGY DEVELOPMENT LLC 2014-06-26 US disclosed
WO-2014096365-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINES-DIMERS FOR USE IN THE TREATMENT OF PROLIFERATIVE AND AUTOIMMUNE DISEASES SPIROGEN SÀRL (CH) 2014-06-26 WO disclosed
WO-2014088555-A1 HIGH PERFORMANCE ACRYLAMIDE ADHESIVES EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2014-06-12 WO disclosed
WO-2014088557-A1 ACRYLAMIDE HYDROGELS FOR TISSUE ENGINEERING EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2014-06-12 WO disclosed
US-20140155563-A1 HIGH PERFORMANCE ACRYLAMIDE ADHESIVES EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2014-06-05 US disclosed
US-20140155563-A1 HIGH PERFORMANCE ACRYLAMIDE ADHESIVES EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2014-06-05 US disclosed
US-20140142090-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN SARL (CH) 2014-05-22 US disclosed
US-8729203-B2 Polymer composition CONTAMAC LIMITED (GB) 2014-05-20 US disclosed
US-20140135315-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2014-05-15 US disclosed
WO-2014067904-A1 NEW ANTIBACTERIAL COMPOUNDS AND BIOLOGICAL APPLICATIONS THEREOF LABORATOIRE BIODIM (FR) 2014-05-08 WO disclosed
WO-2014057122-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES ADC THERAPEUTICS SÀRL (CH) 2014-04-17 WO disclosed
WO-2014057072-A1 SYNTHESIS AND INTERMEDIATES OF PYRROLOBENZODIAZEPINE DERIVATIVES FOR CONJUGATION SPIROGEN SÀRL (CH) 2014-04-17 WO disclosed
WO-2014057115-A1 PYRROLOBENZODIAZEPINE-ANTI-HER2 ANTIBODY CONJUGATES ADC THERAPEUTICS SÀRL (CH) 2014-04-17 WO disclosed
WO-2014057118-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES ADC THERAPEUTICS SARL (CH) 2014-04-17 WO disclosed
US-8697688-B2 Pyrrolobenzodiazepines used to treat proliferative diseases SEATTLE GENETICS INC. (US) 2014-04-15 US disclosed
US-20140080769-A1 SUBSTRATE REDUCTION THERAPY THE CHANCELLOR, MASTERS AND SCHOLARS OF THE UNIVERSITY OF OXFORD (GB) 2014-03-20 US disclosed
US-20140066435-A1 PYRROLOBENZODIAZEPINES USED TO TREAT PROLIFERATIVE DISEASES SPIROGEN SARL (CH) 2014-03-06 US disclosed
US-8664372-B2 Process for producing 1,2-trans-glycoside compound GLYTECH, INC. (JP) 2014-03-04 US disclosed
WO-2014022679-A2 ANTI-ETBR ANTIBODIES AND IMMUNOCONJUGATES GENENTECH, INC. (US) 2014-02-06 WO disclosed
US-20140030279-A1 ANTI-CD22 ANTIBODIES AND IMMUNOCONJUGATES SPIROGEN SARL (CH) 2014-01-30 US disclosed
US-20140031539-A1 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY Biocodex, Inc (US) 2014-01-30 US disclosed
US-20140030280-A1 ANTI-CD79B ANTIBODIES AND IMMUNOCONJUGATES GENENTECH, INC. (US) 2014-01-30 US disclosed
US-8637664-B2 Alkyl 4- [4- (5-oxo-2,3,5, 11a-tetrahydo-5H-pyrrolo [2, 1-c] [1,4] benzodiazepine-8-yloxy)-butyrylamino]-1H-pyrrole-2-carboxylate derivatives and related compounds for the treatment of a proliferative disease SPIROGEN SARL (CH) 2014-01-28 US disclosed
US-8633185-B2 Pyrrolobenzodiazepines SPIROGEN SARL (CH) 2014-01-21 US disclosed
WO-2014011519-A1 IMMUNOCONJUGATES COMPRISING ANTI-CD79B ANTIBODIES GENENTECH, INC. (US) 2014-01-16 WO disclosed
WO-2014011518-A1 IMMUNOCONJUGATES COMPRISING ANTI-CD22 ANTIBODIES GENENTECH, INC. (US) 2014-01-16 WO disclosed
US-20130317237-A1 SYNTEHSIS OF CYCLIC CARBONATES UNIVERSITY OF NEW CASTLE UPON TYNE (GB) 2013-11-28 US disclosed
WO-2013177481-A1 BENZODIAZEPINES AND CONJUGATES THEREOF IMMUNOGEN, INC. (US) 2013-11-28 WO disclosed
US-8592576-B2 Unsymmetrical pyrrolobenzodiazepine-dimers for treatment of proliferative diseases SPIROGEN SARL (CH) 2013-11-26 US disclosed
EP-2662095-A1 Pyrrolobenzodiazepines and conjugates thereof Spirogen Sàrl (CH) 2013-11-13 EP disclosed
WO-2013164593-A1 PYRROLOBENZODIAZEPINES SPIROGEN SÀRL (CH) 2013-11-07 WO disclosed
WO-2013164592-A1 PYRROLOBENZODIAZEPINES UCL BUSINESS PLC (GB) 2013-11-07 WO disclosed
US-8575094-B2 Use of type-B lantibiotic-based compounds having antimicrobial activity NOVACTA BIOSYSTEMS LIMITED (GB) 2013-11-05 US disclosed
US-8557844-B2 Substrate reduction therapy THE CHANCELLOR, MASTERS AND SCHOLARS OF THE UNIVERSITY OF OXFORD (GB) 2013-10-15 US disclosed
US-20130266595-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2013-10-10 US disclosed
US-20130196381-A1 CELL-BASED PRODUCTION OF NANULOSONATES UNIVERSITY OF OTTAWA (CA) 2013-08-01 US disclosed
US-20130190529-A1 Fluorine Radiolabelling Process ISIS INNOVATION LIMITED (GB) 2013-07-25 US disclosed
US-8487092-B2 Pyrrolobenzodiazepines SPIROGEN DEVELOPMENTS SARL (CH) 2013-07-16 US disclosed
EP-2528625-B1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SARL (CH) 2013-07-10 EP disclosed
US-20130172210-A1 METHOD OF DRUG DESIGN ALCHEMIA LIMITED (AU) 2013-07-04 US disclosed
WO-2013095684-A1 GUANINE ANALOGS AS TELOMERASE SUBSTRATES AND TELOMERE LENGTH AFFECTORS GERON CORPORATION (US) 2013-06-27 WO disclosed
EP-2350098-B1 PYRROLOBENZODIAZEPINES SPIROGEN SARL (CH) 2013-05-15 EP disclosed
EP-2590910-A2 FLUORINE RADIOLABELLING PROCESS Isis Innovation Limited (GB) 2013-05-15 EP disclosed
CN-103087847-A Germicidal detergent composition, application thereof, preparation method thereof, and method thereof for cleaning object BEIJING CONFLE TECHNOLOGY CO LTD 2013-05-08 CN disclosed
CN-103087842-A Germicidal detergent composition, application thereof, preparation method thereof, kit thereof and method thereof for cleaning object BEIJING CONFLE TECHNOLOGY CO LTD 2013-05-08 CN disclosed
CN-103087841-A Liquid detergent composition, and use, preparation method, kit and method for washing article thereof BEIJING CONFLE TECHNOLOGY CO LTD 2013-05-08 CN disclosed
US-8435985-B2 Pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors MENEAR KEITH (GB) 2013-05-07 US disclosed
CN-103068405-A Targeted pyrrolobenzodiazepine conjugates SEATTLE GENETICS INC 2013-04-24 CN disclosed
US-8426345-B2 Method of drug design ALCHEMIA LIMITED (AU) 2013-04-23 US disclosed
WO-2013053871-A1 PYRROLOBENZODIAZEPINES SPIROGEN SÀRL (CH) 2013-04-18 WO disclosed
WO-2013055990-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEATTLE GENETICS, INC. (US) 2013-04-18 WO disclosed
WO-2013055993-A1 PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES SEATTLE GENETICS, INC. (US) 2013-04-18 WO disclosed
WO-2013055987-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN SÀRL (CH) 2013-04-18 WO disclosed
WO-2013053872-A1 SYNTHESIS METHOD AND INTERMEDIATES USEFUL IN THE PREPARATION OF PYRROLOBENZODIAZEPINES SPIROGEN SÀRL (CH) 2013-04-18 WO disclosed
WO-2013053873-A1 PYRROLOBENZODIAZEPINES SPIROGEN SÀRL (CH) 2013-04-18 WO disclosed
EP-1720881-B9 11-HYDROXY-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPIN-5-ONE DERIVATIVES AS KEY INTERMEDIATES FOR THE PREPARATION OF C2 SUBSTITUTED PYRROLOBENZODIAZEPINS SPIROGEN SARL (CH) 2013-04-17 EP disclosed
WO-2013041606-A1 PYRROLOBENZODIAZEPINES AS UNSYMMETRICAL DIMERIC PBD COMPOUNDS FOR INCLUSION IN TARGETED CONJUGATES SPIROGEN SÀRL (CH) 2013-03-28 WO disclosed
CN-102971329-A Pyrrolobenzodiazepines for the treatment of proliferative diseases SPIROGEN LTD 2013-03-13 CN disclosed
US-20130059800-A1 PYRROLOBENZODIAZEPINES USED TO TREAT PROLIFERATIVE DISEASES SEATTLE GENETICS INC. (US) 2013-03-07 US disclosed
WO-2013026454-A1 TREATMENT OF CLINICAL CONDITIONS WITH ANTHRACYCLINES VALDERM APS (DK) 2013-02-28 WO disclosed
WO-2013026453-A1 TREATMENT OF INFLAMMATORY DISORDERS WITH ANTHRACYCLINES VALDERM APS (DK) 2013-02-28 WO disclosed
EP-2558445-A1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES Spirogen Sàrl (CH) 2013-02-20 EP disclosed
EP-2558475-A1 PYRROLOBENZODIAZEPINES USED TO TREAT PROLIFERATIVE DISEASES Spirogen Sàrl (CH) 2013-02-20 EP disclosed
EP-2558127-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES Seattle Genetics, Inc. (US) 2013-02-20 EP disclosed
US-20130035484-A1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES SPIROGEN DEVELOPMENTS SÀRL (CH) 2013-02-07 US disclosed
US-20130035414-A1 HIGH REFRACTIVE INDEX POLYMER COMPOSITION FOR OPTHALMIC APPLICATIONS CONTAMAC LIMITED (GB) 2013-02-07 US disclosed
US-20130028917-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN DEVELOPMENTS SÀRL (CH) 2013-01-31 US disclosed
US-20130028919-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES SPIROGEN DEVELOPMENTS SÀRL (CH) 2013-01-31 US disclosed
EP-2542595-A1 HIGH REFRACTIVE INDEX POLYMER COMPOSITION FOR OPTHALMIC APPLICATIONS Contamac Limited (GB) 2013-01-09 EP disclosed
EP-1727808-B3 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LTD (GB) 2013-01-09 EP disclosed
EP-2536275-A1 METHODS OF REDUCING VIRULENCE IN BACTERIA UWM Research Foundation, Inc. (US) 2012-12-26 EP disclosed
US-20120322769-A1 METHODS OF REDUCING VIRULENCE IN BACTERIA DUKE UNIVERSITY (US) 2012-12-20 US disclosed
US-20120321963-A1 GEL POLYMER ELECTROLYTE COMPOSITION KURARAY CO., LTD. (JP) 2012-12-20 US disclosed
EP-1720881-B1 11-HYDROXY-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPIN-5-ONE DERIVATIVES AS KEY INTERMEDIATES FOR THE PREPARATION OF C2 SUBSTITUTED PYRROLOBENZODIAZEPINS SPIROGEN LTD (GB) 2012-12-12 EP disclosed
US-8329644-B2 Lantibiotic-based compounds having antimicrobial activity NOVACTA BIOSYSTEMS LIMITED (GB) 2012-12-11 US disclosed
EP-1934388-B1 METHOD OF DRUG DESIGN ALCHEMIA LTD (AU) 2012-12-05 EP disclosed
EP-2528625-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF Spirogen Developments SARL (CH) 2012-12-05 EP disclosed
CN-102796147-A Compounds library ALCHEMIA LTD 2012-11-28 CN disclosed
EP-2524932-A1 GEL POLYMER ELECTROLYTE COMPOSITION Kuraray Co., Ltd. (JP) 2012-11-21 EP disclosed
EP-2146977-B1 SYNTHESIS OF CYCLIC CARBONATES IN THE PRESENCE OF DIMERIC ALUMINIUM (SALEN) CATALYSTS UNIV NEWCASTLE (GB) 2012-11-14 EP disclosed
EP-1954699-B1 PYRIDO-, PYRAZO- AND PYRIMIDOPYRIMIDINE DERIVATIVES AS mTOR INHIBITORS KUDOS PHARM LTD (GB) 2012-09-19 EP disclosed
CN-101278079-B Drug design method ALCHEMIA LTD 2012-09-19 CN disclosed
US-20120232256-A1 PROCESS FOR PRODUCING 1,2-TRANS-GLYCOSIDE COMPOUND OTSUKA CHEMICAL CO., LTD. 2012-09-13 US disclosed
US-8222381-B2 Derivatives of monosaccharides for drug discovery ALCHEMIA LIMITED (AU) 2012-07-17 US disclosed
US-8212013-B2 Phenyl 3,4,6-tri-O-benzyl-2-O-(1,1,2,2-tetramethyl-dimethylene phosphonoyl)- beta -D-thioglucopyranoside; inhibits formation of o-ester by-product resulting from the conventional glycosilation reaction of pyranose compounds of 1,2-trans form, affording 1,2-transglycoside compounds with high selectivity OTSUKA CHEMICAL CO., LTD. (JP) 2012-07-03 US disclosed
US-20120142673-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2012-06-07 US disclosed
US-20120129855-A1 PHTHALAZINONE DERIVATIVES MENEAR KEITH ALLAN (GB) 2012-05-24 US disclosed
US-8183202-B2 2012-05-22 US disclosed
EP-2013207-B1 IMIDAZO[4,5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS CANCER THERAPEUTIC COMPOUNDS CANCER REC TECH LTD (GB) 2012-04-25 EP disclosed
EP-2427509-A1 POLYMER COMPOSITION Contamac Limited (GB) 2012-03-14 EP disclosed
US-8129380-B2 Phthalazinone derivatives ASTRAZENECA AB (SE) 2012-03-06 US disclosed
US-20120053313-A1 POLYMER COMPOSITION CONTAMAC LIMITED (GB) 2012-03-01 US disclosed
EP-2422183-A2 OXIDATION STATE SENSORS AND METHODS FOR TRANSITION METAL ALLOYS Rolls-Royce PLC (GB) 2012-02-29 EP disclosed
US-20120040467-A1 OXIDATION STATE SENSORS AND METHODS FOR TRANSITION METAL ALLOYS ROLLS-ROYCE PLC 2012-02-16 US disclosed
CN-102356086-A Aluminum complexes and their use in the synthesis of cyclic carbonates UNIV NEWCASTLE 2012-02-15 CN disclosed
EP-1330456-B8 N8,N13 -DISUBSTITUTED QUINO[4,3,2-KL]ACRIDINIUM SALTS AS THERAPEUTIC AGENTS CANCER REC TECH LTD (GB) 2012-02-08 EP disclosed
EP-2270010-B1 11-hydroxy-5h-pyrrolo[2,1-c][1,4]benzodiazepin-5-one derivatives as key intermediates for the preparation of c2 substituted pyrrolobenzodiazepins SPIROGEN LTD (GB) 2012-01-25 EP disclosed
EP-2408784-A1 ALUMINUM COMPLEXES AND THEIR USE IN THE SYNTHESIS OF CYCLIC CARBONATES University Of Newcastle-Upon Tyne (GB) 2012-01-25 EP disclosed
EP-1330456-B9 N8,N13 -DISUBSTITUTED QUINO[4,3,2-KL]ACRIDINIUM SALTS AS THERAPEUTIC AGENTS CANCER REC TECH LTD (GB) 2012-01-25 EP disclosed
US-8101602-B2 Pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as mTOR inhibitors Kudos Pharmaceuticals, Ltd. (GB) 2012-01-24 US disclosed
WO-2012004567-A2 FLUORINE RADIOLABELLING PROCESS ISIS INNOVATION LIMITED (GB) 2012-01-12 WO disclosed
US-20120010204-A1 Phthalazinone Derivatives MAYBRIDGE LIMITED 2012-01-12 US disclosed
US-8093405-B2 Formation of 18F and 19F fluoroarenes bearing reactive functionalities UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2012-01-10 US disclosed
US-20110319634-A1 ALUMINUM COMPLEXES AND THEIR USE IN THE SYNTHESIS OF CYCLIC CARBONATES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2011-12-29 US disclosed
US-8071620-B2 Carbamic acid compounds comprising a bicyclic heteroaryl group as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2011-12-06 US disclosed
US-20110275576-A1 Carbohydrate-Cyclopamine Conjugates as Anticancer Agents UTAH STATE UNIVERSITY (US) 2011-11-10 US disclosed
US-20110275810-A1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2011-11-10 US disclosed
WO-2011128650-A1 INTERMEDIATES USEFUL FOR THE SYNTHESIS OF PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2011-10-20 WO disclosed
WO-2011130613-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES SEATTLE GENETICS, INC. (US) 2011-10-20 WO disclosed
WO-2011130616-A1 PYRROLOBENZODIAZEPINES USED TO TREAT PROLIFERATIVE DISEASES SPIROGEN LIMITED (GB) 2011-10-20 WO disclosed
WO-2011130598-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN LIMITED (GB) 2011-10-20 WO disclosed
US-20110256157-A1 PYRROLOBENZODIAZEPINES AND CONJUGATES THEREOF SPIROGEN LIMITED (GB) 2011-10-20 US disclosed
WO-2011107728-A1 HIGH REFRACTIVE INDEX POLYMER COMPOSITION FOR OPTHALMIC APPLICATIONS CONTAMAC LIMITED (GB) 2011-09-09 WO disclosed
WO-2011103189-A1 METHODS OF REDUCING VIRULENCE IN BACTERIA UWM RESEARCH FOUNDATION, INC. (US) 2011-08-25 WO disclosed
US-20110201803-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2011-08-18 US disclosed
US-20110196148-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN LIMITED (GB) 2011-08-11 US disclosed
EP-2350098-A1 PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2011-08-03 EP disclosed
EP-2350080-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES Spirogen Limited (GB) 2011-08-03 EP disclosed
EP-1974011-B1 CHEMICAL INDUCTION OF QUIESCENCE IN BACTERIA CAMBRIDGE MICROBIAL TECHNOLOGIES LTD (GB) 2011-07-20 EP disclosed
US-7981895-B2 Histone deacetylase inhibitor; anticancer agents; antiproliferative agents; antitumor agents; psoriasis; piperazine compound containing a carbamic acid group TOPOTARGET UK LIMITED (GB) 2011-07-19 US disclosed
US-7981889-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2011-07-19 US disclosed
US-7981890-B2 Phthalazinone derivatives ASTRAZENECA AB (SE) 2011-07-19 US disclosed
EP-2343401-A1 Hydrophobic surface Rolls-Royce plc (GB) 2011-07-13 EP disclosed
EP-2343400-A1 Hydrophobic Surface Rolls-Royce plc (GB) 2011-07-13 EP disclosed
US-20110160192-A1 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LIMITED (GB) 2011-06-30 US disclosed
US-20110150984-A1 METHODS OF INCREASING THE BIOAVAILABILITY AND/OR CELLULAR UPDATE OF DRUGS HET NEDERLANDS KANKER INSTITUUT (NL) 2011-06-23 US disclosed
US-20110147219-A1 HYDROPHOBIC SURFACE ROLLS-ROYCE PLC (GB) 2011-06-23 US disclosed
US-20110151186-A1 HYDROPHOBIC SURFACE ROLLS-ROYCE PLC (GB) 2011-06-23 US disclosed
US-7964643-B2 Biphenyl-4-sulfonic acid-(4-hydroxybutyl)-amide and derivatives; inhibits osteoclast survival, formation, and/or activity and/or inhibits bone resorption; osteoporosis, rheumatoid arthritis, cancer associated bone disease, Paget's disease, antiinflammatory, -carcinogenic agents; immunostimulants THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2011-06-21 US disclosed
EP-1330456-B1 N8,N13 -DISUBSTITUTED QUINO[4,3,2-KL]ACRIDINIUM SALTS AS THERAPEUTIC AGENTS CANCER REC TECH LTD (GB) 2011-06-15 EP disclosed
US-7951819-B2 Imidazo[4, 5-B]pyridin-2-one and oxazolo[4, 5-B] pyridin-2-one compounds and analogs thereof as cancer therapeutic compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-05-31 US disclosed
US-20110124638-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2011-05-26 US disclosed
US-20110105572-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN AMIDE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2011-05-05 US disclosed
EP-1633724-B1 PHTHALAZINONE DERIVATIVES KUDOS PHARM LTD (GB) 2011-05-04 EP disclosed
US-7935836-B2 Compounds comprising a linear series of five fused carbon rings, and preparation thereof FALLIS ALEXANDER GRAHAM 2011-05-03 US disclosed
EP-2310362-A1 FORMATION OF 18F AND 19F FLUOROARENES BEARING REACTIVE FUNCTIONALITIES University Of Newcastle-Upon Tyne (GB) 2011-04-20 EP disclosed
CN-102015639-A Compounds for use in stabilizing p53 mutants MEDICAL RES COUNCIL 2011-04-13 CN disclosed
CN-102015732-A Synthesis of cyclic carbonates UNIV NEWCASTLE 2011-04-13 CN disclosed
US-7915227-B2 Pharmaceutical formulations employing short-chain sphingolipids and their use HET NEDERLANDS KANKER INSTITUUT (NL) 2011-03-29 US disclosed
EP-1432669-B1 4-(C2-6 ALKOXY)-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS SPEAR THERAPEUTICS LTD (GB) 2011-03-23 EP disclosed
US-20110059953-A1 COMPOUNDS FOR USE IN STABILIZING P53 MUTANTS MEDICAL RESEARCH COUNCIL (GB) 2011-03-10 US disclosed
EP-2292593-A2 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TopoTarget UK Limited (GB) 2011-03-09 EP disclosed
US-7902193-B2 Phthalazinone derivatives MAYBRIDGE LIMITED (GB) 2011-03-08 US disclosed
US-7902189-B2 antitumor agent, anticarcinogenic agents; 7-Chloro-2-((2S,6R)-2,6-dimethyl-morpholin-4-yl)-4-morpholin-4-yl-pyrido[2,3-d]pyrimidine; inhibitors of mTOR kinase ASTRAZENECA AB (SE) 2011-03-08 US disclosed
EP-1723151-B1 PYRROLOBENZODIAZEPINES AS KEY INTERMEDIATES IN THE SYNTHESIS OF DIMERIC CYTOTOXIC PYRROLOBENZODIAZEPINES SPIROGEN LTD (GB) 2011-02-16 EP disclosed
EP-1575955-B1 PYRROLOBENZODIAZEPINES FOR THE TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN LTD (GB) 2011-02-09 EP disclosed
EP-1831184-B1 PYRAZINES AND PYRIDINES AND DERIVATIVES THEREOF AS THERAPEUTIC COMPOUNDS WELLCOME TRUST LTD (GB) 2011-02-09 EP disclosed
US-7880020-B2 e.g trichlorostatin A; antiproliferative agent; for treating cancer and psoriasis TOPOTARGET UK LIMITED (GB) 2011-02-01 US disclosed
US-20110015409-A1 SYNTHESIS OF CYCLIC CARBONATES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2011-01-20 US disclosed
EP-2274282-A1 COMPOUNDS FOR USE IN STABILIZING P53 MUTANTS Medical Research Council (GB) 2011-01-19 EP disclosed
EP-2270010-A1 11-HYDROXY-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPIN-5-ONE DERIVATIVES AS KEY INTERMEDIATES FOR THE PREPARATION OF C2 SUBSTITUTED PYRROLOBENZODIAZEPINS Spirogen Limited (GB) 2011-01-05 EP disclosed
EP-2257559-A1 SYNTHESIS OF CYCLIC CARBONATES University Of Newcastle-Upon Tyne (GB) 2010-12-08 EP disclosed
WO-2010133851-A1 PREPARATION OF LABELLED COMPOUNDS ISIS INNOVATION LIMITED (GB) 2010-11-25 WO disclosed
CN-101896180-A Combination 059 ASTRAZENECA AB 2010-11-24 CN disclosed
WO-2010128266-A1 POLYMER COMPOSITION CONTAMAC LIMITED (GB) 2010-11-11 WO disclosed
WO-2010122287-A2 OXIDATION STATE SENSORS AND METHODS FOR TRANSITION METAL ALLOYS ROLLS-ROYCE PLC (GB) 2010-10-28 WO disclosed
US-20100261638-A1 LANTIBIOTIC-BASED COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY NOVACTA BIOSYSTEMS LIMITED (GB) 2010-10-14 US disclosed
CN-101084217-B Imidazo [4,5-B] pyridin-2-ones and oxazolido [4,5-B] pyridin-2-ones and analogues thereof as therapeutic compounds CANCER REC TECH LTD 2010-10-13 CN disclosed
US-20100249112-A1 COMBINATION OF CHK AND PARP INHIBITORS FOR THE TREATMENT OF CANCERS ASTRAZENECA R&D (SE) 2010-09-30 US disclosed
US-20100249197-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN AMIDE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2010-09-30 US disclosed
US-20100249234-A1 METHODS OF REDUCING VIRULENCE IN BACTERIA UWM RESEARCH FOUNDATION, INC. (US) 2010-09-30 US disclosed
EP-2231638-A1 PHTHALAZINONE DERIVATIVES AstraZeneca AB (SE) 2010-09-29 EP disclosed
WO-2010106324-A1 ALUMINUM COMPLEXES AND THEIR USE IN THE SYNTHESIS OF CYCLIC CARBONATES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2010-09-23 WO disclosed
US-7790435-B2 Chemical induction in quiescence in bacteria CAMBRIDGE MICROBIAL TECHNOLOGIES LIMITED (GB) 2010-09-07 US disclosed
US-7781411-B2 Derivatives of avermectin, avermectin monosaccharide and avermectin aglycone SYNGENTA CROP PROTECTION, INC. (US) 2010-08-24 US disclosed
EP-2217234-A2 COMBINATIONS OF MEK INHIBITORS WITH MTOR INHIBITORS AstraZeneca AB (SE) 2010-08-18 EP disclosed
US-20100204162-A1 SUBSTRATE REDUCTION THERAPY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 2010-08-12 US disclosed
US-20100203650-A1 BIOMOLECULE BINDING LIGANDS CAMBRIDGE ENTERPRISE LIMITED (GB) 2010-08-12 US disclosed
CN-101796067-A Lantibiotic-based compounds with antimicrobial activity NOVACTA BIOSYSTEMS LTD 2010-08-04 CN disclosed
CN-101796066-A Biomolecule binding ligands CAMBRIDGE ENTPR LTD 2010-08-04 CN disclosed
WO-2010080817-A2 CARBOHYDRATE-CYCLOPAMINE CONJUGATES AS ANTICANCER AGENTS UTAH STATE UNIVERSITY (US) 2010-07-15 WO disclosed
US-7745424-B2 Alkane diol derivatives as therapeutic agents for the treatment of bone conditions The Univeristy Court of the University of Aberdeen (GB) 2010-06-29 US disclosed
CN-101754769-A Use of type B lantibiotics based on antimicrobial activity NOVACTA BIOSYSTEMS LTD 2010-06-23 CN disclosed
US-7741319-B2 11-hydroxy-5h-pyrrolo[2,1-c][1,4] benzodiazepin-5-one derivatives as key intermediates for the preparation of c2 substituted pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2010-06-22 US disclosed
US-7737152-B2 6-carboaryl-oxy-pyrazin-2-yl-carboaryl-amines and compositions comprising said compounds THE WELLCOME TRUST LIMITED (GB) 2010-06-15 US disclosed
US-20100144651-A1 NOVEL GLUCOPYRANOSE ESTERS AND GLUCOFURANOSE ESTERS OF ALKYL- FUMARATES AND THEIR PHARMACEUTICAL USE ADITECH PHARMA AB (SE) 2010-06-10 US disclosed
US-20100130473-A1 COMPOUNDS HUMMERSONE MARC GEOFFREY 2010-05-27 US disclosed
US-20100130752-A1 SYNTHESIS OF CYCLIC CARBONATES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2010-05-27 US disclosed
EP-2188278-A1 PHTHALAZINONE DERIVATIVES AstraZeneca AB (SE) 2010-05-26 EP disclosed
EP-2186819-A1 Novel glucopyranose esters and glucofuranose esters of alkyl- fumarates and their pharmaceutical use Aditech Pharma AG (CH) 2010-05-19 EP disclosed
EP-2182936-A2 SUBSTRATE REDUCTION THERAPY THE CHANCELLOR, MASTERS AND SCHOLARS OF THE UNIVERSITY OF OXFORD (GB) 2010-05-12 EP disclosed
US-20100113425-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2010-05-06 US disclosed
EP-2178552-A1 THE USE OF TYPE-B LANTIBIOTIC-BASED COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY Novacta Biosystems Limited (GB) 2010-04-28 EP disclosed
WO-2010043880-A1 UNSYMMETRICAL PYRROLOBENZODIAZEPINE-DIMERS FOR TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN LIMITED (GB) 2010-04-22 WO disclosed
WO-2010043877-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2010-04-22 WO disclosed
EP-2176237-A1 PHTHALAZINONE DERIVATIVES AS INHIBITORS OF PARP-1 AstraZeneca AB (SE) 2010-04-21 EP disclosed
US-20100093743-A1 CARBAMIC ACID COMPOUNDS COMPRISING A BICYCLIC HETEROARYL GROUP AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2010-04-15 US disclosed
EP-2170927-A2 BIOMOLECULE BINDING LIGANDS Cambridge Enterprise Limited (GB) 2010-04-07 EP disclosed
EP-2167086-A1 COMBINATION OF CHK AND PARP INHIBITORS FOR THE TREATMENT OF CANCERS AstraZeneca AB (SE) 2010-03-31 EP disclosed
EP-2167527-A2 LANTIBIOTIC-BASED COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY Novacta Biosystems Limited (GB) 2010-03-31 EP disclosed
WO-2010024783-A1 BIARYLRHODANINE AND PYRIDYLRHODANINE COMPOUNDS AND THEIR USE AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2010-03-04 WO disclosed
EP-2155726-A1 PHTHALAZINONE DERIVATIVES AND THEIR USE AS MEDICAMENT TO TREAT CANCER Kudos Pharmaceuticals Limited (GB) 2010-02-24 EP disclosed
US-7666870-B2 Phthalazinone derivatives MAYBRIDGE LIMITED (GB) 2010-02-23 US disclosed
US-7662818-B2 e.g. 4-[5-(piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; and multiple sclerosis KUDOS PHARMACEUTICALS LIMITED (GB) 2010-02-16 US disclosed
EP-1404659-B1 4-ARYL QUINOLS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS CANCER REC TECH LTD (GB) 2010-02-10 EP disclosed
US-20100028262-A1 3,4-METHYLENEDIOXY-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS SPEAR THERAPEUTICS LIMITED (GB) 2010-02-04 US disclosed
US-7655809-B2 Compounds comprising a linear series of five fused carbon rings, and preparation thereof UNIVERSITY OF OTTAWA (CA) 2010-02-02 US disclosed
US-20100022620-A1 EPITOPE REDUCTION THERAPY ISIS INNOVATION LIMITED (GB) 2010-01-28 US disclosed
EP-2146977-A1 SYNTHESIS OF CYCLIC CARBONATES IN THE PRESENCE OF DIMERIC ALUMINIUM (SALEN) CATALYSTS University Of Newcastle-Upon Tyne (GB) 2010-01-27 EP disclosed
US-7652036-B2 Carbamic acid compounds comprising a bicyclic heteroaryl group as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2010-01-26 US disclosed
WO-2010007363-A2 PREPARATION OF FLUORINE-LABELLED COMPOUNDS ISIS INNOVATION LIMITED (GB) 2010-01-21 WO disclosed
EP-1915387-B1 NOVEL GLUCOPYRANOSE ESTERS AND GLUCOFURANOSE ESTERS OF ALKYL- FUMARATES AND THEIR PHARMACEUTICAL USE ADITECH PHARMA AG (CH) 2010-01-20 EP disclosed
US-20100004467-A1 COMPOUNDS COMPRISING A LINEAR SERIES OF FIVE FUSED CARBON RINGS, AND PREPARATION THEREOF FALLIS ALEXANDER GRAHAM 2010-01-07 US disclosed
US-20090325945-A1 IMIDAZO[4, 5-B]PYRIDIN-2-ONE AND OXAZOLO[4, 5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS CANCER THERAPEUTIC COMPOUNDS THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2009-12-31 US disclosed
EP-1664049-B1 SYNTHESIS OF PROTECTED PYRROLOBENZODIAZEPINES SPIROGEN LTD (GB) 2009-12-23 EP disclosed
WO-2009153566-A1 CYP26 INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-12-23 WO disclosed
EP-1879901-B1 PYRROLOBENZODIAZEPINES SPIROGEN LTD (GB) 2009-12-23 EP disclosed
EP-1737812-B1 METHODS OF AMINATION ASTRAZENECA UK LTD (GB) 2009-12-16 EP disclosed
EP-1756046-B1 ARYL ALKYL SULFONAMIDES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS UNIV ABERDEEN (GB) 2009-12-09 EP disclosed
US-7629343-B2 Carbamic acid compounds comprising a piperazine linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2009-12-08 US disclosed
US-7625922-B2 Imidazo[4,5-b]pyridin-2-one and oxazolo[4,5-b]pyridin-2-one compounds and analogs thereof as therapeutic compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-12-01 US disclosed
WO-2009141627-A1 TREATING NIEMANN-PICK DISEASE TYPE C AND RELATED DISORDERS BY ELEVATING INTRACELLULAR CALCIUM ISIS INNOVATION LIMITED (GB) 2009-11-26 WO disclosed
WO-2009138708-A1 BICYCLIC MONOPHOSPHINES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2009-11-19 WO disclosed
WO-2009138763-A1 FORMATION OF 18F AND 19F FLUOROARENES BEARING REACTIVE FUNCTIONALITIES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2009-11-19 WO disclosed
US-20090286992-A1 FORMATION OF 18F AND 19F FLUOROARENES BEARING REACTIVE FUNCTIONALITIES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2009-11-19 US disclosed
US-20090281086-A1 2 -OXYHETEROARYLAMIDE DERIVATIVES AS PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2009-11-12 US disclosed
WO-2009136175-A1 COMPOUNDS FOR USE IN STABILIZING P53 MUTANTS MEDICAL RESEARCH COUNCIL (GB) 2009-11-12 WO disclosed
US-7612062-B2 Pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2009-11-03 US disclosed
US-7598294-B2 Antiproliferative agents; antiinflammatory agents; anticancer agents; diagnosis, therapy SPEAR THERAPEUTICS LIMITED (GB) 2009-10-06 US disclosed
US-7598289-B2 Ketones and reduced ketones as therapeutic agents for the treatment of bone conditions THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2009-10-06 US disclosed
WO-2009109765-A1 SYNTHESIS OF CYCLIC CARBONATES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2009-09-11 WO disclosed
US-20090209520-A1 2 -OXYBENZAMIDE DERIVATIVES AS PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2009-08-20 US disclosed
US-20090209535-A1 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY TOPOTARGET A/S (DK) 2009-08-20 US disclosed
US-20090203583-A1 Use of Type-B Lantibiotic-Based Compounds having Antimicrobial Activity NOVACTA BIOSYSTEMS LIMITED (GB) 2009-08-13 US disclosed
US-7572825-B2 Ketones and reduced ketones as therapeutic agents for the treatment of bone conditions THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2009-08-11 US disclosed
US-7569724-B2 Carbamic acid compounds comprising an amide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2009-08-04 US disclosed
US-20090192156-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2009-07-30 US disclosed
WO-2009093032-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA AB (SE) 2009-07-30 WO disclosed
EP-2083005-A1 Carbamic acid compounds comprising an amide linkage as HDAC inhibitors TopoTarget UK Limited (GB) 2009-07-29 EP disclosed
EP-1572197-B1 4- 1- (SULFONYL) -1H-INDOL-2-YL)-4- (HYDROXY) -CYCLOHEXA-2,5-DIENONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS CANCER REC TECH LTD (GB) 2009-07-29 EP disclosed
US-20090186897-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2009-07-23 US disclosed
US-20090181951-A1 PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2009-07-16 US disclosed
US-7557140-B2 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2009-07-07 US disclosed
US-7557099-B2 Pyrrolobenzodiazepines as key intermediates in the synthesis of dimeric cytotoxic pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2009-07-07 US disclosed
US-20090163477-A1 PHTHALAZINONE DERIVATIVES MAYBRIDGE LIMITED (GB) 2009-06-25 US disclosed
US-20090163373-A1 Method of Drug Design ALCHEMIA LIMITED (AU) 2009-06-25 US disclosed
EP-1686959-B1 PHARMACEUTICAL FORMULATIONS EMPLOYING SHORT-CHAIN SPHINGOLIPIDS AND THEIR USE HET NL KANKER I THE NETHERLAND (NL) 2009-06-24 EP disclosed
WO-2009060208-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2009-05-14 WO disclosed
WO-2009060215-A1 POLYAMIDES SPIROGEN LIMITED (GB) 2009-05-14 WO disclosed
EP-2057156-A1 2-METHYLMORPHOLINE PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS Kudos Pharmaceuticals Limited (GB) 2009-05-13 EP disclosed
EP-1598067-B1 Carbamic acid compounds comprising an amide linkage for the treatment of malaria TOPOTARGET UK LTD (GB) 2009-05-06 EP disclosed
US-7528126-B2 Pyrrolobenzodiazepines SPIROGEN LIMITED 2009-05-05 US disclosed
EP-2051708-A2 EPITOPE REDUCTION THERAPY ISIS Innovation Limited (GB) 2009-04-29 EP disclosed
WO-2009050506-A2 COMBINATION 059 ASTRAZENECA AB (SE) 2009-04-23 WO disclosed
US-20090099174-A1 COMBINATION 059 ASTRAZENECA AB (SE) 2009-04-16 US disclosed
WO-2009044130-A1 BIARYL DIPHOSPHINES UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2009-04-09 WO disclosed
EP-1931671-B1 ALKYL 4- [4- (5-OXO-2, 3, 5, 11A-TETRAHYD0-5H-PYRR0L0 [2, 1-C][1, 4]BENZODIAZEPINE-8-YLOXY) -BUTYRYLAMINO]-1H-PYRROLE-2-CARBOXYLATE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF A PROLIFERATIVE DISEASE SPIROGEN LTD (GB) 2009-04-08 EP disclosed
EP-2041087-A1 2 -OXYBENZAMIDE DERIVATIVES AS PARP INHIBITORS Kudos Pharmaceuticals Limited (GB) 2009-04-01 EP disclosed
EP-2041110-A1 2 -OXYHETEROARYLAMIDE DERIVATIVES AS PARP INHIBITORS Kudos Pharmaceuticals Limited (GB) 2009-04-01 EP disclosed
WO-2009034326-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA AB (SE) 2009-03-19 WO disclosed
EP-2035380-A2 PARP INHIBITORS Kudos Pharmaceuticals Limited (GB) 2009-03-18 EP disclosed
US-7504397-B2 mTOR inhibitor compounds KUDOS PHARMACEUTICALS LTD. (GB) 2009-03-17 US disclosed
US-20090069303-A1 PHTHALAZINONE DERIVATIVES MAYBRIDGE LIMITED (GB) 2009-03-12 US disclosed
US-20090023727-A1 PHTHALAZINONE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 2009-01-22 US disclosed
WO-2009010763-A1 THE USE OF TYPE-B LANTIBIOTIC-BASED COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY NOVACTA BIOSYSTEMS LIMITED (GB) 2009-01-22 WO disclosed
WO-2009010765-A2 LANTIBIOTIC-BASED COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY NOVACTA BIOSYSTEMS LIMITED (GB) 2009-01-22 WO disclosed
WO-2009007676-A2 BIOMOLECULE BINDING LIGANDS CAMBRIDGE ENTERPRISE LIMITED (GB) 2009-01-15 WO disclosed
EP-2013207-A1 IMIDAZO[4, 5-B]PYRIDIN-2-ONE AND OXAZOLO[4, 5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS CANCER THERAPEUTIC COMPOUNDS Cancer Research Technology Limited (GB) 2009-01-14 EP disclosed
WO-2009004356-A1 PHTHALAZINONE DERIVATIVES AS INHIBITORS OF PARP-1 ASTRAZENECA AB (SE) 2009-01-08 WO disclosed
US-20090004700-A1 Chemical Induction in Quiescence in Bacteria CAMBRIDGE MICROBIAL TECHNOLOGIES LIMITED (GB) 2009-01-01 US disclosed
WO-2009001097-A2 SUBSTRATE REDUCTION THERAPY ISIS INNOVATION LIMITED (GB) 2008-12-31 WO disclosed
US-7470688-B2 Phthalazinone derivatives MAYBRIDGE LIMITED (GB) 2008-12-30 US disclosed
US-20080319001-A1 Cancer Treatment Using Specific 3,6,9-Substituted Acridines CANCER RESEARCH TECHNOLOGY LTD (GB) 2008-12-25 US disclosed
US-20080312186-A1 KETONES AND REDUCED KETONES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2008-12-18 US disclosed
US-7465719-B2 Carbamic acid compounds comprising an ester or ketone linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2008-12-16 US disclosed
US-20080300134-A1 Derivatives of Avermectin, Avermectin Monosaccharide and Avermectin Aglycone SYNGENTA CROP PROTECTION, INC. (US) 2008-12-04 US disclosed
WO-2008146035-A1 COMBINATION OF CHK AND PARP INHIBITORS FOR THE TREATMENT OF CANCERS ASTRAZENECA AB (SE) 2008-12-04 WO disclosed
US-20080280910-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2008-11-13 US disclosed
EP-1727808-B1 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LTD (GB) 2008-11-12 EP disclosed
US-7449464-B2 4-{3-[4-(6-Chlorobenzothiazol-2-yl)-1,4-diazepan-1-ylcarbonyl]benzyl}-1(2H)-phthalazinone; Cancer, BRCA deficient KUDOS PHARMACEUTICALS LIMITED (GB) 2008-11-11 US disclosed
WO-2008132474-A1 SYNTHESIS OF CYCLIC CARBONATES IN THE PRESENCE OF DIMERIC ALUMINIUM (SALEN) CATALYSTS UNIVERSITY OF NEWCASTLE UPON TYNE (GB) 2008-11-06 WO disclosed
US-20080267903-A1 Cationic polyamines and dendrimeric polymers; anti-proliferative agents; for treatment of neoplasms and tumours, inflammatory disorders, autoimmune disorders, psoriasis, and atherosclerosis; gene therapy UNIVERSITY COLLEGE LONDON (GB) 2008-10-30 US disclosed
US-20080269237-A1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2008-10-30 US disclosed
US-20080255128-A1 e.g. 4-[5-(Piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; multiple sclerosis KUDOS PHARMACEUTICALS LIMITED (GB) 2008-10-16 US disclosed
WO-2008122810-A1 PHTHALAZINONE DERIVATIVES AND THEIR USE AS MEDICAMENT TO TREAT CANCER KUDOS PHARMACEUTICALS LIMITED (GB) 2008-10-16 WO disclosed
WO-2008124836-A2 METHODS OF REDUCING VIRULENCE IN BACTERIA UWM RESEARCH FOUNDATION, INC. (US) 2008-10-16 WO disclosed
EP-1974011-A1 CHEMICAL INDUCTION OF QUIESCENCE IN BACTERIA Cambridge Microbial Technologies LTD (GB) 2008-10-01 EP disclosed
CN-101278079-A Drug design method ALCHEMIA LTD (AU) 2008-10-01 CN disclosed
US-7429658-B2 Synthesis of protected pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2008-09-30 US disclosed
WO-2008114023-A2 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2008-09-25 WO disclosed
US-20080214525-A1 Alkyl 4- [4- (5-Oxo-2,3,5, 11A-Tetrahydo-5H-Pyrrolo [2, 1-C] [1,4] Benzodiazepine-8-Yloxy) -Butyrylamino]-1H-Pyrrole-2-Carboxylate Derivatives and Related Compounds For the Treatment of a Proliferative Disease SPIROGEN LIMITED (GB) 2008-09-04 US disclosed
US-20080200469-A1 e.g. 4-[5-(Piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; multiple sclerosis KUDOS PHARMACEUTICALS LIMITED 2008-08-21 US disclosed
US-20080194546-A1 Pyrido-, Pyrazo- and Pyrimido-Pyrimidine Derivatives as mTOR Inhibitors KUDOS PHARMACEUTICALS LIMITED (GB) 2008-08-14 US disclosed
EP-1954699-A1 PYRIDO-,PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS Kudos Pharmaceuticals Ltd (GB) 2008-08-13 EP disclosed
US-7407988-B2 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2008-08-05 US disclosed
US-7407951-B2 Pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2008-08-05 US disclosed
US-7407957-B2 e.g. 4-[5-(piperazine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent; septic shock; ischemic injury; reperfusion injury; hemorrhagic shock; and multiple sclerosis MAYBRIDGE LIMITED (GB) 2008-08-05 US disclosed
EP-1948642-A1 4-HETEROARYMETHYL SUBSTITUTED PHTHALAZINONE DERIVATIVES Kudos Pharmaceuticals Ltd (GB) 2008-07-30 EP disclosed
US-20080177049-A1 Process for Producing 1,2-Trans-Glycoside Compound GLYTECH, INC. (JP) 2008-07-24 US disclosed
US-20080167293-A1 Pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2008-07-10 US disclosed
US-20080161401-A1 CARBAMIC ACID COMPOUNDS COMPRISING A SULFONAMIDE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2008-07-03 US disclosed
EP-1934388-A1 METHOD OF DRUG DESIGN Alchemia Ltd (AU) 2008-06-25 EP disclosed
EP-1492534-B1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LTD (GB) 2008-06-25 EP disclosed
EP-1931671-A1 ALKYL 4- [4- (5-OXO-2, 3, 5, 11A-TETRAHYD0-5H-PYRR0L0 [2, 1-C][1, 4]BENZODIAZEPINE-8-YLOXY) -BUTYRYLAMINO]-1H-PYRROLE-2-CARBOXYLATE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF A PROLIFERATIVE DISEASE Spirogen Limited (GB) 2008-06-18 EP disclosed
US-20080119555-A1 Aryl Alkyl Sulfonamides As Therapeutic Agents For The Treatment Of Bone Conditions THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2008-05-22 US disclosed
EP-1915387-A1 NOVEL GLUCOPYRANOSE ESTERS AND GLUCOFURANOSE ESTERS OF ALKYL- FUMARATES AND THEIR PHARMACEUTICAL USE Aditech Pharma AB (SE) 2008-04-30 EP disclosed
US-20080090812-A1 Pyrrolobenzodiazepine Therapeutic Agents Useful in the Treatment of Leukemias SPIROGEN LIMITED (GB) 2008-04-17 US disclosed
US-7358398-B2 of aromatic groups using transition metal catalysis in compressed carbon dioxide; intermediates ASTRAZENECA UK LIMITED (GB) 2008-04-15 US disclosed
US-20080081809-A1 Novel Compounds KUDOS PHARMACEUTICALS LIMITED (GB) 2008-04-03 US disclosed
WO-2008023161-A1 2-METHYLMORPHOLINE PYRIDO-, PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2008-02-28 WO disclosed
WO-2008012555-A2 EPITOPE REDUCTION THERAPY ISIS INNOVATION LIMITED (GB) 2008-01-31 WO disclosed
EP-1879901-A1 PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2008-01-23 EP disclosed
US-20080015191-A1 Pyrazines and Pyridines and Derivatives Thereof as Therapeutic Compounds THE WELLCOME TRUST LIMITED (UK) 2008-01-17 US disclosed
EP-1877388-A2 HYDRAZINOMETHYL, HYDRAZONOMETHYL AND 5-MEMBERED HETEROCYLIC COMPOUNDS WHICH ACT AS MTOR INHIBITORS AND THEIR USE AS ANTI CANCER AGENTS Kudos Pharmaceuticals Ltd (GB) 2008-01-16 EP disclosed
US-20080009418-A1 Selective Inhibitors ALCHEMIA LTD. (AU) 2008-01-10 US disclosed
EP-1871377-A1 2,4-DIAMINO-PYRIDOPYRIMIDINE DERIVATIVES AND THEIR USE AS MTOR INHIBITORS Kudos Pharmaceuticals Ltd (GB) 2008-01-02 EP disclosed
WO-2007144637-A1 2 -OXYHETEROARYLAMIDE DERIVATIVES AS PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2007-12-21 WO disclosed
WO-2007144652-A2 PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2007-12-21 WO disclosed
WO-2007144639-A1 2 -OXYBENZAMIDE DERIVATIVES AS PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2007-12-21 WO disclosed
US-20070287838-A1 Imidazo[4,5-B]Pyridin-2-One and Oxazolo[4,5-B]Pyridin-2-One Compounds and Analogs Thereof as Therapeutic Compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-12-13 US disclosed
US-7307099-B2 4-(1-(sulfonyl)-1h-indol-2-yl)-4-(hydroxy)-cyclohexa-2,5-dienone compounds and analogs thereof as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-12-11 US disclosed
EP-1638544-B1 KETONES AND REDUCED KETONES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS UNIV ABERDEEN (GB) 2007-12-05 EP disclosed
CN-101084217-A Imidazo[4,5-b]pyridin-2-one and oxazolo[4,5-b]pyridin-2-one compounds and analogs thereof as therapeutic compounds CANCER REC TECH LTD (GB) 2007-12-05 CN disclosed
EP-1858856-A2 CANCER TREATMENT USING SPECIFIC 3,6,9-SUBSTITUTED ACRIDINES Antisoma PLC (GB) 2007-11-28 EP disclosed
US-7300930-B2 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-11-27 US disclosed
WO-2007125330-A1 IMIDAZO[4, 5-B]PYRIDIN-2-ONE AND OXAZOLO[4, 5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS CANCER THERAPEUTIC COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-11-08 WO disclosed
EP-1848717-A2 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY Topotarget A/S (DK) 2007-10-31 EP disclosed
EP-1849794-A1 PROCESS FOR PRODUCING 1,2-TRANS-GLYCOSIDE COMPOUND Otsuka Chemical Co., Ltd. (JP) 2007-10-31 EP disclosed
US-20070249591-A1 Biaryl Amino Acids and Their Use in Dna Binding Oligomers SPIROGEN LIMITED (GB) 2007-10-25 US disclosed
CN-100341885-C Process for selective production of aryl 5-thio-beta-d-aldohexopyranosides TAISHO PHARMACEUTICAL CO LTD (JP) 2007-10-10 CN disclosed
EP-1456180-B1 3-(2,4)DIHYDROXYPHENYL-4-PHENYLPYRAZOLES AND THEIR MEDICAL USE VERNALIS CAMBRIDGE LTD (GB) 2007-10-03 EP disclosed
EP-1518823-B1 METAL OXIDE NANOTUBE AND PROCESS FOR PRODUCTION THEREOF JAPAN SCIENCE & TECH AGENCY (JP) 2007-09-26 EP disclosed
EP-1831184-A2 PYRAZINES AND PYRIDINES AND DERIVATIVES THEREOF AS THERAPEUTIC COMPOUNDS The Wellcome Trust Limited (GB) 2007-09-12 EP disclosed
CN-101036057-A Selective inhibitors ALCHEMIA LTD (AU) 2007-09-12 CN disclosed
EP-1828118-A1 PARP INHIBITORS Kudos Pharmaceuticals Ltd (GB) 2007-09-05 EP disclosed
US-20070191309-A1 Pyrrolobenzodiazepines as key intermediates in the synthesis of dimeric cytotoxic pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2007-08-16 US disclosed
US-20070191349-A1 C8, c8' linked 5-oxo-1,2,3,11a-tetrahydro-5h-pyrrolo[2,1-c][1,4] benzodiazepine dimers with 1h-pyrrole-dicarboxylic acid amide linkers and oligomeric analogs therof as well as related compounds for the treatment of proliferative diseases SPIROGEN LIMITED (GB) 2007-08-16 US disclosed
WO-2007088559-A1 PROCESS FOR PRODUCING SUBSTITUTED SULPHOXIDES JUBILANT ORGANOSYS LIMITED (IN) 2007-08-09 WO disclosed
US-20070185073-A1 Pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2007-08-09 US disclosed
US-20070179315-A1 Methods of amination ASTRAZENECA UK LIMITED (GB) 2007-08-02 US disclosed
EP-1812433-A1 IMIDAZO[4,5-B]PYRIDIN-2-ONE AND OXAZOLO[4,5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC COMPOUNDS Cancer Research Technology Limited (GB) 2007-08-01 EP disclosed
US-20070173497-A1 11-Hydroxy-5h-pyrrolo[2,1-c][1,4] benzodiazepin-5-one derivatives as key intermediates for the preparation of c2 substituted pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2007-07-26 US disclosed
US-7247734-B2 3,4-diarylpyrazoles and their use in the therapy of cancer VERNALIS (CAMBRIDGE) LIMITED (GB) 2007-07-24 US disclosed
EP-1807096-A1 BIOACTIVE POLYMERS THE UNIVERSITY COURT OF THE UNIVERSITY OF GLASGOW (GB) 2007-07-18 EP disclosed
WO-2007071959-A1 CHEMICAL INDUCTION OF QUIESCENCE IN BACTERIA CAMBRIDGE MICROBIAL TECHNOLOGIES LTD (GB) 2007-06-28 WO disclosed
EP-1797428-A1 SELECTIVE INHIBITORS Alchemia Pty Ltd (AU) 2007-06-20 EP disclosed
EP-1791827-A1 4-HETEROARYLMETHYL SUBSTITUTED PHTHALAZINONE DERIVATIVES Kudos Pharmaceuticals Limited (GB) 2007-06-06 EP disclosed
WO-2007060404-A1 PYRIDO-,PYRAZO- AND PYRIMIDO-PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2007-05-31 WO disclosed
EP-1789430-A2 DERIVATES OF AVERMECTIN,AVERMECTIN MONOSACCHARIDE AND AVERMECTIN AGLYCONE Syngenta Participations AG (CH) 2007-05-30 EP disclosed
WO-2007045877-A1 4-HETEROARYMETHYL SUBSTITUTED PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2007-04-26 WO disclosed
US-20070093489-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2007-04-26 US disclosed
US-7205311-B2 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED 2007-04-17 US disclosed
WO-2007039752-A1 ALKYL 4- [4- (5-OXO-2, 3, 5, 11A-TETRAHYD0-5H-PYRR0L0 [2, 1-C] [1, 4] BENZODIAZEPINE-8-YLOXY) -BUTYRYLAMINO]-1H-PYRROLE-2-CARBOXYLATE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF A PROLIFERATIVE DISEASE SPIROGEN LIMITED (GB) 2007-04-12 WO disclosed
WO-2007038829-A1 METHOD OF DRUG DESIGN ALCHEMIA LTD (AU) 2007-04-12 WO disclosed
US-20070082855-A1 Pharmaceutical formulations employing short-chain sphingolipids and their use HET NEDERLANDS KANKER INSTITUUT (NL) 2007-04-12 US disclosed
WO-2007029021-A1 1,5-SUBSTITUTED TETRAZOLES AS THERAPEUTIC COMPOUNDS THE UNIVERSITY OF EDINBURGH (GB) 2007-03-15 WO disclosed
EP-1755612-A2 PYRROLOBENZODIAZEPINE THERAPEUTIC AGENTS USEFUL IN THE TREATMENT OF LEUKAEMIAS Spirogen Limited (GB) 2007-02-28 EP disclosed
EP-1756046-A2 ARYL ALKYL SULFONAMIDES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS The University Court of The University of Aberdeen (GB) 2007-02-28 EP disclosed
US-7183298-B2 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2007-02-27 US disclosed
US-7172747-B2 Metal oxide nanotube and process for production thereof JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2007-02-06 US disclosed
US-20070027112-A1 Ketones and reduced ketones as therapeutic agents for the treatment of bone conditions UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN, THE (GB) 2007-02-01 US disclosed
US-20070015799-A1 Glyoxalase inhibitors CHROMA THERAPEUTICS LIMITED (GB) 2007-01-18 US disclosed
WO-2007006308-A1 NOVEL GLUCOPYRANOSE ESTERS AND GLUCOFURANOSE ESTERS OF ALKYL- FU MARATES AND THEIR PHARMACEUTICAL USE ADITECH PHARMA AB (SE) 2007-01-18 WO disclosed
WO-2007007054-A1 PHTHALAMIDES, SUCCINIMIDES AND RELATED COMPOUNDS AND THEIR USE AS PHARMACEUTICALS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-01-18 WO disclosed
US-7160896-B2 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2007-01-09 US disclosed
US-20070004806-A1 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2007-01-04 US disclosed
EP-1737812-A1 METHODS OF AMINATION AstraZeneca UK Limited (GB) 2007-01-03 EP disclosed
US-20060287396-A1 4-aryl quinols and analogs thereof as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-12-21 US disclosed
EP-1727808-A2 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS Spirogen Limited (GB) 2006-12-06 EP disclosed
US-7144893-B2 4-aryl quinols and analogs thereof as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-12-05 US disclosed
US-20060267004-A1 Compounds comprising a linear series of five fused carbon rings, and preparation thereof UNIVERSITY OF OTTAWA (CA) 2006-11-30 US disclosed
US-20060264622-A1 Synthesis of protected pyrrolobenzodiazepines SPIROGEN LIMITED (GB) 2006-11-23 US disclosed
EP-1723152-A1 PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2006-11-22 EP disclosed
EP-1723151-A2 PYRROLOBENZODIAZEPINES AS KEY INTERMEDIATES IN THE SYNTHESIS OF DIMERIC CYTOTOXIC PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2006-11-22 EP disclosed
EP-1720880-A1 C8, C8' LINKED 5-OXO-1,2,3,11A-TETRAHYDRO-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPINE DIMERS WITH 1H-PYRROLE-DICARBOXYLIC ACID AMIDE LINKERS AND OLIGOMERIC ANALOGS THEREOF AS WELL AS RELATED COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES Spirogen Limited (GB) 2006-11-15 EP disclosed
EP-1720881-A1 11-HYDROXY-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPIN-5-ONE DERIVATIVES AS KEY INTERMEDIATES FOR THE PREPARATION OF C2 SUBSTITUTED PYRROLOBENZODIAZEPINS Spirogen Limited (GB) 2006-11-15 EP disclosed
WO-2006111759-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2006-10-26 WO disclosed
US-20060240527-A1 Process for producing fine self-aggregates JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2006-10-26 US disclosed
US-7115619-B2 N8, N13 -disubstituted quino[4,3,2-kl]acridinium salts as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-10-03 US disclosed
US-7112698-B2 4-(c2-6alkoxy)-substituted chalcones as therapeutic agents SPEAR THERAPEUTICS LIMITED (GB) 2006-09-26 US disclosed
US-7109189-B2 Mitochondrially targeted antioxidants UNIVERSITY OF OTAGO (NZ) 2006-09-19 US disclosed
WO-2006095139-A2 CANCER TREATMENT USING SPECIFIC 3,6,9-SUBSTITUTED ACRIDINES ANTISOMA PLC (GB) 2006-09-14 WO disclosed
US-20060199804-A1 Compounds KUDOS PHARMACEUTICALS LTD (GB) 2006-09-07 US disclosed
US-20060199803-A1 Compounds KUDOS PHARMACEUTICALS LTD (GB) 2006-09-07 US disclosed
WO-2006090167-A2 HYDRAZINOMETHYL, HYDR ZONOMETHYL AND 5-MEMBERED HETEROCYLIC COMPOUNDS WHICH ACT AS MTOR INHIBITORS AND THEIR USE AS ANTI CANCER AGENTS KUDOS PHARMACEUTICALS LIMITED (GB) 2006-08-31 WO disclosed
WO-2006090169-A1 2,4-DIAMINO-PYRIDOPYRIMIDINE DERIVATIVES AND THEIR USE AS MTOR INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2006-08-31 WO disclosed
WO-2006085219-A2 6-ETHER/THIOETHER-PURINES AS TOPOISOMERASE II CATALYTIC INHIBITORS AND THEIR USE IN THERAPY TOPOTARGET A/S (DK) 2006-08-17 WO disclosed
EP-1686959-A2 PHARMACEUTICAL FORMULATIONS EMPLOYING SHORT-CHAIN SPHINGOLIPIDS AND THEIR USE HET NEDERLANDS KANKER INSTITUUT (The Netherlands Cancer Institute) (NL) 2006-08-09 EP disclosed
US-20060172019-A1 Cannabinoid receptor inverse agonists and neutral antagonists as therapeutic agents for the treatment of bone disorders ABERDEEN, THE UNIVERSITY COURT OF THE UNIVERSITY OF (GB) 2006-08-03 US disclosed
US-20060167237-A1 Derivatives of monosaccharides for drug discovery ALCHEMIA LIMITED (AU) 2006-07-27 US disclosed
US-20060149059-A1 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2006-07-06 US disclosed
WO-2006067466-A2 PYRAZINES AND PYRIDINES AND DERIVATIVES THEREOF AS THERAPEUTIC COMPOUNDS THE WELLCOME TRUST LIMITED (GB) 2006-06-29 WO disclosed
WO-2006067472-A1 PARP INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2006-06-29 WO disclosed
US-20060135770-A1 PARP inhibitors KUDOS PHARMACEUTICALS LTD. (GB) 2006-06-22 US disclosed
US-20060128693-A1 Pyrrolobenzodiazepines MEDIMMUNE LIMITED (GB) 2006-06-15 US disclosed
EP-1664049-A1 SYNTHESIS OF PROTECTED PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2006-06-07 EP disclosed
EP-1441716-B1 ALKANE DIOL DERIVATIVES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS UNIV ABERDEEN (GB) 2006-05-31 EP disclosed
US-20060111389-A1 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-05-25 US disclosed
US-20060100265-A1 4-(1-(sulfonyl)-1h-indol-2-yl)-4-(hydroxy)-cyclohexa-2,5-dienone compounds and analogs thereof as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-05-11 US disclosed
WO-2006043090-A1 IMIDAZO[4,5-B]PYRIDIN-2-ONE AND OXAZOLO[4,5-B]PYRIDIN-2-ONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-04-27 WO disclosed
WO-2006040579-A1 BIOACTIVE POLYMERS THE UNIVERSITY COURT OF THE UNIVERSITY OF GLASGOW (GB) 2006-04-20 WO disclosed
WO-2006037159-A1 SELECTIVE INHIBITORS ALCHEMIA LIMITED (AU) 2006-04-13 WO disclosed
US-20060079528-A1 (E)-3-(1,3-Benzoxazol-2-yl)-N-hydroxy-2-propenamide; Methyl (E)-3-(2-quinolinyl)-2-propenoate; histone deacetylase inhibitors; inflammatory disease; cancer TOPOTARGET UK LIMITED (GB) 2006-04-13 US disclosed
EP-1638544-A2 KETONES AND REDUCED KETONES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS The University Court of The University of Aberdeen (GB) 2006-03-29 EP disclosed
US-20060063767-A1 Phthalazinone derivatives KUDOS PHARMACEUTICALS LTD (GB) 2006-03-23 US disclosed
US-20060058282-A1 Carbamic acid compounds comprising an ester or ketone linkage as hdac inhibitors TOPOTARGET UK LIMITED (GB) 2006-03-16 US disclosed
EP-1633724-A1 PHTHALAZINONE DERIVATIVES Kudos Pharmaceuticals Limited (GB) 2006-03-15 EP disclosed
WO-2006024405-A2 DERIVATIVES OF AVERMECTIN, AVERMECTIN MONOSACCHARIDE AND AVERMECTIN AGLYCONE SYNGENTA PARTICIPATIONS AG (CH) 2006-03-09 WO disclosed
EP-1632498-A1 Derivatives of avermectin, avermectin monosaccharide and avermectin aglycone Syngenta Participations AG (CH) 2006-03-08 EP disclosed
WO-2006021801-A1 4-HETEROARYLMETHYL SUBSTITUTED PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2006-03-02 WO disclosed
EP-1622869-A1 GLYOXALASE INHIBITORS Chroma Therapeutics Limited (GB) 2006-02-08 EP disclosed
US-6984636-B2 Mitochondrially targeted antioxidants MEDICAL RESEARCH COUNCIL (GB) 2006-01-10 US disclosed
EP-1606019-A1 CANNABINOID RECEPTOR INVERSE AGONISTS AND NEUTRAL ANTAGONISTS AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE DISORDERS The University Court of The University of Aberdeen (GB) 2005-12-21 EP disclosed
US-20050274945-A1 Compounds comprising a linear series of five fused carbon rings, and preparation thereof UNIVERSITY OF OTTAWA (CA) 2005-12-15 US disclosed
WO-2005118528-A2 ARYL ALKYL SULFONAMIDES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2005-12-15 WO disclosed
EP-1599449-A2 CARBAMIC ACID COMPOUNDS COMPRISING A BICYCLIC HETEROARYL GROUP AS HDAC INHIBITORS TopoTarget UK Limited (GB) 2005-11-30 EP disclosed
WO-2005110423-A2 PYRROLOBENZODIAZEPINE THERAPEUTIC AGENTS USEFUL IN THE TREATMENT OF LEUKAEMIAS SPIROGEN LIMITED (GB) 2005-11-24 WO disclosed
EP-1335898-B1 CARBAMIC ACID COMPOUNDS COMPRISING AN AMIDE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LTD (GB) 2005-11-23 EP disclosed
EP-1598067-A1 Carbamic acid compounds comprising an amide linkage as HDAC inhibitors TopoTarget UK Limited (GB) 2005-11-23 EP disclosed
US-6960685-B2 Carbamic acid compounds comprising an ether linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2005-11-01 US disclosed
US-20050227957-A1 Mitochondrially targeted antioxidants MEDICAL RESEARCH COUNCIL (GB) 2005-10-13 US disclosed
EP-1583736-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN ESTER OR KETONE LINKAGE AS HDAC INHIBITORS TopoTarget UK Limited (GB) 2005-10-12 EP disclosed
US-20050222230-A1 3,4-diarylpyrazoles and their use in the therapy of cancer VERNALIS (CAMBRIDGE) LIMITED (GB) 2005-10-06 US disclosed
WO-2005090283-A1 METHODS OF AMINATION ASTRAZENECA UK LIMITED (GB) 2005-09-29 WO disclosed
CN-1675233-A Process for selective production of aryl 5-thio-beta-d-aldohexopyranosides TAISHO PHARMACEUTICAL CO LTD (JP) 2005-09-28 CN disclosed
EP-1575955-A1 PYRROLOBENZODIAZEPINES Spirogen Limited (GB) 2005-09-21 EP disclosed
WO-2005085251-A1 11-HYDROXY-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPIN-5-ONE DERIVATIVES AS KEY INTERMEDIATES FOR THE PREPARATION OF C2 SUBSTITUTED PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed
WO-2005085260-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed
WO-2005085177-A2 BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed
WO-2005085259-A2 PYRROLOBENZODIAZEPINES AS KEY INTERMEDIATES IN THE SYNTHESIS OF DIMERIC CYTOTOXIC PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed
WO-2005085250-A1 C8, C8' LINKED 5-OXO-1,2,3,11A-TETRAHYDRO-5H-PYRROLO[2,1-C][1,4]BENZODIAZEPINE DIMERS WITH 1H-PYRROLE-DICARBOXYLIC ACID AMIDE LINKERS AND OLIGOMERIC ANALOGS THEROF AS WELL AS RELATED COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES SPIROGEN LIMITED (GB) 2005-09-15 WO disclosed
EP-1572197-A1 4- 1- (SULFONYL) -1H-INDOL-2-YL)-4- (HYDROXY) -CYCLOHEXA-2,5-DIENONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2005-09-14 EP disclosed
US-20050143385-A1 Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors TOPOTARGET UK LIMITED (GB) 2005-06-30 US disclosed
EP-1539780-A1 DERIVATIVES OF MONOSACCHARIDES FOR DRUG DISCOVERY Alchemia Limited (AU) 2005-06-15 EP disclosed
EP-1186688-B1 Hollow fibrous organic nanotube and method for producing the same NAT INST OF ADVANCED IND SCIEN (JP) 2005-06-15 EP disclosed
EP-1534720-A1 MITOCHONDRIALLY TARGETED ANTIOXIDANTS Medical Research Council (GB) 2005-06-01 EP disclosed
WO-2005046637-A2 PHARMACEUTICAL FORMULATIONS EMPLOYING SHORT-CHAIN SPHINGOLIPIDS AND THEIR USE HET NEDERLANDS KANKER INSTITUUT (NL) 2005-05-26 WO disclosed
US-20050107445-A1 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors PROLIFIX LIMITED (GB) 2005-05-19 US disclosed
US-6888027-B2 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2005-05-03 US disclosed
US-20050085515-A1 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors TOPO TARGET UK LIMITED, (GB) 2005-04-21 US disclosed
US-20050077496-A1 Metal oxide nanotube and process for production thereof JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2005-04-14 US disclosed
US-20050070568-A1 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2005-03-31 US disclosed
EP-1518823-A1 METAL OXIDE NANOTUBE AND PROCESS FOR PRODUCTION THEREOF Japan Science and Technology Agency (JP) 2005-03-30 EP disclosed
WO-2005023814-A1 SYNTHESIS OF PROTECTED PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2005-03-17 WO disclosed
US-20050059663-A1 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2005-03-17 US disclosed
EP-1512750-A1 PROCESS FOR PRODUCING FINE SELF-AGGREGATE Japan Science and Technology Agency (JP) 2005-03-09 EP disclosed
US-20050014937-A1 Fibrous nano self-assemblies JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2005-01-20 US disclosed
EP-1492534-A1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TopoTarget UK Limited (GB) 2005-01-05 EP disclosed
US-20040259957-A1 4-(c2-6alkoxy)-substituted chalcones as therapeutic agents SPEAR THERAPEUTICS LIMITED (GB) 2004-12-23 US disclosed
US-20040254149-A1 3, 4-Methylenedioxy-substituted chalcones as therapeutic agents SPEAR THERAPEUTICS LIMITED (GB) 2004-12-16 US disclosed
US-20040254151-A1 Alkane diol derivatives as therapeutic agents for the treatment of bone conditions UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN, THE (GB) 2004-12-16 US disclosed
WO-2004101506-A1 GLYOXALASE INHIBITORS CHROMA THERAPEUTICS LIMITED (GB) 2004-11-25 WO disclosed
EP-1479799-A1 FIBROUS NANO SELF-ASSEMBLIES Japan Science and Technology Agency (JP) 2004-11-24 EP disclosed
WO-2004098582-A2 KETONES AND REDUCED KETONES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2004-11-18 WO disclosed
EP-1474397-A1 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS Cancer Research Technology Limited (GB) 2004-11-10 EP disclosed
US-20040220236-A1 4-Aryl quinols and analogs thereof as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2004-11-04 US disclosed
US-20040198830-A1 Carbamic acid compounds comprising an ether linkage as hdac inhibitors TOPOTARGET UK LIMITED (GB) 2004-10-07 US disclosed
WO-2004080976-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2004-09-23 WO disclosed
WO-2004078261-A1 CANNABINOID RECEPTOR INVERSE AGONISTS AND NEUTRAL ANTAGONISTS AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE DISORDERS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2004-09-16 WO disclosed
EP-1456180-A1 3,4-DIARYLPYRAZOLES AND THEIR USE IN THE THERAPY OF CANCER Vernalis (Oxford) Ltd (GB) 2004-09-15 EP disclosed
WO-2004076386-A2 CARBAMIC ACID COMPOUNDS COMPRISING A BICYCLIC HETEROARYL GROUP AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2004-09-10 WO disclosed
WO-2004065354-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN ESTER OR KETONE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2004-08-05 WO disclosed
EP-1441716-A1 ALKANE DIOL DERIVATIVES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS The University Court of The University of Aberdeen (GB) 2004-08-04 EP disclosed
WO-2004056361-A1 4-(1-(SULFONYL)-1H-INDOL-2-YL)-4-(HYDROXY)-CYCLOHEXA-2,5-DIENONE COMPOUNDS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2004-07-08 WO disclosed
EP-1432413-A2 3,4-METHYLENEDIOXY-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2004-06-30 EP disclosed
EP-1432669-A1 4-(C2-6 ALKOXY)-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2004-06-30 EP disclosed
WO-2004043963-A1 PYRROLOBENZODIAZEPINES SPIROGEN LIMITED (GB) 2004-05-27 WO disclosed
US-20040092598-A1 Carbamic acid compounds comprising an amide linkage as hdac inhibitors TOPOTARGET UK LIMITED (GB) 2004-05-13 US disclosed
US-20040077726-A1 Carbamic acid compounds comprising a sulfonamide linkage as hdac inhibitors SWK FUNDING LLC 2004-04-22 US disclosed
EP-1404659-A1 4-ARYL QUINOLS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2004-04-07 EP disclosed
US-20040063739-A1 N8, n13 -disubstituted quino[4,3,2-kl]acridinium salts as therapeutic agents CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2004-04-01 US disclosed
WO-2004014929-A1 DERIVATIVES OF MONOSACCHARIDES FOR DRUG DISCOVERY ALCHEMIA LIMITED (AU) 2004-02-19 WO disclosed
WO-2004014927-A1 MITOCHONDRIALLY TARGETED ANTIOXIDANTS MEDICAL RESEARCH COUNCIL (GB) 2004-02-19 WO disclosed
US-20040029851-A1 Mitochondrially targeted antioxidants MEDICAL RESEARCH COUNCIL (GB) 2004-02-12 US disclosed
EP-1363888-A2 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS Cancer Research Technology Limited (GB) 2003-11-26 EP disclosed
US-20030207909-A1 Therapeutic acridone and acridine compounds CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-11-06 US disclosed
US-6632497-B2 The hollow fibrous organic nanotube having an inner pore diameter of 10 to 20 nm and outer diameter of 40-80 nm, comprising an O-glycoside type glycolipid having aldose residue as glycosyl group NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 2003-10-14 US disclosed
WO-2003082288-A1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LIMITED (GB) 2003-10-09 WO disclosed
EP-1335898-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN AMIDE LINKAGE AS HDAC INHIBITORS Prolifix Limited (GB) 2003-08-20 EP disclosed
EP-1333842-A2 USE OF CORTISOL-SEQUESTERING AGENTS FOR THE TREATMENT OF HYPERCORTISOLAEMIA RELATED DISORDERS Akzo Nobel N.V. (NL) 2003-08-13 EP disclosed
EP-1330456-A2 N8,N13 -DISUBSTITUTED QUINO 4,3,2-KL]ACRIDINIUM SALTS AS THERAPEUTIC AGENTS Cancer Research Technology Limited (GB) 2003-07-30 EP disclosed
WO-2003059885-A1 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-07-24 WO disclosed
EP-1328510-A2 CARBAMIC ACID COMPOUNDS COMPRISING A SULFONAMIDE LINKAGE AS HDAC INHIBITORS PROLIFIX LTD. (GB) 2003-07-23 EP disclosed
WO-2003055860-A1 3,4-DIARYLPYRAZOLES AND THEIR USE IN THE THERAPY OF CANCER VERNALIS (CAMBRIDGE) LIMITED (GB) 2003-07-10 WO disclosed
WO-2003037321-A1 ALKANE DIOL DERIVATIVES AS THERAPEUTIC AGENTS FOR THE TREATMENT OF BONE CONDITIONS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2003-05-08 WO disclosed
WO-2003029176-A1 4-(C2-6ALKOXY)-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-04-10 WO disclosed
WO-2003028713-A2 3,4-METHYLENEDIOXY-SUBSTITUTED CHALCONES AS THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-04-10 WO disclosed
WO-2003004479-A1 4-ARYL QUINOLS AND ANALOGS THEREOF AS THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-01-16 WO disclosed
EP-1210090-A2 USE OF CHEMICAL CHELATORS AS REVERSAL AGENTS FOR DRUG-INDUCED NEUROMUSCULAR BLOCK Akzo Nobel N.V. (NL) 2002-06-05 EP disclosed
WO-2002036105-A2 USE OF CORTISOL-SEQUESTERING AGENTS FOR THE TREATMENT OF HYPERCORTISOLAEMIA RELATED DISORDERS AKZO NOBEL N.V. (US) 2002-05-10 WO disclosed
US-20020051881-A1 Hollow fibrous organic nanotube and method for producing the same NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 2002-05-02 US disclosed
WO-2002030879-A2 CARBAMIC ACID COMPOUNDS COMPRISING A SULFONAMIDE LINKAGE AS HDAC INHIBITORS PROLIFIX LIMITED (GB) 2002-04-18 WO disclosed
WO-2002030932-A2 N8,N13-DISUBSTITUTED QUINO[4,3,2-KL]ACRIDINIUM SALTS AS THERAPEUTIC AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2002-04-18 WO disclosed
WO-2002026696-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN AMIDE LINKAGE AS HDAC INHIBITORS PROLIFIX LIMITED (GB) 2002-04-04 WO disclosed
WO-2002026703-A1 CARBAMIC ACID COMPOUNDS COMPRISING AN ETHER LINKAGE AS HDAC INHIBITORS PROLIFIX LIMITED (GB) 2002-04-04 WO disclosed
EP-1186688-A1 Hollow fibrous organic nanotube and method for producing the same National Institute of Advanced Industrial Science and Technology (JP) 2002-03-13 EP disclosed
WO-2002008193-A2 THERAPEUTIC ACRIDONE AND ACRIDINE COMPOUNDS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2002-01-31 WO disclosed
WO-2001012202-A2 USE OF CHEMICAL CHELATORS AS REVERSAL AGENTS FOR DRUG-INDUCED NEUROMUSCULAR BLOCK AKZO NOBEL N.V. (NL) 2001-02-22 WO disclosed
EP-0973534-A1 PHARMACEUTICAL COMPOSITIONS HAVING APPETITE SUPPRESSANT ACTIVITY CSIR (ZA) 2000-01-26 EP disclosed
WO-1998046243-A2 PHARMACEUTICAL COMPOSITIONS HAVING APPETITE SUPPRESSANT ACTIVITY CSIR (ZA) 1998-10-22 WO disclosed
WO-1998024792-A1 ANTICOAGULANT GLYCOSIDES AND PHARMACEUTICAL COMPOSITIONS THEREOF Richter Gedeon Vegyészeti Gyár Rt. (HU) 1998-06-11 WO disclosed
WO-1998024792-A1 ANTICOAGULANT GLYCOSIDES AND PHARMACEUTICAL COMPOSITIONS THEREOF Richter Gedeon Vegyészeti Gyár Rt. (HU) 1998-06-11 WO disclosed
EP-0730601-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTIONS WASHINGTON UNIVERSITY (US) 1996-09-11 EP disclosed
EP-0505573-B1 PROCESS FOR PRODUCING D-ALTROSE JAPAN TOBACCO INC (JP) 1996-03-27 EP disclosed
WO-1995014028-A9 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTIONS 1995-08-10 WO disclosed
WO-1995014028-A2 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTIONS WASHINGTON UNIVERSITY (US) 1995-05-26 WO disclosed
US-5410038-A method of preparing D-altrose JAPAN TOBACCO INC. (JP) 1995-04-25 US disclosed
EP-0505573-A1 PROCESS FOR PRODUCING D-ALTROSE Japan Tobacco Inc. (JP) 1992-09-30 EP disclosed
US-5066645-A Antitumor agents BRISTOL-MYERS COMPANY (US) 1991-11-19 US disclosed
EP-0415453-A2 Epipodophyllotoxin altroside derivatives Bristol-Myers Squibb Company (US) 1991-03-06 EP disclosed
US-4593090-A Containing perhydrofuran or pyran ring structure GOGO KIMURA (JP) 1986-06-03 US disclosed
EP-0067019-B1 NOVEL NITROSOUREA COMPOUND, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME Kimura, Goro (JP) 1986-03-19 EP disclosed
EP-0067019-A1 Novel nitrosourea compound, method for preparing same, and pharmaceutical composition containing same Kimura, Goro (JP) 1982-12-15 EP disclosed
US-4350811-A Chiral sugar complexes IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1982-09-21 US disclosed
EP-0002046-B1 PROCESS FOR THE PREPARATION OF (1S,2S,6R)-2-METHYL-3,7-DIOXABICYCLO(4,1,0)HEPTAN-4-OL AND ITS METHYL ETHER F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-02-10 EP disclosed
EP-0002046-B1 PROCESS FOR THE PREPARATION OF (1S,2S,6R)-2-METHYL-3,7-DIOXABICYCLO(4,1,0)HEPTAN-4-OL AND ITS METHYL ETHER F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-02-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
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US-20220288221-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES EGFR, ERBB2, ERBB3 LGALS3 1610/4885LGALS1 2642/4885LGALS9 1366/4885
US-20090163477-A1 PHTHALAZINONE DERIVATIVES PARP1, PARP2, PARP11 LGALS3 4101/4885LGALS1 3682/4885LGALS9 4580/4885
US-20140303367-A1 Methods for Synthesizing Molybdopterin Precursor Z Derivatives MTHFD2, ADH1B, DPYD LGALS3 4736/4885LGALS1 4712/4885LGALS9 4287/4885
US-20130317237-A1 SYNTEHSIS OF CYCLIC CARBONATES CA12, SUCLA2, LMNA LGALS3 2089/4885LGALS1 1720/4885LGALS9 2035/4885
US-20140378442-A1 PHTHALAZINONE DERIVATIVES NR0B1, NR0B2, NR2E1 LGALS3 4221/4885LGALS1 2781/4885LGALS9 4247/4885
US-20210284613-A1 RADIOLABELLED COMPOUND PARP3, PARP2, PARP1 LGALS3 1132/4885LGALS1 1629/4885LGALS9 1030/4885
US-20160129013-A1 TARGETED PYRROLOBENZODIAZAPINE CONJUGATES QDPR, SBDS, DNPEP LGALS3 3736/4885LGALS1 4207/4885LGALS9 2225/4885
US-10287220-B2 Fluorination method F13B, PPARG, PGC LGALS3 952/4885LGALS1 1424/4885LGALS9 1241/4885
US-11466032-B2 Cytotoxic agents MKI67, TP53, NFATC1 LGALS3 2118/4885LGALS1 1964/4885LGALS9 3017/4885
US-20070191349-A1 C8, c8' linked 5-oxo-1,2,3,11a-tetrahydro-5h-pyrrolo[2,1-c][1,4] benzodiazepine dimers with 1h-pyrrole-dicarboxylic acid amide linkers and oligomeric analogs therof as well as related compounds for the treatment of proliferative diseases TSPO, GABRD, BCOR LGALS3 4803/4885LGALS1 4764/4885LGALS9 4816/4885
US-20200345861-A1 PYRROLOBENZODIAZEPINE-ANTIBODY CONJUGATES CD79B, BCL6B, BCL6 LGALS3 3180/4885LGALS1 3599/4885LGALS9 1791/4885
US-20210371413-A1 POLYCYCLIC AMIDES AS CYTOTOXIC AGENTS PBRM1, NFATC1, ACIN1 LGALS3 4165/4885LGALS1 3872/4885LGALS9 4417/4885
US-20210171637-A1 ANTI-B7-H3 ANTIBODIES AND ANTIBODY DRUG CONJUGATES HRH3, H1-3, CD274 LGALS3 568/4885LGALS1 2094/4885LGALS9 1295/4885
US-11690918-B2 Pyrrolobenzodiazepine-anti-CD22 antibody conjugates CD22, CD2, CD2BP2 LGALS3 1065/4885LGALS1 1398/4885LGALS9 460/4885
US-20040254149-A1 3, 4-Methylenedioxy-substituted chalcones as therapeutic agents OXER1, CCNO, CCNB3 LGALS3 1959/4885LGALS1 2581/4885LGALS9 4255/4885
US-11524969-B2 Pyrrolobenzodiazepines and conjugates thereof as antitumour agents PBRM1, HDAC6, NPM1 LGALS3 3197/4885LGALS1 4031/4885LGALS9 3688/4885
US-20190218291-A1 COMBINATION THERAPY WITH AN ANTI-AXL ANTIBODY-DRUG CONJUGATE ERBB2, ERBB3, AXL LGALS3 255/4885LGALS1 324/4885LGALS9 229/4885
US-20140323726-A1 Methods for synthesizing molybdopterin precursor Z derivatives MTHFD2, ADH1B, DPYD LGALS3 4736/4885LGALS1 4712/4885LGALS9 4287/4885
US-20060100265-A1 4-(1-(sulfonyl)-1h-indol-2-yl)-4-(hydroxy)-cyclohexa-2,5-dienone compounds and analogs thereof as therapeutic agents TXNRD1, TXNRD3, TXNRD2 LGALS3 4077/4885LGALS1 3726/4885LGALS9 4409/4885
US-20060079528-A1 (E)-3-(1,3-Benzoxazol-2-yl)-N-hydroxy-2-propenamide; Methyl (E)-3-(2-quinolinyl)-2-propenoate; histone deacetylase inhibitors; inflammatory disease; cancer HDAC1, HDAC11, HDAC5 LGALS3 3420/4885LGALS1 3961/4885LGALS9 3978/4885
US-10576164-B2 Pyrrolobenzodiazepines and conjugates thereof CHRM1, NPSR1, CHRM4 LGALS3 3462/4885LGALS1 4533/4885LGALS9 3185/4885
US-20200399365-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES SBDS, DCTD, DRD1 LGALS3 4474/4885LGALS1 4509/4885LGALS9 3223/4885
US-20150307541-A1 WATER-SOLUBLE PHOTOCHROMIC MOLECULES SLC2A3, CCND3, MRPS23 LGALS3 215/4885LGALS1 828/4885LGALS9 2612/4885
US-20070191309-A1 Pyrrolobenzodiazepines as key intermediates in the synthesis of dimeric cytotoxic pyrrolobenzodiazepines CBR3, CBR1, CYCS LGALS3 4373/4885LGALS1 4750/4885LGALS9 4454/4885
US-20170226124-A1 PHTHALAZINONE DERIVATIVES NR0B1, NR0B2, NR2E1 LGALS3 4380/4885LGALS1 3053/4885LGALS9 4359/4885
US-20060058282-A1 Carbamic acid compounds comprising an ester or ketone linkage as hdac inhibitors HDAC1, HDAC7, HDAC11 LGALS3 4046/4885LGALS1 3527/4885LGALS9 3477/4885
US-20090281086-A1 2 -OXYHETEROARYLAMIDE DERIVATIVES AS PARP INHIBITORS PARP2, PARP3, PARP11 LGALS3 4649/4885LGALS1 4455/4885LGALS9 4769/4885
US-12398162-B2 Guanine analogs as telomerase substrates and telomere length affectors TERT, POT1, TERF2 LGALS3 2578/4885LGALS1 1788/4885LGALS9 2878/4885
US-20060172019-A1 Cannabinoid receptor inverse agonists and neutral antagonists as therapeutic agents for the treatment of bone disorders CNR2, CNR1, GPER1 LGALS3 2214/4885LGALS1 2160/4885LGALS9 2578/4885
US-20180169258-A1 PYRROLOBENZODIAZEPINE-ANTI-CD22 ANTIBODY CONJUGATES CD22, CD2, CD2BP2 LGALS3 1133/4885LGALS1 1403/4885LGALS9 518/4885
US-20050107445-A1 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors HDAC1, HDAC11, HDAC3 LGALS3 4614/4885LGALS1 4181/4885LGALS9 4502/4885
US-20180092986-A1 SITE-SPECIFIC ANTIBODY-DRUG CONJUGATES CD22, SBDS, CD2 LGALS3 3313/4885LGALS1 3170/4885LGALS9 2054/4885
US-20060135770-A1 PARP inhibitors PARP2, PARP1, PARP3 LGALS3 4077/4885LGALS1 3918/4885LGALS9 4383/4885
US-20230135723-A1 ANTI-CD98 ANTIBODIES AND ANTIBODY DRUG CONJUGATES CD99, SLC3A2, CD63 LGALS3 1076/4885LGALS1 2150/4885LGALS9 1101/4885
US-20040092598-A1 Carbamic acid compounds comprising an amide linkage as hdac inhibitors HDAC1, HDAC11, HDAC3 LGALS3 4589/4885LGALS1 4283/4885LGALS9 4646/4885
US-20100113425-A1 PYRROLOBENZODIAZEPINES CNR1, MC3R, NPSR1 LGALS3 3390/4885LGALS1 4770/4885LGALS9 3134/4885
US-10561739-B2 Targeted pyrrolobenzodiazapine conjugates QDPR, SBDS, DNPEP LGALS3 3736/4885LGALS1 4207/4885LGALS9 2225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.