Perflubutane

Perflubutane

SCHEMBL73685

FC(F)(F)C(F)(F)C(F)(F)C(F)(F)F.O=S(=O)(F)F

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 7/20 0.48
CA1 P00915 6/20 0.46
MMP1 P03956 4/20 0.46
MMP2 P08253 4/20 0.46
MMP9 P14780 4/20 0.46
MMP8 P22894 4/20 0.46
MMP13 P45452 4/20 0.46
F2 P00734 4/20 0.40
PRSS1 P07477 4/20 0.40
PRSS2 P07478 4/20 0.40
PRSS3 P35030 4/20 0.40
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.38
CA7 P43166 1/20 0.35
CA13 Q8N1Q1 1/20 0.35
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474710 0.96 CA2 (0.52) CA2CA1MMP1MMP2MMP9
Perflenapent SCHEMBL14763328 0.96 CA2 (0.52) CA2CA1MMP1MMP2MMP9
SCHEMBL9505503 0.96 CA2 (0.52) CA2CA1MMP1MMP2MMP9
Perflexane SCHEMBL3192336 0.96 CA2 (0.52) CA2CA1MMP1MMP2MMP9
Perflutren SCHEMBL1470237 0.92 CA2 (0.41) CA2CA1MMP1MMP2MMP9
Perflubutane SCHEMBL6557063 0.85 TSHR (0.57) CA2CA1MMP1MMP2MMP9
SCHEMBL6898759 0.84 CA2 (0.50) CA2CA1MMP1MMP2MMP9
SCHEMBL1469649 0.82 CA2 (0.40) CA2CA1MMP1MMP2MMP9
SCHEMBL11563004 0.82 TSHR (0.53) CA2CA1MMP1MMP2MMP9
Perflubutane SCHEMBL4458683 0.80 CA2 (0.50) CA2CA1MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 177 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118852101-A Sulfonyloxy high-valence iodized salt and preparation method thereof 中国人民解放军军事科学院防化研究院 2024-10-29 CN claimed
WO-2024064745-A1 SYNTHESIS OF RELDESEMTIV CYTOKINETICS, INCORPORATED (US) 2024-03-28 WO claimed
CN-117619175-A Nanofiltration membrane and preparation method and application thereof 清华大学 2024-03-01 CN claimed
CN-116675861-A Preparation method of modified polyethersulfone/polyetherimide polymer alloy 深圳先进技术研究院 2023-09-01 CN claimed
CN-116457335-A Process for preparing 3-fluoro-5- (((1S, 2 aR) -1,3, 4-pentafluoro-2 a-hydroxy-2, 2a,3, 4-tetrahydro-1H-cyclopenta [ cd ] inden-7-yl) oxy) benzonitrile and polymorphs thereof 尼坎治疗公司 2023-07-18 CN claimed
US-10794853-B2 Methods for depositing polymer layer for sensor applications via hot wire chemical vapor deposition APPLIED MATERIALS, INC. (US) 2020-10-06 US claimed
EP-3551780-A1 METHODS FOR DEPOSITING POLYMER LAYER FOR SENSOR APPLICATIONS VIA HOT WIRE CHEMICAL VAPOR DEPOSITION Applied Materials, Inc. (US) 2019-10-16 EP claimed
US-20180164245-A1 METHODS FOR DEPOSITING POLYMER LAYER FOR SENSOR APPLICATIONS VIA HOT WIRE CHEMICAL VAPOR DEPOSITION APPLIED MATERIALS, INC. 2018-06-14 US claimed
US-8906454-B2 Methods for depositing metal-polymer composite materials atop a substrate APPLIED MATERIALS, INC. (US) 2014-12-09 US claimed
WO-2013039862-A2 METHODS FOR DEPOSITING METAL-POLYMER COMPOSITE MATERIALS ATOP A SUBSTRATE APPLIED MATERIALS, INC. (US) 2013-03-21 WO claimed
US-20130065401-A1 METHODS FOR DEPOSITING METAL-POLYMER COMPOSITE MATERIALS ATOP A SUBSTRATE APPLIED MATERIALS, INC. (US) 2013-03-14 US claimed
US-8324417-B2 Process for the preparation of (S)-2-amino-5-cyclopropyl-4,4-difluoropentanoic acid and alkyl esters and acid salts thereof VIROBAY, INC. (US) 2012-12-04 US claimed
WO-2011022429-A2 PROCESS FOR THE PREPARATION OF (S)-2-AMINO-5-CYCLOPROPYL-4,4-DIFLUOROPENTANOIC ACID AND ALKYL ESTERS AND ACID SALTS THEREOF VIROBAY, INC. (US) 2011-02-24 WO claimed
US-20110046406-A1 PROCESS FOR THE PREPARATION OF (S)-2-AMINO-5-CYCLOPROPYL-4,4-DIFLUOROPENTANOIC ACID AND ALKYL ESTERS AND ACID SALTS THEREOF VIROBAY, INC. (US) 2011-02-24 US claimed
US-7429628-B2 Method of making a thermoplastic composition containing an antistatic agent SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2008-09-30 US claimed
US-20080081857-A1 METHOD OF MAKING A THERMOPLASTIC COMPOSITION CONTAINING AN ANTISTATIC AGENT SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2008-04-03 US claimed
US-6566542-B2 Such as 17-alpha-fluoro-11-beta-(4-(2-(1-piperidinyl) ethoxy) phenyl)-estra-1,3,5(10)-trien-3-ol for treatment of osteoporosis and cardiovascular protection; side effect reduction; provides alternative to estradiol AVENTIS PHARMA S.A. (FR) 2003-05-20 US claimed
EP-1090027-B1 NOVEL 17-HALOGENATED 19-NOR STEROIDS, METHOD AND INTERMEDIATES FOR PREPARING SAME, USE AS MEDICINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AVENTIS PHARMA SA (FR) 2003-04-16 EP claimed
US-20030022874-A1 New 17-halogenated 19-nor steroids, preparation process and intermediates, use as medicaments and the pharmaceutical compositions containing them BOUALI YASMINA (FR) 2003-01-30 US claimed
EP-4665332-A2 CYCLIN DEPENDENT KINASE DEGRADERS AND METHODS OF USE THEREOF Differentiated Therapeutics Inc (US) 2025-12-24 EP disclosed
CN-120072800-A Microelectronic assembly with through-glass via stress relief in glass core 英特尔公司 2025-05-30 CN disclosed
CN-119585258-A Novel 7-substituted indole sulfonamide derivatives 豪夫迈·罗氏有限公司 2025-03-07 CN disclosed
CN-113228335-B Organic light emitting device 株式会社LG化学 2024-11-29 CN disclosed
CN-118852101-A Sulfonyloxy high-valence iodized salt and preparation method thereof 中国人民解放军军事科学院防化研究院 2024-10-29 CN disclosed
CN-112868111-B Organic light emitting device 株式会社LG化学 2024-09-06 CN disclosed
WO-2024173412-A2 CYCLIN DEPENDENT KINASE DEGRADERS AND METHODS OF USE THEREOF DIFFERENTIATED THERAPEUTICS, INC. (US) 2024-08-22 WO disclosed
CN-118510783-A Spiro modulators of cholesterol biosynthesis and their use for promoting remyelination 基因泰克公司 2024-08-16 CN disclosed
CN-113228331-B Organic light emitting device 株式会社LG化学 2024-08-02 CN disclosed
CN-118201642-A Linker for antibody drug conjugates 奥隆制药 2024-06-14 CN disclosed
WO-2024064745-A1 SYNTHESIS OF RELDESEMTIV CYTOKINETICS, INCORPORATED (US) 2024-03-28 WO disclosed
CN-113646915-B Organic light emitting device 株式会社LG化学 2024-03-19 CN disclosed
CN-117619175-A Nanofiltration membrane and preparation method and application thereof 清华大学 2024-03-01 CN disclosed
CN-112469719-B Heterocondensed pyridone compounds and their use as IDH inhibitors 内尔维亚诺医疗科学公司 2024-01-23 CN disclosed
WO-2023242598-A1 BIFUNCTIONAL MOLECULES FOR TARGETED PROTEIN DEGRADATION AMPHISTA THERAPEUTICS LIMITED (GB) 2023-12-21 WO disclosed
CN-117098762-A Process for preparing bicyclic ketone compounds 基因泰克公司 2023-11-21 CN disclosed
CN-111936506-B Compound and organic light-emitting element comprising same 株式会社LG化学 2023-11-07 CN disclosed
CN-116940354-A Fused heteroaryl compounds and their use as CaMKII inhibitors 卡都瑞恩医药股份有限公司 2023-10-24 CN disclosed
CN-113924665-B Organic light emitting device 株式会社LG化学 2023-09-29 CN disclosed
CN-116675861-A Preparation method of modified polyethersulfone/polyetherimide polymer alloy 深圳先进技术研究院 2023-09-01 CN disclosed
CN-116457335-A Process for preparing 3-fluoro-5- (((1S, 2 aR) -1,3, 4-pentafluoro-2 a-hydroxy-2, 2a,3, 4-tetrahydro-1H-cyclopenta [ cd ] inden-7-yl) oxy) benzonitrile and polymorphs thereof 尼坎治疗公司 2023-07-18 CN disclosed
CN-111655697-B Compound and organic light-emitting diode comprising same 株式会社LG化学 2023-05-19 CN disclosed
CN-111479857-B Multilayer composite material comprising a specific polycarbonate composition as matrix material 科思创德国股份有限公司 2023-04-04 CN disclosed
CN-111465635-B Multilayer composite material comprising a specific polycarbonate composition as matrix material 科思创德国股份有限公司 2023-04-04 CN disclosed
US-20220145037-A1 METHODS OF PREPARATION OF OMNIPHOBIC SURFACES NUTECH VENTURES (US) 2022-05-12 US disclosed
US-11312688-B2 Pyrazole compound SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-04-26 US disclosed
CN-109851531-B Preparation method of (N-methyl perfluoroalkyl sulfonamide) ethyl acrylate 武汉松石科技股份有限公司 2021-06-08 CN disclosed
WO-2021030670-A1 ARTICLE INCLUDING ELASTOMERIC CORE AND VAPOR DEPOSITED FLUOROELASTOMERIC COATING QUADION LLC (US) 2021-02-18 WO disclosed
EP-3638654-B1 MELT ADDITIVE COMPOUNDS, METHODS OF USING THE SAME, AND ARTICLES AND COMPOSITIONS INCLUDING THE SAME 3M INNOVATIVE PROPERTIES CO (US) 2021-01-27 EP disclosed
CN-112028902-A Novel heterocyclic compound and organic light-emitting element using same 株式会社LG化学 2020-12-04 CN disclosed
US-10794853-B2 Methods for depositing polymer layer for sensor applications via hot wire chemical vapor deposition APPLIED MATERIALS, INC. (US) 2020-10-06 US disclosed
US-20200308119-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2020-10-01 US disclosed
US-10723703-B2 Pyrazole compound SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-07-28 US disclosed
CN-111349103-A Heterocyclic compound and organic light-emitting element using same 株式会社LG化学 2020-06-30 CN disclosed
EP-3551780-A1 METHODS FOR DEPOSITING POLYMER LAYER FOR SENSOR APPLICATIONS VIA HOT WIRE CHEMICAL VAPOR DEPOSITION Applied Materials, Inc. (US) 2019-10-16 EP disclosed
US-20190218203-A1 Neuroprotective Compounds and Use Thereof UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2019-07-18 US disclosed
US-20190084938-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2019-03-21 US disclosed
US-10183913-B2 Pyrazole compound SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2019-01-22 US disclosed
EP-3050872-B1 Fluorinated sulfonamide as electrolyte (co-)solvent for lithium-ion batteries UNIV MUENSTER WESTFAELISCHE WILHELMS (DE) 2018-10-03 EP disclosed
US-10087146-B2 Pyrazole compound SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2018-10-02 US disclosed
US-20180273489-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2018-09-27 US disclosed
US-20180164245-A1 METHODS FOR DEPOSITING POLYMER LAYER FOR SENSOR APPLICATIONS VIA HOT WIRE CHEMICAL VAPOR DEPOSITION APPLIED MATERIALS, INC. 2018-06-14 US disclosed
US-9976165-B2 Methods for increasing molecular diversity of polyketides and non-ribosomal proteins ISOMERASE THERAPEUTICS, LTD. (GB) 2018-05-22 US disclosed
US-9902713-B2 Neuroprotective compounds and use thereof BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2018-02-27 US disclosed
US-9828722-B2 Blends of fluoroalkyl-containing ester oligomers with polycarbodiimide(s) 3M INNOVATIVE PROPERTIES COMPANY (US) 2017-11-28 US disclosed
WO-2017189215-A1 ARTICLES SUBJECT TO ICE FORMATION COMPRISING A REPELLENT SURFACE COMPRISING A FLUOROCHEMICAL MATERIAL 3M INNOVATIVE PROPERTIES COMPANY (US) 2017-11-02 WO disclosed
US-20170217902-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2017-08-03 US disclosed
US-9663472-B2 Pyrazole compound SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-05-30 US disclosed
US-20170101659-A1 METHODS FOR INCREASING MOLECULAR DIVERSITY OF POLYKETIDES AND NON-RIBOSOMAL PROTEINS Isomerase Therapeutics Ltd. (GB) 2017-04-13 US disclosed
WO-2017016943-A1 METHOD FOR RECOVERING SULFONIC ESTERS OR SULFONYL HALIDES FROM SALTS OF SULFONIC ACIDS SOLVAY SPECIALTY POLYMERS ITALY S.P.A. (IT) 2017-02-02 WO disclosed
US-9505773-B2 Rapamycin analogues and their pharmaceutical use Isomerase Therapeutics Ltd. (GB) 2016-11-29 US disclosed
US-20160272619-A1 Neuroprotective Compounds and Use Thereof UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2016-09-22 US disclosed
EP-3068388-A2 NEUROPROTECTIVE COMPOUNDS AND USE THEREOF Board of Regents of the University of Texas System (US) 2016-09-21 EP disclosed
EP-3050872-A1 Fluorinated sulfonamide as electrolyte (co-)solvent for lithium-ion batteries Westfälische Wilhelms-Universität Münster (DE) 2016-08-03 EP disclosed
US-20160176893-A1 RAPAMYCIN ANALOGUES AND THEIR PHARMACEUTICAL USE ISOMERASE THERAPEUTICS, LTD. (GB) 2016-06-23 US disclosed
EP-2594559-B1 PYRAZOLE COMPOUND SUMITOMO DAINIPPON PHARMA CO LTD (JP) 2016-02-24 EP disclosed
EP-2417184-B1 PROCESS FOR THE MANUFACTURE OF FUNCTIONAL PFPE DERIVATIVE SOLVAY SPECIALTY POLYMERS IT (IT) 2016-01-06 EP disclosed
WO-2015070234-A9 NEUROPROTECTIVE COMPOUNDS AND USE THEREOF BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-12-10 WO disclosed
EP-2091926-B1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG (CH) 2015-10-21 EP disclosed
EP-2638116-B1 OPTICAL DEVICE SURFACE TREATMENT PROCESS AND SMUDGE-RESISTANT ARTICLE PRODUCED THEREBY 3M INNOVATIVE PROPERTIES CO (US) 2015-08-12 EP disclosed
US-8993116-B2 Blends of fluoroalkyl-containing ester oligomers with polydicarbodiimide(S) 3M INNOVATIVE PROPERTIES COMPANY (US) 2015-03-31 US disclosed
US-8975445-B2 Process for the manufacture of functional PFPE derivative SOLVAY SPECIALTY POLYMERS ITALY S.P.A. (IT) 2015-03-10 US disclosed
US-8906454-B2 Methods for depositing metal-polymer composite materials atop a substrate APPLIED MATERIALS, INC. (US) 2014-12-09 US disclosed
US-20140315971-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2014-10-23 US disclosed
US-8809383-B2 Pyrazole compound DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2014-08-19 US disclosed
US-20140227191-A1 L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2014-08-14 US disclosed
US-8735599-B2 Substituted imidazole derivates NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2014-05-27 US disclosed
US-20140031406-A1 PYRAZOLE COMPOUND DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2014-01-30 US disclosed
US-8569353-B2 Pyrazole compound DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-10-29 US disclosed
EP-2638116-A1 OPTICAL DEVICE SURFACE TREATMENT PROCESS AND SMUDGE-RESISTANT ARTICLE PRODUCED THEREBY 3M Innovative Properties Company (US) 2013-09-18 EP disclosed
EP-2396431-B1 LEATHER ARTICLE HAVING IMPROVED SOIL RESISTANCE AND METHOD OF MAKING SAME 3M INNOVATIVE PROPERTIES CO (US) 2013-09-11 EP disclosed
US-20130229378-A1 OPTICAL DEVICE SURFACE TREATMENT PROCESS AND SMUDGE-RESISTANT ARTICLE PRODUCED THEREBY 3M INNOVATIVE PROPERTIES COMPANY 2013-09-05 US disclosed
EP-2594559-A1 PYRAZOLE COMPOUND Dainippon Sumitomo Pharma Co., Ltd. (JP) 2013-05-22 EP disclosed
US-20130116296-A1 PYRAZOLE COMPOUND NEUROINNOVATECH APS (DK) 2013-05-09 US disclosed
WO-2013039862-A2 METHODS FOR DEPOSITING METAL-POLYMER COMPOSITE MATERIALS ATOP A SUBSTRATE APPLIED MATERIALS, INC. (US) 2013-03-21 WO disclosed
US-20130065401-A1 METHODS FOR DEPOSITING METAL-POLYMER COMPOSITE MATERIALS ATOP A SUBSTRATE APPLIED MATERIALS, INC. (US) 2013-03-14 US disclosed
EP-1765789-B1 N-(1-(1-BENZYL-4-PHENYL-1H-IMIDAZOL-2-YL)-2,2-DIMETHYLPROPYL)BENZAMIDE DERIVATIVES AND RELATED COMPOUNDS AS KINESIN SPINDLE PROTEIN (KSP) INHIBITORS FOR THE TREATMENT OF CANCER NOVARTIS AG (CH) 2013-02-27 EP disclosed
US-20130017196-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES CHIRON CORPORATION 2013-01-17 US disclosed
US-8324417-B2 Process for the preparation of (S)-2-amino-5-cyclopropyl-4,4-difluoropentanoic acid and alkyl esters and acid salts thereof VIROBAY, INC. (US) 2012-12-04 US disclosed
US-8318791-B2 Substituted imidazole derivatives NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2012-11-27 US disclosed
WO-2012105586-A1 PERFLUOROBUTANE SULFONYL FLUORIDE, POTASSIUM PERFLUOROBUTANE SULFONATE SALT, AND METHOD FOR PRODUCING PERFLUOROBUTANE SULFONYL FLUORIDE 三菱マテリアル株式会社 (JP) 2012-08-09 WO disclosed
EP-1743014-B1 FLUORINATED SULFONAMIDE SURFACTANTS FOR AQUEOUS CLEANING SOLUTIONS 3M INNOVATIVE PROPERTIES CO (US) 2012-06-27 EP disclosed
WO-2012064649-A1 OPTICAL DEVICE SURFACE TREATMENT PROCESS AND SMUDGE-RESISTANT ARTICLE PRODUCED THEREBY 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-05-18 WO disclosed
US-8129358-B2 Substituted pyrazole and triazole compounds as KSP inhibitors NOVARTIS AG (CH) 2012-03-06 US disclosed
EP-2417184-A1 PROCESS FOR THE MANUFACTURE OF FUNCTIONAL PFPE DERIVATIVE Solvay Solexis S.p.A. (IT) 2012-02-15 EP disclosed
US-20120028858-A1 Process for the manufacture of functional PFPE derivative SOLVAY SOLEXIS S.P.A. (IT) 2012-02-02 US disclosed
EP-1912972-B1 SUBSTITUTED IMIDAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG (CH) 2011-09-28 EP disclosed
EP-1832574-B1 Methods of making an antistatic agent SABIC INNOVATIVE PLASTICS IP (NL) 2011-08-10 EP disclosed
US-7985723-B2 Fluorinated sulfonamide surfactants for aqueous cleaning solutions 3M INNOVATIVE PROPERTIES COMPANY (US) 2011-07-26 US disclosed
US-20110064673-A1 New L-Glutamic acid and L-Glutamine derivative (III), use thereof and method for obtaining them PIRAMAL IMAGING SA (CH) 2011-03-17 US disclosed
US-7902240-B2 Kinesin spindle protein (KSP); anticancer agents; antiproliferative agents; e.g. N-((S)-3-amino-4-fluorobutyl)-N ((R)-1-(1-benzyl-3-(2,5-difluorophenyl)-1H-1,2,4-triazol-5-yl)-2,2-dimethylpropyl)nicotinamide NOVARTIS AG (CH) 2011-03-08 US disclosed
WO-2011022429-A2 PROCESS FOR THE PREPARATION OF (S)-2-AMINO-5-CYCLOPROPYL-4,4-DIFLUOROPENTANOIC ACID AND ALKYL ESTERS AND ACID SALTS THEREOF VIROBAY, INC. (US) 2011-02-24 WO disclosed
US-20110046406-A1 PROCESS FOR THE PREPARATION OF (S)-2-AMINO-5-CYCLOPROPYL-4,4-DIFLUOROPENTANOIC ACID AND ALKYL ESTERS AND ACID SALTS THEREOF VIROBAY, INC. (US) 2011-02-24 US disclosed
EP-2282981-A1 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM Bayer Schering Pharma Aktiengesellschaft (DE) 2011-02-16 EP disclosed
US-20100320416-A1 FLUORINATED SULFONAMIDE SURFACTANTS FOR AQUEOUS CLEANING SOLUTIONS 3M INNOVATIVE PROPERTIES COMPANY 2010-12-23 US disclosed
US-20100278751-A1 RADIOLABELED 2-AMINO-4-ALKYL-6-(HALOALKYL)PYRIDINE COMPOUNDS AND THEIR USE IN DIAGNOSTIC IMAGING WASHINGTON UNIVERSITY (US) 2010-11-04 US disclosed
WO-2010115855-A1 PROCESS FOR THE MANUFACTURE OF FUNCTIONAL PFPE DERIVATIVE SOLVAY SOLEXIS S.P.A. (IT) 2010-10-14 WO disclosed
US-7811978-B2 Fluorinated sulfonamide surfactants for aqueous cleaning solutions 3M INNOVATIVE PROPERTIES COMPANY (US) 2010-10-12 US disclosed
US-20100227148-A1 WATER- AND OIL-REPELLENCY IMPARTING ESTER OLIGOMERS COMPRISING PERFLUOROALKYL MOIETIES 3M INNOVATIVE PROPERTIES COMPANY 2010-09-09 US disclosed
EP-1737814-B1 METHODS OF MAKING AN ANTISTATIC AGENT SABIC INNOVATIVE PLASTICS IP (NL) 2010-06-09 EP disclosed
EP-2167462-A2 WATER- AND OIL-REPELLENCY IMPARTING ESTER OLIGOMERS COMPRISING PERFLUOROALKYL MOIETIES 3M Innovative Properties Company (US) 2010-03-31 EP disclosed
WO-2009141090-A9 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-03-25 WO disclosed
US-20100034813-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG (CH) 2010-02-11 US disclosed
US-7626040-B2 Substituted imidazole compounds as KSP inhibitors NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2009-12-01 US disclosed
WO-2009141090-A1 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-11-26 WO disclosed
US-20090258016-A1 Substituted imidazole derivatives WANG WEIBO 2009-10-15 US disclosed
EP-2091926-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS Novartis AG (CH) 2009-08-26 EP disclosed
US-7576221-B2 N-(3-aminopropyl)-N-[(1R)-1-(1-benzyl-4-phenyl-1H-imidazol-2-yl)-2-methylpropyl]-4-methylbenzamide; kinesin-related proteins (KRP) inhibitors; anticarcinogenic agent NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2009-08-18 US disclosed
WO-2008154414-A2 WATER- AND OIL-REPELLENCY IMPARTING ESTER OLIGOMERS COMPRISING PERFLUOROALKYL MOIETIES 3M INNOVATIVE PROPERTIES COMPANY (US) 2008-12-18 WO disclosed
US-20080306238-A1 WATER- AND OIL-REPELLENCY IMPARTING ESTER OLIGOMERS COMPRISING PERFLUOROALKYL MOIETIES 3M INNOVATIVE PROPERTIES COMPANY 2008-12-11 US disclosed
US-7449572-B2 Process and intermediates for preparing 17-halogenated 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2008-11-11 US disclosed
US-20080269526-A1 METHODS OF MAKING AN ANTISTATIC AGENT SAIC INNOVATIVE PLASTICS, IP B.V. (NL) 2008-10-30 US disclosed
WO-2008122611-A1 PROCESS FOR THE MANUFACTURE OF FLUORINATED COMPOUNDS Solvay (Société Anonyme) (BE) 2008-10-16 WO disclosed
US-7429628-B2 Method of making a thermoplastic composition containing an antistatic agent SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2008-09-30 US disclosed
US-20080200462-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG 2008-08-21 US disclosed
WO-2008063912-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG (CH) 2008-05-29 WO disclosed
EP-1912972-A1 SUBSTITUTED IMIDAZOLE COMPOUNDS AS KSP INHIBITORS Novartis AG (CH) 2008-04-23 EP disclosed
US-20080081857-A1 METHOD OF MAKING A THERMOPLASTIC COMPOSITION CONTAINING AN ANTISTATIC AGENT SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2008-04-03 US disclosed
US-20080078747-A1 FLUORINATED SULFONAMIDE SURFACTANTS FOR AQUEOUS CLEANING SOLUTIONS 3M INNOVATIVE PROPERTIES COMPANY 2008-04-03 US disclosed
US-20080015377-A1 METHODS OF MAKING AN ANTISTATIC AGENT GENERAL ELECTRIC COMPANY (US) 2008-01-17 US disclosed
US-7309735-B2 One-step, phosphonium haloalkylsulfonate antistatic agent by combining an alkyl sulfonate salt of lithium or Sodium with a tetraalkylphosphonium halogen in an aqueous medium; simple mixing of the reactants results in a precipitation of the anti-static molecule in high yield GENERAL ELECTRIC COMPANY (US) 2007-12-18 US disclosed
US-7294610-B2 Fluorinated sulfonamide surfactants for aqueous cleaning solutions 3M INNOVATIVE PROPERTIES COMPANY (US) 2007-11-13 US disclosed
EP-1832574-A2 Methods of making an antistatic agent General Electric Company (US) 2007-09-12 EP disclosed
EP-1812502-A2 METHODS OF MAKING AN ANTISTATIC AGENT General Electric Company (US) 2007-08-01 EP disclosed
US-20070129472-A1 METHOD OF MAKING A THERMOPLASTIC COMPOSITION CONTAINING AN ANTISTATIC AGENT SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2007-06-07 US disclosed
US-7211690-B2 Methods of making an antistatic agent GENERAL ELECTRIC COMPANY (US) 2007-05-01 US disclosed
EP-1765789-A1 N-(1-(1-BENZYL-4-PHENYL-1H-IMIDAZOL-2-YL)-2,2-DIMETHYLPROPYL)BENZAMIDE DERIVATIVES AND RELATED COMPOUNDS AS KINESIN SPINDLE PROTEIN (KSP) INHIBITORS FOR THE TREATMENT OF CANCER Novartis Vaccines and Diagnostics, Inc. (US) 2007-03-28 EP disclosed
WO-2007021794-A1 SUBSTITUTED IMIDAZOLE COMPOUNDS AS KSP INHIBITORS NOVARTIS AG (CH) 2007-02-22 WO disclosed
US-20070037853-A1 N-(3-aminopropyl)-N-{1-[1-benzyl-4-(3-chlorophenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholine-4-carboxamide and derivatives; kinesin spindle protein (KSP) inhibitors; anticarcinogenic agents; antimiotic; gene expression inhibition NOVARTIS VACCINES AND DIAGNOSTICS INC. 2007-02-15 US disclosed
EP-1743014-A1 FLUORINATED SULFONAMIDE SURFACTANTS FOR AQUEOUS CLEANING SOLUTIONS 3M Innovative Properties Company (US) 2007-01-17 EP disclosed
EP-1737814-A2 METHODS OF MAKING AN ANTISTATIC AGENT GENERAL ELECTRIC COMPANY (US) 2007-01-03 EP disclosed
WO-2006052522-A2 METHODS OF MAKING AN ANTISTATIC AGENT GENERAL ELECTRIC COMPANY (US) 2006-05-18 WO disclosed
US-20060100327-A1 Methods of making an antistatic agent CITIBANK, N.A., AS COLLATERAL AGENT 2006-05-11 US disclosed
US-20060009472-A1 Substituted imidazole derivatives CHIRON CORPORATION 2006-01-12 US disclosed
WO-2006002236-A1 N- (1- (1-BENZYL -4-PHENYL-1H-IMIDAZOL-2-YL) -2,2-DYMETHYLPROPYL) BENZAMIDE DERIVATIVES AND RELATED COMPOUNDS AS KINESIN SPINDLE PROTEIN (KSP) INHIBITORS FOR THE TREATMENT OF CANCER NOVARTIS VACCINES AND DIAGNOSTICS INC. (US) 2006-01-05 WO disclosed
WO-2005100307-A2 METHODS OF MAKING AN ANTISTATIC AGENT GENERAL ELECTRIC COMPANY (US) 2005-10-27 WO disclosed
US-20050228194-A1 Methods of making an antistatic agent SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2005-10-13 US disclosed
WO-2005095567-A1 FLUORINATED SULFONAMIDE SURFACTANTS FOR AQUEOUS CLEANING SOLUTIONS 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-10-13 WO disclosed
US-20050197273-A1 Fluorinated sulfonamide surfactants for aqueous cleaning solutions 3M INNOVATIVE PROPERTIES COMPANY 2005-09-08 US disclosed
US-20040224933-A1 Novel process and intermediates for preparing 17-halogenated 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2004-11-11 US disclosed
EP-1131270-B1 PROCESS FOR CONVERTING AN ALCOHOL TO THE CORRESPONDING FLUORIDE 3M INNOVATIVE PROPERTIES CO (US) 2004-04-07 EP disclosed
US-6566542-B2 Such as 17-alpha-fluoro-11-beta-(4-(2-(1-piperidinyl) ethoxy) phenyl)-estra-1,3,5(10)-trien-3-ol for treatment of osteoporosis and cardiovascular protection; side effect reduction; provides alternative to estradiol AVENTIS PHARMA S.A. (FR) 2003-05-20 US disclosed
US-20030031844-A1 Layer of perfluoroalkyl sulfonic ammonium acid salts, phosphonium acid salts and sulfonium acid salts and polycarbonate (co)polymers BAYER AKTIENGESELLSCHAFT (DE) 2003-02-13 US disclosed
US-20030022874-A1 New 17-halogenated 19-nor steroids, preparation process and intermediates, use as medicaments and the pharmaceutical compositions containing them BOUALI YASMINA (FR) 2003-01-30 US disclosed
US-6423700-B1 17-halogenated 19-nor steroids, method and intermediates for preparing same, use as medicines and pharmaceutical compositions containing same AVENTIS PHARMA S.A. (FR) 2002-07-23 US disclosed
US-6365068-B1 IN SOLVENT HYDRO-QUEBEC (CA) 2002-04-02 US disclosed
EP-1131270-A1 PROCESS FOR CONVERTING AN ALCOHOL TO THE CORRESPONDING FLUORIDE 3M Innovative Properties Company (US) 2001-09-12 EP disclosed
US-6248889-B1 FORMING MIXTURE COMPRISING AT LEAST ONE FLUORINATED, SATURATED ALIPHATIC OR ALICYCLIC SULFONYL FLUORIDE AND AT LEAST ONE PRIMARY OR SECONDARY ALCOHOL, ADDING MOLAR EXCESS OF STRONG, APROTIC, NON-NUCLEOPHILIC HINERED ORGANIC BASE 3M INNOVATIVE PROPERTIES COMPANY 2001-06-19 US disclosed
US-6171522-B1 Heterocyclic aromatic anion salts, and their uses as ionic conducting materials Hydro-Qu{acute over (e)}bec (CA) 2001-01-09 US disclosed
EP-0735992-B1 METHOD OF CONVERTING HYDROXYL GROUPS INTO CORRESPONDING FLUORO COMPOUNDS BAYER AG (DE) 2001-01-03 EP disclosed
WO-2000031003-A1 PROCESS FOR CONVERTING AN ALCOHOL TO THE CORRESPONDING FLUORIDE 3M INNOVATIVE PROPERTIES COMPANY (US) 2000-06-02 WO disclosed
EP-0735992-A1 METHOD OF CONVERTING HYDROXYL GROUPS INTO CORRESPONDING FLUORO COMPOUNDS BAYER AG (DE) 1996-10-09 EP disclosed
WO-1996013474-A1 METHOD OF CONVERTING HYDROXYL GROUPS INTO CORRESPONDING FLUORO COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 1996-05-09 WO disclosed
EP-0339284-B1 Fluorine-containing dielectric media and capacitors employing such media ATOCHEM NORTH AMERICA (US) 1994-06-29 EP disclosed
US-4899249-A Fluorine-containing dielectric media and capacitors employing such media PENNWALT CORPORATION (US) 1990-02-06 US disclosed
EP-0339284-A1 Fluorine-containing dielectric media and capacitors employing such media ATOCHEM NORTH AMERICA, INC. (a Pennsylvania corp.) (US) 1989-11-02 EP disclosed
US-4168277-A QUATERNIZATION OF TRIETHYLAMINE WITH AN ETHOXY SILANE, SALT FORMAT BAYER AKTIENGESELLSCHAFT (DE) 1979-09-18 US disclosed
US-3970586-A Perfluoroalkane sulfonamido-alkane phosphonic and phosphonic acid derivatives BAYER AKTIENGESELLSCHAFT (DT) 1976-07-20 US disclosed
US-3970586-A Perfluoroalkane sulfonamido-alkane phosphonic and phosphonic acid derivatives BAYER AKTIENGESELLSCHAFT (DT) 1976-07-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (31 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070129472-A1 METHOD OF MAKING A THERMOPLASTIC COMPOSITION CONTAINING AN ANTISTATIC AGENT LBR, RPS4X, RER1 CA2 251/4885CA1 113/4885MMP1 1501/4885
US-20190218203-A1 Neuroprotective Compounds and Use Thereof NLN, GAP43, BDNF CA2 3901/4885CA1 793/4885MMP1 2735/4885
US-20110046406-A1 PROCESS FOR THE PREPARATION OF (S)-2-AMINO-5-CYCLOPROPYL-4,4-DIFLUOROPENTANOIC ACID AND ALKYL ESTERS AND ACID SALTS THEREOF DNPEP, CTRL, CTSS CA2 398/4885CA1 118/4885MMP1 498/4885
US-20140315971-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20070037853-A1 N-(3-aminopropyl)-N-{1-[1-benzyl-4-(3-chlorophenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholine-4-carboxamide and derivatives; kinesin spindle protein (KSP) inhibitors; anticarcinogenic agents; antimiotic; gene expression inhibition KIF5B, KIF2C, KIF18B CA2 2598/4885CA1 4331/4885MMP1 3040/4885
US-20120028858-A1 Process for the manufacture of functional PFPE derivative PF4, PFAS, PFKP CA2 1127/4885CA1 1650/4885MMP1 3312/4885
US-20060009472-A1 Substituted imidazole derivatives ABCG2, CYP2C19, AADAC CA2 1526/4885CA1 3855/4885MMP1 3200/4885
US-20040224933-A1 Novel process and intermediates for preparing 17-halogenated 19-norsteroid compounds CYP17A1, HSD17B7, HSD3B1 CA2 4805/4885CA1 3084/4885MMP1 4443/4885
US-10183913-B2 Pyrazole compound HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20100034813-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS CYP3A43, ABCG2, CYP3A7 CA2 3748/4885CA1 3975/4885MMP1 4370/4885
US-20170217902-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20030022874-A1 New 17-halogenated 19-nor steroids, preparation process and intermediates, use as medicaments and the pharmaceutical compositions containing them HSD17B7, CYP11B1, CYP11B2 CA2 4293/4885CA1 3926/4885MMP1 4380/4885
US-11312688-B2 Pyrazole compound HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20130116296-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20200308119-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20110064673-A1 New L-Glutamic acid and L-Glutamine derivative (III), use thereof and method for obtaining them GLUL, GATD3, QPCT CA2 981/4885CA1 231/4885MMP1 4724/4885
US-20140227191-A1 L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM GLUL, GATD3, QPCT CA2 905/4885CA1 203/4885MMP1 4614/4885
US-20080200462-A1 SUBSTITUTED PYRAZOLE AND TRIAZOLE COMPOUNDS AS KSP INHIBITORS CYP3A43, ABCG2, CYP3A7 CA2 3748/4885CA1 3975/4885MMP1 4370/4885
US-20090258016-A1 Substituted imidazole derivatives ABCG2, CYP2C19, AADAC CA2 1526/4885CA1 3855/4885MMP1 3200/4885
US-20080015377-A1 METHODS OF MAKING AN ANTISTATIC AGENT GPX1, GPX4, PRDX1 CA2 14/4885CA1 12/4885MMP1 273/4885
US-20160272619-A1 Neuroprotective Compounds and Use Thereof NLN, BDNF, CASP3 CA2 4010/4885CA1 1358/4885MMP1 2318/4885
US-20050228194-A1 Methods of making an antistatic agent MTX1, GPX4, CA2 CA2 3/4885CA1 16/4885MMP1 522/4885
US-10723703-B2 Pyrazole compound HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20160176893-A1 RAPAMYCIN ANALOGUES AND THEIR PHARMACEUTICAL USE FKBP1A, FKBP1B, FKBP2 CA2 3673/4885CA1 4726/4885MMP1 1564/4885
US-20180273489-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20080269526-A1 METHODS OF MAKING AN ANTISTATIC AGENT PGM2, CA6, NHERF1 CA2 7/4885CA1 38/4885MMP1 886/4885
US-20130017196-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES ABCG2, CYP2C19, AADAC CA2 1526/4885CA1 3855/4885MMP1 3200/4885
US-20100278751-A1 RADIOLABELED 2-AMINO-4-ALKYL-6-(HALOALKYL)PYRIDINE COMPOUNDS AND THEIR USE IN DIAGNOSTIC IMAGING NOS2, NOS3, NOS1 CA2 739/4885CA1 1937/4885MMP1 1706/4885
US-20190084938-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-10087146-B2 Pyrazole compound HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885
US-20140031406-A1 PYRAZOLE COMPOUND HTR2C, HTR3B, HTR3A CA2 2270/4885CA1 1971/4885MMP1 4534/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.