Metogest

Metogest

SCHEMBL121047

CC1(C)C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@@H]4[C@H]3CC[C@]2(C)[C@H]1O

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
▸ ALDH1A1 P00352 3/20 0.70
▸ SERPINA6 P08185 2/20 0.70
▸ SHBG P04278 2/20 0.70
▸ SLC22A1 O15245 1/20 0.70
▸ THRB P10828 1/20 0.70
▸ CYP19A1 P11511 2/20 0.60
▸ PGR P06401 3/20 0.55
▸ LMNA P02545 2/20 0.55
▸ CYP3A4 P08684 2/20 0.55
▸ ABCB11 O95342 2/20 0.55
▸ HIF1A Q16665 2/20 0.55
▸ TSHR P16473 1/20 0.55
▸ CYP2C19 P33261 1/20 0.55
▸ ESR1 P03372 1/20 0.55
▸ NR3C1 P04150 1/20 0.55
▸ ADRA2A P08913 1/20 0.55
▸ SLC6A4 P31645 1/20 0.55
▸ MCL1 Q07820 1/20 0.53
▸ CYP1A2 P05177 1/20 0.53
▸ HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10380000 0.89 ALDH1A1 (0.69) ALDH1A1SERPINA6SHBGSLC22A1THRB
SCHEMBL13474805 0.89 ALDH1A1 (0.69) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL17831191 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL22739132 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL11977556 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL11872554 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL5017882 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL11736454 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL12101449 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB
Nandrolone SCHEMBL5021656 0.82 ALDH1A1 (1.00) ALDH1A1SERPINA6SHBGSLC22A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 276 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180177759-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA-GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CEMM - FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GMBH (AT) 2018-06-28 — — US claimed
EP-3285753-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA -GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CeMM - Forschungszentrum für Molekulare Medizin GmbH (AT) 2018-02-28 — — EP claimed
WO-2016170102-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA -GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CEMM - FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GMBH (AT) 2016-10-27 — — WO claimed
WO-2016005599-A1 COMPOSITIONS, METHODS AND USES FOR TREATING GENDER-BIASED IMMUNE DISORDERS BIOCOPEA LIMITED (GB) 2016-01-14 — — WO claimed
US-20160008376-A1 Compositions, Methods and Uses for Treating Gender-Biased Immune Disorders BIOCOPEA LIMITED (GB) 2016-01-14 — — US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 — — US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 — — US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 — — US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 — — US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 — — CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 — — EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 — — WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 — — US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 — — US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
EP-1549292-A2 PHARMACEUTICAL PREPARATIONS, USE OF SAID PREPARATIONS AND METHOD FOR INCREASING THE BIOAVAILABILITY OF MEDICAMENTS FOR PERORAL ADMINISTRATION Schering Aktiengesellschaft (DE) 2005-07-06 — — EP claimed
US-20040223983-A1 Pharmaceutical preparations, use of these preparations and process for increasing the biovailability of pharmaceutical substances to be administered perorally BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2004-11-11 — — US claimed
WO-2004032897-A2 PHARMACEUTICAL PREPARATIONS, USE OF SAID PREPARATIONS AND METHOD FOR INCREASING THE BIOAVAILABILITY OF MEDICAMENTS FOR PERORAL ADMINISTRATION SCHERING AKTIENGESELLSCHAFT (DE) 2004-04-22 — — WO claimed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 — — EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 — — US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 — — US disclosed
US-20250339367-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-06 — — US disclosed
US-12403090-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-09-02 — — US disclosed
US-20250255780-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2025-08-14 — — US disclosed
US-12310922-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2025-05-27 — — US disclosed
US-12290597-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-05-06 — — US disclosed
US-12171723-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2024-12-24 — — US disclosed
EP-4422607-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2024-09-04 — — EP disclosed
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2024-07-25 — — US disclosed
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2024-02-20 — — US disclosed
US-20240050317-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2024-02-15 — — US disclosed
EP-4304554-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES Aquestive Therapeutics, Inc. (US) 2024-01-17 — — EP disclosed
US-20230414452-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2023-12-28 — — US disclosed
EP-4277611-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2023-11-22 — — EP disclosed
US-11806311-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2023-11-07 — — US disclosed
CN-116940351-A Prodrug compositions and methods of treatment 阿奎斯蒂弗医疗股份有限公司 2023-10-24 — — CN disclosed
US-20230295617-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2023-09-21 — — US disclosed
US-20230277448-A1 CHEWABLE FORMULATIONS ELANCO TIERGESUNDHEIT AG (CH) 2023-09-07 — — US disclosed
EP-4208155-A1 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2023-07-12 — — EP disclosed
US-20230149304-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-18 — — US disclosed
US-20230145752-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-11 — — US disclosed
WO-2023076281-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-04 — — WO disclosed
US-20230131450-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2023-04-27 — — US disclosed
WO-2023039125-A1 ADENOSINE RECEPTOR AGONISTS FOR USE IN THE TREATMENT OF CANCER TEON THERAPEUTICS, INC. (US) 2023-03-16 — — WO disclosed
US-20230059204-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PHARMACEUTICAL AGENTS Pike Therapeutics Inc. (CA) 2023-02-23 — — US disclosed
EP-4135712-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES Pike Therapeutics, Inc. (CA) 2023-02-22 — — EP disclosed
WO-2023012691-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PHARMACEUTICAL AGENTS PIKE THERAPEUTICS, INC. (CA) 2023-02-09 — — WO disclosed
US-11541002-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2023-01-03 — — US disclosed
US-20220347117-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES U.S. BANK TRUST COMPANY, NATIONAL ASSOCIATION 2022-11-03 — — US disclosed
EP-4058029-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2022-09-21 — — EP disclosed
WO-2022192476-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2022-09-15 — — WO disclosed
WO-2022187556-A1 THERAPEUTIC METHODS AND COMPOSITIONS COMPRISING MAGNETIZABLE NANOPARTICLES VRG STEM CELL SERVICES INC. (US) 2022-09-09 — — WO disclosed
EP-4051235-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2022-09-07 — — EP disclosed
US-20220233471-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2022-07-28 — — US disclosed
WO-2022155544-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2022-07-21 — — WO disclosed
WO-2022049149-A1 CHEWABLE FORMULATIONS ELANCO TIERGESUNDHEIT AG (CH) 2022-03-10 — — WO disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 — — US disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 — — US disclosed
WO-2021209815-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES PIKE THERAPEUTICS, INC. (CA) 2021-10-21 — — WO disclosed
US-20210322447-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES PIKE THERAPEUTICS INC (CA) 2021-10-21 — — US disclosed
US-20210301346-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2021-09-30 — — US disclosed
US-20210290771-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-09-23 — — US disclosed
EP-3846778-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES Aquestive Therapeutics, Inc. (US) 2021-07-14 — — EP disclosed
EP-3258958-B1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIV VIRGINIA PATENT FOUNDATION (US) 2021-05-26 — — EP disclosed
US-20210145731-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-20 — — US disclosed
WO-2021097247-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-20 — — WO disclosed
US-11000597-B2 Engineered receptor/ligand system for delivery of therapeutic agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-05-11 — — US disclosed
US-20210128511-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-06 — — US disclosed
WO-2021087359-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-06 — — WO disclosed
US-10995374-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2021-05-04 — — US disclosed
EP-3811371-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES Aquestive Therapeutics, Inc. (US) 2021-04-28 — — EP disclosed
WO-2021050564-A2 THERAPEUTIC AGENTS AND METHODS FOR TREATMENT OF LYME DISEASE AND LYME DISEASE-RELATED DISORDERS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2021-03-18 — — WO disclosed
US-10864190-B2 Combination of an antiandrogen with a vitamin K antagonist or with a gamma-glutamyl carboxylase inhibitor for the therapy of androgen receptor positive cancer CeMM—FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GmbH (AT) 2020-12-15 — — US disclosed
US-20200345624-A1 Nanopore Delivery Device HUDSON LEE EDWARD (US) 2020-11-05 — — US disclosed
WO-2020163425-A1 AZLOCILLIN AND DISULFIRAM-BASED FORMULATIONS AND METHODS OF USE FLIGHTPATH BIOSCIENCES, INC. (US) 2020-08-13 — — WO disclosed
EP-3692989-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2020-08-12 — — EP disclosed
US-20200199679-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA 2020-06-25 — — US disclosed
US-10619209-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-04-14 — — US disclosed
US-20200101009-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES U.S. BANK TRUST COMPANY, NATIONAL ASSOCIATION 2020-04-02 — — US disclosed
US-10463611-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2019-11-05 — — US disclosed
US-20190249255-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-08-15 — — US disclosed
US-20190249173-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2019-08-15 — — US disclosed
US-10369340-B2 Device and method for sustained release of low water solubility therapeutic agent in solubilizer NANOMEDICAL SYSTEMS, INC. (US) 2019-08-06 — — US disclosed
US-10363299-B2 Compositions and methods for preventing and treating rhinovirus infections UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2019-07-30 — — US disclosed
EP-2419091-B1 NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS (US) 2019-06-26 — — EP disclosed
EP-3452597-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS Wave Life Sciences Ltd. (SG) 2019-03-13 — — EP disclosed
CN-109462995-A The method and composition of bioactivator 波涛生命科学有限公司 2019-03-12 — — CN disclosed
US-20190021998-A1 TOPICAL NANOEMULSION THERAPY FOR WOUNDS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2019-01-24 — — US disclosed
US-20190002984-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2019-01-03 — — US disclosed
US-20180251840-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIV VIRGINIA PATENT FOUNDATION (US) 2018-09-06 — — US disclosed
US-20180177759-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA-GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CEMM - FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GMBH (AT) 2018-06-28 — — US disclosed
US-20180098970-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS, INC. (US) 2018-04-12 — — US disclosed
EP-3285753-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA -GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CeMM - Forschungszentrum für Molekulare Medizin GmbH (AT) 2018-02-28 — — EP disclosed
US-20180043006-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2018-02-15 — — US disclosed
US-20180015172-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2018-01-18 — — US disclosed
CN-104546669-B Nanochannel device and correlation technique 得克萨斯大学体系董事会 2018-01-05 — — CN disclosed
EP-3258958-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS University Of Virginia Patent Foundation (US) 2017-12-27 — — EP disclosed
WO-2017192679-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2017-11-09 — — WO disclosed
US-20170319698-A1 GASTRORETENTIVE GEL FORMULATIONS JAGOTEC AG (CH) 2017-11-09 — — US disclosed
EP-3212167-A1 GASTRORETENTIVE GEL FORMULATIONS Jagotec AG (CH) 2017-09-06 — — EP disclosed
CN-107106484-A Gastric retention gel preparation 雅戈泰克股份公司 2017-08-29 — — CN disclosed
US-20170226585-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2017-08-10 — — US disclosed
US-20170216314-A1 TOPICAL FORMULATIONS NUVO RESEARCH INC. (CA) 2017-08-03 — — US disclosed
US-9642912-B2 Topical formulations for treating skin conditions CRESCITA THERAPEUTICS INC. (CA) 2017-05-09 — — US disclosed
EP-3156053-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2017-04-19 — — EP disclosed
US-20170100335-A1 TOPICAL NANOEMULSION THERAPY FOR WOUNDS NANOBIO CORPORATION 2017-04-13 — — US disclosed
US-20160376658-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2016-12-29 — — US disclosed
US-9526824-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-12-27 — — US disclosed
EP-2307011-B1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS INC (US) 2016-11-30 — — EP disclosed
EP-2355864-B1 NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS (US) 2016-11-09 — — EP disclosed
WO-2016170102-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA -GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CEMM - FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GMBH (AT) 2016-10-27 — — WO disclosed
WO-2016134288-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2016-08-25 — — WO disclosed
WO-2016118787-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2016-07-28 — — WO disclosed
CN-105744983-A Device and method for sustained release of low water solubility therapeutic agent in solubilizer 纳米医学系统公司 2016-07-06 — — CN disclosed
US-20160175572-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER NANOMEDICAL SYSTEMS, INC. (US) 2016-06-23 — — US disclosed
EP-3033138-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER Nanomedical Systems Inc. (US) 2016-06-22 — — EP disclosed
US-20160139161-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2016-05-19 — — US disclosed
WO-2016066256-A1 GASTRORETENTIVE GEL FORMULATIONS JAGOTEC AG (CH) 2016-05-06 — — WO disclosed
US-9308181-B2 Topical formulations, systems and methods NUVO RESEARCH INC. (CA) 2016-04-12 — — US disclosed
US-9308162-B2 Biocompatible oligomer-polymer compositions TOLMAR THERAPEUTICS, INC. (US) 2016-04-12 — — US disclosed
US-9278134-B2 Dual functioning ionic liquids and salts thereof THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2016-03-08 — — US disclosed
WO-2016005599-A1 COMPOSITIONS, METHODS AND USES FOR TREATING GENDER-BIASED IMMUNE DISORDERS BIOCOPEA LIMITED (GB) 2016-01-14 — — WO disclosed
US-20160008376-A1 Compositions, Methods and Uses for Treating Gender-Biased Immune Disorders BIOCOPEA LIMITED (GB) 2016-01-14 — — US disclosed
WO-2015167760-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF CELANESE ACETATE LLC (US) 2015-11-05 — — WO disclosed
US-20150306230-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF CELANESE ACETATE LLC (US) 2015-10-29 — — US disclosed
US-20150297723-A1 TOPICAL FORMULATIONS FOR TREATING SKIN CONDITIONS NUVO RESEARCH INC. (CA) 2015-10-22 — — US disclosed
WO-2015143386-A1 TOPICAL NANOEMULSION THERAPY FOR WOUNDS THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2015-09-24 — — WO disclosed
US-20150246174-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-09-03 — — US disclosed
EP-2912070-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO Celanese Acetate LLC (US) 2015-09-02 — — EP disclosed
US-9096743-B2 Process for forming films, fibers, and beads from chitinous biomass THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2015-08-04 — — US disclosed
CN-104812777-A Polysaccharide ester microspheres and methods and articles related thereto CELANESE ACETATE LLC 2015-07-29 — — CN disclosed
CN-104546669-A NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS 2015-04-29 — — CN disclosed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 — — US disclosed
US-9005185-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-04-14 — — US disclosed
WO-2015023557-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER NANOMEDICAL SYSTEMS, INC. (US) 2015-02-19 — — WO disclosed
EP-2291174-B1 FLOWABLE COMPOSITION COMPRISING BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS TOLMAR THERAPEUTICS INC (US) 2015-01-28 — — EP disclosed
CN-102271732-B Nanochannel devices and related methods UNIV TEXAS 2014-12-31 — — CN disclosed
CN-104203220-A Device and method for sustained release of therapeutic agent UNIV TEXAS 2014-12-10 — — CN disclosed
US-20140348936-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMOPLASTIC POLYURETHANES CELANESE EVA PERFORMANCE POLYMERS, INC. 2014-11-27 — — US disclosed
US-20140328884-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES CELANESE EVA PERFORMANCE POLYMERS, INC. 2014-11-06 — — US disclosed
US-20140315720-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-10-23 — — US disclosed
EP-2790678-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMPOPLASTIC POLYURETHANES Celanese Eva Performance Polymers, Inc. (US) 2014-10-22 — — EP disclosed
EP-2790677-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES Celanese Eva Performance Polymers, Inc. (US) 2014-10-22 — — EP disclosed
EP-2770984-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-09-03 — — EP disclosed
US-8802596-B2 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2014-08-12 — — US disclosed
US-20140206734-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2014-07-24 — — US disclosed
US-20140180251-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2014-06-26 — — US disclosed
US-20140154313-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2014-06-05 — — US disclosed
WO-2014066463-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-05-01 — — WO disclosed
US-20140113826-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-04-24 — — US disclosed
EP-2717860-A1 CONTROLLED ABSORPTION WATER-SOLUBLE PHARMACEUTICALLY ACTIVE ORGANIC COMPOUND FORMULATION FOR ONCE-DAILY ADMINISTRATION STI Pharma, LLC (US) 2014-04-16 — — EP disclosed
US-8697361-B2 Serotonin transporter gene and treatment of alcoholism UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2014-04-15 — — US disclosed
WO-2014031398-A1 BIOMEDICAL DEVICES COMPRISING MOLDED POLYETHYLENE COMPONENTS TICONA LLC (US) 2014-02-27 — — WO disclosed
US-20140051771-A1 Biomedical Devices Comprising Molded Polyethylene Components TICONA LLC (US) 2014-02-20 — — US disclosed
US-20140052264-A1 Porous, Stabilized Craniomaxillofacial Implants and Methods and Kits Relating Thereto TICONA LLC (US) 2014-02-20 — — US disclosed
US-8632510-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-01-21 — — US disclosed
US-20130337031-A1 TOPICAL FORMULATIONS, SYSTEMS AND METHODS NUVO RESEARCH INC. (CA) 2013-12-19 — — US disclosed
US-20130240483-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2013-09-19 — — US disclosed
CN-103271083-A Multi-functional ionic liquid compositions UNIV ALABAMA 2013-09-04 — — CN disclosed
US-8513304-B2 Topical formulation NUVO RESEARCH INC. (CA) 2013-08-20 — — US disclosed
US-8480637-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-07-09 — — US disclosed
WO-2013090893-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMPOPLASTIC POLYURETHANES CELANESE EVA PERFORMANCE POLYMERS, INC. (US) 2013-06-20 — — WO disclosed
WO-2013090891-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES CELANESE EVA PERFORMANCE POLYMERS, INC. (US) 2013-06-20 — — WO disclosed
CN-101326275-B Multifunctional ionic liquid composition UNIV ALABAMA 2013-06-05 — — CN disclosed
US-8454582-B2 Methods and devices for the treatment of ocular conditions SURMODICS, INC. (US) 2013-06-04 — — US disclosed
US-20130131628-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-23 — — US disclosed
WO-2013063004-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-02 — — WO disclosed
EP-2255184-B1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM Univ Virginia Patent Found (US) 2013-04-24 — — EP disclosed
US-20130079404-A1 TOPICAL FORMULATION NUVO RESEARCH INC. (CA) 2013-03-28 — — US disclosed
EP-2556830-A1 Combined effects of topiramate, ondansetron and naltrexone on alcohol consumption UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2013-02-13 — — EP disclosed
US-8343962-B2 Topical formulation NUVO RESEARCH INC. (CA) 2013-01-01 — — US disclosed
WO-2012170676-A1 CONTROLLED ABSORPTION WATER-SOLUBLE PHARMACEUTICALLY ACTIVE ORGANIC COMPOUND FORMULATION FOR ONCE-DAILY ADMINISTRATION STI PHARMA, LLC (US) 2012-12-13 — — WO disclosed
US-20120302592-A1 TOPIRAMATE PLUS NALTREXONE FOR THE TREATMENT OF ADDICTIVE DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-11-29 — — US disclosed
US-8314077-B2 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. (US) 2012-11-20 — — US disclosed
US-20120264605-A1 Multi-Functional Ionic Liquid Compositions for Overcoming Polymorphism and Imparting Improved Properties for Active Pharmaceutical, Biological, Nutritional, and Energetic Ingredients THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-10-18 — — US disclosed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 — — US disclosed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 — — US disclosed
US-8232265-B2 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-07-31 — — US disclosed
US-20120115729-A1 PROCESS FOR FORMING FILMS, FIBERS, AND BEADS FROM CHITINOUS BIOMASS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-05-10 — — US disclosed
US-20120115149-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-05-10 — — US disclosed
US-20120095443-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-04-19 — — US disclosed
US-8158152-B2 Preparing lyophilizates, especially those free of undesired extra components such as mono- or disaccharides; dosage forms of a wide variety of over 2000 drugs, such as rapidly dissolving tablets SCIDOSE LLC (US) 2012-04-17 — — US disclosed
EP-2425013-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM University Of Virginia Patent Foundation (US) 2012-03-07 — — EP disclosed
US-20120046244-A1 DUAL FUNCTIONING IONIC LIQUIDS AND SALTS THEREOF THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-02-23 — — US disclosed
EP-2419091-A2 NANOCHANNELED DEVICE AND RELATED METHODS The Board of Regents of The University of Texas System (US) 2012-02-22 — — EP disclosed
US-20110245172-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS TOLMAR THERAPEUTICS, INC. (US) 2011-10-06 — — US disclosed
EP-2355864-A2 NANOCHANNELED DEVICE AND RELATED METHODS The Board of Regents of The University of Texas System (US) 2011-08-17 — — EP disclosed
US-7976871-B2 Modified release composition of highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2011-07-12 — — US disclosed
US-20110159073-A1 METHODS AND DEVICES FOR THE TREATMENT OF OCULAR CONDITIONS DEJUAN EUGENE 2011-06-30 — — US disclosed
US-7951398-B2 Pharmaceutical preparation comprising an active dispersed on a matrix NYCOMED GMBH (DE) 2011-05-31 — — US disclosed
US-20110112159-A1 SEROTONIN TRANSPORTER GENE AND TREAMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2011-05-12 — — US disclosed
EP-2307011-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2011-04-13 — — EP disclosed
CN-102016571-A Serotonin transporter gene and treatment of alcoholism UNIV VIRGINIA 2011-04-13 — — CN disclosed
US-20110065628-A1 Medication Combinations for the Treatment of Alcoholism and Drug Addiction UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2011-03-17 — — US disclosed
US-7905852-B2 Skin-contacting-adhesive free dressing JENNINGS-SPRING BARBARA 2011-03-15 — — US disclosed
EP-2291174-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS Tolmar Therapeutics, Inc. (US) 2011-03-09 — — EP disclosed
US-20110028460-A1 TOPICAL FORMULATION FQUBED, INC. 2011-02-03 — — US disclosed
WO-2010141470-A2 PROCESS FOR FORMING FILMS, FIBERS, AND BEADS FROM CHITINOUS BIOMASS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2010-12-09 — — WO disclosed
EP-2255184-A2 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM University Of Virginia Patent Foundation (US) 2010-12-01 — — EP disclosed
WO-2010126603-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-11-04 — — WO disclosed
WO-2010120817-A2 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-10-21 — — WO disclosed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 — — US disclosed
CN-101810592-A Contain the pharmaceutical preparation that is dispersed in the active matter in the substrate ALTANA PHARMA AG 2010-08-25 — — CN disclosed
WO-2010078300-A1 DUAL FUNCTIONING IONIC LIQUIDS AND SALTS THEREOF THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2010-07-08 — — WO disclosed
US-20100152699-A1 Nanochanneled Device and Related Methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-06-17 — — US disclosed
WO-2010056986-A2 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-05-20 — — WO disclosed
US-20100076006-A1 Topiramate Plus Naltrexone for the Treatment of Addictive Disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-03-25 — — US disclosed
WO-2010024870-A1 SKIN-CONTACTING-ADHESIVE FREE DRESSING JENNINGS-SPRING BARBARA BROOKE (US) 2010-03-04 — — WO disclosed
CN-101663028-A Combined effect of topiramate and ondansetron on alcohol consumption UNIV VIRGINIA 2010-03-03 — — CN disclosed
US-20100041689-A1 Combined Effects of Topiramate and Ondansetron on Alcohol Consumption UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-02-18 — — US disclosed
US-20090318520-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS DRIVE (US) 2009-12-24 — — US disclosed
WO-2009155139-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS, INC. (US) 2009-12-23 — — WO disclosed
WO-2009148581-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS QLT USA, INC. (US) 2009-12-10 — — WO disclosed
EP-2124909-A2 COMBINED EFFECTS OF TOPIRAMATE AND ONDANSETRON ON ALCOHOL CONSUMPTION University Of Virginia Patent Foundation (US) 2009-12-02 — — EP disclosed
CN-100548290-C Sulfamate derivatives is used for the treatment of the purposes of impulse control disorder UNIV CINCINNATI (US) 2009-10-14 — — CN disclosed
WO-2009108837-A2 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2009-09-03 — — WO disclosed
WO-2009029308-A1 MEDICATION COMBINATIONS FOR THE TREATMENT OF ALCOHOLISM AND DRUG ADDICTION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2009-03-05 — — WO disclosed
US-20090005722-A1 Skin-contacting-adhesive free dressing JENNLNGS-SPRING BARBARA 2009-01-01 — — US disclosed
US-20080319092-A1 Transdermal Drug Delivery Formulation NUVO RESEARCH INC. (CA) 2008-12-25 — — US disclosed
CN-101326275-A Multifunctional ionic liquid composition UNIV ALABAMA (US) 2008-12-17 — — CN disclosed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 — — EP disclosed
WO-2008095086-A2 TOPIRAMATE PLUS NALTREXONE FOR THE TREATMENT OF ADDICTIVE DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-08-07 — — WO disclosed
WO-2008077092-A2 COMBINED EFFECTS OF TOPIRAMATE AND ONDANSETRON ON ALCOHOL CONSUMPTION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-06-26 — — WO disclosed
EP-1931760-A2 MULTI-FUNCTIONAL IONIC LIQUID COMPOSITIONS The University of Alabama (US) 2008-06-18 — — EP disclosed
EP-1909772-A1 TRANSDERMAL DRUG DELIVERY FORMULATION Nuvo Research Inc. (CA) 2008-04-16 — — EP disclosed
US-20070269379-A1 Penetration Enhancer Combinations for Transdermal Delivery REGENTS OF THE UNIVERSITY OF CALIFORNIA, THE 2007-11-22 — — US disclosed
US-20070122474-A1 Pharmaceutical preparation comprising an active dispersed on a matrix ALTANA PHARMA AG 2007-05-31 — — US disclosed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 — — WO disclosed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 — — US disclosed
US-20070093462-A1 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA 2007-04-26 — — US disclosed
WO-2007044693-A2 MULTI-FUNCTIONAL IONIC LIQUID COMPOSITIONS THE UNIVERSITY OF ALABAMA (US) 2007-04-19 — — WO disclosed
US-7199151-B2 DHA-pharmaceutical agent conjugates of taxanes LUITPOLD PHARMACEUTICALS, INC. (US) 2007-04-03 — — US disclosed
WO-2007016766-A1 TRANSDERMAL DRUG DELIVERY FORMULATION NUVO RESEARCH INC. (CA) 2007-02-15 — — WO disclosed
US-7175854-B2 Pharmaceutical preparation comprising an active dispersed on a matrix ALTANA PHARMA AG (DE) 2007-02-13 — — US disclosed
US-20060110428-A1 Methods and devices for the treatment of ocular conditions SURMODICS MD, LLC 2006-05-25 — — US disclosed
WO-2006014484-A2 METHODS AND DEVICES FOR THE TREATMENT OF OCULAR CONDITIONS SURMODICS, INC. (US) 2006-02-09 — — WO disclosed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 — — US disclosed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US disclosed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US disclosed
US-20050250709-A1 Anti-neoplastic agents, combination therapies and related methods BIONAUT PHARMACEUTICALS (US) 2005-11-10 — — US disclosed
WO-2005060951-A2 ANTI-NEOPLASTIC AGENTS, COMBINATION THERAPIES AND RELATED METHODS BIONAUT PHARMACEUTICALS, INC. (US) 2005-07-07 — — WO disclosed
EP-1549292-A2 PHARMACEUTICAL PREPARATIONS, USE OF SAID PREPARATIONS AND METHOD FOR INCREASING THE BIOAVAILABILITY OF MEDICAMENTS FOR PERORAL ADMINISTRATION Schering Aktiengesellschaft (DE) 2005-07-06 — — EP disclosed
EP-1158973-B1 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIV CINCINNATI (US) 2005-05-04 — — EP disclosed
WO-2005009510-A2 PENETRATION ENHANCER COMBINATIONS FOR TRANSDERMAL DELIVERY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2005-02-03 — — WO disclosed
US-20050002865-A1 Diagnostic/therapeutic agents AMERSHAM HEALTH AS (NO) 2005-01-06 — — US disclosed
US-20040223983-A1 Pharmaceutical preparations, use of these preparations and process for increasing the biovailability of pharmaceutical substances to be administered perorally BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2004-11-11 — — US disclosed
EP-1466628-A1 DHA-pharmaceutical agent conjugates Luitpold Pharmaceuticals, Inc. (US) 2004-10-13 — — EP disclosed
US-20040180949-A1 conjugates of pharmaceutical agents and a highly lipphilic group, a C22 unbranched carbon chain; render the activity of these compounds selective for colon tissue, breast tissue and central nervous system tissue PROTARGA, INC. 2004-09-16 — — US disclosed
CN-1523980-A Pharmaceutical formulations containing an active dispersed in a matrix ��̹��ҽҩ��˾ 2004-08-25 — — CN disclosed
US-20040141922-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2004-07-22 — — US disclosed
US-20040106589-A1 Fatty acid-pharmaceutical agent conjugates PROTARGA PHARMACEUTICALS, INC. 2004-06-03 — — US disclosed
WO-2004032897-A2 PHARMACEUTICAL PREPARATIONS, USE OF SAID PREPARATIONS AND METHOD FOR INCREASING THE BIOAVAILABILITY OF MEDICAMENTS FOR PERORAL ADMINISTRATION SCHERING AKTIENGESELLSCHAFT (DE) 2004-04-22 — — WO disclosed
US-20040058896-A1 Pharmaceutical preparation comprising an active dispersed on a matrix ASTRAZENECA AB (SE) 2004-03-25 — — US disclosed
US-6680047-B2 FOR USE IN ULTRASOUND IMAGING, CONTRAST AGENTS AMERSHAM HEALTH AS (NO) 2004-01-20 — — US disclosed
EP-1341527-A1 PHARMACEUTICAL PREPARATION COMPRISING AN ACTIVE DISPERSED ON A MATRIX ALTANA Pharma AG (DE) 2003-09-10 — — EP disclosed
US-6602902-B2 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid PROTARGA, INC. 2003-08-05 — — US disclosed
US-6576636-B2 Treating a noncentral nervous system by administering a covalent conjugate of a C8-26, unbranched, naturally occurring fatty acid and a drug, provided the drug is not an adenosine receptor agonist/antagonist; anticarcinogenics PROTARGA, INC. 2003-06-10 — — US disclosed
US-20030059471-A1 Oral delivery formulation COMPTON BRUCE JON (US) 2003-03-27 — — US disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 — — US disclosed
US-20020102217-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 — — US disclosed
CN-1360500-A Use of sulfamate derivatives for the treatment of impulse control disorders UNIV CINCINNATI (US) 2002-07-24 — — CN disclosed
WO-2002045693-A1 PHARMACEUTICAL PREPARATION COMPRISING AN ACTIVE DISPERSED ON A MATRIX ALTANA PHARMA AG (DE) 2002-06-13 — — WO disclosed
US-20020010208-A1 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid LUITPOLD PHARMACEUTICALS, INC. 2002-01-24 — — US disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 — — US disclosed
EP-1158973-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2001-12-05 — — EP disclosed
US-6323236-B2 PSYCHOLOGICAL DISORDERS UNIVERSITY OF CINCINNATI 2001-11-27 — — US disclosed
US-20010023254-A1 Psychological disorders CINCINNATI, UNIVERSITY OF 2001-09-20 — — US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 — — US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 — — US disclosed
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. 2001-05-31 — — US disclosed
WO-2000050020-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2000-08-31 — — WO disclosed
WO-1999030690-A1 ORAL DELIVERY FORMULATION AXIA THERAPEUTICS, INC. (US) 1999-06-24 — — WO disclosed
EP-0909183-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES Neuromedica, Inc. (US) 1999-04-21 — — EP disclosed
US-5795909-A ANTICARCINOGENIC AND ANTITUMOR AGENTS; BREAST, COLON, OVARIANCANCERS NEUROMEDICA, INC. (US) 1998-08-18 — — US disclosed
WO-1997044063-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES NEUROMEDICA, INC. (US) 1997-11-27 — — WO disclosed
WO-1997044063-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES NEUROMEDICA, INC. (US) 1997-11-27 — — WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120264605-A1 Multi-Functional Ionic Liquid Compositions for Overcoming Polymorphism and Imparting Improved Properties for Active Pharmaceutical, Biological, Nutritional, and Energetic Ingredients SLC5A6, PNLIP, IPMK ALDH1A1 2937/4885SERPINA6 1294/4885SHBG 3301/4885
US-20150306230-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF PGRMC2, PGRMC1, CYP3A43 ALDH1A1 3882/4885SERPINA6 963/4885SHBG 18/4885
US-20040141922-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 ALDH1A1 4549/4885SERPINA6 97/4885SHBG 1029/4885
US-20180043006-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS CD4, HLA-DRB1, CD74 ALDH1A1 4488/4885SERPINA6 120/4885SHBG 2791/4885
US-20110245172-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS BMP2, CHERP, PUF60 ALDH1A1 3666/4885SERPINA6 2960/4885SHBG 1599/4885
US-10619209-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20070093462-A1 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients SLC5A6, PNLIP, IPMK ALDH1A1 2937/4885SERPINA6 1294/4885SHBG 3301/4885
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20190021998-A1 TOPICAL NANOEMULSION THERAPY FOR WOUNDS CUTA, MMP8, DSG1 ALDH1A1 2106/4885SERPINA6 723/4885SHBG 4597/4885
US-20020010208-A1 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid FABP7, FADS2, ALOX5 ALDH1A1 1451/4885SERPINA6 999/4885SHBG 1819/4885
US-20180251840-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 427/4885SERPINA6 1315/4885SHBG 2146/4885
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20110065628-A1 Medication Combinations for the Treatment of Alcoholism and Drug Addiction SLC6A3, SLC6A4, ADH5 ALDH1A1 210/4885SERPINA6 2016/4885SHBG 2655/4885
US-20210128511-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT ADRA2C, ADRB3, ADRA2B ALDH1A1 559/4885SERPINA6 433/4885SHBG 362/4885
US-20190249255-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 427/4885SERPINA6 1315/4885SHBG 2146/4885
US-20230277448-A1 CHEWABLE FORMULATIONS SI, TAS2R39, TAS2R31 ALDH1A1 4640/4885SERPINA6 2353/4885SHBG 2746/4885
US-20100041689-A1 Combined Effects of Topiramate and Ondansetron on Alcohol Consumption SLC6A3, SLC6A4, HTR5A ALDH1A1 176/4885SERPINA6 1425/4885SHBG 2735/4885
US-20050002865-A1 Diagnostic/therapeutic agents FUS, HNRNPF, HNRNPR ALDH1A1 3855/4885SERPINA6 35/4885SHBG 137/4885
US-20220233471-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT CYP2C19, PAICS, CYP2B6 ALDH1A1 1571/4885SERPINA6 1234/4885SHBG 1958/4885
US-20140206734-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 427/4885SERPINA6 1315/4885SHBG 2146/4885
US-20200199679-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20210322447-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES OPRL1, OPRM1, HTR2A ALDH1A1 2870/4885SERPINA6 2790/4885SHBG 773/4885
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates FABP7, FFAR2, FFAR4 ALDH1A1 615/4885SERPINA6 1732/4885SHBG 2636/4885
US-10995374-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20040180949-A1 conjugates of pharmaceutical agents and a highly lipphilic group, a C22 unbranched carbon chain; render the activity of these compounds selective for colon tissue, breast tissue and central nervous system tissue ALOX12, FABP2, ALOX15B ALDH1A1 1137/4885SERPINA6 1065/4885SHBG 2348/4885
US-20170226585-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 427/4885SERPINA6 1315/4885SHBG 2146/4885
US-20110112159-A1 SEROTONIN TRANSPORTER GENE AND TREAMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 281/4885SERPINA6 1680/4885SHBG 2547/4885
US-20100076006-A1 Topiramate Plus Naltrexone for the Treatment of Addictive Disorders SLC6A3, SLC6A4, SLC6A2 ALDH1A1 156/4885SERPINA6 3030/4885SHBG 1866/4885
US-20230295617-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS ELOVL6, ELOVL5, ELOVL1 ALDH1A1 2846/4885SERPINA6 1899/4885SHBG 420/4885
US-20130337031-A1 TOPICAL FORMULATIONS, SYSTEMS AND METHODS SMURF1, SMURF2, SMS ALDH1A1 3386/4885SERPINA6 3668/4885SHBG 1630/4885
US-20190002984-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 ALDH1A1 427/4885SERPINA6 1315/4885SHBG 2146/4885
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES SORD, SLC6A13, CACNA1A ALDH1A1 683/4885SERPINA6 2915/4885SHBG 527/4885
US-20110028460-A1 TOPICAL FORMULATION SPTLC1, SPTSSB, SPTLC3 ALDH1A1 4194/4885SERPINA6 3170/4885SHBG 4106/4885
US-10363299-B2 Compositions and methods for preventing and treating rhinovirus infections CD4, HLA-DRB1, CD74 ALDH1A1 4488/4885SERPINA6 120/4885SHBG 2791/4885
US-20040106589-A1 Fatty acid-pharmaceutical agent conjugates FABP7, FFAR2, FFAR4 ALDH1A1 615/4885SERPINA6 1732/4885SHBG 2636/4885
US-20120046244-A1 DUAL FUNCTIONING IONIC LIQUIDS AND SALTS THEREOF SLC6A6, SLC10A2, CLK2 ALDH1A1 3146/4885SERPINA6 1274/4885SHBG 793/4885
US-20210301346-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 ALDH1A1 718/4885SERPINA6 1665/4885SHBG 2104/4885
US-20050250709-A1 Anti-neoplastic agents, combination therapies and related methods HRAS, TP53, MYC ALDH1A1 2439/4885SERPINA6 2458/4885SHBG 4787/4885
US-20150297723-A1 TOPICAL FORMULATIONS FOR TREATING SKIN CONDITIONS SMURF1, SGMS1, SMURF2 ALDH1A1 3339/4885SERPINA6 461/4885SHBG 903/4885
US-20010023254-A1 Psychological disorders DRD2, DRD3, DRD1 ALDH1A1 606/4885SERPINA6 3310/4885SHBG 804/4885
US-20170216314-A1 TOPICAL FORMULATIONS SMURF1, SGMS1, SPTLC1 ALDH1A1 3342/4885SERPINA6 2888/4885SHBG 2311/4885
US-20230059204-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PHARMACEUTICAL AGENTS OPRM1, OPRL1, OPRK1 ALDH1A1 3472/4885SERPINA6 3301/4885SHBG 749/4885
US-20180098970-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS INMT, PNMT, SLC6A2 ALDH1A1 617/4885SERPINA6 2000/4885SHBG 2793/4885
US-20090318520-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS INMT, PNMT, SLC6A2 ALDH1A1 814/4885SERPINA6 1870/4885SHBG 2957/4885
US-20190249173-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS ELOVL6, ELOVL5, ELOVL1 ALDH1A1 2811/4885SERPINA6 1972/4885SHBG 423/4885
US-20130079404-A1 TOPICAL FORMULATION SPTLC1, SPTLC3, SARAF ALDH1A1 4496/4885SERPINA6 2761/4885SHBG 3706/4885
US-20120302592-A1 TOPIRAMATE PLUS NALTREXONE FOR THE TREATMENT OF ADDICTIVE DISORDERS SLC6A3, SLC6A4, SLC6A2 ALDH1A1 156/4885SERPINA6 3030/4885SHBG 1866/4885
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 ALDH1A1 4459/4885SERPINA6 109/4885SHBG 951/4885
US-20170100335-A1 TOPICAL NANOEMULSION THERAPY FOR WOUNDS CUTA, MMP8, DSG1 ALDH1A1 2106/4885SERPINA6 723/4885SHBG 4597/4885
US-20120115729-A1 PROCESS FOR FORMING FILMS, FIBERS, AND BEADS FROM CHITINOUS BIOMASS CHIA, CHIT1, CHI3L1 ALDH1A1 4300/4885SERPINA6 2118/4885SHBG 3554/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.

Send feedback