Prinoxodan

Prinoxodan

SCHEMBL122042

CN1Cc2cc(C3=NNC(=O)CC3)ccc2NC1=O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
▸ PDE3B Q13370 14/20 0.55
▸ PDE3A Q14432 14/20 0.55
▸ PDE4A P27815 7/20 0.55
▸ PDE4B Q07343 7/20 0.55
▸ PDE4C Q08493 7/20 0.55
▸ PDE4D Q08499 7/20 0.55
▸ BRD4 O60885 3/20 0.55
▸ CREBBP Q92793 2/20 0.52
▸ BRD2 P25440 1/20 0.52
▸ SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10595977 0.81 PDE3B (0.64) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL2930091 0.80 PDE3B (0.63) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL7417981 0.76 PDE3B (0.57) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10835125 0.74 PDE3B (0.59) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL20889281 0.74 BRD4 (0.60) PDE3BPDE3ABRD4CREBBPBRD2
SCHEMBL7420928 0.73 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL7414950 0.73 PDE3B (0.61) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10597216 0.73 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11317512 0.73 PDE3B (0.68) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10596133 0.72 PDE3B (0.61) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 285 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3621593-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2020-03-18 — — EP claimed
WO-2019194866-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2019-10-10 — — WO claimed
US-20190231786-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES CARDIX Therapeutics, LLC 2019-08-01 — — US claimed
US-20190070184-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2019-03-07 — — US claimed
US-20180325907-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES CARDIX Therapeutics, LLC 2018-11-15 — — US claimed
WO-2018208723-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2018-11-15 — — WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 — — US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 — — US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 — — US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 — — US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 — — EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 — — WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 — — US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 — — US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US claimed
EP-0247177-A4 BENZODIAZINONE-PYRIDAZINONE AND HYDROXY-PYRAZOLYL COMPOUNDS, CARDIOTONIC COMPOSITIONS INCLUDING THE SAME, AND THEIR USES. RORER INTERNAT OVERSEAS INC (US) 1988-04-06 — — EP claimed
EP-0247177-A1 BENZODIAZINONE-PYRIDAZINONE AND HYDROXY-PYRAZOLYL COMPOUNDS, CARDIOTONIC COMPOSITIONS INCLUDING THE SAME, AND THEIR USES RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1987-12-02 — — EP claimed
WO-1987003201-A1 BENZODIAZINONE-PYRIDAZINONE AND HYDROXY-PYRAZOLYL COMPOUNDS, CARDIOTONIC COMPOSITIONS INCLUDING THE SAME, AND THEIR USES RORER INTERNATIONAL (OVERSEAS) INC. (US) 1987-06-04 — — WO claimed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 — — EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 — — US disclosed
US-12472186-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases Cardix Therapeutics LLC (US) 2025-11-18 — — US disclosed
US-20250345308-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS ANSELLA THERAPEUTICS INC (US) 2025-11-13 — — US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 — — US disclosed
US-20250339367-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-06 — — US disclosed
US-12403090-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-09-02 — — US disclosed
US-20250255780-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2025-08-14 — — US disclosed
US-12310922-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2025-05-27 — — US disclosed
US-12290597-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-05-06 — — US disclosed
US-12201607-B2 Compositions and methods for preventing and treating conditions Ansella Therapeutics, Inc. (US) 2025-01-21 — — US disclosed
US-12171723-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2024-12-24 — — US disclosed
EP-4422607-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2024-09-04 — — EP disclosed
US-20240285639-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2024-08-29 — — US disclosed
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2024-07-25 — — US disclosed
US-20240207279-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2024-06-27 — — US disclosed
US-11951107-B2 Deuterated pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2024-04-09 — — US disclosed
US-11911389-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases Cardix Therapeutics LLC (US) 2024-02-27 — — US disclosed
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2024-02-20 — — US disclosed
US-20240050317-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2024-02-15 — — US disclosed
US-11878017-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2024-01-23 — — US disclosed
EP-4304554-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES Aquestive Therapeutics, Inc. (US) 2024-01-17 — — EP disclosed
US-20230414452-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES AQUESTIVE THERAPEUTICS, INC. (US) 2023-12-28 — — US disclosed
EP-4277611-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2023-11-22 — — EP disclosed
US-11806311-B2 System and method for making personalized individual unit doses containing pharmaceutical actives AQUESTIVE THERAPEUTICS, INC. (US) 2023-11-07 — — US disclosed
US-20230295617-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2023-09-21 — — US disclosed
US-20230277448-A1 CHEWABLE FORMULATIONS ELANCO TIERGESUNDHEIT AG (CH) 2023-09-07 — — US disclosed
EP-4208155-A1 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2023-07-12 — — EP disclosed
US-20230149304-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-18 — — US disclosed
US-20230145752-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-11 — — US disclosed
WO-2023076281-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2023-05-04 — — WO disclosed
US-20230131450-A1 ORAL AND NASAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2023-04-27 — — US disclosed
US-20230107723-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2023-04-06 — — US disclosed
US-20230071157-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2023-03-09 — — US disclosed
US-20230059204-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PHARMACEUTICAL AGENTS Pike Therapeutics Inc. (CA) 2023-02-23 — — US disclosed
EP-4135712-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES Pike Therapeutics, Inc. (CA) 2023-02-22 — — EP disclosed
WO-2023012691-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PHARMACEUTICAL AGENTS PIKE THERAPEUTICS, INC. (CA) 2023-02-09 — — WO disclosed
US-11541002-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2023-01-03 — — US disclosed
US-11510924-B2 Deuterated pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2022-11-29 — — US disclosed
US-11491159-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2022-11-08 — — US disclosed
US-20220347117-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES U.S. BANK TRUST COMPANY, NATIONAL ASSOCIATION 2022-11-03 — — US disclosed
EP-4058029-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2022-09-21 — — EP disclosed
WO-2022192476-A1 DOSAGE FORMS HAVING EQUIVALENT BIOCOMPARABLE PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2022-09-15 — — WO disclosed
WO-2022187556-A1 THERAPEUTIC METHODS AND COMPOSITIONS COMPRISING MAGNETIZABLE NANOPARTICLES VRG STEM CELL SERVICES INC. (US) 2022-09-09 — — WO disclosed
EP-4051235-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT Aquestive Therapeutics, Inc. (US) 2022-09-07 — — EP disclosed
US-20220233471-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2022-07-28 — — US disclosed
WO-2022155544-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2022-07-21 — — WO disclosed
US-20220184089-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2022-06-16 — — US disclosed
WO-2022049149-A1 CHEWABLE FORMULATIONS ELANCO TIERGESUNDHEIT AG (CH) 2022-03-10 — — WO disclosed
US-11266651-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2022-03-08 — — US disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 — — US disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 — — US disclosed
US-20210322447-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES PIKE THERAPEUTICS INC (CA) 2021-10-21 — — US disclosed
WO-2021209815-A1 TRANSDERMAL MICRO-DOSING DELIVERY OF PSYCHEDELICS DERIVATIVES PIKE THERAPEUTICS, INC. (CA) 2021-10-21 — — WO disclosed
US-20210301346-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2021-09-30 — — US disclosed
US-20210290771-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-09-23 — — US disclosed
EP-3846778-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES Aquestive Therapeutics, Inc. (US) 2021-07-14 — — EP disclosed
EP-3258958-B1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIV VIRGINIA PATENT FOUNDATION (US) 2021-05-26 — — EP disclosed
US-20210145731-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-20 — — US disclosed
WO-2021097247-A1 MULTIMODAL COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-20 — — WO disclosed
US-11000597-B2 Engineered receptor/ligand system for delivery of therapeutic agents UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2021-05-11 — — US disclosed
US-20210128511-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-06 — — US disclosed
WO-2021087359-A1 PRODRUG COMPOSITIONS AND METHODS OF TREATMENT AQUESTIVE THERAPEUTICS, INC. (US) 2021-05-06 — — WO disclosed
US-10995374-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2021-05-04 — — US disclosed
EP-3811371-A1 SYSTEM AND METHOD FOR MAKING PERSONALIZED INDIVIDUAL UNIT DOSES CONTAINING PHARMACEUTICAL ACTIVES Aquestive Therapeutics, Inc. (US) 2021-04-28 — — EP disclosed
CN-109890366-B Combination medicine for treating cardiovascular diseases and preparation and use methods thereof 美进医药公司 2020-12-25 — — CN disclosed
US-20200397793-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2020-12-24 — — US disclosed
US-20200360340-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS ANSELLA THERAPEUTICS INC (US) 2020-11-19 — — US disclosed
US-20200345624-A1 Nanopore Delivery Device HUDSON LEE EDWARD (US) 2020-11-05 — — US disclosed
EP-3727382-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS Ansella Therapeutics, Inc. (US) 2020-10-28 — — EP disclosed
US-10758544-B2 Pharmaceutical compositions and methods of treating cardiovascular diseases CARDIX Therapeutics, LLC (US) 2020-09-01 — — US disclosed
EP-3692989-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2020-08-12 — — EP disclosed
US-20200199679-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA 2020-06-25 — — US disclosed
US-10668046-B2 Compositions and methods for preventing and treating conditions Ansella Therapeutics, Inc. (US) 2020-06-02 — — US disclosed
US-10619209-B2 Serotonin transporter gene and treatment of opioid-related disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-04-14 — — US disclosed
US-20200101009-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES U.S. BANK TRUST COMPANY, NATIONAL ASSOCIATION 2020-04-02 — — US disclosed
EP-3621593-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2020-03-18 — — EP disclosed
US-10463611-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2019-11-05 — — US disclosed
WO-2019194866-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2019-10-10 — — WO disclosed
US-20190249173-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2019-08-15 — — US disclosed
US-20190249255-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-08-15 — — US disclosed
US-10369340-B2 Device and method for sustained release of low water solubility therapeutic agent in solubilizer NANOMEDICAL SYSTEMS, INC. (US) 2019-08-06 — — US disclosed
US-20190231786-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES CARDIX Therapeutics, LLC 2019-08-01 — — US disclosed
US-10363299-B2 Compositions and methods for preventing and treating rhinovirus infections UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2019-07-30 — — US disclosed
EP-2419091-B1 NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS (US) 2019-06-26 — — EP disclosed
US-20190183854-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING CONDITIONS Ansella Therapeutics, Inc. 2019-06-20 — — US disclosed
CN-109890366-A Combination medicine for treating cardiovascular diseases and preparation and use methods thereof 美进医药公司 2019-06-14 — — CN disclosed
EP-3452597-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS Wave Life Sciences Ltd. (SG) 2019-03-13 — — EP disclosed
CN-109462995-A The method and composition of bioactivator 波涛生命科学有限公司 2019-03-12 — — CN disclosed
US-20190070184-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2019-03-07 — — US disclosed
US-20190002984-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2019-01-03 — — US disclosed
US-20180325907-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES CARDIX Therapeutics, LLC 2018-11-15 — — US disclosed
WO-2018208723-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES Cardix Therapeutics LLC (US) 2018-11-15 — — WO disclosed
US-20180251840-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIV VIRGINIA PATENT FOUNDATION (US) 2018-09-06 — — US disclosed
US-20180098970-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS, INC. (US) 2018-04-12 — — US disclosed
WO-2018055211-A1 NOVEL COMPOUNDS AND METHODS FOR MODULATING UBIQUITINATION Johann Wolfgang Goethe-Universität Frankfurt am Main (DE) 2018-03-29 — — WO disclosed
EP-3299460-A1 NOVEL COMPOUNDS AND METHODS FOR MODULATING UBIQUITINATION Johann Wolfgang Goethe-Universität Frankfurt am Main (DE) 2018-03-28 — — EP disclosed
US-20180043006-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2018-02-15 — — US disclosed
US-20180015172-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2018-01-18 — — US disclosed
CN-104546669-B Nanochannel device and correlation technique 得克萨斯大学体系董事会 2018-01-05 — — CN disclosed
EP-3258958-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS University Of Virginia Patent Foundation (US) 2017-12-27 — — EP disclosed
US-20170319698-A1 GASTRORETENTIVE GEL FORMULATIONS JAGOTEC AG (CH) 2017-11-09 — — US disclosed
WO-2017192679-A1 METHODS AND COMPOSITIONS OF BIOLOGICALLY ACTIVE AGENTS WAVE LIFE SCIENCES LTD. (SG) 2017-11-09 — — WO disclosed
EP-3212167-A1 GASTRORETENTIVE GEL FORMULATIONS Jagotec AG (CH) 2017-09-06 — — EP disclosed
CN-107106484-A Gastric retention gel preparation 雅戈泰克股份公司 2017-08-29 — — CN disclosed
US-20170226585-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2017-08-10 — — US disclosed
US-20170216314-A1 TOPICAL FORMULATIONS NUVO RESEARCH INC. (CA) 2017-08-03 — — US disclosed
US-9642912-B2 Topical formulations for treating skin conditions CRESCITA THERAPEUTICS INC. (CA) 2017-05-09 — — US disclosed
EP-3156053-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2017-04-19 — — EP disclosed
US-20160376658-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2016-12-29 — — US disclosed
US-9526824-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-12-27 — — US disclosed
EP-2307011-B1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS INC (US) 2016-11-30 — — EP disclosed
EP-2355864-B1 NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS (US) 2016-11-09 — — EP disclosed
WO-2016134288-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2016-08-25 — — WO disclosed
WO-2016118787-A1 ENGINEERED RECEPTOR/LIGAND SYSTEM FOR DELIVERY OF THERAPEUTIC AGENTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2016-07-28 — — WO disclosed
US-20160175572-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER NANOMEDICAL SYSTEMS, INC. (US) 2016-06-23 — — US disclosed
EP-3033138-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER Nanomedical Systems Inc. (US) 2016-06-22 — — EP disclosed
US-20160139161-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA 2016-05-19 — — US disclosed
WO-2016066256-A1 GASTRORETENTIVE GEL FORMULATIONS JAGOTEC AG (CH) 2016-05-06 — — WO disclosed
US-9308181-B2 Topical formulations, systems and methods NUVO RESEARCH INC. (CA) 2016-04-12 — — US disclosed
US-9308162-B2 Biocompatible oligomer-polymer compositions TOLMAR THERAPEUTICS, INC. (US) 2016-04-12 — — US disclosed
US-9278134-B2 Dual functioning ionic liquids and salts thereof THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2016-03-08 — — US disclosed
WO-2015167760-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF CELANESE ACETATE LLC (US) 2015-11-05 — — WO disclosed
US-20150306230-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF CELANESE ACETATE LLC (US) 2015-10-29 — — US disclosed
US-20150297723-A1 TOPICAL FORMULATIONS FOR TREATING SKIN CONDITIONS NUVO RESEARCH INC. (CA) 2015-10-22 — — US disclosed
US-20150246174-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-09-03 — — US disclosed
EP-2912070-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO Celanese Acetate LLC (US) 2015-09-02 — — EP disclosed
US-9096743-B2 Process for forming films, fibers, and beads from chitinous biomass THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2015-08-04 — — US disclosed
CN-104812777-A Polysaccharide ester microspheres and methods and articles related thereto CELANESE ACETATE LLC 2015-07-29 — — CN disclosed
CN-104546669-A NANOCHANNELED DEVICE AND RELATED METHODS UNIV TEXAS 2015-04-29 — — CN disclosed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 — — US disclosed
US-9005185-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-04-14 — — US disclosed
WO-2015023557-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF LOW WATER SOLUBILITY THERAPEUTIC AGENT IN SOLUBILIZER NANOMEDICAL SYSTEMS, INC. (US) 2015-02-19 — — WO disclosed
EP-2291174-B1 FLOWABLE COMPOSITION COMPRISING BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS TOLMAR THERAPEUTICS INC (US) 2015-01-28 — — EP disclosed
CN-102271732-B Nanochannel devices and related methods UNIV TEXAS 2014-12-31 — — CN disclosed
CN-104203220-A Device and method for sustained release of therapeutic agent UNIV TEXAS 2014-12-10 — — CN disclosed
US-20140348936-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMOPLASTIC POLYURETHANES CELANESE EVA PERFORMANCE POLYMERS, INC. 2014-11-27 — — US disclosed
US-20140328884-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES CELANESE EVA PERFORMANCE POLYMERS, INC. 2014-11-06 — — US disclosed
US-20140315720-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-10-23 — — US disclosed
EP-2790677-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES Celanese Eva Performance Polymers, Inc. (US) 2014-10-22 — — EP disclosed
EP-2790678-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMPOPLASTIC POLYURETHANES Celanese Eva Performance Polymers, Inc. (US) 2014-10-22 — — EP disclosed
EP-2770984-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-09-03 — — EP disclosed
US-8802596-B2 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2014-08-12 — — US disclosed
US-20140206734-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2014-07-24 — — US disclosed
US-20140180251-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2014-06-26 — — US disclosed
US-20140154313-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2014-06-05 — — US disclosed
WO-2014066463-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-05-01 — — WO disclosed
US-20140113826-A1 POLYSACCHARIDE ESTER MICROSPHERES AND METHODS AND ARTICLES RELATING THERETO CELANESE ACETATE LLC (US) 2014-04-24 — — US disclosed
EP-2717860-A1 CONTROLLED ABSORPTION WATER-SOLUBLE PHARMACEUTICALLY ACTIVE ORGANIC COMPOUND FORMULATION FOR ONCE-DAILY ADMINISTRATION STI Pharma, LLC (US) 2014-04-16 — — EP disclosed
US-8697361-B2 Serotonin transporter gene and treatment of alcoholism UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2014-04-15 — — US disclosed
WO-2014031398-A1 BIOMEDICAL DEVICES COMPRISING MOLDED POLYETHYLENE COMPONENTS TICONA LLC (US) 2014-02-27 — — WO disclosed
US-20140051771-A1 Biomedical Devices Comprising Molded Polyethylene Components TICONA LLC (US) 2014-02-20 — — US disclosed
US-20140052264-A1 Porous, Stabilized Craniomaxillofacial Implants and Methods and Kits Relating Thereto TICONA LLC (US) 2014-02-20 — — US disclosed
US-8632510-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-01-21 — — US disclosed
US-20130337031-A1 TOPICAL FORMULATIONS, SYSTEMS AND METHODS NUVO RESEARCH INC. (CA) 2013-12-19 — — US disclosed
US-20130240483-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2013-09-19 — — US disclosed
CN-103271083-A Multi-functional ionic liquid compositions UNIV ALABAMA 2013-09-04 — — CN disclosed
US-8513304-B2 Topical formulation NUVO RESEARCH INC. (CA) 2013-08-20 — — US disclosed
US-8480637-B2 Nanochanneled device and related methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-07-09 — — US disclosed
WO-2013090891-A1 CONTROLLED RELEASE VEHICLES HAVING DESIRED VOID VOLUME ARCHITECTURES CELANESE EVA PERFORMANCE POLYMERS, INC. (US) 2013-06-20 — — WO disclosed
WO-2013090893-A1 GASTRORETENTIVE CONTROLLED RELEASE VEHICLES THAT INCLUDE ETHYLENE COPOLYMERS, ETHYL CELLULOSES, AND/OR THERMPOPLASTIC POLYURETHANES CELANESE EVA PERFORMANCE POLYMERS, INC. (US) 2013-06-20 — — WO disclosed
CN-101326275-B Multifunctional ionic liquid composition UNIV ALABAMA 2013-06-05 — — CN disclosed
US-20130131628-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-23 — — US disclosed
WO-2013063004-A1 DEVICE AND METHOD FOR SUSTAINED RELEASE OF THERAPEUTIC AGENT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2013-05-02 — — WO disclosed
EP-2255184-B1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM Univ Virginia Patent Found (US) 2013-04-24 — — EP disclosed
US-20130079404-A1 TOPICAL FORMULATION NUVO RESEARCH INC. (CA) 2013-03-28 — — US disclosed
EP-2556830-A1 Combined effects of topiramate, ondansetron and naltrexone on alcohol consumption UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2013-02-13 — — EP disclosed
US-8343962-B2 Topical formulation NUVO RESEARCH INC. (CA) 2013-01-01 — — US disclosed
WO-2012170676-A1 CONTROLLED ABSORPTION WATER-SOLUBLE PHARMACEUTICALLY ACTIVE ORGANIC COMPOUND FORMULATION FOR ONCE-DAILY ADMINISTRATION STI PHARMA, LLC (US) 2012-12-13 — — WO disclosed
US-20120302592-A1 TOPIRAMATE PLUS NALTREXONE FOR THE TREATMENT OF ADDICTIVE DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-11-29 — — US disclosed
US-8314077-B2 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. (US) 2012-11-20 — — US disclosed
US-20120264605-A1 Multi-Functional Ionic Liquid Compositions for Overcoming Polymorphism and Imparting Improved Properties for Active Pharmaceutical, Biological, Nutritional, and Energetic Ingredients THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-10-18 — — US disclosed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 — — US disclosed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 — — US disclosed
US-8232265-B2 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-07-31 — — US disclosed
US-20120115149-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-05-10 — — US disclosed
US-20120115729-A1 PROCESS FOR FORMING FILMS, FIBERS, AND BEADS FROM CHITINOUS BIOMASS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-05-10 — — US disclosed
US-20120095443-A1 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-04-19 — — US disclosed
US-8158152-B2 Preparing lyophilizates, especially those free of undesired extra components such as mono- or disaccharides; dosage forms of a wide variety of over 2000 drugs, such as rapidly dissolving tablets SCIDOSE LLC (US) 2012-04-17 — — US disclosed
EP-2425013-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM University Of Virginia Patent Foundation (US) 2012-03-07 — — EP disclosed
US-20120046244-A1 DUAL FUNCTIONING IONIC LIQUIDS AND SALTS THEREOF THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2012-02-23 — — US disclosed
EP-2419091-A2 NANOCHANNELED DEVICE AND RELATED METHODS The Board of Regents of The University of Texas System (US) 2012-02-22 — — EP disclosed
CN-102225046-A Transdermal drug delivery formulation NUVO RES INC 2011-10-26 — — CN disclosed
US-20110245172-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS TOLMAR THERAPEUTICS, INC. (US) 2011-10-06 — — US disclosed
US-20110224128-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF MUSCULAR DYSTROPHY WHALEN ANNE 2011-09-15 — — US disclosed
US-20110201665-A1 Compositions, Methods, and Kits for Treating Influenza Viral Infections COMBINATORX (SINGAPORE) PTE. LTD. (SG) 2011-08-18 — — US disclosed
EP-2355864-A2 NANOCHANNELED DEVICE AND RELATED METHODS The Board of Regents of The University of Texas System (US) 2011-08-17 — — EP disclosed
CN-101296691-B Transdermal drug delivery dosage form NUVO RES INC 2011-07-27 — — CN disclosed
US-7976871-B2 Modified release composition of highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2011-07-12 — — US disclosed
US-7951398-B2 Pharmaceutical preparation comprising an active dispersed on a matrix NYCOMED GMBH (DE) 2011-05-31 — — US disclosed
US-20110112159-A1 SEROTONIN TRANSPORTER GENE AND TREAMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2011-05-12 — — US disclosed
EP-2307011-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS Afecta Pharmaceuticals, Inc. (US) 2011-04-13 — — EP disclosed
CN-102016571-A Serotonin transporter gene and treatment of alcoholism UNIV VIRGINIA 2011-04-13 — — CN disclosed
US-20110065628-A1 Medication Combinations for the Treatment of Alcoholism and Drug Addiction UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2011-03-17 — — US disclosed
US-7905852-B2 Skin-contacting-adhesive free dressing JENNINGS-SPRING BARBARA 2011-03-15 — — US disclosed
EP-2291174-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS Tolmar Therapeutics, Inc. (US) 2011-03-09 — — EP disclosed
US-20110028510-A1 Compositions, Methods, and Kits for Treating Influenza Viral Infections COMBINATORX (SINGAPORE) PTE. LTD. (SG) 2011-02-03 — — US disclosed
US-20110028460-A1 TOPICAL FORMULATION FQUBED, INC. 2011-02-03 — — US disclosed
WO-2010141470-A2 PROCESS FOR FORMING FILMS, FIBERS, AND BEADS FROM CHITINOUS BIOMASS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2010-12-09 — — WO disclosed
EP-2255184-A2 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM University Of Virginia Patent Foundation (US) 2010-12-01 — — EP disclosed
WO-2010126603-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-11-04 — — WO disclosed
WO-2010120817-A2 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-10-21 — — WO disclosed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 — — US disclosed
CN-101810592-A Contain the pharmaceutical preparation that is dispersed in the active matter in the substrate ALTANA PHARMA AG 2010-08-25 — — CN disclosed
WO-2010078300-A1 DUAL FUNCTIONING IONIC LIQUIDS AND SALTS THEREOF THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA (US) 2010-07-08 — — WO disclosed
US-20100152699-A1 Nanochanneled Device and Related Methods THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-06-17 — — US disclosed
WO-2010056986-A2 NANOCHANNELED DEVICE AND RELATED METHODS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-05-20 — — WO disclosed
CN-101685733-A High-temperature thermal fuse device THERM O DISC INC 2010-03-31 — — CN disclosed
US-20100076006-A1 Topiramate Plus Naltrexone for the Treatment of Addictive Disorders UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-03-25 — — US disclosed
WO-2010024870-A1 SKIN-CONTACTING-ADHESIVE FREE DRESSING JENNINGS-SPRING BARBARA BROOKE (US) 2010-03-04 — — WO disclosed
CN-101663028-A Combined effect of topiramate and ondansetron on alcohol consumption UNIV VIRGINIA 2010-03-03 — — CN disclosed
US-20100041689-A1 Combined Effects of Topiramate and Ondansetron on Alcohol Consumption UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2010-02-18 — — US disclosed
US-20100009934-A1 BETA ADRENERGIC RECEPTOR AGONISTS FOR THE TREATMENT OF B-CELL PROLIFERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2010-01-14 — — US disclosed
US-20090318520-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS DRIVE (US) 2009-12-24 — — US disclosed
WO-2009155139-A1 USE OF ISOINDOLES FOR THE TREATMENT OF NEUROBEHAVIORAL DISORDERS AFECTA PHARMACEUTICALS, INC. (US) 2009-12-23 — — WO disclosed
WO-2009148581-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS QLT USA, INC. (US) 2009-12-10 — — WO disclosed
EP-2124909-A2 COMBINED EFFECTS OF TOPIRAMATE AND ONDANSETRON ON ALCOHOL CONSUMPTION University Of Virginia Patent Foundation (US) 2009-12-02 — — EP disclosed
CN-100548290-C Sulfamate derivatives is used for the treatment of the purposes of impulse control disorder UNIV CINCINNATI (US) 2009-10-14 — — CN disclosed
WO-2009108837-A2 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2009-09-03 — — WO disclosed
WO-2009029308-A1 MEDICATION COMBINATIONS FOR THE TREATMENT OF ALCOHOLISM AND DRUG ADDICTION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2009-03-05 — — WO disclosed
US-20090053168-A1 TREATMENTS OF B-CELL PROLIFERATIVE DISORDERS ZALICUS INC. 2009-02-26 — — US disclosed
US-20090047243-A1 COMBINATIONS FOR THE TREATMENT OF B-CELL PROLIFERATIVE DISORDERS ZALICUS INC. 2009-02-19 — — US disclosed
US-20090005722-A1 Skin-contacting-adhesive free dressing JENNLNGS-SPRING BARBARA 2009-01-01 — — US disclosed
US-20080319092-A1 Transdermal Drug Delivery Formulation NUVO RESEARCH INC. (CA) 2008-12-25 — — US disclosed
CN-101326275-A Multifunctional ionic liquid composition UNIV ALABAMA (US) 2008-12-17 — — CN disclosed
CN-101296691-A transdermal drug delivery dosage form NUVO RES INC (CA) 2008-10-29 — — CN disclosed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 — — EP disclosed
WO-2008095086-A2 TOPIRAMATE PLUS NALTREXONE FOR THE TREATMENT OF ADDICTIVE DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-08-07 — — WO disclosed
WO-2008077092-A2 COMBINED EFFECTS OF TOPIRAMATE AND ONDANSETRON ON ALCOHOL CONSUMPTION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2008-06-26 — — WO disclosed
EP-1931760-A2 MULTI-FUNCTIONAL IONIC LIQUID COMPOSITIONS The University of Alabama (US) 2008-06-18 — — EP disclosed
EP-1909772-A1 TRANSDERMAL DRUG DELIVERY FORMULATION Nuvo Research Inc. (CA) 2008-04-16 — — EP disclosed
US-20070269379-A1 Penetration Enhancer Combinations for Transdermal Delivery REGENTS OF THE UNIVERSITY OF CALIFORNIA, THE 2007-11-22 — — US disclosed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 — — WO disclosed
US-20070122474-A1 Pharmaceutical preparation comprising an active dispersed on a matrix ALTANA PHARMA AG 2007-05-31 — — US disclosed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 — — US disclosed
US-20070093462-A1 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA 2007-04-26 — — US disclosed
WO-2007044693-A2 MULTI-FUNCTIONAL IONIC LIQUID COMPOSITIONS THE UNIVERSITY OF ALABAMA (US) 2007-04-19 — — WO disclosed
US-7199151-B2 DHA-pharmaceutical agent conjugates of taxanes LUITPOLD PHARMACEUTICALS, INC. (US) 2007-04-03 — — US disclosed
WO-2007016766-A1 TRANSDERMAL DRUG DELIVERY FORMULATION NUVO RESEARCH INC. (CA) 2007-02-15 — — WO disclosed
US-7175854-B2 Pharmaceutical preparation comprising an active dispersed on a matrix ALTANA PHARMA AG (DE) 2007-02-13 — — US disclosed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 — — US disclosed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US disclosed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 — — US disclosed
EP-1158973-B1 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIV CINCINNATI (US) 2005-05-04 — — EP disclosed
WO-2005009510-A2 PENETRATION ENHANCER COMBINATIONS FOR TRANSDERMAL DELIVERY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2005-02-03 — — WO disclosed
EP-1466628-A1 DHA-pharmaceutical agent conjugates Luitpold Pharmaceuticals, Inc. (US) 2004-10-13 — — EP disclosed
US-20040180949-A1 conjugates of pharmaceutical agents and a highly lipphilic group, a C22 unbranched carbon chain; render the activity of these compounds selective for colon tissue, breast tissue and central nervous system tissue PROTARGA, INC. 2004-09-16 — — US disclosed
CN-1523980-A Pharmaceutical formulations containing an active dispersed in a matrix ��̹��ҽҩ��˾ 2004-08-25 — — CN disclosed
US-20040106589-A1 Fatty acid-pharmaceutical agent conjugates PROTARGA PHARMACEUTICALS, INC. 2004-06-03 — — US disclosed
US-20040058896-A1 Pharmaceutical preparation comprising an active dispersed on a matrix ASTRAZENECA AB (SE) 2004-03-25 — — US disclosed
EP-1341527-A1 PHARMACEUTICAL PREPARATION COMPRISING AN ACTIVE DISPERSED ON A MATRIX ALTANA Pharma AG (DE) 2003-09-10 — — EP disclosed
US-6602902-B2 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid PROTARGA, INC. 2003-08-05 — — US disclosed
US-6576636-B2 Treating a noncentral nervous system by administering a covalent conjugate of a C8-26, unbranched, naturally occurring fatty acid and a drug, provided the drug is not an adenosine receptor agonist/antagonist; anticarcinogenics PROTARGA, INC. 2003-06-10 — — US disclosed
US-20030059471-A1 Oral delivery formulation COMPTON BRUCE JON (US) 2003-03-27 — — US disclosed
CN-1360500-A Use of sulfamate derivatives for the treatment of impulse control disorders UNIV CINCINNATI (US) 2002-07-24 — — CN disclosed
WO-2002045693-A1 PHARMACEUTICAL PREPARATION COMPRISING AN ACTIVE DISPERSED ON A MATRIX ALTANA PHARMA AG (DE) 2002-06-13 — — WO disclosed
US-20020010208-A1 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid LUITPOLD PHARMACEUTICALS, INC. 2002-01-24 — — US disclosed
EP-1158973-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2001-12-05 — — EP disclosed
US-6323236-B2 PSYCHOLOGICAL DISORDERS UNIVERSITY OF CINCINNATI 2001-11-27 — — US disclosed
US-20010023254-A1 Psychological disorders CINCINNATI, UNIVERSITY OF 2001-09-20 — — US disclosed
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. 2001-05-31 — — US disclosed
WO-2000050020-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2000-08-31 — — WO disclosed
WO-1999030690-A1 ORAL DELIVERY FORMULATION AXIA THERAPEUTICS, INC. (US) 1999-06-24 — — WO disclosed
EP-0909183-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES Neuromedica, Inc. (US) 1999-04-21 — — EP disclosed
US-5795909-A ANTICARCINOGENIC AND ANTITUMOR AGENTS; BREAST, COLON, OVARIANCANCERS NEUROMEDICA, INC. (US) 1998-08-18 — — US disclosed
WO-1997044063-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES NEUROMEDICA, INC. (US) 1997-11-27 — — WO disclosed
WO-1997044063-A2 DHA-PHARMACEUTICAL AGENT CONJUGATES NEUROMEDICA, INC. (US) 1997-11-27 — — WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120264605-A1 Multi-Functional Ionic Liquid Compositions for Overcoming Polymorphism and Imparting Improved Properties for Active Pharmaceutical, Biological, Nutritional, and Energetic Ingredients SLC5A6, PNLIP, IPMK PDE3B 451/4885PDE3A 677/4885PDE4A 1105/4885
US-11951107-B2 Deuterated pharmaceutical compositions and methods of treating cardiovascular diseases ADRB2, ADRA2C, ADRB1 PDE3B 84/4885PDE3A 81/4885PDE4A 49/4885
US-20150306230-A1 DRUG DELIVERY VEHICLES COMPRISING CELLULOSE DERIVATIVES, STARCH DERIVATIVES, AND COMBINATIONS THEREOF PGRMC2, PGRMC1, CYP3A43 PDE3B 649/4885PDE3A 354/4885PDE4A 477/4885
US-20180043006-A1 COMPOSITIONS AND METHODS FOR PREVENTING AND TREATING RHINOVIRUS INFECTIONS CD4, HLA-DRB1, CD74 PDE3B 4631/4885PDE3A 4705/4885PDE4A 4142/4885
US-20110245172-A1 BIOCOMPATIBLE OLIGOMER-POLYMER COMPOSITIONS BMP2, CHERP, PUF60 PDE3B 452/4885PDE3A 348/4885PDE4A 1493/4885
US-10619209-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 PDE3B 881/4885PDE3A 961/4885PDE4A 645/4885
US-20070093462-A1 Multi-functional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional, and energetic ingredients SLC5A6, PNLIP, IPMK PDE3B 451/4885PDE3A 677/4885PDE4A 1105/4885
US-11905562-B2 Serotonin transporter gene and treatment of opioid-related disorders SLC6A4, SLC6A3, SLC6A2 PDE3B 881/4885PDE3A 961/4885PDE4A 645/4885
US-20020010208-A1 Targeting a pharmaceutical agent to a noncentral nervous system tissue by administering a covalent conjugate of the drug and cis-docosahexanoic acid FABP7, FADS2, ALOX5 PDE3B 2617/4885PDE3A 2123/4885PDE4A 1506/4885
US-20230107723-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES ADRB2, ADRA2C, ADRB1 PDE3B 84/4885PDE3A 81/4885PDE4A 49/4885
US-20180251840-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF ALCOHOLISM SLC6A4, SLC6A3, SLC6A2 PDE3B 587/4885PDE3A 723/4885PDE4A 459/4885
US-20240285639-A1 DEUTERATED PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING CARDIOVASCULAR DISEASES ADRB2, ADRA2C, ADRB1 PDE3B 84/4885PDE3A 81/4885PDE4A 49/4885
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“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.

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