Ibacitabine

Ibacitabine

SCHEMBL225403

Nc1nc(=O)n([C@H]2CC(O)[C@@H](CO)O2)cc1I

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 6/20 0.63
ADRB1 P08588 1/20 0.63
TK1 P04183 2/20 0.60
DNMT3B Q9UBC3 2/20 0.54
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
PNP P00491 1/20 0.49
TP53 P04637 1/20 0.49
HTT P42858 1/20 0.49
PDE4D Q08499 1/20 0.49
PDE3A Q14432 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
FPR2 P25090 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ibacitabine SCHEMBL5981937 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL21423094 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL5981939 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL13812993 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL887475 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL225402 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
Ibacitabine SCHEMBL244921 1.00 DNMT1 (0.63) DNMT1ADRB1TK1DNMT3BLMNA
SCHEMBL1635378 0.91 DNMT1 (0.52) DNMT1ADRB1TK1DNMT3BFPR2
SCHEMBL1635376 0.91 DNMT1 (0.52) DNMT1ADRB1TK1DNMT3BFPR2
Ibacitabine SCHEMBL9710365 0.91 DNMT1 (0.54) DNMT1ADRB1TK1DNMT3BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 508 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4271389-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA Rejuvenation Technologies Inc. (US) 2023-11-08 EP claimed
WO-2022147039-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES INC. (US) 2022-07-07 WO claimed
US-20220096649-A1 IMMUNOMODULATING POLYNUCLEOTIDE CONJUGATES AND METHODS OF USE HORIZON TECHNOLOGY FINANCE CORPORATION 2022-03-31 US claimed
US-11203611-B2 Immunomodulating polynucleotides, antibody conjugates thereof, and methods of their use TOLLNINE, INC. (US) 2021-12-21 US claimed
US-11021497-B2 Compositions and methods for synthesis of phosphorylated molecules THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-06-01 US claimed
US-20200239500-A1 Compositions and Methods for Synthesis of Phosphorylated Molecules THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-07-30 US claimed
WO-2020081744-A1 IMMUNOMODULATING POLYNUCLEOTIDE CONJUGATES AND METHODS OF USE TOLLNINE, INC. (US) 2020-04-23 WO claimed
EP-3610022-A1 IMMUNOMODULATING POLYNUCLEOTIDES, ANTIBODY CONJUGATES THEREOF, AND METHODS OF THEIR USE Tollnine, Inc. (US) 2020-02-19 EP claimed
CN-110770345-A Immunomodulatory polynucleotides, antibody conjugates, and methods of use thereof 托尔奈公司 2020-02-07 CN claimed
WO-2019195494-A1 COMPOSITIONS AND METHODS FOR SYNTHESIS OF PHOSPHORYLATED MOLECULES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-10-10 WO claimed
WO-2018189382-A1 IMMUNOMODULATING POLYNUCLEOTIDES, ANTIBODY CONJUGATES THEREOF, AND METHODS OF THEIR USE SOLSTICE BIOLOGICS, LTD. (IE) 2018-10-18 WO claimed
EP-3186387-A1 METHOD OF DETERMINING THE ACTIVITY OF ENZYMES CONVERTING CYTOSINE DERIVATIVES TO URACIL DERIVATIVES IN CELLS, TISSUES AND ORGANISMS Univerzita Palackého v Olomouci (CZ) 2017-07-05 EP claimed
WO-2016029889-A1 METHOD OF DETERMINING THE ACTIVITY OF ENZYMES CONVERTING CYTOSINE DERIVATIVES TO URACIL DERIVATIVES IN CELLS, TISSUES AND ORGANISMS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-03-03 WO claimed
US-20090325897-A1 DESIGNER THERAPY OF PANCREATIC TUMORS UNIVERSITY OF MIAMI (US) 2009-12-31 US claimed
US-7598230-B2 For the treatment of viral infections, microbial infections, and proliferative disorders; contain di- or triphosphate moeity mimetics, such as those containing boron anions BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2009-10-06 US claimed
WO-2008085611-A2 DESIGNER THERAPHY OF PANCREATIC TUMORS UNIVERSITY OF MIAMI (US) 2008-07-17 WO claimed
US-20070259832-A1 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2007-11-08 US claimed
US-20040059104-A1 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2004-03-25 US claimed
EP-0806956-B1 USE OF 5'SUBSTITUTED NUCLEOSIDES TO PROVIDE RESISTANCE IN CYTOSTATIC TREATMENT RESPROTECT GMBH (DE) 2002-08-28 EP claimed
EP-4746905-A1 RSV VACCINE Astrazeneca AB (SE) 2026-05-27 EP disclosed
WO-2026104647-A1 VACCINE ASTRAZENECA AB (SE) 2026-05-21 WO disclosed
WO-2026106815-A1 Z-INDUCING CHIMERA COMPOSITION RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2026-05-21 WO disclosed
US-20260109728-A1 IMMUNOMODULATING POLYNUCLEOTIDES, ANTIBODY CONJUGATES THEREOF, AND METHODS OF THEIR USE TALLAC THERAPEUTICS INC (US) 2026-04-23 US disclosed
US-12605397-B2 Deoxy-cytidine or uridine derivatives for use in cancer therapies TETRAGON BIOSCIENCE LTD. (IL) 2026-04-21 US disclosed
US-12606863-B2 Bioluminescent detection of DNA synthesis PROMEGA CORPORATION (US) 2026-04-21 US disclosed
US-12584168-B2 Sample preparation method OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2026-03-24 US disclosed
US-20260066042-A1 METHODS AND SYSTEMS FOR HIGH-THROUGHPUT MOLECULAR ANALYSIS OPENTRONS LABWORKS INC (US) 2026-03-05 US disclosed
US-12503730-B2 Detectable nucleotide analogues THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-12-23 US disclosed
US-20250313889-A1 SAMPLE PREPARATION METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2025-10-09 US disclosed
US-20250283094-A1 Modified Nucleosides SOMALOGIC OPERATING CO., INC. (US) 2025-09-11 US disclosed
EP-4611757-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS Ramirez, Christina, M. (US) 2025-09-10 EP disclosed
US-20250263678-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES, INC. (US) 2025-08-21 US disclosed
EP-4591940-A2 DEOXY- CYTIDINE DERIVATIVES FOR USE IN CANCER THERAPIES Hemispherian AS (NO) 2025-07-30 EP disclosed
US-20250236911-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-07-24 US disclosed
EP-4233879-B1 DEOXY- CYTIDINE DERIVATIVES FOR USE IN CANCER THERAPIES HEMISPHERIAN AS (NO) 2025-07-23 EP disclosed
US-12351598-B2 Immunomodulating polynucleotides, antibody conjugates thereof, and methods of their use Tallac Therapeutics, Inc. (US) 2025-07-08 US disclosed
WO-2025125630-A1 METHOD FOR BIOPROTAC DESIGN MEDIMMUNE LIMITED (GB) 2025-06-19 WO disclosed
EP-3443001-B1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS INC (US) 2025-04-30 EP disclosed
US-20250041400-A1 RSV VACCINE ASTRAZENECA PHARMACEUTICALS LP 2025-02-06 US disclosed
WO-2025017142-A1 RSV VACCINE ASTRAZENECA AB (SE) 2025-01-23 WO disclosed
WO-2024238558-A1 USE OF IMMUNOMODULATING TARGETED POLYNUCLEOTIDE CONJUGATES FOR USE WITH IMMUNE HONING AGENT Tallac Therapeutics, Inc. (US) 2024-11-21 WO disclosed
US-20240382610-A1 NECTIN-4 ANTIBODIES AND CONJUGATES HORIZON TECHNOLOGY FINANCE CORPORATION 2024-11-21 US disclosed
US-20240376536-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-11-14 US disclosed
US-20240374746-A1 SIRP-ALPHA ANTIBODIES AND CONJUGATES HORIZON TECHNOLOGY FINANCE CORPORATION 2024-11-14 US disclosed
US-20240342182-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS ELIAN LLC (US) 2024-10-17 US disclosed
US-20240342200-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS ELIAN LLC (US) 2024-10-17 US disclosed
US-20240343753-A1 THERAPEUTIC COMPOUNDS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2024-10-17 US disclosed
US-20240287528-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2024-08-29 US disclosed
US-12054768-B2 Methods for detecting agglutination and compositions for use in practicing the same THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-08-06 US disclosed
US-20240218374-A1 Nucleic Acid Compounds That Bind Coronavirus Proteins SOMALOGIC OPERATING CO., INC. (US) 2024-07-04 US disclosed
US-20240216415-A1 DEOXY-CYTIDINE OR URIDINE DERIVATIVES FOR USE IN CANCER THERAPIES TETRAGON BIOSCIENCES LTD. (IL) 2024-07-04 US disclosed
EP-4392076-A1 SIRP-ALPHA ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2024-07-03 EP disclosed
EP-4388103-A1 NECTIN-4 ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2024-06-26 EP disclosed
CN-118239996-A Application of fluorescent labeled nucleotide in DNA synthesis sequencing and single molecule sequencing 上海交通大学 2024-06-25 CN disclosed
US-20240191242-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2024-06-13 US disclosed
US-12006540-B2 Synthesis of novel disulfide linker based nucleotides as reversible terminators for DNA sequencing by synthesis THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-06-11 US disclosed
US-11999999-B2 Synthesis of novel disulfide linker based nucleotides as reversible terminators for DNA sequencing by synthesis THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-06-04 US disclosed
WO-2024097158-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS RAMIREZ CHRISTINA M (US) 2024-05-10 WO disclosed
US-11963973-B2 Deoxy-cytidine or uridine derivatives for use in cancer therapies HEMISPHERIAN AS (NO) 2024-04-23 US disclosed
US-11959137-B2 Synthesis of novel disulfide linker based nucleotides as reversible terminators for DNA sequencing by synthesis THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-04-16 US disclosed
US-20240117337-A1 METHODS AND POLYNUCLEOTIDES FOR AMPLIFYING A TARGET POLYNUCLEOTIDE OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2024-04-11 US disclosed
EP-4342545-A2 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS Elian LLC (US) 2024-03-27 EP disclosed
EP-4337646-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS Promega Corporation (US) 2024-03-20 EP disclosed
US-20240076719-A9 METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2024-03-07 US disclosed
WO-2024050372-A2 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES INC. (US) 2024-03-07 WO disclosed
US-11920136-B2 Transglutaminase-mediated conjugation Tallac Therapeutics, Inc. (US) 2024-03-05 US disclosed
EP-4323374-A1 MODIFIED NUCLEOSIDES SomaLogic Operating Co., Inc. (US) 2024-02-21 EP disclosed
CN-117567536-A Application of fluorescent labeled nucleotide in DNA synthesis sequencing and single molecule sequencing 上海交通大学 2024-02-20 CN disclosed
EP-4312942-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA Rejuvenation Technologies Inc. (US) 2024-02-07 EP disclosed
CN-117343990-A Method and kit for determining target polynucleotide and probe set 牛津纳米孔科技公开有限公司 2024-01-05 CN disclosed
US-11858953-B2 Compositions and methods for synthesis of phosphorylated molecules THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-01-02 US disclosed
CN-117242085-A Modified nucleosides 私募蛋白质体操作有限公司 2023-12-15 CN disclosed
US-20230364255-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2023-11-16 US disclosed
EP-3166680-B1 ANTI-HSV PRE-EXPOSURE PROPHYLAXIS ELIAN LLC (US) 2023-11-15 EP disclosed
EP-4271389-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA Rejuvenation Technologies Inc. (US) 2023-11-08 EP disclosed
US-11795463-B2 Transglutaminase-mediated conjugation Tallac Therapeutics, Inc. (US) 2023-10-24 US disclosed
US-20230310439-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS ELIAN LLC 2023-10-05 US disclosed
US-20230295694-A1 METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2023-09-21 US disclosed
EP-4233879-A1 DEOXY- CYTIDINE DERIVATIVES FOR USE IN CANCER THERAPIES Hemispherian AS (NO) 2023-08-30 EP disclosed
CN-116670161-A Methods of preventing or treating viral-induced organ injury or failure using IL-22 dimers 亿一生物医药开发(上海)有限公司 2023-08-29 CN disclosed
US-20230257414-A1 NUCLEOTIDE ANALOGUES FIRST-CITIZENS BANK & TRUST COMPANY 2023-08-17 US disclosed
US-20230257414-A1 NUCLEOTIDE ANALOGUES FIRST-CITIZENS BANK & TRUST COMPANY 2023-08-17 US disclosed
US-11725205-B2 Methods and polynucleotides for amplifying a target polynucleotide OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2023-08-15 US disclosed
US-20230250474-A1 SAMPLE PREPARATION METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2023-08-10 US disclosed
WO-2023147565-A2 METHODS AND SYSTEMS FOR HIGH-THROUGHPUT MOLECULAR ANALYSIS Opentrons LabWorks Inc. (US) 2023-08-03 WO disclosed
US-20230233608-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. (US) 2023-07-27 US disclosed
EP-3917538-B1 DEOXY- CYTIDINE DERIVATIVES FOR USE IN CANCER THERAPIES HEMISPHERIAN AS (NO) 2023-07-12 EP disclosed
US-11696918-B2 Viral prophylaxis treatment methods and pre-exposure prophylaxis kits ELIAN LLC (US) 2023-07-11 US disclosed
US-20230160000-A1 SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-05-25 US disclosed
US-20230160000-A1 SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-05-25 US disclosed
US-20230160000-A1 SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-05-25 US disclosed
US-11649451-B2 Evolution of bioactive sequence-defined synthetic polymers using DNA-templated polymerization PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-05-16 US disclosed
US-11649451-B2 Evolution of bioactive sequence-defined synthetic polymers using DNA-templated polymerization PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-05-16 US disclosed
US-20230130194-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2023-04-27 US disclosed
US-11633385-B2 Combination compositions for treatment of cancer REDHILL BIOPHARMA LTD. (IL) 2023-04-25 US disclosed
US-20230079150-A1 METHODS FOR PREVENTION OR TREATMENT OF VIRUS-INDUCED ORGAN INJURY OR FAILURE WITH IL-22 DIMER Evive Biotechnology (Shanghai) Ltd (CN) 2023-03-16 US disclosed
WO-2023028511-A1 SIRP-ALPHA ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2023-03-02 WO disclosed
WO-2023023659-A1 NECTIN-4 ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2023-02-23 WO disclosed
US-20230046363-A1 METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2023-02-16 US disclosed
US-20230028388-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-01-26 US disclosed
US-20230028388-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-01-26 US disclosed
EP-4123031-A1 METHODS FOR DETECTING AGGLUTINATION AND COMPOSITIONS FOR USE IN PRACTICING THE SAME The Regents of The University of California (US) 2023-01-25 EP disclosed
EP-4110830-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION Tallac Therapeutics, Inc. (US) 2023-01-04 EP disclosed
US-11542551-B2 Sample preparation method OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2023-01-03 US disclosed
US-20220411860-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2022-12-29 US disclosed
US-20220411860-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2022-12-29 US disclosed
EP-4103219-A1 METHODS FOR PREVENTION OR TREATMENT OF VIRUS-INDUCED ORGAN INJURY OR FAILURE WITH IL-22 DIMER Evive Biotechnology (Shanghai) Ltd (CN) 2022-12-21 EP disclosed
US-20220396830-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS PROMEGA CORPORATION 2022-12-15 US disclosed
EP-3529373-B1 METHOD FOR DETERMINING THE PRESENCE, ABSENCE OR AMOUNT OF TWO OR MORE TARGET POLYNUCLEOTIDES OXFORD NANOPORE TECH PLC (GB) 2022-12-07 EP disclosed
US-20220380768-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2022-12-01 US disclosed
WO-2022241249-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS PROMEGA CORPORATION (US) 2022-11-17 WO disclosed
US-20220347112-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES, INC. 2022-11-03 US disclosed
WO-2022221241-A1 MODIFIED NUCLEOSIDES SOMALOGIC OPERATING CO., INC. (US) 2022-10-20 WO disclosed
WO-2022212576-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES INC. (US) 2022-10-06 WO disclosed
US-11446398-B2 Regulated biocircuit systems OBSIDIAN THERAPEUTICS, INC. (US) 2022-09-20 US disclosed
CN-114989235-A Design and synthesis of nucleotides based on novel disulfide linkers for use as reversible terminators for DNA sequencing by synthesis 哥伦比亚大学董事会 2022-09-02 CN disclosed
US-20220257629-A1 COMPOSITIONS AND METHODS FOR UPREGULATION OF HUMAN FETAL HEMOGLOBIN THE UAB RESEARCH FOUNDATION 2022-08-18 US disclosed
US-11390904-B2 Nanopore-based method and double stranded nucleic acid construct therefor OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2022-07-19 US disclosed
US-11390910-B2 Method OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2022-07-19 US disclosed
US-20220213541-A1 METHOD FOR DETERMINING A POLYMER SEQUENCE OXFORD NANOPORE TECHNOLOGIES LIMITED (GB) 2022-07-07 US disclosed
WO-2022147039-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA REJUVENATION TECHNOLOGIES INC. (US) 2022-07-07 WO disclosed
EP-3283499-B1 DUAL QUENCHER PROBES BIOSEARCH TECH INC (US) 2022-07-06 EP disclosed
CN-108779138-B Design and synthesis of nucleotides based on novel disulfide linkers for use as reversible terminators for DNA sequencing by synthesis 哥伦比亚大学董事会 2022-06-17 CN disclosed
EP-3283638-B1 METHODS FOR DETECTING AGGLUTINATION AND USE OF KITS IN PRACTICING THE SAME UNIV CALIFORNIA (US) 2022-06-08 EP disclosed
CN-114469958-A Method for prophylactic treatment of viruses and pre-exposure prophylactic kit 艾利安有限责任公司 2022-05-13 CN disclosed
US-20220127299-A1 NUCLEOTIDE CLEAVABLE LINKERS AND USES THEREOF LG ELECTRONICS INC. (KR) 2022-04-28 US disclosed
US-20220117992-A1 DEOXY-CYTIDINE OR URIDINE DERIVATIVES FOR USE IN CANCER THERAPIES TETRAGON BIOSCIENCES LTD. (IL) 2022-04-21 US disclosed
US-20220096649-A1 IMMUNOMODULATING POLYNUCLEOTIDE CONJUGATES AND METHODS OF USE HORIZON TECHNOLOGY FINANCE CORPORATION 2022-03-31 US disclosed
WO-2022040173-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION Tallac Therapeutics, Inc. (US) 2022-02-24 WO disclosed
US-20220056069-A1 IMMUNOMODULATING POLYNUCLEOTIDES, ANTIBODY CONJUGATES THEREOF, AND METHODS OF THEIR USE HORIZON TECHNOLOGY FINANCE CORPORATION 2022-02-24 US disclosed
CN-111732623-B Tri-isopropyl silaacetylene modified deoxycytidine phosphoramidite monomer and preparation method and application thereof 中国科学院化学研究所 2022-01-18 CN disclosed
CN-106794336-B Method for prophylactic treatment of viruses and pre-exposure prophylactic kit 艾利安有限责任公司 2022-01-11 CN disclosed
EP-3930721-A1 TREATMENT OF HERPES SIMPLEX WITH A COMBINATION OF VALACYCLOVIR AND FAMCICLOVIR Elian LLC (US) 2022-01-05 EP disclosed
US-20210403978-A1 METHODS FOR DETECTING AGGLUTINATION AND COMPOSITIONS FOR USE IN PRACTICING THE SAME THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2021-12-30 US disclosed
US-11203611-B2 Immunomodulating polynucleotides, antibody conjugates thereof, and methods of their use TOLLNINE, INC. (US) 2021-12-21 US disclosed
EP-3917538-A1 DEOXY- CYTIDINE OR URIDINE DERIVATIVES FOR USE IN CANCER THERAPIES Hemispherian AS (NO) 2021-12-08 EP disclosed
CN-113727715-A Treatment of herpes simplex with a combination of valacyclovir and famciclovir 艾利安有限责任公司 2021-11-30 CN disclosed
US-11180522-B2 Disulfide-linked reversible terminators CENTRILLION TECHNOLOGY HOLDINGS CORPORATION (KY) 2021-11-23 US disclosed
US-11180523-B2 Design, synthesis and use of synthetic nucleotides comprising charge mass tags QUANTUMDX GROUP LIMITED (GB) 2021-11-23 US disclosed
US-20210346410-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS ELIAN LLC (US) 2021-11-11 US disclosed
US-20210332070-A1 Compositions and Methods for Synthesis of Phosphorylated Molecules UNIV CALIFORNIA (US) 2021-10-28 US disclosed
CN-107922454-B Dual quencher probes 生物检索技术股份有限公司 2021-10-22 CN disclosed
US-11149296-B2 Methods for detecting agglutination and compositions for use in practicing the same THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-10-19 US disclosed
WO-2021160163-A1 METHODS FOR PREVENTION OR TREATMENT OF VIRUS-INDUCED ORGAN INJURY OR FAILURE WITH IL-22 DIMER Evive Biotechnology (Shanghai) Ltd (CN) 2021-08-19 WO disclosed
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CN-107109483-B Method for modifying template double-stranded polynucleotide 牛津纳米孔技术公司 2021-07-20 CN disclosed
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EP-3363809-B1 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING ILLUMINA CAMBRIDGE LTD (GB) 2020-04-08 EP disclosed
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EP-3363809-A1 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING Illumina Cambridge Limited (GB) 2018-08-22 EP disclosed
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US-9938314-B2 Cytidine-5-carboxamide modified nucleotide compositions and methods related thereto SOMALOGIC, INC. (US) 2018-04-10 US disclosed
US-9938314-B2 Cytidine-5-carboxamide modified nucleotide compositions and methods related thereto SOMALOGIC, INC. (US) 2018-04-10 US disclosed
EP-3002289-B1 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING ILLUMINA CAMBRIDGE LTD (GB) 2018-02-28 EP disclosed
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EP-3186387-A1 METHOD OF DETERMINING THE ACTIVITY OF ENZYMES CONVERTING CYTOSINE DERIVATIVES TO URACIL DERIVATIVES IN CELLS, TISSUES AND ORGANISMS Univerzita Palackého v Olomouci (CZ) 2017-07-05 EP disclosed
EP-2757091-B1 Stabilized Nucleic Acid Dark Quencher-Fluorophore Probes BIOSEARCH TECH INC (US) 2017-06-28 EP disclosed
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US-9688980-B2 Templated molecules and methods for using such molecules NUEVOLUTION (DK) 2017-06-27 US disclosed
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EP-3166680-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS Prophylaxis, LLC (US) 2017-05-17 EP disclosed
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EP-3126517-A1 MODIFIED CYTOSINE POLYNUCLEOTIDE OLIGOMERS AND METHODS Cepheid (US) 2017-02-08 EP disclosed
EP-3108010-A1 SAMPLE PREPARATION METHOD Oxford Nanopore Technologies Limited (GB) 2016-12-28 EP disclosed
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CN-105658658-A Cytidine-5-carboxamide modified nucleotide compositions and methods related thereto 私募蛋白质体公司 2016-06-08 CN disclosed
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WO-2016059363-A1 METHOD OXFORD NANOPORE TECHNOLOGIES LIMITED (GB) 2016-04-21 WO disclosed
EP-3002289-A1 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING Illumina Cambridge Limited (GB) 2016-04-06 EP disclosed
WO-2016029889-A1 METHOD OF DETERMINING THE ACTIVITY OF ENZYMES CONVERTING CYTOSINE DERIVATIVES TO URACIL DERIVATIVES IN CELLS, TISSUES AND ORGANISMS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-03-03 WO disclosed
WO-2016029889-A1 METHOD OF DETERMINING THE ACTIVITY OF ENZYMES CONVERTING CYTOSINE DERIVATIVES TO URACIL DERIVATIVES IN CELLS, TISSUES AND ORGANISMS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2016-03-03 WO disclosed
EP-2305808-B1 Templated molecules and methods for using such molecules NUEVOLUTION AS (DK) 2016-03-02 EP disclosed
EP-2305808-B1 Templated molecules and methods for using such molecules NUEVOLUTION AS (DK) 2016-03-02 EP disclosed
EP-1905829-B1 Templated molecules and methods for using such molecules NUEVOLUTION AS (DK) 2016-02-17 EP disclosed
US-20160032378-A1 MODIFIED NUCLEOTIDES SOLEXA LIMITED (GB) 2016-02-04 US disclosed
WO-2016007538-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS PROPHYLAXIS, LLC (US) 2016-01-14 WO disclosed
US-20160000797-A1 VIRAL PROPHYLAXIS TREATMENT METHODS AND PRE-EXPOSURE PROPHYLAXIS KITS ELIAN LLC 2016-01-07 US disclosed
WO-2015172134-A1 COSMIC QUENCHERS BIOSEARCH TECHNOLOGIES, INC. (US) 2015-11-12 WO disclosed
US-20150315567-A1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION A/S (DK) 2015-11-05 US disclosed
US-20150315567-A1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION A/S (DK) 2015-11-05 US disclosed
US-20150315567-A1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION A/S (DK) 2015-11-05 US disclosed
WO-2015153510-A1 MODIFIED CYTOSINE POLYNUCLEOTIDE OLIGOMERS AND METHODS CEPHEID (US) 2015-10-08 WO disclosed
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EP-2607369-B1 Modified nucleotides for polynucleotide sequencing ILLUMINA CAMBRIDGE LTD (GB) 2015-09-23 EP disclosed
US-9121060-B2 Modified nucleotides ILLUMINA CAMBRIDGE LIMITED (GB) 2015-09-01 US disclosed
WO-2015124935-A1 SAMPLE PREPARATION METHOD OXFORD NANOPORE TECHNOLOGIES LIMITED (GB) 2015-08-27 WO disclosed
WO-2015077292-A1 CYTIDINE-5-CARBOXAMIDE MODIFIED NUCLEOTIDE COMPOSITIONS AND METHODS RELATED THERETO SOMALOGIC, INC. (US) 2015-05-28 WO disclosed
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US-8921124-B2 Pyrazole-based cyanine dye WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2014-12-30 US disclosed
US-20140315191-A1 FOUR-COLOR DNA SEQUENCING BY SYNTHESIS USING CLEAVABLE FLUORESCENT NUCLEOTIDE REVERSIBLE TERMINATORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2014-10-23 US disclosed
EP-2770058-A1 Ligand and method for detection of okadaic acid Université de Perpignan (FR) 2014-08-27 EP disclosed
US-20140221639-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF INSTITUTE OF NUCLEAR ENERGY RESEARCH ATOMIC ENERGY COUNCIL, EXECUTIVE YUAN (TW) 2014-08-07 US disclosed
US-20140221639-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF INSTITUTE OF NUCLEAR ENERGY RESEARCH ATOMIC ENERGY COUNCIL, EXECUTIVE YUAN (TW) 2014-08-07 US disclosed
EP-2757091-A1 Stabilized Nucleic Acid Dark Quencher-Fluorophore Probes Biosearch Technologies, Inc. (US) 2014-07-23 EP disclosed
US-20140194611-A1 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES BIOSEARCH TECHNOLOGIES, INC. (US) 2014-07-10 US disclosed
US-8674094-B2 Stabilized nucleic acid dark quencher-fluorophore probes BIOSEARCH TECHNOLOGIES, INC. (US) 2014-03-18 US disclosed
US-8614312-B2 Method for preparing nucleotides and related analogues by synthesis on soluble substrate, and biological tools thus prepared CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2013-12-24 US disclosed
US-8597881-B2 Modified nucleotides ILLUMINA CAMBRIDGE LIMITED (GB) 2013-12-03 US disclosed
US-20130280700-A1 FOUR-COLOR DNA SEQUENCING BY SYNTHESIS USING CLEAVABLE FLUORESCENT NUCLEOTIDE REVERSIBLE TERMINATORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2013-10-24 US disclosed
US-8512559-B2 Device, method, and system for separation and detection of biomolecules and cells INTEL CORPORATION (US) 2013-08-20 US disclosed
US-20130197209-A1 MODIFIED NUCLEOTIDES ILLUMINA CAMBRIDGE LIMITED (GB) 2013-08-01 US disclosed
EP-2607369-A1 Modified nucleotides for polynucleotide sequencing Illumina Cambridge Limited (GB) 2013-06-26 EP disclosed
US-8466266-B2 Stabilized nucleic acid dark quencher-fluorophore probes BIOSEARCH TECHNOLOGIES, INC. (US) 2013-06-18 US disclosed
US-8410075-B2 Mannich base N-oxide drugs CASCADE PRODRUG INC. (US) 2013-04-02 US disclosed
EP-1530578-B1 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING ILLUMINA CAMBRIDGE LTD (GB) 2013-03-13 EP disclosed
US-8298792-B2 Four-color DNA sequencing by synthesis using cleavable fluorescent nucleotide reversible terminators THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-10-30 US disclosed
US-8298792-B2 Four-color DNA sequencing by synthesis using cleavable fluorescent nucleotide reversible terminators THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-10-30 US disclosed
US-20120225494-A1 DNA LIGANDS FOR AFLATOXIN AND ZEARALENONE LE LINDA CHRYSEIS (CA) 2012-09-06 US disclosed
WO-2012113072-A1 A METHOD FOR THE SELECTION OF DNA LIGANDS FOR A MOLECULAR TARGET NEOVENTURES BIOTECHNOLOGY INC. (CA) 2012-08-30 WO disclosed
US-8252768-B2 Designer therapy of pancreatic tumors UNIVERSITY OF MIAMI (US) 2012-08-28 US disclosed
US-20120178919-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF NATIONAL YANG-MING UNIVERSITY (TW) 2012-07-12 US disclosed
US-20120178919-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF NATIONAL YANG-MING UNIVERSITY (TW) 2012-07-12 US disclosed
US-20120178919-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF NATIONAL YANG-MING UNIVERSITY (TW) 2012-07-12 US disclosed
EP-2467483-A1 DNA LIGANDS FOR AFLATOXIN AND ZEARALENONE Neoventures Biotechnology Inc. (CA) 2012-06-27 EP disclosed
US-8193335-B2 Click chemistry for the production of reporter molecules BASECLICK GMBH (DE) 2012-06-05 US disclosed
WO-2012033298-A3 METHOD FOR MANUFACTURING A NOX GAS SENSOR, AND NOX GAS SENSOR MANUFACTURED USING SAME 일진머티리얼즈 주식회사 (KR) 2012-05-10 WO disclosed
US-20120095201-A1 MODIFIED NUCLEOTIDES ILLUMINA CAMBRIDGE LIMITED (GB) 2012-04-19 US disclosed
US-20120045796-A1 NUCLEIC ACID HOTSTART TECHNOLOGY CO-DIAGNOSTICS, INC. 2012-02-23 US disclosed
US-8105770-B2 Method of detecting amplification or deletion in genomic DNA Fragment WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2012-01-31 US disclosed
US-20120021408-A1 FOUR-COLOR DNA SEQUENCING BY SYNTHESIS USING CLEAVABLE FLUORESCENT NUCLEOTIDE REVERSIBLE TERMINATORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2012-01-26 US disclosed
US-20120021408-A1 FOUR-COLOR DNA SEQUENCING BY SYNTHESIS USING CLEAVABLE FLUORESCENT NUCLEOTIDE REVERSIBLE TERMINATORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2012-01-26 US disclosed
US-20120004391-A2 CYANINE-TYPE COMPOUNDS HAVING AN ALKYNYL LINKER ARM Cyanine Technologies S.p.A. (IT) 2012-01-05 US disclosed
US-8071739-B2 Modified nucleotides ILLUMINA CAMBRIDGE LIMITED (GB) 2011-12-06 US disclosed
EP-2006289-B1 PYRAZOLE-TYPE CYANINE DYE WAKO PURE CHEM IND LTD (JP) 2011-11-30 EP disclosed
US-8062841-B2 Multiplex data collection and analysis in bioanalyte detection INTEL CORPORATION (US) 2011-11-22 US disclosed
US-20110282041-A1 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES BIOSEARCH TECHNOLOGIES, INC. (US) 2011-11-17 US disclosed
EP-2089343-B1 CLICK CHEMISTRY FOR THE PRODUCTION OF REPORTER MOLECULES BASECLICK GMBH (DE) 2011-07-06 EP disclosed
US-20110118438-A1 CYANINE-TYPE COMPOUNDS HAVING AN ALKYNYL LINKER ARM Cyanine Technologies S.p.A. (IT) 2011-05-19 US disclosed
US-20110118454-A1 METHOD FOR PREPARING NUCLEOTIDES AND RELATED ANALOGUES BY SYNTHESIS ON SOLUBLE SUBSTRATE, AND BIOLOGICAL TOOLS THUS PREPARED CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2011-05-19 US disclosed
EP-2305808-A1 Templated molecules and methods for using such molecules Nuevolution A/S (DK) 2011-04-06 EP disclosed
EP-2305808-A1 Templated molecules and methods for using such molecules Nuevolution A/S (DK) 2011-04-06 EP disclosed
WO-2011020198-A1 DNA LIGANDS FOR AFLATOXIN AND ZEARALENONE NEOVENTURES BIOTECHNOLOGY LIMITED (CA) 2011-02-24 WO disclosed
US-7892297-B2 Cyanin-type compounds having an alkynyl linker arm Cyanine Technologies S.p.A. (IT) 2011-02-22 US disclosed
EP-2268608-A2 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES Biosearch Technologies, Inc. (US) 2011-01-05 EP disclosed
US-20100317004-A1 PROBES Life Technologies Corporation (US) 2010-12-16 US disclosed
US-20100290992-A1 NANOPARTICLE NUCLEIC ACID BINDING COMPOUND CONJUGATES FORMING I-MOTIFS ROCHE DIAGNOSTICS GMBH (DE) 2010-11-18 US disclosed
US-20100292452-A1 Modified nucleotides ILLUMINA CAMBRIDGE LTD 2010-11-18 US disclosed
US-20100290992-A1 NANOPARTICLE NUCLEIC ACID BINDING COMPOUND CONJUGATES FORMING I-MOTIFS ROCHE DIAGNOSTICS GMBH (DE) 2010-11-18 US disclosed
EP-2242761-A1 METHOD OF MYCOTOXIN DETECTION Neoventures Biotechnology Inc. (CA) 2010-10-27 EP disclosed
US-7807653-B2 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2010-10-05 US disclosed
US-7771973-B2 sequencing reactions where nucleotide or nucleoside molecules modified by reversible covalent attachment of 3'-OH blocking groups thereto, are used where blocked nucleotide or nucleoside molecules are required ILLUMINA CAMBRIDGE LIMITED (GB) 2010-08-10 US disclosed
US-7727713-B2 Templated molecules and methods for using such molecules NUEVOLUTION A/S (DK) 2010-06-01 US disclosed
US-20100112711-A1 METHOD OF DETECTING AMPLIFICATION OR DELETION IN GENOMIC DNA FRAGMENT WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2010-05-06 US disclosed
US-20100081137-A1 Click Chemistry for the Production of Reporter Molecules BASECLICK GMBH (DE) 2010-04-01 US disclosed
US-20100016252-A1 Mannich Base N-Oxide Drugs State of Oregon Acting By and Through The Oregon State Board of Higher Education On Behalf of The U (US) 2010-01-21 US disclosed
US-20100016177-A1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION A/S (DK) 2010-01-21 US disclosed
US-20090325897-A1 DESIGNER THERAPY OF PANCREATIC TUMORS UNIVERSITY OF MIAMI (US) 2009-12-31 US disclosed
US-20090325172-A1 Modified nucleotides SOLEXA LIMITED 2009-12-31 US disclosed
EP-2136626-A1 MANNICH BASE N-OXIDE DRUGS State of Oregon acting by and through the Oregon State Board of Higher Education on behalf of the University of Oregon (US) 2009-12-30 EP disclosed
EP-2119797-A1 METHOD OF DETECTING AMPLIFICATION OR DELETION IN GENOMIC DNA FRAGMENT Wako Pure Chemical Industries, Ltd. (JP) 2009-11-18 EP disclosed
EP-2119797-A1 METHOD OF DETECTING AMPLIFICATION OR DELETION IN GENOMIC DNA FRAGMENT Wako Pure Chemical Industries, Ltd. (JP) 2009-11-18 EP disclosed
US-20090259030-A1 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES BIOSEARCH TECHNOLOGIES (US) 2009-10-15 US disclosed
WO-2009124150-A2 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES BIOSEARCH TECHNOLOGIES, INC. (US) 2009-10-08 WO disclosed
US-7598230-B2 For the treatment of viral infections, microbial infections, and proliferative disorders; contain di- or triphosphate moeity mimetics, such as those containing boron anions BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2009-10-06 US disclosed
EP-2089343-A2 CLICK CHEMISTRY FOR THE PRODUCTION OF REPORTER MOLECULES baseclick GmbH (DE) 2009-08-19 EP disclosed
WO-2009086621-A1 METHOD OF MYCOTOXIN DETECTION NEOVENTURES BIOTECHNOLOGY INC. (CA) 2009-07-16 WO disclosed
US-7541444-B2 Modified nucleotides ILLUMINA CAMBRIDGE LIMITED (GB) 2009-06-02 US disclosed
EP-2054085-A2 NANOPARTICLE NUCLEIC ACID BONDING COMPOUND CONJUGATES FORMING I-MOTIFS Roche Diagnostics GmbH (DE) 2009-05-06 EP disclosed
US-20090069546-A1 PYRAZOLE-BASED CYANINE DYE WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2009-03-12 US disclosed
US-7488607-B2 Electronically readable microarray with electronic addressing function AGILENT TECHNOLOGIES, INC. (US) 2009-02-10 US disclosed
US-20090005260-A1 MULTIPLEX DATA COLLECTION AND ANALYSIS IN BIOANALYTE DETECTION INTEL CORPORATION 2009-01-01 US disclosed
EP-2006289-A1 PYRAZOLE-TYPE CYANINE DYE Wako Pure Chemical Industries, Ltd. (JP) 2008-12-24 EP disclosed
EP-1985702-A2 CPG-like nucleic acids and methods of use thereof Coley Pharmaceuticals GmbH (DE) 2008-10-29 EP disclosed
US-20080262989-A1 MULTIPLEX DATA COLLECTION AND ANALYSIS IN BIOANALYTE DETECTION INTEL CORPORATION 2008-10-23 US disclosed
WO-2008115499-A1 MANNICH BASE N-OXIDE DRUGS STATE OF OREGON ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION ON BEHALF OF THE UNIVERSITY OF OREGON (US) 2008-09-25 WO disclosed
US-20080226649-A1 CPG-like nucleic acids and methods of use thereof COLEY PHARMACEUTICAL GMBH (DE) 2008-09-18 US disclosed
US-7410763-B2 Multiplex data collection and analysis in bioanalyte detection INTEL CORPORATION (US) 2008-08-12 US disclosed
EP-1952155-A2 METHOD AND CMOS-BASED DEVICE TO ANALYZE MOLECULES AND NANOMATERIALS BASED ON THE ELECTRICAL READOUT OF SPECIFIC BINDING EVENTS ON FUNCTIONALIZED ELECTRODES Intel Corporation (INTEL) (US) 2008-08-06 EP disclosed
WO-2008085611-A2 DESIGNER THERAPHY OF PANCREATIC TUMORS UNIVERSITY OF MIAMI (US) 2008-07-17 WO disclosed
US-7399844-B2 Method and reagents for analyzing the nucleotide sequence of nucleic acids AGILENT TECHNOLOGIES, INC. (US) 2008-07-15 US disclosed
EP-1350262-B1 CPG-LIKE NUCLEIC ACIDS AND METHODS OF USE THEREOF COLEY PHARMACEUTICALS GMBH (DE) 2008-06-11 EP disclosed
EP-1383890-B1 MUTANTS OF DESOXYCYTIDINE KINASE HAVING EXTENDED ENZYMATIC ACTIVITY PASTEUR INSTITUT (FR) 2008-05-14 EP disclosed
WO-2008052775-A2 CLICK CHEMISTRY FOR THE PRODUCTION OF REPORTER MOLECULES BASECLICK GMBH (DE) 2008-05-08 WO disclosed
WO-2008052775-A2 CLICK CHEMISTRY FOR THE PRODUCTION OF REPORTER MOLECULES BASECLICK GMBH (DE) 2008-05-08 WO disclosed
WO-2008048222-A2 METHOD AND CMOS-BASED DEVICE TO ANALYZE MOLECULES AND NANOMATERIALS BASED ON THE ELECTRICAL READOUT OF SPECIFIC BINDING EVENTS ON FUNCTIONALIZED ELECTRODES INTEL CORPORATION (US) 2008-04-24 WO disclosed
EP-1905829-A2 Templated molecules and methods for using such molecules Nuevolution A/S (DK) 2008-04-02 EP disclosed
WO-2008017507-A2 NANOPARTICLE NUCLEIC ACID BONDING COMPOUND CONJUGATES FORMING I-MOTIFS ROCHE DIAGNOSTICS GMBH (DE) 2008-02-14 WO disclosed
US-7323555-B2 Nucleotide derivative and DNA microarray ISAO SAITO (JP) 2008-01-29 US disclosed
US-20070292855-A1 Method and CMOS-based device to analyze molecules and nanomaterials based on the electrical readout of specific binding events on functionalized electrodes INTEL CORPORATION (US) 2007-12-20 US disclosed
US-20070265224-A1 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2007-11-15 US disclosed
US-20070259832-A1 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2007-11-08 US disclosed
US-7285658-B2 Nucleotide mimics and their prodrugs BIOTA, INC. (US) 2007-10-23 US disclosed
EP-1402024-B1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION AS (DK) 2007-08-22 EP disclosed
US-20070166705-A1 Modified nucleotides ILLUMINA CAMBRIDGE LIMITED (GB) 2007-07-19 US disclosed
EP-1251136-B1 Method and reagents for analyzing the nucleotide sequence of nucleic acids AGILENT TECHNOLOGIES INC (US) 2007-06-13 EP disclosed
US-20070114180-A1 Device, method, and system for separation and detection of biomolecules and cells INTEL CORPORATION (US) 2007-05-24 US disclosed
EP-1585835-B1 Nucleic acid probes and method for detecting a target nucleic acid sequence comprising two or more cis-located nucleic acid regions DYNAL BIOTECH LTD (GB) 2007-04-18 EP disclosed
US-20070048746-A1 Beam emitter, microfluidic channel, spectrometer and detector; binding between reporter molecules and analyte; microelectric mechanical system INTEL CORPORATION (US) 2007-03-01 US disclosed
US-20060269916-A1 Probes DYNAL BIOTECH INC. 2006-11-30 US disclosed
US-20060230554-A1 Cyanin-type compounds having an alkynyl linker arm CYANINE TECHNOLOGIES S. P. A. (IT) 2006-10-19 US disclosed
US-20060216312-A1 Mutants of replication competent vaccinia virus ARIZONA BOARD OF REGENTS, ACTING FOR AND ON BEHALF OF, ARIZONA STATE UNIVERSITY 2006-09-28 US disclosed
EP-1689439-A2 SMALL MOLECULE COMPOSITIONS AND METHODS FOR INCREASING DRUG EFFICIENCY USING COMPOSITIONS THEREOF Acidophil LLC (US) 2006-08-16 EP disclosed
US-7057027-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2006-06-06 US disclosed
EP-1654327-A1 CYANIN-TYPE COMPOUNDS HAVING AN ALKYNYL LINKER ARM Caputo, Giuseppe (IT) 2006-05-10 EP disclosed
US-6967079-B2 Pyrimidine derivatives for labeled binding partners ISIS PHARMACEUTICALS, INC. (US) 2005-11-22 US disclosed
US-6962783-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2005-11-08 US disclosed
EP-1585835-A2 NUCLEIC ACID PROBES AND METHOD FOR DETECTING A TARGET NUCLEIC ACID SEQUENCE COMPRISE TWO OR MORE CIS- LOCATED NUCLEIC ACID REGIONS Dynal Biotech Limited (GB) 2005-10-19 EP disclosed
EP-1015643-B1 METHOD AND REAGENTS FOR ANALYZING THE NUCLEOTIDE SEQUENCE OF NUCLEIC ACIDS AGILENT TECHNOLOGIES INC (US) 2005-09-21 EP disclosed
US-20050148534-A1 Small molecule compositions and methods for increasing drug efficiency using compositions thereof ACIDOPHIL LLC 2005-07-07 US disclosed
US-6914148-B2 Guanidinium functionalized intermediates ISIS PHARMACEUTICALS, INC. (US) 2005-07-05 US disclosed
EP-1530578-A2 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING Solexa Limited (GB) 2005-05-18 EP disclosed
US-20050079505-A1 Electronically readable microarray with electronic addressing function AGILENT TECHNOLOGIES INC 2005-04-14 US disclosed
WO-2005030258-A2 SMALL MOLECULE COMPOSITIONS AND METHODS FOR INCREASING DRUG EFFICIENCY USING COMPOSITIONS THEREOF ACIDOPHIL LLC (US) 2005-04-07 WO disclosed
US-6875593-B2 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2005-04-05 US disclosed
US-20050069905-A1 Detection of molecular binding events AGILENT TECHNOLOGIES, INC. 2005-03-31 US disclosed
WO-2005014723-A1 CYANIN-TYPE COMPOUNDS HAVING AN ALKYNYL LINKER ARM CAPUTO GIUSEPPE (IT) 2005-02-17 WO disclosed
US-20040265802-A9 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES FROEHLER BRIAN (US) 2004-12-30 US disclosed
US-20040248104-A1 Methods and reagents for profiling quantities of nucleic acids AGILENT TECHNOLOGIES, INC. 2004-12-09 US disclosed
US-6825331-B2 DIAGNOSTIC HYBRIDIZATION PROBES; BIOCHEMICAL CONJUGATION ISIS PHARMACEUTICALS, INC. 2004-11-30 US disclosed
US-20040220395-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. 2004-11-04 US disclosed
WO-2004087047-A2 MUTANTS OF REPLICATION COMPETENT VACCINIA VIRUS ARIZONA BOARD OF REGENTS (US) 2004-10-14 WO disclosed
WO-2004048611-A2 NUCLEIC ACID PROBES AND METHOD FOR DETECTING A TARGET NUCLEIC ACID SEQUENCE COMPRISE TWO OR MORE CIS- LOCATED NUCLEIC ACID REGIONS DYNAL BIOTECH LIMITED (GB) 2004-06-10 WO disclosed
EP-1404370-A2 OPHTHALMIC COMPOSITIONS COMPRISING HYALURONIC ACID Novartis AG (CH) 2004-04-07 EP disclosed
EP-1402024-A2 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES Nuevolution A/S (DK) 2004-03-31 EP disclosed
EP-1401850-A1 NUCLEOSIDE DERIVATIVES FOR LIBRARY PREPARATION Nuevolution A/S (DK) 2004-03-31 EP disclosed
US-20040059104-A1 Nucleotide mimics and their prodrugs BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2004-03-25 US disclosed
US-20040049008-A1 Templated molecules and methods for using such molecules NUEVOLUTION A/S (DK) 2004-03-11 US disclosed
WO-2004018497-A2 MODIFIED NUCLEOTIDES FOR POLYNUCLEOTIDE SEQUENCING SOLEXA LIMITED (GB) 2004-03-04 WO disclosed
US-20030207824-A1 Pyrimidine derivatives for labeled binding partners MATTEUCCI MARK D (US) 2003-11-06 US disclosed
EP-1350262-A2 CPG-LIKE NUCLEIC ACIDS AND METHODS OF USE THEREOF Coley Pharmaceuticals GmbH (DE) 2003-10-08 EP disclosed
US-6627456-B1 Incorporating into the oligonucleotide analogs that are the components of a library to which in vitro selection methods functionalized standard and non-standard nucleotides, and incorporating functionalized cofactors into the experiment BENNER, STEVEN 2003-09-30 US disclosed
US-20030181406-A1 CpG-like nucleic acids and methods of use thereof PFIZER INC. 2003-09-25 US disclosed
US-20030170680-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines FROEHLER BRIAN (US) 2003-09-11 US disclosed
US-6617437-B1 Modified oligonucleotide of given formula; useful in diagnostics and therapeutics ISIS PHARMACEUTICALS, INC. 2003-09-09 US disclosed
US-20030143561-A1 Nucleoside derivatives for library preparation NUEVOLUTION A/S (DK) 2003-07-31 US disclosed
US-6593466-B1 Monomer of given formula; modified to increase binding affinity to target DNA or RNA and resist nuclease degradation; useful as therapeutics or diagnostics; gene expression inhibition ISIS PHARMACEUTICALS, INC. 2003-07-15 US disclosed
US-6589941-B1 Preventing or reducing formation of resistance in cytostatic treatment comprising combining BVDU, a salt thereof or BVDU in protected form or in prodrug form with at least one cytostatic agent in order to prevent or reduce the formation RESPROTECT GMBH (DE) 2003-07-08 US disclosed
US-20030113769-A1 Aminooxy functionalized oligomers, oligomer arrays and methods of using them IONIS PHARMACEUTICALS, INC. 2003-06-19 US disclosed
US-6576752-B1 Oligonucleotide comprising a plurality of nucleotide units of given structure; useful for diagnostic, therapeutic and investigative purposes ISIS PHARMACEUTICALS, INC. 2003-06-10 US disclosed
US-20030096980-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. 2003-05-22 US disclosed
US-20030092046-A1 Guanidinium functionalized oligomers and methods MANOHARAN MUTHIAH (US) 2003-05-15 US disclosed
EP-0719272-B1 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS ISIS PHARMACEUTICALS INC (US) 2003-05-07 EP disclosed
US-6534639-B1 Useful for diagnostic, therapeutic and investigative purposes; guanidine group gives enhanced DNA-RNA hybrid binding affinity and/or increased nuclease resistance ISIS PHARMACEUTICALS, INC. 2003-03-18 US disclosed
US-20030022150-A1 Detecting preferential bioplymers in sample; obtain nutrient broths inoculate with cells, immerse electrodes, code cells, incubate cells with substrate, monitor response, evaluate response AGILENT TECHNOLOGIES, INC. 2003-01-30 US disclosed
WO-2002102820-A1 NUCLEOSIDE DERIVATIVES FOR LIBRARY PREPARATION NUEVOLUTION A/S (DK) 2002-12-27 WO disclosed
WO-2002103008-A2 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES NUEVOLUTION A/S (DK) 2002-12-27 WO disclosed
WO-2002100436-A2 OPHTHALMIC ONCE-A-DAY COMPOSITION NOVARTIS AG (CH) 2002-12-19 WO disclosed
WO-2002100437-A2 OPHTHALMIC COMPOSITIONS COMPRISING HYALURONIC ACID NOVARTIS AG (CH) 2002-12-19 WO disclosed
US-20020182601-A1 Method and reagents for analyzing the nucleotide sequence of nucleic acids AGILENT TECHNOLOGIES, INC. 2002-12-05 US disclosed
EP-1256589-A2 Oligomers containing modified pyrimidines ISIS PHARMACEUTICALS, INC. (US) 2002-11-13 EP disclosed
EP-1251136-A2 Method and reagents for analyzing the nucleotide sequence of nucleic acids Agilent Technologies, Inc. (US) 2002-10-23 EP disclosed
EP-0637965-B1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES ISIS PHARMACEUTICALS INC (US) 2002-10-16 EP disclosed
EP-1206574-A4 GUANIDINIUM FUNCTIONALIZED OLIGOMERS AND METHODS ISIS PHARMACEUTICALS INC (US) 2002-10-16 EP disclosed
WO-2002069369-A2 CPG-LIKE NUCLEIC ACIDS AND METHODS OF USE THEREOF COLEY PHARMACEUTICAL GMBH (US) 2002-09-06 WO disclosed
EP-0806956-B1 USE OF 5'SUBSTITUTED NUCLEOSIDES TO PROVIDE RESISTANCE IN CYTOSTATIC TREATMENT RESPROTECT GMBH (DE) 2002-08-28 EP disclosed
EP-1206574-A2 GUANIDINIUM FUNCTIONALIZED OLIGOMERS AND METHODS ISIS PHARMACEUTICALS, INC. (US) 2002-05-22 EP disclosed
WO-2001002423-A9 2'-GUANIDINYL-SUBSTITUTED OLIGONUCLEOTIDES AND GENE EXPRESSION MODULATION THEREWITH ISIS PHARMACEUTICALS INC (US) 2002-05-02 WO disclosed
US-6380368-B1 GENETIC ENGINEERING ISIS PHARMACEUTICALS, INC. 2002-04-30 US disclosed
US-6342217-B1 ADMINISTERING 5-HALOGENATED PYRIMIDINE DERIVATIVE TO CONFER RADIATION SENSITIVITY TO TUMOR CELLS, EXPOSING TUMOR CELLS TO RADIATION THERAPY TO KILL TUMOR CELLS HUMAN GENE THERAPY RESEARCH INSTITUTE 2002-01-29 US disclosed
US-6218118-B1 MIXTURE OF NATURAL AND MASS-MODIFIED GENERIC OLIGONUCLEOTIDE PRECURSORS; USING MIXTURE AND ENZYMATIC PROCESSES TO ALTER THE LENGTH, AND THUS THE MASS, OF PRECURSORS THAT ARE COMPLEMENTARY TO TARGET NUCLEIC ACID AGILENT TECHNOLOGIES, INC. 2001-04-17 US disclosed
EP-0923591-A4 NOVEL BORONIC ACID-CONTAINING NUCLEIC ACIDS AND THEIR USE AS DIAGNOSTIC AGENTS PROLINX INC (US) 2001-01-31 EP disclosed
WO-2001002423-A2 2'-GUANIDINYL-SUBSTITUTED OLIGONUCLEOTIDES AND GENE EXPRESSION MODULATION THEREWITH ISIS PHARMACEUTICALS, INC. (US) 2001-01-11 WO disclosed
US-6162459-A Acyclovir transdermal delivery system NATIONAL SCIENCE COUNCIL (TW) 2000-12-19 US disclosed
US-6136332-A NONAQUEOUS, TOPICAL SOCIETE L'OREAL S.A. (FR) 2000-10-24 US disclosed
EP-1015643-A2 METHOD AND REAGENTS FOR ANALYZING THE NUCLEOTIDE SEQUENCE OF NUCLEIC ACIDS Hewlett-Packard Company (US) 2000-07-05 EP disclosed
US-6031086-A HAVING DIMINISHED CHARGE BUT UNDIMINISHED ABILITY TO COMPLEX WITH NATURAL DNA AT LOW IONIC STRENGTHS; PREPARED BY REPLACING NATURAL NUCLEOTIDES WITH UNNATURAL ZWITTERIONIC NUCLEOTIDES; MEMBRANE PERMEABLE AND NUCLEASE RESISTANT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-02-29 US disclosed
EP-0974672-A1 Improved primers for AFLP amplification KEYGENE N.V. (NL) 2000-01-26 EP disclosed
WO-2000003038-A2 METHOD AND REAGENTS FOR ANALYZING THE NUCLEOTIDE SEQUENCE OF NUCLEIC ACIDS HEWLETT-PACKARD COMPANY (US) 2000-01-20 WO disclosed
US-6005096-A FOR OLIGONUCLEOTIDES THAT ARE MODIFIED TO ENHANCE THE BINDING AFFINITY AND TO BEAR DETECTABLE LABELS; FOR DIAGNOSTIC USE GILEAD SCIENCES, INC. (US) 1999-12-21 US disclosed
US-5985266-A SENSITIZE TUMORS, RETROVIRUS COMPRISES OPERATIVELY LINKED TO A PROMOTER A GENE ENCODING A VIRAL THYMIDINE KINASE; SUCH THAT SAID TUMOR CELLS BECOME TRANSDUCED BY SAID RETROVIRUS AND EXPRESS SAID VIRAL THYMIDINE KINASE GENE; HUMAN GENE THERAPY RESEARCH INSTITUTE (US) 1999-11-16 US disclosed
US-5965364-A Method for selecting functional deoxyribonucleotide derivatives BENNER, STEVEN 1999-10-12 US disclosed
EP-0923591-A1 NOVEL BORONIC ACID-CONTAINING NUCLEIC ACIDS AND THEIR USE AS DIAGNOSTIC AGENTS PROLINX, INC. (US) 1999-06-23 EP disclosed
US-5876938-A Use of boron-containing polynucleotides as diagnostic agents PROLINX, INCORPORATED (US) 1999-03-02 US disclosed
US-5831045-A Boronic acid-containing polynucleotides PORLINX, INCORPORATED (US) 1998-11-03 US disclosed
US-5830653-A ABILITY TO INHIBIT GENE EXPRESSION GILEAD SCIENCES, INC. (US) 1998-11-03 US disclosed
US-5831046-A Boronic acid-contaning nucleic acid monomers PROLINX, INCORPORATED (US) 1998-11-03 US disclosed
US-5763588-A Pyrimidine derivatives for labeled binding partners GILEAD SCIENCES, INC. (US) 1998-06-09 US disclosed
WO-1998005672-A1 NOVEL BORONIC ACID-CONTAINING NUCLEIC ACIDS AND THEIR USE AS DIAGNOSTIC AGENTS PROLINX INCORPORATED (US) 1998-02-12 WO disclosed
EP-0806956-A1 USE OF 5'SUBSTITUTED NUCLEOSIDES TO PROVIDE RESISTANCE IN CYTOSTATIC TREATMENT AND MEDICAMENTS CONTAINING SAID NUCLEOSIDES FRAUNHOFER-GESELLSCHAFT ZUR FÖRDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 1997-11-19 EP disclosed
EP-0755675-B1 Dermatological and/or pharmaceutical composition, process of preparation and utilization OREAL (FR) 1997-09-17 EP disclosed
US-5645985-A USED FOR DIAGNOSIS TO DETECT VIRUSES OR DISEASED CONDITIONS GILEAD SCIENCES, INC. (US) 1997-07-08 US disclosed
EP-0755675-A1 Dermatological and/or pharmaceutical composition, process of preparation and utilization L'OREAL (FR) 1997-01-29 EP disclosed
US-5596091-A DNA AND RNA FOR GENE EXPRESSION FOR DIAGNOSIS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-01-21 US disclosed
WO-1996026743-A1 RADIATION ENHANCED GENE THERAPY FOR TREATMENT OF TUMORS HUMAN GENE THERAPY RESEARCH INSTITUTE (US) 1996-09-06 WO disclosed
WO-1996023506-A1 USE OF 5'SUBSTITUTED NUCLEOSIDES TO PROVIDE RESISTANCE IN CYTOSTATIC TREATMENT AND MEDICAMENTS CONTAINING SAID NUCLEOSIDES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 1996-08-08 WO disclosed
EP-0719272-A1 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS GILEAD SCIENCES, INC. (US) 1996-07-03 EP disclosed
US-5502177-A POLYCYCLIC STRUCTURE BOUND TO OLIGONUCLEOTIDE, FLUORESCENT LABEL, IMMUNOASSAY GILEAD SCIENCES, INC. (US) 1996-03-26 US disclosed
EP-0637965-A4 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES. GILEAD SCIENCES INC (US) 1996-01-24 EP disclosed
US-5434257-A Binding compentent oligomers containing unsaturated 3',5' and 2',5' linkages GILEAD SCIENCES, INC. (US) 1995-07-18 US disclosed
WO-1995011911-A1 BINDING COMPETENT OLIGOMERS CONTAINING UNSATURATED 3',5' AND 2',5' LINKAGES GLAXO WELLCOME INC. (US) 1995-05-04 WO disclosed
WO-1995007918-A2 PYRIMIDINE DERIVATIVES FOR LABELED BINDING PARTNERS GILEAD SCIENCES, INC. (US) 1995-03-23 WO disclosed
EP-0637965-A1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES GILEAD SCIENCES, INC. (US) 1995-02-15 EP disclosed
WO-1993018776-A1 COMBINATIONS OF COMPOUNDS HAVING ANTIVIRAL ACTIVITY CHIESI FARMACEUTICI S.P.A. (IT) 1993-09-30 WO disclosed
WO-1993010820-A1 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES GILEAD SCIENCES, INC. (US) 1993-06-10 WO disclosed
US-5213972-A Production of thymidine and deoxyuridine, intermediates for AZT CHEMGEN CORPORATION (US) 1993-05-25 US disclosed
US-5151507-A Alkynylamino-nucleotides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-09-29 US disclosed
US-4975433-A DRUG DELIVERY FOR TREATING SKIN DISORDERS UNIVERSITY OF FLORIDA (US) 1990-12-04 US disclosed
EP-0160079-B1 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION GREER, Sheldon B. (US) 1990-01-31 EP disclosed
US-4894364-A ANTITUMOR AGENTS HALOGENETICS, INC. 1990-01-16 US disclosed
EP-0339161-A1 Novel fluorophosphonate nucleotide derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-11-02 EP disclosed
EP-0335770-A2 Novel fluorophosphonate nucleotide derivatives MERRELL PHARMACEUTICALS INC. (US) 1989-10-04 EP disclosed
US-4845081-A PRODRUGS, URACILS UNIVERSITY OF FLORIDA (US) 1989-07-04 US disclosed
EP-0258412-A1 COMPOSITION FOR AND METHOD OF TREATING AIDS AND CERTAIN RELATED DISEASES GREER, Sheldon B. (US) 1988-03-09 EP disclosed
WO-1987004929-A1 COMPOSITION FOR AND METHOD OF TREATING AIDS AND CERTAIN RELATED DISEASES GREER SHELDON B 1987-08-27 WO disclosed
US-4594339-A Veterinary medicine SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1986-06-10 US disclosed
EP-0160079-A4 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION. GREER SHELDON B 1986-05-14 EP disclosed
EP-0160079-A1 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION. GREER SHELDON B 1985-11-06 EP disclosed
WO-1985001871-A1 METHOD AND MATERIALS FOR SENSITIZING NEOPLASTIC TISSUE TO RADIATION GREER SHELDON B 1985-05-09 WO disclosed
EP-0010205-B1 5-SUBSTITUTED 1-(2'-DEOXY-2'-SUBSTITUTED-BETA-D-ARABINOFURANOSYL) PYRIMIDINE NUCLEOSIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Sloan-Kettering Institute For Cancer Research (US) 1983-05-04 EP disclosed
US-4211773-A VIRICIDES, ANTITUMOR AGENTS SLOAN KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1980-07-08 US disclosed
US-4210638-A 5-TRIFLUOROMETHYL-2'-DEOXYCYCTIDINE AND TETRAHYDROURIDINE OR 2'-DEOXYTETRAHYDROURIDINE PCR, INC. (US) 1980-07-01 US disclosed
EP-0010205-A1 5-Substituted 1-(2'-deoxy-2'-substituted-beta-D-arabinofuranosyl) pyrimidine nucleosides and pharmaceutical compositions containing them Sloan-Kettering Institute For Cancer Research (US) 1980-04-30 EP disclosed
US-4093715-A 5-Iodo-5'-amino-2',5'-dideoxycytidine and the pharmaceutically acceptable salts thereof RESEARCH CORPORATION (US) 1978-06-06 US disclosed
US-4093715-A 5-Iodo-5'-amino-2',5'-dideoxycytidine and the pharmaceutically acceptable salts thereof RESEARCH CORPORATION (US) 1978-06-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11959137-B2 Synthesis of novel disulfide linker based nucleotides as reversible terminators for DNA sequencing by synthesis POLRMT, RNGTT, MTR DNMT1 86/4885ADRB1 4821/4885TK1 78/4885
US-12606863-B2 Bioluminescent detection of DNA synthesis PCNA, MKI67, POLL DNMT1 54/4885ADRB1 1776/4885TK1 6/4885
US-20100292452-A1 Modified nucleotides ADAR, NT5C2, NSUN2 DNMT1 241/4885ADRB1 2083/4885TK1 142/4885
US-12584168-B2 Sample preparation method POLN, POLRMT, POLM DNMT1 274/4885ADRB1 4500/4885TK1 472/4885
US-20210196723-A1 Modulators of DUX4 for Regulation of Muscle Function DDX21, MBNL1, MECP2 DNMT1 199/4885ADRB1 4348/4885TK1 2815/4885
US-20070259832-A1 Nucleotide mimics and their prodrugs NUDT14, ENTPD5, MTAP DNMT1 570/4885ADRB1 3876/4885TK1 62/4885
US-20070265224-A1 Nucleotide mimics and their prodrugs NUDT14, ENTPD5, MTAP DNMT1 570/4885ADRB1 3876/4885TK1 62/4885
US-11858953-B2 Compositions and methods for synthesis of phosphorylated molecules PIK3CA, CHAMP1, TYMP DNMT1 402/4885ADRB1 4637/4885TK1 22/4885
US-20200239500-A1 Compositions and Methods for Synthesis of Phosphorylated Molecules PIK3CA, CHAMP1, TYMP DNMT1 402/4885ADRB1 4637/4885TK1 22/4885
US-20250236911-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS RNGTT, POLRMT, MTR DNMT1 146/4885ADRB1 4776/4885TK1 112/4885
US-20090259030-A1 STABILIZED NUCLEIC ACID DARK QUENCHER-FLUOROPHORE PROBES DDX1, DDX18, DDX3X DNMT1 177/4885ADRB1 4378/4885TK1 344/4885
US-20220117992-A1 DEOXY-CYTIDINE OR URIDINE DERIVATIVES FOR USE IN CANCER THERAPIES UMPS, UPP1, TYMP DNMT1 697/4885ADRB1 1973/4885TK1 19/4885
US-20220411860-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS POLL, POLQ, POLB DNMT1 252/4885ADRB1 2139/4885TK1 54/4885
US-11920136-B2 Transglutaminase-mediated conjugation TGM2, TGM3, TGM1 DNMT1 277/4885ADRB1 4834/4885TK1 310/4885
US-20160326576-A1 DUAL QUENCHER PROBES DNA2, WRN, DDX42 DNMT1 281/4885ADRB1 4693/4885TK1 1366/4885
US-20220056069-A1 IMMUNOMODULATING POLYNUCLEOTIDES, ANTIBODY CONJUGATES THEREOF, AND METHODS OF THEIR USE TYMP, DUT, PAICS DNMT1 197/4885ADRB1 4437/4885TK1 107/4885
US-20090069546-A1 PYRAZOLE-BASED CYANINE DYE CBR3, CYB5R3, TST DNMT1 3683/4885ADRB1 1209/4885TK1 3542/4885
US-20230028388-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS RNGTT, POLRMT, MTR DNMT1 146/4885ADRB1 4794/4885TK1 107/4885
US-20180274024-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS RNGTT, POLRMT, MTR DNMT1 146/4885ADRB1 4794/4885TK1 107/4885
US-20100112711-A1 METHOD OF DETECTING AMPLIFICATION OR DELETION IN GENOMIC DNA FRAGMENT GLB1, GDA, DNTT DNMT1 199/4885ADRB1 4446/4885TK1 7/4885
US-20030170680-A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines NUDT1, DHX15, DDX5 DNMT1 336/4885ADRB1 3612/4885TK1 43/4885
US-20250263678-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF RNA RNASE1, POLRMT, TERT DNMT1 384/4885ADRB1 4067/4885TK1 156/4885
US-10933068-B2 Modulators of DUX4 for regulation of muscle function DDX21, MBNL1, MECP2 DNMT1 200/4885ADRB1 4347/4885TK1 2927/4885
US-20200172896-A1 EVOLUTION OF BIOACTIVE SEQUENCE-DEFINED SYNTHETIC POLYMERS USING DNA-TEMPLATED POLYMERIZATION PCSK9, IL6, PCSK6 DNMT1 473/4885ADRB1 4715/4885TK1 1078/4885
US-20220257629-A1 COMPOSITIONS AND METHODS FOR UPREGULATION OF HUMAN FETAL HEMOGLOBIN HBB, HBG1, HBG2 DNMT1 647/4885ADRB1 4766/4885TK1 1094/4885
US-11180523-B2 Design, synthesis and use of synthetic nucleotides comprising charge mass tags POLM, RNGTT, TYMP DNMT1 119/4885ADRB1 4810/4885TK1 10/4885
US-20240376536-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS RNGTT, POLRMT, MTR DNMT1 146/4885ADRB1 4776/4885TK1 112/4885
US-20040049008-A1 Templated molecules and methods for using such molecules INTS6, ABL1, INMT DNMT1 319/4885ADRB1 4209/4885TK1 772/4885
US-20180125831-A1 COMBINATION THERAPIES FOR TREATING CANCER TPMT, KRAS, ACE DNMT1 1643/4885ADRB1 335/4885TK1 2512/4885
US-20120178919-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF TYMP, TK1, NUDT1 DNMT1 950/4885ADRB1 1825/4885TK1 2/4885
US-20040265802-A9 ENHANCED TRIPLE-HELIX AND DOUBLE-HELIX FORMATION WITH OLIGOMERS CONTAINING MODIFIED PYRIMIDINES NUDT1, DHX15, DDX5 DNMT1 336/4885ADRB1 3612/4885TK1 43/4885
US-20220396830-A1 BIOLUMINESCENT DETECTION OF DNA SYNTHESIS RNGTT, NUDT1, DNTT DNMT1 74/4885ADRB1 3842/4885TK1 44/4885
US-20180201641-A1 Cytidine-5-Carboxamide Modified Nucleotide Compositions and Methods Related Thereto NT5C3B, CDA, RNGTT DNMT1 127/4885ADRB1 4037/4885TK1 80/4885
US-20190004055-A1 DESIGN, SYNTHESIS AND USE OF SYNTHETIC NUCLEOTIDES COMPRISING CHARGE MASS TAGS POLM, RNGTT, TYMP DNMT1 119/4885ADRB1 4810/4885TK1 10/4885
US-20100016177-A1 TEMPLATED MOLECULES AND METHODS FOR USING SUCH MOLECULES INTS6, ABL1, INMT DNMT1 319/4885ADRB1 4209/4885TK1 772/4885
US-20260066042-A1 METHODS AND SYSTEMS FOR HIGH-THROUGHPUT MOLECULAR ANALYSIS POLRMT, POLL, SARS1 DNMT1 1090/4885ADRB1 2217/4885TK1 1713/4885
US-20220380768-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION TGM2, TGM3, TGM1 DNMT1 277/4885ADRB1 4834/4885TK1 310/4885
US-20030143561-A1 Nucleoside derivatives for library preparation PNP, SAMHD1, DCTD DNMT1 340/4885ADRB1 3875/4885TK1 70/4885
US-20240343753-A1 THERAPEUTIC COMPOUNDS TET1, TET2, TET3 DNMT1 20/4885ADRB1 3545/4885TK1 4778/4885
US-20110118438-A1 CYANINE-TYPE COMPOUNDS HAVING AN ALKYNYL LINKER ARM ACR, RNGTT, NCL DNMT1 716/4885ADRB1 1984/4885TK1 126/4885
US-20170114058-A1 COSMIC QUENCHERS APEX1, NQO2, SQOR DNMT1 61/4885ADRB1 4748/4885TK1 1431/4885
US-20160362737-A1 MODIFIED NUCLEOTIDES ADAR, NT5C2, NSUN2 DNMT1 235/4885ADRB1 2081/4885TK1 143/4885
US-20210047646-A1 Compositions Comprising Immune System Activators and Method of Using Same RNASEL, RNASE1, RNASEH1 DNMT1 306/4885ADRB1 4644/4885TK1 347/4885
US-20130197209-A1 MODIFIED NUCLEOTIDES ADAR, NT5C2, NSUN2 DNMT1 241/4885ADRB1 2083/4885TK1 142/4885
US-20100081137-A1 Click Chemistry for the Production of Reporter Molecules DNTT, RNGTT, NSUN3 DNMT1 552/4885ADRB1 4572/4885TK1 313/4885
US-20220127299-A1 NUCLEOTIDE CLEAVABLE LINKERS AND USES THEREOF NUDT21, CPSF7, DCLRE1A DNMT1 200/4885ADRB1 4880/4885TK1 92/4885
US-20240382610-A1 NECTIN-4 ANTIBODIES AND CONJUGATES NECTIN4, FUT4, VCAM1 DNMT1 1146/4885ADRB1 4494/4885TK1 3241/4885
US-20140221639-A1 RADIOLABELED NUCLEOSIDE ANALOGUE, AND PREPARATION METHOD AND USE THEREOF TYMP, TK1, NUDT1 DNMT1 950/4885ADRB1 1825/4885TK1 2/4885
US-10239908-B2 Cytidine-5-carboxamide modified nucleotide compositions and methods related thereto NT5C3B, CDA, RNGTT DNMT1 127/4885ADRB1 4037/4885TK1 80/4885
US-11963973-B2 Deoxy-cytidine or uridine derivatives for use in cancer therapies UMPS, UPP1, TYMP DNMT1 697/4885ADRB1 1973/4885TK1 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.