SCHEMBL761018

SCHEMBL761018

CNc1ccc2ccccc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
CYP1A2 P05177 3/20 0.58
CYP3A4 P08684 2/20 0.58
HSD17B10 Q99714 2/20 0.58
CYP2C19 P33261 2/20 0.58
HIF1A Q16665 2/20 0.58
HPGD P15428 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
L3MBTL1 Q9Y468 3/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 1/20 0.48
RAB9A P51151 5/20 0.48
NPC1 O15118 4/20 0.48
MAPT P10636 2/20 0.48
CYP2A6 P11509 2/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1873124 0.98 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL6759670 0.93 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
Toluene SCHEMBL28366625 0.89 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL8156941 0.89 EGFR (0.48) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL25973229 0.87 EGFR (0.47) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL23192909 0.82 ESR1 (0.55) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL16194105 0.82 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL13562995 0.82 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C19
SCHEMBL16194322 0.81 HPRT1 (0.56) ALDH1A1CYP1A2HSD17B10HIF1AHPGD
SCHEMBL27937772 0.81 ESR1 (0.52) ALDH1A1CYP3A4HSD17B10HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 362 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903518-A Synthesis method of N-methyl-4, 5-benzindole 太原理工大学 2023-10-20 CN claimed
CN-111704591-B Synthesis method of copper-catalyzed thionaphthothiazolone compound 衡阳师范学院 2023-05-16 CN claimed
CN-109336887-B Benzimidazole chiral heterocyclic compound and preparation method and application thereof 中山大学 2021-12-17 CN claimed
US-11066749-B2 Corrosion inhibition of HCL treatment fluids with environmentally compatible solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2021-07-20 US claimed
CN-111704591-A Synthesis method of copper-catalyzed thio-naphthothiazolone compound 衡阳师范学院 2020-09-25 CN claimed
US-20200173034-A1 Corrosion Inhibition of HCL Treatment Fluids with Environmentally Compatible Solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2020-06-04 US claimed
US-10604850-B2 Corrosion inhibition of HCL treatment fluids with environmentally compatible solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2020-03-31 US claimed
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN claimed
US-20180127882-A1 Corrosion Inhibition of HCL Treatment Fluids with Environmentally Compatible Solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2018-05-10 US claimed
WO-2016190865-A1 CORROSION INHIBITION OF HCL TREATMENT FLUIDS WITH ENVIRONMENTALLY COMPATIBLE SOLVENT HALLIBURTON ENERGY SERVICES, INC. (US) 2016-12-01 WO claimed
EP-2646600-A1 CORROSION INHIBITOR COMPOSITIONS COMPRISING REACTION PRODUCTS OF ALDEHYDES AND AMIDES AND RELATED METHODS Halliburton Energy Services, Inc. (US) 2013-10-09 EP claimed
US-8361937-B2 Corrosion inhibitor compositions comprising reaction products of aldehydes and amides and related methods HALLIBURTON ENERGY SERVICES, INC. (US) 2013-01-29 US claimed
WO-2012072986-A1 CORROSION INHIBITOR COMPOSITIONS COMPRISING REACTION PRODUCTS OF ALDEHYDES AND AMIDES AND RELATED METHODS HALLIBURTON ENERGY SERVICES, INC. (US) 2012-06-07 WO claimed
US-20120142563-A1 Corrosion Inhibitor Compositions Comprising Reaction Products of Aldehydes and Amides and Related Methods HALLIBURTON ENERGY SERVICES, INC. (US) 2012-06-07 US claimed
EP-0853618-B1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL -AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2011-08-17 EP claimed
US-6984673-B2 Dental cement composition KURARAY CO., LTD. (JP) 2006-01-10 US claimed
CN-1553897-A Dolastatin 10 derivatives - 2004-12-08 CN claimed
CN-1114669-C Normal temp. solidified conveying band joint chloroprene rubber adhesive HUANG SHIDE (CN) 2003-07-16 CN claimed
CN-1272520-A Normal temp. solidified conveying band joint chloroprene rubber adhesive HUANG HONGXIA (CN) 2000-11-08 CN claimed
US-20260112544-A1 ELECTROLYTIC CAPACITOR PANASONIC IP MAN CO LTD (JP) 2026-04-23 US disclosed
US-12531188-B2 Electrolytic capacitor PANASONIC INTELLECTUAL PROPERTY MANAGEMENT CO., LTD. (JP) 2026-01-20 US disclosed
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2025-11-27 US disclosed
CN-120058683-A SLC6A19 inhibitor compound, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2025-05-30 CN disclosed
CN-116283683-B Method for synthesizing diaryl thioether amine compound by photoinduction catalysis 衡阳师范学院 2025-05-23 CN disclosed
WO-2025089384-A1 PHOTOELECTRIC CONVERSION ELEMENT AND PHOTOELECTRIC CONVERSION DEVICE キヤノン株式会社 2025-05-01 WO disclosed
WO-2025051157-A1 PYRIDINE-2(1H)-KETONE PRMT5-MTA INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 赛诺哈勃药业(成都)有限公司 2025-03-13 WO disclosed
US-20240400568-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2024-12-05 US disclosed
WO-2024241889-A1 CHARGE-TRANSPORTING VARNISH 日産化学株式会社 2024-11-28 WO disclosed
EP-4445902-A2 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS Carna Biosciences, Inc. (JP) 2024-10-16 EP disclosed
EP-4081305-B1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS CARNA BIOSCIENCES INC (JP) 2024-09-18 EP disclosed
US-12075637-B2 Perovskite solar cell and fabrication method thereof CONTEMPORARY AMPEREX TECHNOLOGY CO., LIMITED (CN) 2024-08-27 US disclosed
US-12054490-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-08-06 US disclosed
CN-118324767-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-07-12 CN disclosed
EP-4393923-A1 PYRIDO RING COMPOUND, PREPARATION METHOD THEREFOR, INTERMEDIATE, COMPOSITION, AND APPLICATION Yiyou Biotech (Shanghai) Co., Ltd. (CN) 2024-07-03 EP disclosed
US-20240182476-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2024-06-06 US disclosed
CN-114423742-B Benzotriazole-based compound, light absorber and resin composition 三井化学株式会社 2024-05-28 CN disclosed
CN-115722266-B Azacarbene-amino-ruthenium catalyst, and preparation method and application thereof 广东药科大学 2024-04-05 CN disclosed
CN-117736207-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
CN-115362003-B Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
CN-117623935-A Method for preparing amine compound by reductive amination of molecular sieve-based metal catalyst 浙江大学 2024-03-01 CN disclosed
CN-114409493-B Method for synthesizing 9-aryl fluorene compound 浙江工业大学 2024-02-23 CN disclosed
EP-4320131-A1 PROCESS FOR PREPARING ISOHEXIDE DIAMINES FROM ISOHEXIDE DIOLS Covestro Deutschland AG (DE) 2024-02-14 EP disclosed
CN-117466830-A Benzotriazole-based compound, light absorber and resin composition 三井化学株式会社 2024-01-30 CN disclosed
US-20240024266-A1 Therapeutic Agent or Prophylactic Agent for COVID-19 HIROSHIMA UNIVERSITY (JP) 2024-01-25 US disclosed
US-20240024266-A1 Therapeutic Agent or Prophylactic Agent for COVID-19 HIROSHIMA UNIVERSITY (JP) 2024-01-25 US disclosed
WO-2024005030-A1 DIPHENYLETHENE-BASED COMPOUND, LIGHT ABSORBER, RESIN COMPOSITION, AND USE THEREOF 山本化成株式会社 2024-01-04 WO disclosed
CN-117285504-A Amino phenylacetamide derivative and preparation method and application thereof 桂林医学院 2023-12-26 CN disclosed
US-11845723-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2023-12-19 US disclosed
US-20230403869-A1 PEROVSKITE SOLAR CELL AND FABRICATION METHOD THEREOF CONTEMPORARY AMPEREX TECHNOLOGY (HONG KONG) LIMITED (CN) 2023-12-14 US disclosed
WO-2023222682-A1 PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) LIGANDS Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2023-11-23 WO disclosed
US-20230355609-A1 Spirolactone Compounds QUIXGEN, INC. (US) 2023-11-09 US disclosed
CN-116969930-A Thiazole ring-containing pyrazole carboxamide derivative and preparation method and application thereof 安徽农业大学 2023-10-31 CN disclosed
CN-116903518-A Synthesis method of N-methyl-4, 5-benzindole 太原理工大学 2023-10-20 CN disclosed
CN-116903518-A Synthesis method of N-methyl-4, 5-benzindole 太原理工大学 2023-10-20 CN disclosed
US-20230322656-A1 ORGANIC COMPOUND, AND ELECTRONIC COMPONENT AND ELECTRONIC DEVICE HAVING SAME SHAANXI LIGHTE OPTOELECTRONICS MATERIAL CO., LTD. (CN) 2023-10-12 US disclosed
WO-2022183008-A9 AMINO-BENZIMIDAZOLE CATALYSTS FOR THE PREPARATION OF POLYOLEFINS DOW GLOBAL TECHNOLOGIES LLC (US) 2023-10-12 WO disclosed
WO-2023192960-A1 STAT MODULATORS AND USES THEREOF RECLUDIX PHARMA, INC. (US) 2023-10-05 WO disclosed
US-20230303537-A1 NITROGEN-CONTAINING COMPOUND, AND ELECTRONIC ELEMENT AND ELECTRONIC DEVICE THEREOF SHAANXI LIGHTE OPTOELECTRONICS MATERIAL CO., LTD. (CN) 2023-09-28 US disclosed
US-11767291-B2 Preparation of secondary amines with electrophilic N-linchpin reagents WILLIAM MARSH RICE UNIVERSITY (US) 2023-09-26 US disclosed
US-20230301182-A1 ORGANIC COMPOUND, AND ELECTRONIC ELEMENT AND ELECTRONIC DEVICE USING SAME SHAANXI LIGHTE OPTOELECTRONICS MATERIAL CO., LTD. (CN) 2023-09-21 US disclosed
WO-2023168240-A1 SMALL MOLECULE INHIBITORS OF ENPP1 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-09-07 WO disclosed
WO-2023160187-A1 CARBAZOLE DERIVATIVE AND USE THEREOF 上海八亿时空先进材料有限公司 2023-08-31 WO disclosed
US-20230260716-A1 ELECTROLYTIC CAPACITOR PANASONIC INTELLECTUAL PROPERTY MANAGEMENT CO., LTD. (JP) 2023-08-17 US disclosed
US-20230250048-A1 NITROGEN-CONTAINING COMPOUND, ELECTRONIC ELEMENT AND ELECTRONIC DEVICE SHAANXI LIGHTE OPTOELECTRONICS MATERIAL CO., LTD. (CN) 2023-08-10 US disclosed
WO-2023138254-A1 HETEROCYCLIC COMPOUND, AND ORGANIC ELECTROLUMINESCENT MATERIAL AND ELEMENT 上海八亿时空先进材料有限公司 2023-07-27 WO disclosed
WO-2023133336-A1 STAT MODULATORS AND USES THEREOF RECLUDIX PHARMA, INC. (US) 2023-07-13 WO disclosed
US-20230203048-A1 SPIROPYRROLIDINE DERIVED ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2023-06-29 US disclosed
US-20230203048-A1 SPIROPYRROLIDINE DERIVED ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2023-06-29 US disclosed
CN-116283683-A Method for synthesizing diaryl thioether amine compound by photoinduction catalysis 衡阳师范学院 2023-06-23 CN disclosed
US-20230200209-A1 ORGANOMETALLIC COMPOUND AND ORGANIC LIGHT-EMITTING DIODE INCLUDING THE SAME LG DISPLAY CO., LTD. (KR) 2023-06-22 US disclosed
US-20230200227-A1 ORGANIC ELECTROLUMINESCENT DEVICE Beijing Summer Sprout Technology Co., Ltd. (CN) 2023-06-22 US disclosed
WO-2023087557-A1 ORGANIC ELECTROLUMINESCENT DEVICE AND ELECTRONIC DEVICE 陕西莱特光电材料股份有限公司 2023-05-25 WO disclosed
CN-111704591-B Synthesis method of copper-catalyzed thionaphthothiazolone compound 衡阳师范学院 2023-05-16 CN disclosed
US-20230133581-A1 Novel 3,5-Diaminobenzoic Acid Compound, and PIN1 Inhibitor and Therapeutic Agent for Inflammatory Diseases Using Same HIROSHIMA UNIVERSITY (JP) 2023-05-04 US disclosed
US-20230133581-A1 Novel 3,5-Diaminobenzoic Acid Compound, and PIN1 Inhibitor and Therapeutic Agent for Inflammatory Diseases Using Same HIROSHIMA UNIVERSITY (JP) 2023-05-04 US disclosed
US-20230122957-A1 PSMA LIGANDS FOR IMAGING AND ENDORADIOTHERAPY Technische Universität München (DE) 2023-04-20 US disclosed
CN-115836367-A Electrolytic capacitor 松下知识产权经营株式会社 2023-03-21 CN disclosed
CN-115722266-A Novel aza-carbene-amido-ruthenium catalyst and preparation method and application thereof 广东药科大学 2023-03-03 CN disclosed
EP-4119165-A1 NOVEL 3,5-DIAMINOBENZOIC ACID COMPOUND, AND PIN1 INHIBITOR AND THERAPEUTIC AGENT FOR INFLAMMATORY DISEASES USING SAME Hiroshima University (JP) 2023-01-18 EP disclosed
CN-115362003-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2022-11-18 CN disclosed
EP-4081305-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS Carna Biosciences, Inc. (JP) 2022-11-02 EP disclosed
US-20220324866-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2022-10-13 US disclosed
WO-2022214469-A1 PROCESS FOR PREPARING ISOHEXIDE DIAMINES FROM ISOHEXIDE DIOLS COVESTRO DEUTSCHLAND AG (DE) 2022-10-13 WO disclosed
US-11370740-B2 Method for producing ester group-containing compound DIC CORPORATION (JP) 2022-06-28 US disclosed
CN-114423742-A Benzotriazole compound, light absorber, and resin composition 三井化学株式会社 2022-04-29 CN disclosed
CN-114409493-A Method for synthesizing 9-aryl fluorene compound 浙江工业大学 2022-04-29 CN disclosed
WO-2022025189-A1 ELECTROLYTIC CAPACITOR パナソニックIPマネジメント株式会社 2022-02-03 WO disclosed
CN-109651208-B N-aryl sulfonamide compound, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2022-01-04 CN disclosed
CN-109336887-B Benzimidazole chiral heterocyclic compound and preparation method and application thereof 中山大学 2021-12-17 CN disclosed
US-20210351358-A1 ORGANIC ELECTROLUMINESCENT DEVICE ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2021-11-11 US disclosed
CN-109420525-B Metal iridium catalyst of 2, 2' -bis-benzimidazole ligand and method for synthesizing N-methylated primary amine by using metal iridium catalyst 南京理工大学 2021-10-08 CN disclosed
US-11130780-B2 Inhibitors of growth factor activation enzymes WASHINGTON UNIVERSITY (US) 2021-09-28 US disclosed
WO-2021149767-A1 HETEROCYCLIC DERIVATIVE 大日本住友製薬株式会社 2021-07-29 WO disclosed
US-11066749-B2 Corrosion inhibition of HCL treatment fluids with environmentally compatible solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2021-07-20 US disclosed
US-20210214542-A1 NOVEL AMINE FUNCTIONALIZED POLYMERS AND METHODS OF PREPARATION THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2021-07-15 US disclosed
WO-2021054459-A1 BENZOTRIAZOLE COMPOUND, LIGHT ABSORBER, AND RESIN COMPOSITION 三井化学株式会社 2021-03-25 WO disclosed
CN-109836365-B Amine thioacyl fluoride derivatives and synthetic method thereof 华东师范大学 2021-02-26 CN disclosed
EP-3564249-B1 NOVEL COMPOUND AND ORGANIC LIGHT EMITTING DEVICE USING SAME LG CHEMICAL LTD (KR) 2021-01-20 EP disclosed
US-20200383987-A1 Novel Amide Compound, and Pin1 Inhibitor, Therapeutic Agent for Inflammatory Diseases and Therapeutic Agent for Cancer That Use the Same HIROSHIMA UNIVERSITY (JP) 2020-12-10 US disclosed
EP-3122353-B1 SUBSTITUTED INDOLE MCL-1 INHIBITORS UNIV VANDERBILT (US) 2020-10-28 EP disclosed
CN-111704591-A Synthesis method of copper-catalyzed thio-naphthothiazolone compound 衡阳师范学院 2020-09-25 CN disclosed
US-20200297876-A1 PSMA ligands for imaging and endoradiotherapy Technische Universität München (DE) 2020-09-24 US disclosed
WO-2020165420-A1 PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) LIGANDS WITH IMPROVED TISSUE SPECIFICITY Ruprecht-Karls-Universität Heidelberg (DE) 2020-08-20 WO disclosed
US-20200199453-A1 POLYMERISABLE LIQUID CRYSTAL MATERIAL AND POLYMERISED LIQUID CRYSTAL FILM MERCK PATENT GMBH (DE) 2020-06-25 US disclosed
US-20200173034-A1 Corrosion Inhibition of HCL Treatment Fluids with Environmentally Compatible Solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2020-06-04 US disclosed
CN-107417623-B Method for synthesizing 5-diarylaminobenzimidazole derivative in one step 华南理工大学 2020-05-22 CN disclosed
US-10649124-B2 Composition including compound having mesogenic group, polymer and optically anisotropic body obtained by polymerizing polymerizable composition, and phase difference film DIC CORPORATION (JP) 2020-05-12 US disclosed
EP-3030569-B1 SILANE AND SILICIC ACID (HETERO)POLYCONDENSATE HAVING AROMATIC COMPOUNDS LINKED VIA COUPLING GROUPS WHICH ARE SUITABLE AS OR FOR MATRIX SYSTEMS HAVING HIGH TRANSLUCENCY AND GOOD MECHANICAL PROPERTIES WOLTER HERBERT (DE) 2020-05-06 EP disclosed
US-10604850-B2 Corrosion inhibition of HCL treatment fluids with environmentally compatible solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2020-03-31 US disclosed
WO-2020040157-A1 COMPOSITION FOR DENTAL MATERIAL, DENTAL MATERIAL, AND MICROFIBROUS CELLULOSE USED IN DENTAL MATERIAL 王子ホールディングス株式会社 2020-02-27 WO disclosed
WO-2020017587-A1 PYRIDAZINONE DERIVATIVE 大日本住友製薬株式会社 2020-01-23 WO disclosed
WO-2019147015-A1 EFFICIENT SYNTHESIS METHOD OF C20 POLYENE BIS(PHOSPHONATE) AND CAROTENE COMPOUND USING SAME 명지대학교 산학협력단 2019-08-01 WO disclosed
EP-2551270-B1 PYRAZOLOPYRIMIDINE DERIVATIVES FOR USE AS PI3 KINASE ANTAGONISTS UNIV CALIFORNIA (US) 2019-06-12 EP disclosed
CN-109836365-A The thio acyl fluorides derivative of a kind of amine and its synthetic method 华东师范大学 2019-06-04 CN disclosed
EP-3489390-A1 ELECTROCHEMICAL METHOD FOR O-C COUPLING OF UNPROTECTED PHENOLS WITH OPTICALLY PURE ARYLAMINES Evonik Degussa GmbH (DE) 2019-05-29 EP disclosed
EP-3483146-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT EMITTING DEVICE USING SAME Heesung Material Ltd. (KR) 2019-05-15 EP disclosed
EP-2949655-B1 REACTION CATALYST FOR CROSS COUPLING AND METHOD FOR MANUFACTURING AROMATIC COMPOUND HOKKO CHEM IND CO (JP) 2019-05-15 EP disclosed
CN-109651208-A N- arylsulfonamides compound, medical composition and its use 中国科学院上海药物研究所 2019-04-19 CN disclosed
EP-3212694-B1 SILANES AND SILICIC ACID (HETERO) POLYCONDENSATES SUBSTITUTED WITH AROMATIC RESIDUES AND WITH HYDROXY GROUPS, AND DERIVATIVES THEREOF, WHICH ARE SUITABLE, AS SUCH OR AS COMPOSITES, FOR (MATRIX) SYSTEMS HAVING HIGH TRANSLUCENCE AND GOOD MECHANICAL PROPERTIES WOLTER HERBERT (DE) 2019-03-27 EP disclosed
EP-2427451-B1 ALPHA HELIX MIMETICS AND METHODS RELATING THERETO PRISM BIOLAB CO LTD (JP) 2019-03-20 EP disclosed
US-10227364-B2 Silane and silicic acid (hetero)polycondensate having aromatic compounds linked via coupling groups which are suitable as or for matrix systems having high translucency and good mechanical properties FRAUNHOFER-GESELLSCHAFT ZUR FOERDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 2019-03-12 US disclosed
CN-109420525-A The method of the metal iridium catalyst and its synthesis N- methylation primary amine of 2,2 '-bisbenzimidazole ligands 南京理工大学 2019-03-05 CN disclosed
US-10208000-B2 Eis inhibitors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2019-02-19 US disclosed
CN-109336887-A A kind of benzimidazole and chiral heterocycle class compound and its preparation method and application 中山大学 2019-02-15 CN disclosed
US-10202353-B2 Therapeutic compounds GILEAD SCIENCES, INC. (US) 2019-02-12 US disclosed
US-20190025490-A1 COMPOSITION INCLUDING COMPOUND HAVING MESOGENIC GROUP, POLYMER AND OPTICALLY ANISOTROPIC BODY OBTAINED BY POLYMERIZING POLYMERIZABLE COMPOSITION, AND PHASE DIFFERENCE FILM DIC CORPORATION (JP) 2019-01-24 US disclosed
WO-2018100159-A1 BACTERIAL GLUTAMINYL CYCLASES AND INHIBITORS THEREOF FOR USE IN THE TREATMENT OF PERIODONTITIS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2018-06-07 WO disclosed
CN-105008378-B The manufacturing method of cross-coupling catalysts and aromatic compound 北兴化学工业株式会社 2018-05-18 CN disclosed
US-20180127882-A1 Corrosion Inhibition of HCL Treatment Fluids with Environmentally Compatible Solvent HALLIBURTON ENERGY SERVICES, INC. (US) 2018-05-10 US disclosed
US-20180066015-A1 INHIBITORS OF GROWTH FACTOR ACTIVATION ENZYMES WASHINGTON UNIVERSITY (US) 2018-03-08 US disclosed
CN-107417623-A A kind of method of the diarylamino benzimidizole derivatives of one-step synthesis 5 华南理工大学 2017-12-01 CN disclosed
US-9809556-B2 Treatment of amyotrophic lateral sclerosis NORTHWESTERN UNIVERSITY (US) 2017-11-07 US disclosed
EP-3225619-A1 2-AMINOPYRIMIDINE COMPOUND AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Shanghai Institute Of Materia Medica Chinese Academy of Sciences (CN) 2017-10-04 EP disclosed
EP-3212694-A1 SILANES AND SILICIC ACID (HETERO) POLYCONDENSATES SUBSTITUTED WITH AROMATIC RESIDUES AND WITH HYDROXY GROUPS, AND DERIVATIVES THEREOF, WHICH ARE SUITABLE, AS SUCH OR AS COMPOSITES, FOR (MATRIX) SYSTEMS HAVING HIGH TRANSLUCENCE AND GOOD MECHANICAL PROPERTIES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2017-09-06 EP disclosed
US-9707551-B2 Reaction catalyst for cross-coupling and method for manufacturing aromatic compound HOKKO CHEMICAL INDUSTRY CO., LTD. (JP) 2017-07-18 US disclosed
CN-106928037-A A kind of preparation method of carvol 万华化学集团股份有限公司 2017-07-07 CN disclosed
US-20170189410-A1 Amino Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2017-07-06 US disclosed
US-9695191-B2 Conformationally constrained, fully synthetic macrocyclic compounds POLYPHOR AG (CH) 2017-07-04 US disclosed
US-9688646-B2 Process for producing N-methyl or N,N-dimethyl amines Lanxhou Institute of Chemical Physics, Chinese Academy of Sciences (CN) 2017-06-27 US disclosed
US-20170174639-A1 EIS INHIBITORS UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION 2017-06-22 US disclosed
WO-2017070560-A1 COMPOSITIONS AND METHODS OF PROMOTING ORGANIC PHOTOCATALYSIS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2017-04-27 WO disclosed
US-9598446-B2 Amino compounds for treatment of complement mediated disorders ACHILLION PHARMACEUTICALS, INC. (US) 2017-03-21 US disclosed
CN-106458868-A Guanidine compounds and uses thereof 伊谬诺米特医疗有限公司 2017-02-22 CN disclosed
EP-2499148-B1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2017-01-18 EP disclosed
US-20160368881-A1 THERAPEUTIC COMPOUNDS GILEAD SCIENCES, INC. 2016-12-22 US disclosed
US-9512139-B2 Conformationally constrained, fully synthetic macrocyclic compounds POLYPHOR AG (CH) 2016-12-06 US disclosed
WO-2016190865-A1 CORROSION INHIBITION OF HCL TREATMENT FLUIDS WITH ENVIRONMENTALLY COMPATIBLE SOLVENT HALLIBURTON ENERGY SERVICES, INC. (US) 2016-12-01 WO disclosed
US-9499474-B2 Process for producing arylamines MERCK PATENT GMBH (DE) 2016-11-22 US disclosed
US-20160194284-A1 ALLOSTERIC MODULATORS OF THE CANNABINOID 1 RECEPTOR NORTHEASTERN UNIVERSITY (US) 2016-07-07 US disclosed
US-20160185804-A1 SILANE AND SILICIC ACID (HETERO)POLYCONDENSATE HAVING AROMATIC COMPOUNDS LINKED VIA COUPLING GROUPS WHICH ARE SUITABLE AS OR FOR MATRIX SYSTEMS HAVING HIGH TRANSLUCENCY AND GOOD MECHANICAL PROPERTIES FRAUNHOFER-GESELLSCHAFT ZUR FOERDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 2016-06-30 US disclosed
EP-3030569-A1 SILANE AND SILICIC ACID (HETERO)POLYCONDENSATE HAVING AROMATIC COMPOUNDS LINKED VIA COUPLING GROUPS WHICH ARE SUITABLE AS OR FOR MATRIX SYSTEMS HAVING HIGH TRANSLUCENCY AND GOOD MECHANICAL PROPERTIES Fraunhofer Gesellschaft zur Förderung der angewandten Forschung E.V. (DE) 2016-06-15 EP disclosed
WO-2016066653-A1 SILANES AND SILICIC ACID (HETERO) POLYCONDENSATES SUBSTITUTED WITH AROMATIC RESIDUES AND WITH HYDROXY GROUPS, AND DERIVATIVES THEREOF, WHICH ARE SUITABLE, AS SUCH OR AS COMPOSITES, FOR (MATRIX) SYSTEMS HAVING HIGH TRANSLUCENCE AND GOOD MECHANICAL PROPERTIES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2016-05-06 WO disclosed
US-20150360214-A1 REACTION CATALYST FOR CROSS-COUPLING AND METHOD FOR MANUFACTURING AROMATIC COMPOUND HOKKO CHEMICAL INDUSTRY CO., LTD. (JP) 2015-12-17 US disclosed
EP-2949655-A1 REACTION CATALYST FOR CROSS COUPLING AND METHOD FOR MANUFACTURING AROMATIC COMPOUND Hokko Chemical Industry Co., Ltd. (JP) 2015-12-02 EP disclosed
CN-105008378-A Reaction catalyst for cross coupling and method for manufacturing aromatic compound HOKKO CHEM IND CO 2015-10-28 CN disclosed
CN-104922117-A BETA-LACTAMYLALKANOIC ACIDS FOR TREATING PREMENSTRUAL DISORDERS AZEVAN PHARMACEUTICALS INC 2015-09-23 CN disclosed
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders ACHILLION PHARMACEUTICALS, INC. (US) 2015-08-27 US disclosed
CN-103298772-B Method for producing aromatic alcohol or heterocyclic aromatic alcohol MITSUBISHI GAS CHEMICAL CO 2015-06-24 CN disclosed
US-9012166-B2 Method for assaying histone methylation enzyme activity KYUSHU INSTITUTE OF TECHNOLOGY (JP) 2015-04-21 US disclosed
US-9012166-B2 Method for assaying histone methylation enzyme activity KYUSHU INSTITUTE OF TECHNOLOGY (JP) 2015-04-21 US disclosed
US-8962244-B2 Compounds for modulating RNA binding proteins and uses therefor UNIVERSITY OF MASSACHUSETTS (US) 2015-02-24 US disclosed
WO-2015018906-A1 SILANE AND SILICIC ACID (HETERO)POLYCONDENSATE HAVING AROMATIC COMPOUNDS LINKED VIA COUPLING GROUPS WHICH ARE SUITABLE AS OR FOR MATRIX SYSTEMS HAVING HIGH TRANSLUCENCY AND GOOD MECHANICAL PROPERTIES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2015-02-12 WO disclosed
CN-104334528-A (2-heteroarylamino) succinic acid derivatives DAIICHI SANKYO CO LTD 2015-02-04 CN disclosed
EP-2562264-B1 METHOD FOR ASSAYING HISTONE METHYLATION ENZYME ACTIVITY KYUSHU INST TECHNOLOGY (JP) 2015-01-14 EP disclosed
EP-2810944-A1 HETEROCYCLIC COMPOUND HAVING ANTI-HIV ACTIVITY Toyama Chemical Co., Ltd. (JP) 2014-12-10 EP disclosed
US-20140309458-A1 PROCESS FOR PRODUCING ARYLAMINES MERCK PATENT GMBH (DE) 2014-10-16 US disclosed
EP-2435423-B1 SUBSTITUTED BENZOTRIAZINES AND QUINOXALINES AS INHIBITORS OF P70S6 KINASE SENTINEL ONCOLOGY LTD (GB) 2014-10-15 EP disclosed
US-8716473-B2 Substituted benzotriazines and quinoxalines as inhibitors of P7OS6 kinase SENTINEL ONCOLOGY LIMITED (GB) 2014-05-06 US disclosed
WO-2014015276-A1 α-AND γ-TRUXILLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2014-01-23 WO disclosed
CN-103459372-A Process for preparing cyclic amine compounds KANEKA CORP 2013-12-18 CN disclosed
US-8569505-B2 Aminotetralin-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA, NV (BE) 2013-10-29 US disclosed
EP-2646600-A1 CORROSION INHIBITOR COMPOSITIONS COMPRISING REACTION PRODUCTS OF ALDEHYDES AND AMIDES AND RELATED METHODS Halliburton Energy Services, Inc. (US) 2013-10-09 EP disclosed
CN-103298772-A Method for producing aromatic alcohol or heterocyclic aromatic alcohol MITSUBISHI GAS CHEMICAL CO 2013-09-11 CN disclosed
CN-103269584-A Methods for treating post-traumatic stress disorder AZEVAN PHARMACEUTICALS INC 2013-08-28 CN disclosed
US-20130217685-A1 COMPOUNDS FOR MODULATING RNA BINDING PROTEINS AND USES THEREFOR UNIVERSITY OF MASSACHUSETTS (US) 2013-08-22 US disclosed
US-8377639-B2 Compounds for modulating RNA binding proteins and uses therefor UNIVERSITY OF MASSACHUSETTS (US) 2013-02-19 US disclosed
US-20130029878-A1 Method for Assaying Histone Methylation Enzyme Activity KYUSHU INSTITUTE OF TECHNOLOGY (JP) 2013-01-31 US disclosed
US-20130029878-A1 Method for Assaying Histone Methylation Enzyme Activity KYUSHU INSTITUTE OF TECHNOLOGY (JP) 2013-01-31 US disclosed
US-8361937-B2 Corrosion inhibitor compositions comprising reaction products of aldehydes and amides and related methods HALLIBURTON ENERGY SERVICES, INC. (US) 2013-01-29 US disclosed
US-20120202821-A1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2012-08-09 US disclosed
WO-2012072986-A1 CORROSION INHIBITOR COMPOSITIONS COMPRISING REACTION PRODUCTS OF ALDEHYDES AND AMIDES AND RELATED METHODS HALLIBURTON ENERGY SERVICES, INC. (US) 2012-06-07 WO disclosed
US-20120142563-A1 Corrosion Inhibitor Compositions Comprising Reaction Products of Aldehydes and Amides and Related Methods HALLIBURTON ENERGY SERVICES, INC. (US) 2012-06-07 US disclosed
US-20120071478-A1 SUBSTITUTED BENZOTRIAZINES AND QUINOXALINES AS INHIBITORS OF P7OS6 KINASE SENTINEL ONCOLOGY LIMITED (GB) 2012-03-22 US disclosed
US-20120053345-A1 Indazole Compounds ABBOTT LABORATORIES (US) 2012-03-01 US disclosed
EP-1506166-B1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA NV (BE) 2011-11-16 EP disclosed
WO-2011131712-A1 METAL HYBRID COMPOSITE CASTING Rheinisch-Westfälische Technische Hochschule Aachen (DE) 2011-10-27 WO disclosed
US-8008481-B2 Indazole compounds ABBVIE INC. 2011-08-30 US disclosed
EP-0853618-B1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL -AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2011-08-17 EP disclosed
EP-2357169-A1 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators AstraZeneca AB (SE) 2011-08-17 EP disclosed
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND NAKAMOTO KAZUTAKA 2011-08-11 US disclosed
CN-101001886-B Redox curing-type nonaqueous curable composition KURARAY MEDICAL INC 2011-07-13 CN disclosed
US-7968570-B2 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators ASTRAZENECA AB (SE) 2011-06-28 US disclosed
US-7932272-B2 Antifungal agent containing heterocyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-04-26 US disclosed
CN-1863784-B 2-naphthylimino-1,3-thiazine derivative SHIONOGI & CO 2010-11-17 CN disclosed
EP-1028942-B1 DIPEPTIDE NITRILES NOVARTIS AG (CH) 2010-09-01 EP disclosed
US-20100125140-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR CODD ELLEN 2010-05-20 US disclosed
US-7678812-B2 Aminotetralin-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA NV (BE) 2010-03-16 US disclosed
US-7662960-B2 Beta-strand mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2010-02-16 US disclosed
EP-1919896-B1 AMINOARYL SULPHONAMIDE DERIVATIVES AS FUNCTIONAL 5-HT6 LIGANDS. SUVEN LIFE SCIENCES LTD (IN) 2009-12-23 EP disclosed
US-20090275578-A1 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators ASTRAZENECA AB (SE) 2009-11-05 US disclosed
US-20090227799-A1 Novel Antimalarial Agent Containing Heterocyclic Compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-09-10 US disclosed
US-7553340-B2 Reactive dyes, a process for their preparation and their use HUNTSMAN INTERNATIONAL, LLC (US) 2009-06-30 US disclosed
CN-100467458-C Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB CO LTD (FR) 2009-03-11 CN disclosed
WO-2008098857-A1 2-AMINOOXAZOLINES AS TAAR1 LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2008-08-21 WO disclosed
US-7399884-B2 Histone deacetylase inhibitors TAKEDA SAN DIEGO, INC. (US) 2008-07-15 US disclosed
CN-101208010-A Beta-lactamylalkanoic acids for the treatment of premenstrual disorders AZEVAN PHARMACEUTICALS INC (US) 2008-06-25 CN disclosed
US-7390822-B2 Substituted 4-phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives for reducing ischaemic damage JANSSEN PHARMACEUTICA, N.V. (BE) 2008-06-24 US disclosed
US-7390822-B2 Substituted 4-phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives for reducing ischaemic damage JANSSEN PHARMACEUTICA, N.V. (BE) 2008-06-24 US disclosed
US-20080097102-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR CODD ELLEN 2008-04-24 US disclosed
US-20080096925-A1 Novel Substituted 4-Phenyl-4[H-Imidazol-2-YL]-Piperidine Derivatived And Their Use As Selective Non-Peptide Delta Opioid Agonists JANSSEN PHARMACEUTICA N.V. (BE) 2008-04-24 US disclosed
US-20080096925-A1 Novel Substituted 4-Phenyl-4[H-Imidazol-2-YL]-Piperidine Derivatived And Their Use As Selective Non-Peptide Delta Opioid Agonists JANSSEN PHARMACEUTICA N.V. (BE) 2008-04-24 US disclosed
US-20080027060-A1 DIPEPTIDE NITRILES ALTMANN EVA 2008-01-31 US disclosed
US-20080027060-A1 DIPEPTIDE NITRILES ALTMANN EVA 2008-01-31 US disclosed
EP-1549598-A4 NAPTHTHALENE DERIVATIVES WHICH INHIBIT THE CYTOKINE OR BIOLOGICAL ACTIVITY OF MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF) CORTICAL PTY LTD (AU) 2008-01-23 EP disclosed
US-20070294842-A1 Reactive Dyes, a Process for Their Preparation and Their Use HUNTSMAN INTERNATIONAL LLC 2007-12-27 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed
US-7282508-B2 Substituted 4-phenyl-4-(1H-imidazol-2-yl)-piperidine derivatives and their use as selective non-peptide delta opioid agonists JANSSEN PHARMACEUTICA N.V. (BE) 2007-10-16 US disclosed
US-7282508-B2 Substituted 4-phenyl-4-(1H-imidazol-2-yl)-piperidine derivatives and their use as selective non-peptide delta opioid agonists JANSSEN PHARMACEUTICA N.V. (BE) 2007-10-16 US disclosed
CN-101001886-A Redox curing-type nonaqueous curable composition KURARAY MEDICAL INC (JP) 2007-07-18 CN disclosed
US-20070149495-A1 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2007-06-28 US disclosed
US-20070105943-A1 Novel antifungal agent containing heterocyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2007-05-10 US disclosed
EP-1782811-A1 NOVEL ANTIMALARIA AGENT CONTAINING HETEROCYCLIC COMPOUND Eisai R&D Management Co., Ltd. (JP) 2007-05-09 EP disclosed
EP-1778634-A1 ISOINDOLONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS AstraZeneca AB (SE) 2007-05-02 EP disclosed
US-7173032-B2 Methods and compositions of novel triazine compounds REDDY US THERAPEUTICS, INC. (US) 2007-02-06 US disclosed
US-7173032-B2 Methods and compositions of novel triazine compounds REDDY US THERAPEUTICS, INC. (US) 2007-02-06 US disclosed
CN-1874991-A Compounds capable of binding to the S1P receptor and pharmaceutical uses thereof ONO PHARMACEUTICAL CO (JP) 2006-12-06 CN disclosed
CN-1867339-A Novel use of cannabinoid receptor antagonists SHIONOGI & CO (JP) 2006-11-22 CN disclosed
CN-1863784-A 2-naphthylimino-1,3-thiazine derivative SHIONOGI & CO (JP) 2006-11-15 CN disclosed
EP-1194144-B1 ANTIBACTERIAL COMPOUNDS AFFINIUM PHARM INC (CA) 2006-11-02 EP disclosed
CN-1840527-A Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2006-10-04 CN disclosed
EP-1669348-A1 NOVEL ANTIFUNGAL AGENT COMPRISING HETEROCYCLIC COMPOUND Eisai Co., Ltd. (JP) 2006-06-14 EP disclosed
CN-1255386-C Substituted fused heterocyclic compound SANKYO CO (JP) 2006-05-10 CN disclosed
CN-1250189-C Tooth cement agent composition KURARAY CO (JP) 2006-04-12 CN disclosed
CN-1247553-C 2-imino-1,3-thiazine derivs. SHIONOGI & CO (JP) 2006-03-29 CN disclosed
CN-1245931-C Composition reagent box for dentistry KURARAY CO (JP) 2006-03-22 CN disclosed
WO-2006020879-A1 ISOINDOLONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2006-02-23 WO disclosed
CN-1729159-A Amide compounds and methods for controlling plant diseases SUMITOMO CHEMICAL CO (JP) 2006-02-01 CN disclosed
EP-1615890-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY (US) 2006-01-18 EP disclosed
US-6984647-B2 Aminotetralin-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2006-01-10 US disclosed
US-6984673-B2 Dental cement composition KURARAY CO., LTD. (JP) 2006-01-10 US disclosed
WO-2004089903-A9 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER LAMBERT CO (US) 2005-10-27 WO disclosed
EP-1269968-B1 Dental cement composition KURARAY CO (JP) 2005-10-12 EP disclosed
EP-1577290-A1 AMIDE COMPOUND AND METHOD OF CONTROLLING PLANT DISEASE WITH THE SAME Sumitomo Chemical Company, Limited (JP) 2005-09-21 EP disclosed
US-6943256-B2 Chiral organic compounds and metal coordination complexes thereof INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2005-09-13 US disclosed
US-20050187291-A1 use of 2-(urea or thiourea)tetralins as analgesic or to treat pulmonary dysfunction JANSSEN PHARMACEUTICA, N.V. (BE) 2005-08-25 US disclosed
EP-1549598-A1 NAPTHTHALENE DERIVATIVES WHICH INHIBIT THE CYTOKINE OR BIOLOGICAL ACTIVITY OF MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF) Cortical Pty Ltd (AU) 2005-07-06 EP disclosed
EP-1269967-B1 Dental composition kit KURARAY CO (JP) 2005-05-18 EP disclosed
US-6869984-B2 Dental composition kit KURARAY CO., LTD. (JP) 2005-03-22 US disclosed
EP-1506166-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-16 EP disclosed
CN-1188407-C Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof LG CHEMICAL LTD (KR) 2005-02-09 CN disclosed
CN-1553897-A Dolastatin 10 derivatives - 2004-12-08 CN disclosed
WO-2004089903-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY LLC (US) 2004-10-21 WO disclosed
US-20040204455-A1 Piperidine derivative rennin inhibitors WARNER-LAMBERT COMPANY LLC 2004-10-14 US disclosed
CN-1161356-C Puring inhibitors of cylin dependent kinase 2 and I'kappa'beta-'alpha' CV���ƹ�˾ 2004-08-11 CN disclosed
US-20040143118-A1 Chiral organic compounds and metal coordination complexes thereof ADVANCED RESEARCH & TECHNOLOGY INSTITUTE, INC. 2004-07-22 US disclosed
US-6673941-B2 Disubstituted imidazoles useful in the treatment of bacterial infections AFFINIUM PHARMACEUTICALS, INC. (CA) 2004-01-06 US disclosed
US-20030236280-A1 Aminotetralin-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA, N.V. (BE) 2003-12-25 US disclosed
WO-2003104178-A1 NAPTHTHALENE DERIVATIVES WHICH INHIBIT THE CYTOKINE OR BIOLOGICAL ACTIVITY OF MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF) CORTICAL PTY LTD (AU) 2003-12-18 WO disclosed
WO-2003097586-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2003-11-27 WO disclosed
US-6653321-B1 Stimulating kinase activity of insulin receptor; type II diabetes; hyperglycemia TELIK, INC. 2003-11-25 US disclosed
EP-0878196-B1 KAINIC ACID NEURONOTOXICITY INHIBITORS AND PYRIDOTHIAZINE DERIVATIVES YAMANOUCHI PHARMA CO LTD (JP) 2003-09-03 EP disclosed
US-20030149089-A1 Antibacterial compounds SMITHKLINE BEECHAM CORPORATION 2003-08-07 US disclosed
US-6559172-B1 Treatment of bacterial infections, particularly through the inhibition of FAB I. and antiobiotics SMITHKLINE BEECHAM CORPORATION 2003-05-06 US disclosed
US-20030083398-A1 Dental composition kit KURARAY CO. LTD. (JP) 2003-05-01 US disclosed
CN-1104413-C Phenylalkylcarboxylic acid derivatives SANKYO CO (JP) 2003-04-02 CN disclosed
US-20030055123-A1 Dental cement composition KURARAY CO. LTD, (JP) 2003-03-20 US disclosed
CN-1101380-C 4-mercaptopyrrolidine derivatives as farnesyl transferase inhibitors ZENECA LTD (GB) 2003-02-12 CN disclosed
CN-1394567-A Composition reagent box for dentistry KURARAY CO (JP) 2003-02-05 CN disclosed
CN-1394566-A Tooth cement agent composition KURARAY CO (JP) 2003-02-05 CN disclosed
CN-1391484-A Methods for enhancing chemotherapeutic efficacy and treating solid tumors HEW CORP (US) 2003-01-15 CN disclosed
EP-1269967-A1 Dental composition kit KURARAY CO., LTD. (JP) 2003-01-02 EP disclosed
EP-1269968-A1 Dental cement composition KURARAY CO., LTD. (JP) 2003-01-02 EP disclosed
EP-1261327-A2 ADENOSINE RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2002-12-04 EP disclosed
CN-1377647-A 4-mercaptopyrrolidinyl derivative as fernesyl transferase inhibitor ZENECA LTD (GB) 2002-11-06 CN disclosed
WO-2002085820-A2 CHIRAL ORGANIC COMPOUNDS AND METAL COORDINATION COMPLEXES THEREOF INDIANA UNIVERSITY (US) 2002-10-31 WO disclosed
EP-1194144-A4 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-08-07 EP disclosed
CN-1353713-A Purine inhibitors of cyclin dependent kinase 2 and IK B-alpha CV THERAPEUTICS INC (US) 2002-06-12 CN disclosed
EP-0923551-B1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PROD (US) 2002-06-05 EP disclosed
EP-1194144-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-10 EP disclosed
CN-1079391-C Preparation of N-alkyl naphthylamines CHINA PETRO CHEM GROUP CORP (CN) 2002-02-20 CN disclosed
EP-1177175-A2 HETEROSUBSTITUTED PYRIDINE DERIVATIVES AS PDE 4 INHIBITORS MERCK FROSST CANADA INC. (CA) 2002-02-06 EP disclosed
WO-2001062233-A2 ADENOSINE RECEPTOR MODULATORS F. HOFFMANN LA ROCHE AG (CH) 2001-08-30 WO disclosed
CN-1065532-C Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO CO (JP) 2001-05-09 CN disclosed
US-6200993-B1 ASTHMA; ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-03-13 US disclosed
CN-1280570-A Substituted fused heterocyclic compounds SANKYO CO (JP) 2001-01-17 CN disclosed
CN-1279680-A Imidazole derivatives having farnesyl transferase inhibitory activity and process for producing the same LG CHEMICAL LTD (KR) 2001-01-10 CN disclosed
WO-2000071120-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-11-30 WO disclosed
WO-2000068198-A2 HETEROSUBSTITUTED PYRIDINE DERIVATIVES AS PDE 4 INHIBITORS MERCK FROSST CANADA & CO. (CA) 2000-11-16 WO disclosed
US-6133258-A PYRIDOTHIAZINE DERIVATIVE; FOR TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS, MULTIPLE SCLEROSIS, PAIN, GLAUCOMA YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-17 US disclosed
US-6114310-A THERAPY FOR MICROBIAL INFECTIONS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-09-05 US disclosed
CN-1234024-A 4-aminoethoxy indolone derivatives AMERICAN HOME PROD (US) 1999-11-03 CN disclosed
CN-1231611-A Puring inhibitors of cylin dependent kinase 2 and I'kappa'beta-'alpha' CV THERAPEUTIC INC (US) 1999-10-13 CN disclosed
EP-0923551-A1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-06-23 EP disclosed
EP-0918757-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1999-06-02 EP disclosed
CN-1214338-A Preparation of N-alkyl naphthylamines CHINA PETROCHEMICAL CORP (CN) 1999-04-21 CN disclosed
CN-1202109-A Kainic acid neuronotoxicity inhibitors and pyridothioazine derivatives YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 CN disclosed
EP-0878196-A1 KAINIC ACID NEURONOTOXICITY INHIBITORS AND PYRIDOTHIAZINE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-11-18 EP disclosed
CN-1197453-A 4-mercaptopyrrolidine derivatives as farnesyl transferase inhibitors ZENECA LTD (GB) 1998-10-28 CN disclosed
US-5817690-A ANTIDOPAMINE AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-10-06 US disclosed
WO-1998008819-A1 4-AMINOETHOXY INDOLONE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-05 WO disclosed
WO-1997043268-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1997-11-20 WO disclosed
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US disclosed
EP-0540673-B1 ACETYLENE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1996-10-16 EP disclosed
CN-1132750-A Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO CO (JP) 1996-10-09 CN disclosed
US-5559144-A LIPOXYGENASE INHIBITORS, INHIBITORS OF BIOSYNTHESIS OF LEUKOTRIENES ABBOTT LABORATORIES (US) 1996-09-24 US disclosed
US-5476873-A Inhibit biosynthesis of leukotrienes ABBOTT LABORATORIES (US) 1995-12-19 US disclosed
WO-1994014762-A1 OXIME ETHER DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LABORATORIES (US) 1994-07-07 WO disclosed
US-5326883-A Oxime ether derivatives having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1994-07-05 US disclosed
US-5288743-A Lipoxygenase inhibitors ABBOTT LABORATORIES (US) 1994-02-22 US disclosed
US-5250565-A Must incorporate a metabolically cleavable leaving group; pro-drugs; administering to mammals ABBOTT LABORATORIES (US) 1993-10-05 US disclosed
US-5204453-A Process for the preparation of 1:2 metal complex azo compounds by carrying out diazotization and coupling in the presence of a metal donor CIBA-GEIGY CORPORATION (US) 1993-04-20 US disclosed
EP-0278910-B1 HEAVY METAL COMPLEX DYESTUFFS, THEIR PREPARATION AND THEIR USE CIBA-GEIGY AG (CH) 1992-01-22 EP disclosed
EP-0241414-B1 PROCESS FOR THE PREPARATION OF 1:2 METAL COMPLEX AZO DYES CIBA-GEIGY AG (CH) 1991-05-08 EP disclosed
US-5001227-A Fibre-reactive 1:1 chromium complex azo or azomethine dyes having a bidentate chelating group and a monofunctional neutral ligand CIBA-GEIGY CORPORATION (US) 1991-03-19 US disclosed
US-4990598-A Colorfastness CIBA-GEIGY CORPORATION, A CORP. OF NEW YORK 1991-02-05 US disclosed
US-4960870-A DYEING WOOL, POLYAMIDES; FIBER REACTIVE DYES CIBA-GEIGY CORPORATION (US) 1990-10-02 US disclosed
EP-0142104-B1 FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE CIBA-GEIGY AG (CH) 1990-01-03 EP disclosed
US-4889946-A Phenoxybenzoic acid compounds and herbicidal and plant growth regulant compositions BAYER AKTIENGESELLSCHAFT (DE) 1989-12-26 US disclosed
US-4874391-A USING WATER SOLUBLE COPPER COMPLEX AZO DYE, LIGHT STABILIZER AND ANTIOXIDANT CIBA-GEIGY CORPORATION (US) 1989-10-17 US disclosed
EP-0144776-B1 FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE CIBA-GEIGY AG (CH) 1989-10-11 EP disclosed
EP-0141416-B1 FIBRE-REACTIVE CHROMIUM COMPLEXES, THEIR PREPARATION AND THEIR USE CIBA-GEIGY AG (CH) 1989-08-16 EP disclosed
US-4833243-A BENZOOXAZOLES OR BENZOTHIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1989-05-23 US disclosed
US-4813972-A USING LEVELING DYES, COLORFASTNESS CIBA-GEIGY CORPORATION (US) 1989-03-21 US disclosed
EP-0159962-B1 FIBRE-REACTIVE CHROMIUM OR COBALT COMPLEXES, THEIR PREPARATION AND THEIR USE CIBA-GEIGY AG (CH) 1989-02-08 EP disclosed
EP-0185611-B1 PROCESS FOR THE PHOTOCHEMICAL STABILISATION OF SYNTHETIC FIBROUS MATERIALS CONTAINING POLYAMIDE FIBRES CIBA-GEIGY AG (CH) 1988-09-21 EP disclosed
EP-0278910-A2 Heavy metal complex dyestuffs, their preparation and their use CIBA-GEIGY AG (CH) 1988-08-17 EP disclosed
US-4756741-A Azolyloxy-carboxylic acid amide compounds and herbicidal compositions BAYER AKTIENGESELLSCHAFT (DE) 1988-07-12 US disclosed
EP-0255481-A1 Process for the photochemical stabilisation of a fibrous polyamide material and its mixtures with other fibres CIBA-GEIGY AG (CH) 1988-02-03 EP disclosed
US-4723001-A Fibre-reactive chromium complexes and their preparation and use CIBA-GEIGY CORPORATION (US) 1988-02-02 US disclosed
US-4719053-A FOR DYES HOECHST AKTIENGESELLSCHAFT (DE) 1988-01-12 US disclosed
US-4704133-A FIBER-REACTIVE CIBA-GEIGY CORPORATION (US) 1987-11-03 US disclosed
EP-0241414-A2 Process for the preparation of 1:2 metal complex azo dyes CIBA-GEIGY AG (CH) 1987-10-14 EP disclosed
US-4680385-A Metal dye complexes containing an azo or azomethine dye and a colorless ligand with the C═N--N═C group CIBA-GEIGY CORPORATION (US) 1987-07-14 US disclosed
US-4678851-A FIBER-RACTIVE CIBA-GEIGY CORPORATION (US) 1987-07-07 US disclosed
US-4645525-A Azolyoxy-carboxylic acid amide compounds and herbicidal compositions BAYER AKTIENGESELLSCHAFT (DE) 1987-02-24 US disclosed
US-4585471-A PREEMERGENCE BAYER AKTIENGESELLSCHAFT (DE) 1986-04-29 US disclosed
EP-0159962-A2 Fibre-reactive chromium or cobalt complexes, their preparation and their use CIBA-GEIGY AG (CH) 1985-10-30 EP disclosed
US-4549899-A Hericidally active novel substituted 3-trihalogenomethyl-1,2,4-thiadiazol-5-yl-oxyacetamides BAYER AKTIENGESELLSCHAFT (DE) 1985-10-29 US disclosed
US-4540430-A Herbicidally active novel substituted 3-trichloromethyl-1,2,4-thiadiazol-5-yl-oxyacetamides BAYER AKTIENGESELLSCHAFT (DE) 1985-09-10 US disclosed
EP-0045488-B1 WATER-SOLUBLE FIBRE-REACTIVE COMPOUNDS AND THEIR USE IN FINISHING TEXTILES, AS WELL AS THE BETA-CHLOROETHYL-SULFONYL-METHYL-BENZOIC-ACID HALOGENIDES, AND THEIR USE AS A FIBRE-REACTIVE ANCHOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-06-19 EP disclosed
EP-0144776-A2 Fibre-reactive chromium complexes, their preparation and their use CIBA-GEIGY AG (CH) 1985-06-19 EP disclosed
EP-0142104-A2 Fibre-reactive chromium complexes, their preparation and their use CIBA-GEIGY AG (CH) 1985-05-22 EP disclosed
EP-0141416-A2 Fibre-reactive chromium complexes, their preparation and their use CIBA-GEIGY AG (CH) 1985-05-15 EP disclosed
US-4509971-A Benzothiazole substituted carboxylic acid amide compounds and herbicidal methods compositions thereof BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed
US-4473498-A Water-soluble, fiber-reactive organic dyestuffs containing a β-chloro-ethylsulfonyl-methyl-benzoic acid amide group HOECHST AKTIENGESELLSCHAFT (DE) 1984-09-25 US disclosed
US-4455428-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1984-06-19 US disclosed
US-4399285-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1983-08-16 US disclosed
EP-0012969-B1 WATER-SOLUBLE FIBRE-REACTIVE COMPOUNDS AND THEIR USE IN FIBRE FINISHING,ESPECIALLY AS DYESTUFFS,AND DIHALOGENO-PYRIDAZONYL-CARBOXYLIC AND SULFONIC ACID HALIDES AND THEIR USE AS FIBRE-REACTIVE ANCHORS,AS WELL AS PROCESS FOR THE PREPARATION OF THESE COMPOUND HOECHST AKTIENGESELLSCHAFT (DE) 1983-06-08 EP disclosed
US-4334073-A BASIC CATALYSTS, DEACETYLATION, ESTERIFICATION BAYER AKTIENGESELLSCHAFT (DE) 1982-06-08 US disclosed
EP-0045488-A2 Water-soluble fibre-reactive compounds and their use in finishing textiles, as well as the beta-chloroethyl-sulfonyl-methyl-benzoic-acid halogenides, and their use as a fibre-reactive anchor HOECHST AKTIENGESELLSCHAFT (DE) 1982-02-10 EP disclosed
EP-0030676-A1 Derivatives of phenoxybenzoic acid, process for their preparation and their use as herbicides and as plant growth regulators BAYER AG (DE) 1981-06-24 EP disclosed
EP-0030287-A1 1-Aminocyclopropanecarboxylic acid derivatives, methods for their production, their use as plant-growth regulators and compositions containing such derivatives BAYER AG (DE) 1981-06-17 EP disclosed
EP-0012969-A2 Water-soluble fibre-reactive compounds and their use in fibre finishing,especially as dyestuffs,and dihalogeno-pyridazonyl-carboxylic and sulfonic acid halides and their use as fibre-reactive anchors,as well as process for the preparation of these compound HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-09 EP disclosed
US-4116952-A POLYAMIDES CIBA-GEIGY CORPORATION (US) 1978-09-26 US disclosed
US-RE29585-E DYEING WOOL CIBA-GEIGY CORPORATION (US) 1978-03-21 US disclosed
US-4067903-A Manufacture of arylamines BASF AKTIENGESELLSCHAFT (DT) 1978-01-10 US disclosed
US-4065492-A Process for preparing aminonaphthalene derivatives in a titanium or titanium alloy reactor BAYER AKTIENGESELLSCHAFT (DT) 1977-12-27 US disclosed
US-4033942-A Chromium complex dye, including azo and azo methine dye compounds CIBA-GEIGY AG (CH) 1977-07-05 US disclosed
US-4002606-A FIBER-REACTIVE DYES HOECHST AKTIENGESELLSCHAFT (DT) 1977-01-11 US disclosed
US-3978037-A POLYAMIDES CIBA-GEIGY CORPORATION (US) 1976-08-31 US disclosed
US-3971738-A Heavy metal complexes of azo compounds containing a halogeno-2,3-dihydroxy pyridine coupling component CIBA-GEIGY AG (CH) 1976-07-27 US disclosed
US-3933785-A Azo compounds CIBA-GEIGY AG (CH) 1976-01-20 US disclosed
US-3933785-A Azo compounds CIBA-GEIGY AG (CH) 1976-01-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160194284-A1 ALLOSTERIC MODULATORS OF THE CANNABINOID 1 RECEPTOR CNR1, CNR2, GPR119 ALDH1A1 2771/4885CYP1A2 1120/4885CYP3A4 1339/4885
US-20130217685-A1 COMPOUNDS FOR MODULATING RNA BINDING PROTEINS AND USES THEREFOR TIA1, ZFP3, RBM3 ALDH1A1 3135/4885CYP1A2 4801/4885CYP3A4 4278/4885
US-20120202821-A1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS HTR2B, MC1R, HTR1A ALDH1A1 4268/4885CYP1A2 882/4885CYP3A4 1869/4885
US-20070294842-A1 Reactive Dyes, a Process for Their Preparation and Their Use CBR3, ARSA, CBR1 ALDH1A1 397/4885CYP1A2 1208/4885CYP3A4 625/4885
US-20230122957-A1 PSMA LIGANDS FOR IMAGING AND ENDORADIOTHERAPY KLK3, FOLH1, EEA1 ALDH1A1 1331/4885CYP1A2 4483/4885CYP3A4 4103/4885
US-20100125140-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR UTS2R, TRPV1, GPR17 ALDH1A1 1211/4885CYP1A2 1934/4885CYP3A4 1496/4885
US-20230133581-A1 Novel 3,5-Diaminobenzoic Acid Compound, and PIN1 Inhibitor and Therapeutic Agent for Inflammatory Diseases Using Same PIN1, DUSP15, FKBP1A ALDH1A1 2183/4885CYP1A2 1141/4885CYP3A4 1308/4885
US-20240400568-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20230203048-A1 SPIROPYRROLIDINE DERIVED ANTIVIRAL AGENTS ACE, ACE2, PKD1 ALDH1A1 319/4885CYP1A2 1377/4885CYP3A4 221/4885
US-20170174639-A1 EIS INHIBITORS ABCC1, ATP5ME, ABCG2 ALDH1A1 819/4885CYP1A2 2393/4885CYP3A4 2869/4885
US-20080097102-A1 AMINOTETRALIN-DERIVED UREA MODULATORS OF VANILLOID VR1 RECEPTOR UTS2R, TRPV1, GPR17 ALDH1A1 1211/4885CYP1A2 1934/4885CYP3A4 1496/4885
US-20070282101-A1 Indazole compounds CYP3A43, CYP3A7, UGT1A1 ALDH1A1 89/4885CYP1A2 15/4885CYP3A4 5/4885
US-11370740-B2 Method for producing ester group-containing compound COASY, TAF5, TAF9 ALDH1A1 1667/4885CYP1A2 1185/4885CYP3A4 673/4885
US-20260112544-A1 ELECTROLYTIC CAPACITOR ASIC1, SLC9A2, SLC25A13 ALDH1A1 508/4885CYP1A2 1225/4885CYP3A4 1967/4885
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND ERG28, CYP51A1, XPO1 ALDH1A1 1677/4885CYP1A2 147/4885CYP3A4 61/4885
US-20120071478-A1 SUBSTITUTED BENZOTRIAZINES AND QUINOXALINES AS INHIBITORS OF P7OS6 KINASE CDK1, CDK2, CDK6 ALDH1A1 4137/4885CYP1A2 1508/4885CYP3A4 2000/4885
US-20220324866-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20230250048-A1 NITROGEN-CONTAINING COMPOUND, ELECTRONIC ELEMENT AND ELECTRONIC DEVICE NOS1, NOM1, NCF1 ALDH1A1 1717/4885CYP1A2 1640/4885CYP3A4 1315/4885
US-20090227799-A1 Novel Antimalarial Agent Containing Heterocyclic Compound XPO1, THPO, G6PD ALDH1A1 1926/4885CYP1A2 1886/4885CYP3A4 1535/4885
US-20230301182-A1 ORGANIC COMPOUND, AND ELECTRONIC ELEMENT AND ELECTRONIC DEVICE USING SAME OR10J3, ESR1, EPCAM ALDH1A1 496/4885CYP1A2 428/4885CYP3A4 309/4885
US-20230322656-A1 ORGANIC COMPOUND, AND ELECTRONIC COMPONENT AND ELECTRONIC DEVICE HAVING SAME PIEZO1, OR10J3, ODC1 ALDH1A1 237/4885CYP1A2 213/4885CYP3A4 133/4885
US-20160368881-A1 THERAPEUTIC COMPOUNDS HAVCR2, SARS1, RPL35 ALDH1A1 429/4885CYP1A2 782/4885CYP3A4 358/4885
US-20090275578-A1 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators GRM1, GRIN1, GRM3 ALDH1A1 1582/4885CYP1A2 1256/4885CYP3A4 1095/4885
US-10227364-B2 Silane and silicic acid (hetero)polycondensate having aromatic compounds linked via coupling groups which are suitable as or for matrix systems having high translucency and good mechanical properties NR4A1, SMC4, NR4A2 ALDH1A1 4377/4885CYP1A2 4394/4885CYP3A4 2510/4885
US-20050187291-A1 use of 2-(urea or thiourea)tetralins as analgesic or to treat pulmonary dysfunction TMEM109, UTS2R, GPR17 ALDH1A1 1133/4885CYP1A2 1823/4885CYP3A4 2581/4885
US-20080096925-A1 Novel Substituted 4-Phenyl-4[H-Imidazol-2-YL]-Piperidine Derivatived And Their Use As Selective Non-Peptide Delta Opioid Agonists OPRD1, OPRK1, OPRL1 ALDH1A1 1647/4885CYP1A2 1627/4885CYP3A4 1049/4885
US-11767291-B2 Preparation of secondary amines with electrophilic N-linchpin reagents PNMT, NCL, NPM1 ALDH1A1 1805/4885CYP1A2 2396/4885CYP3A4 3968/4885
US-20200383987-A1 Novel Amide Compound, and Pin1 Inhibitor, Therapeutic Agent for Inflammatory Diseases and Therapeutic Agent for Cancer That Use the Same PIN1, FKBP1A, FKBP5 ALDH1A1 3518/4885CYP1A2 2435/4885CYP3A4 3220/4885
US-12054490-B2 Diacylglycerol kinase modulating compounds DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20040143118-A1 Chiral organic compounds and metal coordination complexes thereof ORC3, SOD1, SLC39A3 ALDH1A1 3442/4885CYP1A2 1967/4885CYP3A4 1059/4885
US-20130029878-A1 Method for Assaying Histone Methylation Enzyme Activity EHMT1, DOT1L, EHMT2 ALDH1A1 1742/4885CYP1A2 3922/4885CYP3A4 3405/4885
US-20070105943-A1 Novel antifungal agent containing heterocyclic compound ERG28, DPM1, CYP51A1 ALDH1A1 1459/4885CYP1A2 187/4885CYP3A4 104/4885
US-20200297876-A1 PSMA ligands for imaging and endoradiotherapy KLK3, FOLH1, EEA1 ALDH1A1 1331/4885CYP1A2 4483/4885CYP3A4 4103/4885
US-12531188-B2 Electrolytic capacitor ASIC1, SLC1A2, HCN2 ALDH1A1 1325/4885CYP1A2 2181/4885CYP3A4 2762/4885
US-11845723-B2 Diacylglycerol kinase modulating compounds DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20230200209-A1 ORGANOMETALLIC COMPOUND AND ORGANIC LIGHT-EMITTING DIODE INCLUDING THE SAME CRY1, ZFX, PPOX ALDH1A1 315/4885CYP1A2 523/4885CYP3A4 237/4885
US-20040204455-A1 Piperidine derivative rennin inhibitors REN, ACE, HPN ALDH1A1 921/4885CYP1A2 2821/4885CYP3A4 2949/4885
US-20030149089-A1 Antibacterial compounds MRPL21, MRPS28, SPOUT1 ALDH1A1 388/4885CYP1A2 742/4885CYP3A4 698/4885
US-11130780-B2 Inhibitors of growth factor activation enzymes HDGF, MMP7, HGF ALDH1A1 2862/4885CYP1A2 977/4885CYP3A4 1459/4885
US-20230303537-A1 NITROGEN-CONTAINING COMPOUND, AND ELECTRONIC ELEMENT AND ELECTRONIC DEVICE THEREOF NPM1, NFE2L2, MNS1 ALDH1A1 2635/4885CYP1A2 1184/4885CYP3A4 2158/4885
US-20160185804-A1 SILANE AND SILICIC ACID (HETERO)POLYCONDENSATE HAVING AROMATIC COMPOUNDS LINKED VIA COUPLING GROUPS WHICH ARE SUITABLE AS OR FOR MATRIX SYSTEMS HAVING HIGH TRANSLUCENCY AND GOOD MECHANICAL PROPERTIES NR4A1, SMC4, NR4A2 ALDH1A1 4377/4885CYP1A2 4394/4885CYP3A4 2510/4885
US-20150239894-A1 Amino Compounds for Treatment of Complement Mediated Disorders CFD, TFPI, C9 ALDH1A1 3450/4885CYP1A2 4580/4885CYP3A4 4463/4885
US-10202353-B2 Therapeutic compounds RPL35, SARS1, HAVCR2 ALDH1A1 424/4885CYP1A2 903/4885CYP3A4 488/4885
US-20240182476-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK ALDH1A1 4095/4885CYP1A2 4595/4885CYP3A4 4334/4885
US-20230355609-A1 Spirolactone Compounds ACACA, AKR1C2, AKR1A1 ALDH1A1 40/4885CYP1A2 204/4885CYP3A4 1349/4885
US-20070149495-A1 HISTONE DEACETYLASE INHIBITORS HDAC1, HDAC3, HDAC11 ALDH1A1 2744/4885CYP1A2 4543/4885CYP3A4 4453/4885
US-20080027060-A1 DIPEPTIDE NITRILES CTSL, CTSS, CTSB ALDH1A1 4249/4885CYP1A2 3454/4885CYP3A4 895/4885
US-20150360214-A1 REACTION CATALYST FOR CROSS-COUPLING AND METHOD FOR MANUFACTURING AROMATIC COMPOUND ALK, HRH4, HRH3 ALDH1A1 2351/4885CYP1A2 516/4885CYP3A4 237/4885
US-20240024266-A1 Therapeutic Agent or Prophylactic Agent for COVID-19 PIN1, ACE2, ACE ALDH1A1 4006/4885CYP1A2 4049/4885CYP3A4 3976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.