Itraconazole

Itraconazole

SCHEMBL95627

CCC(C)n1ncn(-c2ccc(N3CCN(c4ccc(OCC5COC(Cn6cncn6)(c6ccc(Cl)cc6Cl)O5)cc4)CC3)cc2)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Itraconazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 19/20 1.00
ABCG2 Q9UNQ0 3/20 1.00
LMNA P02545 3/20 1.00
CYP51A1 Q16850 3/20 1.00
FYN P06241 2/20 1.00
MEN1 O00255 2/20 1.00
ABCB11 O95342 2/20 1.00
ABCB1 P08183 2/20 1.00
MAPT P10636 2/20 1.00
MAPK1 P28482 2/20 1.00
KMT2A Q03164 2/20 1.00
HIF1A Q16665 2/20 1.00
CYP8B1 Q9UNU6 2/20 1.00
CXCR1 P25024 1/20 1.00
TACR1 P25103 1/20 1.00
AVPR2 P30518 1/20 1.00
CCR4 P51679 1/20 1.00
PDE4D Q08499 1/20 1.00
NR1I2 O75469 2/20 0.75
HSP90AA1 P07900 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Itraconazole SCHEMBL14875797 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL16984893 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL14875705 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL18073409 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL23934 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL15948108 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL18241650 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL20464865 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL14875903 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN
Itraconazole SCHEMBL64913 1.00 CYP3A4 (1.00) CYP3A4ABCG2LMNACYP51A1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 577 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3813799-B1 PHARMACEUTICAL FORMULATION WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY CONSEJO SUPERIOR INVESTIGACION (ES) 2024-02-21 EP claimed
CN-116925052-A Synthesis method of optically pure itraconazole 上海现代哈森(商丘)药业有限公司 2023-10-24 CN claimed
US-20230158259-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS TOPELIA AUST LIMITED (652 771 670) (AU) 2023-05-25 US claimed
CN-115955965-A Products of manufacture and methods for treating, ameliorating or preventing microbial infections 拓比利亚欧斯特有限公司 2023-04-11 CN claimed
EP-4138832-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS Topelia Aust Limited (AU) 2023-03-01 EP claimed
US-20220401579-A1 INCLUSION COMPLEXES OF PHARMACEUTICALS AND CYCLIC OLIGOMERS DISPERSOL TECHNOLOGIES, LLC (US) 2022-12-22 US claimed
US-20220378861-A1 COMPOSITIONS AND METHODS FOR DELIVERING CANNABINOIDS USING MICRONEEDLE DEVICES TO THE SKIN AQUAVIT PHARMACEUTICALS INC (US) 2022-12-01 US claimed
CN-115219611-A Kit for determining 7 antifungal drugs in serum by ultra-high performance liquid chromatography-tandem mass spectrometry and application thereof 上海义准生物有限公司 2022-10-21 CN claimed
CN-114660200-A Method for simultaneously measuring 4 triazole antifungal drugs in blood plasma by high performance liquid chromatography tandem mass spectrometry technology 中国人民解放军总医院 2022-06-24 CN claimed
EP-3753966-B1 AMPHIPHILIC BLOCK COPOLYMER, PREPARATION METHOD THEREOF AND NANOMICELLE DRUG-LOADING SYSTEM SHANGHAI BEST LINK BIOSCIENCE LLC (CN) 2022-05-25 EP claimed
US-20220143143-A1 USE OF ACTIVATORS OF THE ARYL HYDROCARBON RECEPTOR FOR TREATING GLUTEN-INDUCED GASTROINTESTINAL DISEASES UNIV MCMASTER (CA) 2022-05-12 US claimed
WO-2022094174-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ESOPHAGEAL CONDITIONS CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-05-05 WO claimed
EP-1511490-A4 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS TRANSFORM PHARMACEUTICALS INC (US) 2009-03-11 EP claimed
US-20080305173-A1 AMORPHOUS DRUG BEADS BOGUE BEUFORD ARLIE 2008-12-11 US claimed
EP-1511490-A2 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS Transform Pharmaceuticals, Inc. (US) 2005-03-09 EP claimed
WO-2004108114-A2 ANTI-FUNGAL COMPOSITION AND A PROCESS FOR ITS MANUFACTURE PATEL DINESH SHANTILAL (IN) 2004-12-16 WO claimed
WO-2003101392-A2 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS TRANSFORM PHARMACEUTICALS, INC. (US) 2003-12-11 WO claimed
US-20030026843-A1 Amorphous drug beads CAPRICORN PHARMA INC. 2003-02-06 US claimed
US-4988697-A Alpha-demethylase inhibiting azole compound and a beta-lactone MERCK & CO., INC. (US) 1991-01-29 US claimed
CN-122031617-A Traditional Chinese medicine composition and traditional Chinese medicine preparation for preventing and treating invasive aspergillosis as well as preparation method and application of traditional Chinese medicine composition and traditional Chinese medicine preparation 淮北市中医医院 2026-05-15 CN disclosed
US-20260102391-A1 INHIBITION OF A TRIPARTITE VOR PROTEIN COMPLEX IN MULTICELLULAR ORGANISMS LORICO AURELIO (US) 2026-04-16 US disclosed
US-20260091097-A1 COMBINATION TREATMENT REGIMES FOR TREATING CANCER BARINTHUS BIOTHERAPEUTICS NORTH AMERICA INC (US) 2026-04-02 US disclosed
US-12582717-B2 Protein based excipient for active pharmaceutical ingredients DISPERSOME IP APS (NL) 2026-03-24 US disclosed
US-20260076977-A1 METHODS FOR TREATMENT OF DISEASES GALERA LABS LLC (US) 2026-03-19 US disclosed
EP-4709721-A1 DUAL EZH2-HSP90 INHIBITORS Taipei Medical University (TW) 2026-03-18 EP disclosed
US-12569482-B2 Methods and compositions for treating idiopathic pulmonary fibrosis LIANG GUI BAI (US) 2026-03-10 US disclosed
US-20260066250-A1 METHOD AND DEVICE FOR THE QUANTIFICATION OF TARGET ION SPECIES BRUKER DALTONICS GMBH & CO KG (DE) 2026-03-05 US disclosed
US-20260048013-A1 PHARMACEUTICAL FORMULATION WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY CONSEJO SUPERIOR INVESTIGACION (ES) 2026-02-19 US disclosed
US-20260047266-A1 ORGANIC ELECTROLUMINESCENT ELEMENT NIPPON STEEL CHEMICAL & MATERIAL CO., LTD. (JP) 2026-02-12 US disclosed
US-20260041734-A1 M-CSF FOR USE IN THE PROPHYLAXIS AND/OR TREATMENT OF VIRAL INFECTIONS IN STATES OF IMMUNOSUPPRESSION UNIV DRESDEN TECH (DE) 2026-02-12 US disclosed
US-12527789-B2 Inhibition of a tripartite VOR protein complex in multicellular organisms LORICO, Aurelio (US) 2026-01-20 US disclosed
US-12508248-B2 Therapeutic agent for prototheca disease SEREN PHARMACEUTICALS INC. (JP) 2025-12-30 US disclosed
US-20250387326-A1 CRYSTALLINE PHARMACEUTICAL COMPOSITION FOR INHALATION COMPRISING SUGAR AND LIPID COMPOSITE PARTICLES AND PROCESS FOR MANUFACTURE HOVIONE SCIENTIA LTD (IE) 2025-12-25 US disclosed
US-12494355-B2 Method and device for the quantification of target ion species BRUKER DALTONICS GMBH & CO KG (DE) 2025-12-09 US disclosed
EP-4651898-A1 STABILIZED BIOPOLYMER COMPOSITION, THEIR MANUFACTURE AND USE BASF SE (DE) 2025-11-26 EP disclosed
CN-121005819-A Biocompatible antibacterial composite material and preparation method thereof 中国科学院化学研究所 2025-11-25 CN disclosed
EP-4642465-A1 A CANCER ASSOCIATED FIBROBLAST (CAF) INHIBITOR FOR USE WITH AN ALTERNATING ELECTRIC FIELD IN A METHOD OF TREATING DISEASES SUCH AS CANCER Novocure GmbH (CH) 2025-11-05 EP disclosed
EP-4641223-A1 SYSTEM FOR DETECTING LEAKAGE CURRENTS FOR DRIVE SYSTEMS OF VEHICLES WITH AN ELECTRIC DRIVE SYSTEM CAF Power & Automation, S.L.U. (ES) 2025-10-29 EP disclosed
US-20250325494-A1 COMPOSITION FOR ORGAN-SPECIFIC DELIVERY OF NUCLEIC ACID THEMEDIUM THERAPEUTICS CO., LTD. (CN) 2025-10-23 US disclosed
US-12435067-B2 Truncated itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2025-10-07 US disclosed
US-12419838-B2 Pharmaceutical formulation with improved solubility and bioavailability CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS (CSIC) (ES) 2025-09-23 US disclosed
EP-3522902-B1 PROBIOTIC BACTERIA PRODUCING AN AHR AGONIST AND THEIR USE IN THE TREATMENT OF METABOLIC SYNDROME AND OBESITY INSTITUT NATIONAL DE RECH POUR LAGRICULTURE LALIMENTATION ET LENVIRONNEMENT (FR) 2025-09-03 EP disclosed
EP-4608437-A2 COMBINATION TREATMENT REGIMES FOR TREATING CANCER Barinthus Biotherapeutics North America, Inc. (US) 2025-09-03 EP disclosed
EP-4608455-A1 SELF-ASSEMBLING NANOPARTICLES Barinthus Biotherapeutics North America, Inc. (US) 2025-09-03 EP disclosed
US-20250248986-A1 ANTIFUNGAL DRUG INHALATION FORMULATIONS Hefei Cosource Pharmaceuticals Co., Ltd (CN) 2025-08-07 US disclosed
US-20250243176-A1 (S)-1-(1-ACRYLOYLPIPERIDIN-3-YL)-2-FLUORO-5,6,7,8,9,10-HEXAHYDROCYCLO HEPTA[B]INDOLE-4-CARBOXAMIDE, AND RELATED CRYSTALLINE FORMS, COMPOSITIONS, AND METHODS THEREOF VIDYA THERAPEUTICS, INC. 2025-07-31 US disclosed
US-20250242015-A1 SELF-ASSEMBLING NANOPARTICLES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 2025-07-31 US disclosed
EP-4592677-A1 METHOD FOR ASSISTING IN DETERMINING TREATMENT PLAN FOR DOG HAVING SKIN CONDITION Nippon Zenyaku Kogyo Co., Ltd. (JP) 2025-07-30 EP disclosed
US-20250235422-A1 DODECA-2,4,6,8,10-PENTAENOIC ACID COMPOSITIONS AND USES THEREOF BIOMEDIT, INC. 2025-07-24 US disclosed
US-20250228788-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-07-17 US disclosed
US-20250188013-A1 LIPID COMPOUND AND USE THEREOF THEMEDIUM THERAPEUTICS CO., LTD. (CN) 2025-06-12 US disclosed
EP-4558161-A1 M-CSF FOR USE IN THE PROPHYLAXIS AND/OR TREATMENT OF VIRAL INFECTIONS IN STATES OF IMMUNOSUPPRESSION Technische Universität Dresden (DE) 2025-05-28 EP disclosed
US-20250161386-A1 METHOD OF IMPROVING COGNITIVE FUNCTION IN ADULTS SEMPERA ORGANICS, INC. 2025-05-22 US disclosed
CN-119950465-A Application of carbonyl cyanide-4-trifluoromethoxy phenylhydrazone in aspergillus fumigatus infection prevention and treatment 安徽中医药大学 2025-05-09 CN disclosed
US-12290538-B2 Methods and products for treatment of gastrointestinal disorders FINCH THERAPEUTICS HOLDINGS LLC (US) 2025-05-06 US disclosed
EP-4545147-A2 PHOTOPROTECTIVE COMPOSITIONS CONTAINING MALASSEZIA-DERIVED COMPOUNDS AND/OR CHEMICAL ANALOGS THEREOF VERSICOLOR TECHNOLOGIES, LLC (US) 2025-04-30 EP disclosed
US-12285522-B2 Thermally gelling drug formulations UNM RAINFOREST INNOVATIONS (US) 2025-04-29 US disclosed
US-20250127717-A1 COMPOSITIONS AND METHODS OF MAKING BRITTLE-MATRIX PARTICLES THROUGH BLISTER PACK FREEZING UNIV TEXAS (US) 2025-04-24 US disclosed
US-20250127887-A1 Self-Assembling Nanoparticles Based On Amphiphilic Peptides BARINTHUS BIOTHERAPEUTICS NORTH AMERICA, INC. (US) 2025-04-24 US disclosed
EP-4539821-A1 CRYSTALLINE PHARMACEUTICAL COMPOSITION FOR INHALATION COMPRISING SUGAR AND LIPID COMPOSITE PARTICLES AND PROCESS FOR MANUFACTURE Hovione Scientia Limited (IE) 2025-04-23 EP disclosed
CN-119856599-A Organic electroluminescent element 日铁化学材料株式会社 2025-04-18 CN disclosed
CN-119798484-A Retinoyl hyaluronic acid sodium acid and composition thereof 山东省药学科学院 2025-04-11 CN disclosed
US-12263243-B2 Templated open flocs of anisotropic particles for enhanced pulmonary delivery BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-04-01 US disclosed
WO-2025043394-A1 KIT FOR FORMING SUPRAMOLECULAR SELF-ASSEMBLY COMPLEX AND USE THEREOF 北京睿创康泰医药研究院有限公司 2025-03-06 WO disclosed
CN-112996519-B Compositions and methods for organ-specific delivery of nucleic acids 德克萨斯大学系统董事会 2025-02-28 CN disclosed
US-20250060358-A1 DIAGNOSIS AND TREATMENT OF HISTOPLASMOSIS THE BRIGHAM AND WOMEN’S HOSPITAL INC (US) 2025-02-20 US disclosed
US-12226404-B2 Methods for making compositions for pulmonary administration BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-02-18 US disclosed
US-20250051519-A1 SOLUTION ELECTROSPUN FIBERS, COMPOSITIONS COMPRISING THE SAME AND A PROCESS OF MANUFACTURING THEREOF UNIVERSITEIT GENT (BE) 2025-02-13 US disclosed
CN-119421870-A Lipid compound and application thereof 传信生物医药(苏州)有限公司 2025-02-11 CN disclosed
CN-119384273-A Organ-specific delivery compositions for nucleic acids 传信生物医药(苏州)有限公司 2025-01-28 CN disclosed
US-12203124-B2 Methods for improved rapid antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2025-01-21 US disclosed
US-20250017944-A1 METHODS FOR TREATMENT OF DISEASES GALERA LABS, LLC 2025-01-16 US disclosed
US-20250000800-A1 METHODS OF PREPARING DOSAGE FORMS USING 3D PRINTING CONTAINING AMORPHOUS SOLID DISPERSIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2025-01-02 US disclosed
EP-3774811-B1 PHOTOPROTECTIVE COMPOSITIONS CONTAINING MALASSEZIA-DERIVED COMPOUNDS AND/OR CHEMICAL ANALOGS THEREOF VERSICOLOR TECH LLC (US) 2024-12-18 EP disclosed
US-20240398760-A1 CHELATED, STABLE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF SOMERSET THERAPEUTICS, LLC 2024-12-05 US disclosed
WO-2024249959-A1 COMPOSITIONS REDUCING THE EXPRESSION OR ACTIVITY OF C1 GALT1 FOR TREATING EWING SARCOMA UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL (US) 2024-12-05 WO disclosed
US-20240390271-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-28 US disclosed
US-20240390272-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-28 US disclosed
CN-116064571-B Mango salt-tolerant gene and identification method and application thereof 中国热带农业科学院三亚研究院 2024-11-26 CN disclosed
WO-2024238381-A1 DUAL EZH2-HSP90 INHIBITORS TAIPEI MEDICAL UNIVERSITY (TW) 2024-11-21 WO disclosed
US-20240374512-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-14 US disclosed
US-20240374513-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-14 US disclosed
US-20240374511-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-14 US disclosed
US-20240374514-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2024-11-14 US disclosed
EP-3998109-B1 NOVEL THERAPEUTIC AGENT FOR PROTOTHECA DISEASE SEREN PHARMACEUTICALS INC (JP) 2024-11-13 EP disclosed
EP-3152321-B1 DIAGNOSIS AND TREATMENT OF INVASIVE ASPERGILLOSIS BRIGHAM & WOMENS HOSPITAL INC (US) 2024-11-13 EP disclosed
CN-118903162-A Application of forsythoside A in preparation of medicines and method for screening active components in medicines 闽江学院 2024-11-08 CN disclosed
CN-115845069-B Combined medicine, application and kit for treating oral squamous cell carcinoma 四川大学 2024-11-08 CN disclosed
EP-4456921-A2 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-11-06 EP disclosed
US-12133924-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-11-05 US disclosed
US-20240358718-A1 CONCOMITANT ADMINISTRATION OF GLUCOCORTICOID RECEPTOR MODULATORS AND CYP3A INHIBITORS CORCEPT THERAPEUTICS, INC. (US) 2024-10-31 US disclosed
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EP-4453292-A1 SOLUTION ELECTROSPUN FIBERS, COMPOSITIONS COMPRISING THE SAME AND A PROCESS OF MANUFACTURING THEREOF Universiteit Gent (BE) 2024-10-30 EP disclosed
CN-116077499-B Anti-azole aspergillus fumigatus pharmaceutical composition and application thereof 徐州医科大学 2024-10-29 CN disclosed
US-12121512-B2 Anti-fungal agent SEREN PHARMACEUTICALS INC. (JP) 2024-10-22 US disclosed
US-12121610-B2 Compositions and methods for targeted delivery to cells RECODE THERAPEUTICS, INC. (US) 2024-10-22 US disclosed
WO-2024216136-A1 COMBINATION THERAPY FOR THE TREATMENT OF HEMATOLOGICAL CANCERS FOGHORN THERAPEUTICS INC. (US) 2024-10-17 WO disclosed
WO-2024216151-A1 COMBINATION THERAPY FOR TREATING HEMATOLOGICAL CANCERS FOGHORN THERAPEUTICS INC. (US) 2024-10-17 WO disclosed
US-12102632-B2 Quinolone dispersions SOMERSET THERAPEUTICS, LLC (US) 2024-10-01 US disclosed
US-12097210-B2 Concomitant administration of glucocorticoid receptor modulators and CYP3A inhibitors CORCEPT THERAPEUTICS, INC. (US) 2024-09-24 US disclosed
CN-118660721-A Compositions and methods for targeted delivery to cells 德克萨斯大学系统董事会 2024-09-17 CN disclosed
US-20240301498-A1 DIAGNOSTIC METHOD FOR CANCER EVOLUTION PREDICTION, AND USES THEREOF INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2024-09-12 US disclosed
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WO-2024177494-A1 SYSTEM FOR SECURING PHOTOVOLTAIC MODULES TO TRAPEZOIDAL SHEET ROOFS SANTANA CISNEROS ARTURO JAVIER (MX) 2024-08-29 WO disclosed
EP-4419532-A1 FUSED BICYCLIC HETEROARYL COMPOUNDS USEFUL AS NLRP3 INHIBITORS F. Hoffmann-La Roche AG (CH) 2024-08-28 EP disclosed
US-12071430-B2 Itraconazole analogs and use thereof THE JOHNS HOPKINS UNIVERSITY (US) 2024-08-27 US disclosed
US-20240269269-A1 Self-Assembling Nanoparticles VACCITECH NORTH AMERICA, INC. (US) 2024-08-15 US disclosed
US-20240272140-A1 DIAGNOSIS AND TREATMENT OF FUSARIOSIS AND SCEDOSPORIOSIS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2024-08-15 US disclosed
EP-3626242-B1 ITRACONAZOLE ANALOGS AS INHIBITORS OF FIBROSIS SCRIPPS RESEARCH INST (US) 2024-08-07 EP disclosed
EP-3641822-B1 DRY-BINDERS FOR TABLETS BASED ON POLYETHYLENE GLYCOL-POLYVINYL ALCOHOL GRAFT POLYMERS, THE PRODUCTION AND USE THEREOF BASF SE (DE) 2024-08-07 EP disclosed
US-20240255506-A1 PAIRED-CELL PROFILING SYSTEMS FOR HIGH-THROUGHPUT SCREENING SYNCYTIUM FORMATION VERSITECH LIMITED (CN) 2024-08-01 US disclosed
US-20240252449-A1 STABILISED COMPOSITIONS Rumin8 Pty Ltd (AU) 2024-08-01 US disclosed
CN-118406679-A Paired cell assay system for high throughput screening syncytia formation 港大科桥有限公司 2024-07-30 CN disclosed
CN-118401506-A (S) -1- (1-propenylpiperidin-3-yl) -2-fluoro-5, 6,7,8,9, 10-hexahydrocyclohepta [ b ] indole-4-carboxamide and related crystalline forms, compositions and methods GB005股份有限公司 2024-07-26 CN disclosed
US-20240245618-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-25 US disclosed
WO-2024153789-A1 STABILIZED BIOPOLYMER COMPOSITION, THEIR MANUFACTURE AND USE BASF SE (DE) 2024-07-25 WO disclosed
US-20240245620-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-25 US disclosed
EP-4402278-A1 DIAGNOSIS AND TREATMENT OF HISTOPLASMOSIS The Brigham & Women's Hospital, Inc. (US) 2024-07-24 EP disclosed
WO-2024151838-A1 CO-CRYSTALS WITH THIN-FILM FREEZE-DRYING PROCESS TO ENHANCE DELIVERY BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-18 WO disclosed
EP-4400491-A1 NOVEL LIPIDS USED FOR NUCLEIC ACID DELIVERY AND LIPID NANOPARTICLE COMPOSITION Themedium Therapeutics Co., Ltd (CN) 2024-07-17 EP disclosed
EP-3968964-B1 METHOD FOR PRODUCING NANOPARTICLES LEON NANODRUGS GMBH (DE) 2024-07-10 EP disclosed
US-12029816-B2 Compositions and methods of making brittle-matrix particles through blister pack freezing BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-09 US disclosed
US-12029729-B2 Chelated, stable ophthalmological compositions of ketorolac and phenylephrine and applications thereof SOMERSET THERAPEUTICS, LLC (US) 2024-07-09 US disclosed
US-20240216515-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2024-07-04 US disclosed
WO-2024141952-A1 A CANCER ASSOCIATED FIBROBLAST (CAF) INHIBITOR FOR USE WITH AN ALTERNATING ELECTRIC FIELD IN A METHOD OF TREATING DISEASES SUCH AS CANCER NOVOCURE GMBH (CH) 2024-07-04 WO disclosed
US-20240216403-A1 METHODS AND COMPOSITIONS FOR INHIBITING FIBROBLAST ACTIVATION BIOPHARMA CREDIT PLC (GB) 2024-07-04 US disclosed
EP-4393511-A1 LIPID COMPOUND AND USE THEREOF Themedium Therapeutics Co., Ltd. (CN) 2024-07-03 EP disclosed
EP-4393484-A1 COMPOSITION FOR ORGAN-SPECIFIC DELIVERY OF NUCLEIC ACID Themedium Therapeutics Co., Ltd. (CN) 2024-07-03 EP disclosed
EP-4393513-A1 DRY SUSPENSION PARTICLES FOR DRY SUSPENSION, PREPARATION METHOD THEREFOR AND USE THEREOF Livzon Pharmaceutical Group Inc. (CN) 2024-07-03 EP disclosed
US-12023343-B2 Thermo-kinetic mixing for pharmaceutical applications AustinPx, LLC (US) 2024-07-02 US disclosed
WO-2024133992-A1 SYSTEM FOR DETECTING LEAKAGE CURRENTS FOR DRIVE SYSTEMS OF VEHICLES WITH AN ELECTRIC DRIVE SYSTEM CAF POWER & AUTOMATION, S.L.U. (ES) 2024-06-27 WO disclosed
US-20240207178-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-06-27 US disclosed
WO-2024136219-A1 INHALATION FORMULATION COMPRISING NANOPARTICLES AND PREPARATION METHOD THEREFOR 주식회사 포스테라헬스사이언스 2024-06-27 WO disclosed
US-12016855-B2 Prednisolone and moxifloxacin compositions and methods SOMERSET THERAPEUTICS, LLC (US) 2024-06-25 US disclosed
US-20240201166-A1 DIAGNOSIS AND TREATMENT OF CONGESTIVE COLON FAILURE (CCF) KHURANA VIKAS (US) 2024-06-20 US disclosed
US-20240197641-A1 COMPOSITIONS AND METHODS FOR TARGETED SYSTEMIC DELIVERY TO CELLS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-06-20 US disclosed
US-20240189239-A1 PROCESS FOR CONTINUOUS HOT MELT GRANULATION OF LOW SOLUBLE PHARMACEUTICALS MERCK PATENT GMBH (DE) 2024-06-13 US disclosed
EP-3322814-B1 METHOD FOR DETERMINING THE DEGREE OF SENSITIVITY OF A STRAIN OF FUNGUS TO AN ANTIFUNGAL AGENT UNIV GRENOBLE ALPES (FR) 2024-06-12 EP disclosed
EP-4380553-A1 STABILISED COMPOSITIONS Rumin8 Pty Ltd (AU) 2024-06-12 EP disclosed
WO-2024109794-A1 NOVEL LIPIDS USED FOR NUCLEIC ACID DELIVERY AND LIPID NANOPARTICLE COMPOSITION 传信生物医药(苏州)有限公司 2024-05-30 WO disclosed
EP-3954370-B1 ANTI-FUNGAL AGENT SEREN PHARMACEUTICALS INC (JP) 2024-05-29 EP disclosed
US-11994510-B2 Diagnosis and treatment of Fusariosis and Scedosporiosis THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2024-05-28 US disclosed
CN-118103059-A Self-assembled nanoparticles based on amphiphilic peptides 巴林萨斯生物疗法北美公司 2024-05-28 CN disclosed
US-20240156920-A1 COMPOSITIONS COMPRISING HYALURONIDASE AND/OR COLLAGENASE AND/OR 4-METHYLUMBELLIFERONE (4-MU) AND METHODS OF TREATMENT USING SAME STANDARD OF CARE CORPORATION 2024-05-16 US disclosed
US-20240148666-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-05-09 US disclosed
WO-2024092030-A1 SELF-ASSEMBLING NANOPARTICLES VACCITECH NORTH AMERICA, INC. (US) 2024-05-02 WO disclosed
WO-2024092028-A2 COMBINATION TREATMENT REGIMES FOR TREATING CANCER VACCITECH NORTH AMERICA, INC. (US) 2024-05-02 WO disclosed
US-11969435-B2 Concomitant administration of glucocorticoid receptor modulators and CYP3A inhibitors CORCEPT THERAPEUTICS, INC. (US) 2024-04-30 US disclosed
CN-115381797-B Preparation and application of itraconazole sustained-release microspheres 江南大学 2024-04-30 CN disclosed
CN-117843659-A Rapamycin analogues and uses thereof 詹森药业有限公司 2024-04-09 CN disclosed
CN-117835967-A Compositions and methods for targeted delivery to cells 瑞科德治疗公司 2024-04-05 CN disclosed
US-20240108639-A1 COMPOSITIONS AND METHODS OF MAKING COCRYSTALS USING DIELECTRIC HEATING WITH DISPERSIVE AND DISTRIBUTIVE MIXING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-04-04 US disclosed
US-20240110192-A1 BACTERIA ENGINEERED TO TREAT DISEASES THAT BENEFIT FROM REDUCED GUT INFLAMMATION AND/OR TIGHTENED GUT MUCOSAL BARRIER SYNLOGIC OPERATING COMPANY, INC. (US) 2024-04-04 US disclosed
US-20240108684-A1 DOSING REGIMENS FOR TREATMENT OF FUNGAL INFECTIONS NAPP PHARMACEUTICAL GROUP LIMITED (GB) 2024-04-04 US disclosed
CN-117750948-A Compositions and methods for targeted systemic delivery to cells 瑞科德治疗公司 2024-03-22 CN disclosed
WO-2024048537-A1 ORGANIC ELECTROLUMINESCENT ELEMENT 日鉄ケミカル&マテリアル株式会社 2024-03-07 WO disclosed
US-20240076689-A1 VIRAL VECTORS AND NUCLEIC ACIDS FOR REGULATED GENE THERAPY BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-03-07 US disclosed
CN-117643590-A Combined medicine composition for treating candida infection and application thereof 宁夏大学 2024-03-05 CN disclosed
US-20240058350-A1 Methods of Treatment ARENA PHARMACEUTICALS, INC. (US) 2024-02-22 US disclosed
EP-3813799-B1 PHARMACEUTICAL FORMULATION WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY CONSEJO SUPERIOR INVESTIGACION (ES) 2024-02-21 EP disclosed
CN-117561081-A Application of CYP450 inhibitor in inhibiting or killing mites and treating xerophthalmia 广州珍实视界生物医药科技有限公司 2024-02-13 CN disclosed
US-11896627-B2 Bacteria engineered to treat metabolic diseases SYNLOGIC OPERATING COMPANY, INC. (US) 2024-02-13 US disclosed
EP-4312990-A1 PROCESS FOR CONTINUOUS HOT MELT GRANULATION OF LOW SOLUBLE PHARMACEUTICALS Merck Patent GmbH (DE) 2024-02-07 EP disclosed
EP-4313004-A1 COMPOSITIONS AND METHODS FOR TARGETED SYSTEMIC DELIVERY TO CELLS Recode Therapeutics, Inc. (US) 2024-02-07 EP disclosed
EP-4313001-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-02-07 EP disclosed
EP-4312987-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS Recode Therapeutics, Inc. (US) 2024-02-07 EP disclosed
WO-2024026412-A1 THIN FILM FREEZING METHODS AND COMPOSITIONS FORMULATED FROM DISPERSED ACTIVE AGENTS TFF PHARMACEUTICALS, INC. (US) 2024-02-01 WO disclosed
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WO-2024017998-A1 M-CSF FOR USE IN THE PROPHYLAXIS AND/OR TREATMENT OF VIRAL INFECTIONS IN STATES OF IMMUNOSUPPRESSION Technische Universität Dresden (DE) 2024-01-25 WO disclosed
WO-2024020592-A1 COSMETIC OR PERSONAL CARE COMPOSITION COMPRISING RECOMBINANT MILK PROTEIN Perfect Day, Inc. (US) 2024-01-25 WO disclosed
EP-4309666-A1 M-CSF FOR USE IN THE PROPHYLAXIS AND/OR TREATMENT OF VIRAL INFECTIONS IN STATES OF IMMUNOSUPPRESSION Technische Universität Dresden (DE) 2024-01-24 EP disclosed
CN-114668849-B Shh pathway for modulating biological rhythms and related applications thereof 中国人民解放军军事科学院军事医学研究院 2024-01-23 CN disclosed
WO-2024012270-A1 COMPOSITION FOR ORGAN-SPECIFIC DELIVERY OF NUCLEIC ACID 传信生物医药(苏州)有限公司 2024-01-18 WO disclosed
EP-4304562-A1 METHODS TO PREPARE DRY POWDERS USING SUSPENSION BASED THIN FILM FREEZING Board of Regents, The University of Texas System (US) 2024-01-17 EP disclosed
US-11858917-B2 Bifunctional molecules with antibody-recruiting and entry inhibitory activity against the human immunodeficiency virus YALE UNIVERSITY (US) 2024-01-02 US disclosed
CN-114126609-B Novel therapeutic agent for prototheca 株式会社赛轮制药 2024-01-02 CN disclosed
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WO-2023247952-A1 CRYSTALLINE PHARMACEUTICAL COMPOSITION FOR INHALATION COMPRISING SUGAR AND LIPID COMPOSITE PARTICLES AND PROCESS FOR MANUFACTURE HOVIONE SCIENTIA LIMITED (IE) 2023-12-28 WO disclosed
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EP-4294431-A1 SELF-ASSEMBLING NANOPARTICLES BASED ON AMPHIPHILIC PEPTIDES Vaccitech North America, Inc. (US) 2023-12-27 EP disclosed
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CN-117241786-A Method for preparing dry powder by using film freezing based on suspension 德克萨斯大学系统董事会 2023-12-15 CN disclosed
US-20230398222-A1 METHOD FOR PRODUCING AN AMORPHOUSE SOLID DISPERSION AND PHARMACEUTICAL COMPOSITION FOR STABILIZING ACTIVE PHARMACEUTICAL INGREDIENTS MERCK PATENT GMBH (DE) 2023-12-14 US disclosed
US-20230390204-A1 PHARMACEUTICAL COMPOSITION AND METHOD FOR ENHANCING SOLUBILITY OF POORLY SOLUBLE ACTIVE PHARMACEUTICAL INGREDIENTS MERCK PATENT GMBH (DE) 2023-12-07 US disclosed
US-11826373-B2 Methods for treatment of diseases GALERA LABS, LLC (US) 2023-11-28 US disclosed
CN-117120036-A Continuous hot melt granulation process for low-solubility pharmaceutical 默克专利股份公司 2023-11-24 CN disclosed
EP-4279071-A2 NOVEL CANNABINOID FORMULATIONS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD (IL) 2023-11-22 EP disclosed
CN-117070374-A Construction method of aspergillus fumigatus in-vitro bone invasion model 荆州市中心医院(长江大学附属荆州医院) 2023-11-17 CN disclosed
EP-4271375-A1 METHODS OF TREATMENT Arena Pharmaceuticals, Inc. (US) 2023-11-08 EP disclosed
EP-4268896-A2 DOSING REGIMENS FOR TREATMENT OF FUNGAL INFECTIONS Cidara Therapeutics, Inc. (US) 2023-11-01 EP disclosed
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CN-116925052-A Synthesis method of optically pure itraconazole 上海现代哈森(商丘)药业有限公司 2023-10-24 CN disclosed
CN-116925052-A Synthesis method of optically pure itraconazole 上海现代哈森(商丘)药业有限公司 2023-10-24 CN disclosed
EP-4259143-A1 COMPOSITIONS AND METHODS OF MAKING COCRYSTALS USING DIELECTRIC HEATING WITH DISPERSIVE AND DISTRIBUTIVE MIXING Board of Regents, The University of Texas System (US) 2023-10-18 EP disclosed
EP-4259829-A1 DIAGNOSTIC METHOD FOR CANCER EVOLUTION PREDICTION, AND USES THEREOF Institut National de la Santé et de la Recherche Médicale (FR) 2023-10-18 EP disclosed
CN-116870166-A Shh pathway for modulating biological rhythms and related applications thereof 中国人民解放军军事科学院军事医学研究院 2023-10-13 CN disclosed
EP-3368014-B1 NOVEL CANNABINOID FORMULATIONS YISSUM RES DEV CO OF HEBREW UNIV JERUSALEM LTD (IL) 2023-10-04 EP disclosed
US-20230302138-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2023-09-28 US disclosed
US-11766408-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-09-26 US disclosed
US-20230293429-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. 2023-09-21 US disclosed
US-20230295220-A1 C-3 AND C-17 MODIFIED TRITERPENOIDS AS HIV-1 INHIBITORS VIIV HEALTHCARE UK NO 5 LTD (GB) 2023-09-21 US disclosed
US-20230295277-A1 UNIVERSAL CAR-NK CELL TARGETING VARIOUS EPITOPES OF HIV-1 GP160 UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2023-09-21 US disclosed
CN-110662756-B Dimer-avoiding multiplex polymerase chain reaction for multi-target amplification 艾瑞普特公司 2023-09-15 CN disclosed
EP-4236919-A1 PHARMACEUTICAL COMPOSITION AND METHOD FOR ENHANCING SOLUBILITY OF POORLY SOLUBLE ACTIVE PHARMACEUTICAL INGREDIENTS Merck Patent GmbH (DE) 2023-09-06 EP disclosed
EP-4236920-A1 METHOD FOR PRODUCING AN AMORPHOUS SOLID DISPERSION AND PHARMACEUTICAL COMPOSITION FOR STABILIZING ACTIVE PHARMACEUTICAL INGREDIENTS Merck Patent GmbH (DE) 2023-09-06 EP disclosed
US-11737981-B2 Cellulosic polymer nanoparticles and methods of forming them THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2023-08-29 US disclosed
EP-4230619-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2023-08-23 EP disclosed
EP-4230619-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2023-08-23 EP disclosed
CN-116617150-A Antifungal microneedle patch and preparation method and application thereof 中山大学·深圳 2023-08-22 CN disclosed
US-11712459-B2 Dosing regimens for treatment of fungal infections CIDARA THERAPEUTICS, INC. (US) 2023-08-01 US disclosed
EP-3831839-B1 C-3 AND C-17 MODIFIED TRITERPENOIDS AS HIV-1 INHIBITORS VIIV HEALTHCARE UK NO 5 LTD (GB) 2023-07-26 EP disclosed
CN-113637603-B Lactobacillus entericus and application thereof 南京大学 2023-07-25 CN disclosed
CN-115463218-B Shh pathway for modulating biological rhythms and related applications thereof 中国人民解放军军事科学院军事医学研究院 2023-07-14 CN disclosed
US-20230219936-A1 PROCESS FOR THE PREPARATION SALTS OF TRIAZOLE COMPOUNDS CELLIX BIO PRIVATE LIMITED (IN) 2023-07-13 US disclosed
US-20230219936-A1 PROCESS FOR THE PREPARATION SALTS OF TRIAZOLE COMPOUNDS CELLIX BIO PRIVATE LIMITED (IN) 2023-07-13 US disclosed
US-20230218533-A1 3D LASER SINTERING PROCESSES FOR IMPROVED DRUG DELIVERY BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-07-13 US disclosed
US-11696910-B2 Buffer-free, stable ophthalmological compositions of ketorolac and phenylephrine and applications thereof SOMERSET THERAPEUTICS, LLC (US) 2023-07-11 US disclosed
CN-116406257-A Pharmaceutical compositions and methods for increasing the solubility of poorly soluble active pharmaceutical ingredients 默克专利股份有限公司 2023-07-07 CN disclosed
WO-2023129915-A2 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-07-06 WO disclosed
CN-116390717-A Method for preparing amorphous solid dispersions and pharmaceutical compositions for stabilizing active pharmaceutical ingredients 默克专利股份有限公司 2023-07-04 CN disclosed
CN-116376937-A Aspergillus fumigatus monocarboxylic acid transporter MFSmt gene and application thereof 荆州市中心医院(长江大学附属荆州医院) 2023-07-04 CN disclosed
US-11692212-B2 Diagnosis and treatment of invasive aspergillosis THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2023-07-04 US disclosed
WO-2023117590-A1 SOLUTION ELECTROSPUN FIBERS, COMPOSITIONS COMPRISING THE SAME AND A PROCESS OF MANUFACTURING THEREOF UNIVERSITEIT GENT (BE) 2023-06-29 WO disclosed
EP-4202036-A1 METHODS AND COMPOSITIONS FOR STEM CELL TRANSPLANTATION Angiocrine Bioscience, Inc. (US) 2023-06-28 EP disclosed
US-11685925-B2 Bacteria engineered to treat diseases that benefit from reduced gut inflammation and/or tightened gut mucosal barrier SYNLOGIC OPERATING COMPANY, INC. (US) 2023-06-27 US disclosed
CN-116323949-A Compositions and methods for treating ocular disorders 方拓生物科技公司 2023-06-23 CN disclosed
EP-3430400-B1 DOSING REGIMENS FOR TREATMENT OF FUNGAL INFECTIONS CIDARA THERAPEUTICS INC (US) 2023-06-21 EP disclosed
EP-4196110-A1 PHARMACEUTICAL COMPOSITION CONTAINING COCRYSTALS FOR ADDITIVE MANUFACTURING Board of Regents, The University of Texas System (US) 2023-06-21 EP disclosed
US-20230181689-A1 SINGLE DOSE METHODS FOR PREVENTING AND TREATING FUNGAL INFECTIONS CIDARA THERAPEUTICS, INC. 2023-06-15 US disclosed
US-20230172949-A1 THERMO-KINETIC MIXING FOR PHARMACEUTICAL APPLICATIONS BOARD OF REGENTS, THE UNIVERISTY OF TEXAS SYSTEM (US) 2023-06-08 US disclosed
US-20230167181-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF MANUFACTURE USING THERMALLY CONDUCTIVE EXCIPIENTS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-06-01 US disclosed
CN-116162175-A Influenza virus vaccine and application thereof 西奈山伊坎医学院 2023-05-26 CN disclosed
US-20230158259-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS TOPELIA AUST LIMITED (652 771 670) (AU) 2023-05-25 US disclosed
WO-2023086832-A1 METHODS OF PREPARING DOSAGE FORMS USING 3D PRINTING CONTAINING AMORPHOUS SOLID DISPERSIONS BOARD OF REGENTS, THE UNIVERSITY OFTEXAS SYSTEM (US) 2023-05-19 WO disclosed
EP-4178626-A2 UNIVERSAL CAR-NK CELL TARGETING VARIOUS EPITOPES OF HIV-1 GP160 University of Southern California (US) 2023-05-17 EP disclosed
US-11649477-B2 Assays and reagents for antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2023-05-16 US disclosed
US-11648210-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-05-16 US disclosed
US-11649215-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2023-05-16 US disclosed
US-11649215-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2023-05-16 US disclosed
US-11649215-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2023-05-16 US disclosed
US-11648209-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-05-16 US disclosed
CN-116077499-A Anti-azole aspergillus fumigatus pharmaceutical composition and application thereof 徐州医科大学 2023-05-09 CN disclosed
CN-116064571-A Mango salt-tolerant gene and identification method and application thereof 中国热带农业科学院三亚研究院 2023-05-05 CN disclosed
US-20230138752-A1 PLASTICIZERS TO IMPROVE RELEASE PERFORMANCE OF AMORPHOUS SOLID DISPERSIONS PURDUE RESEARCH FOUNDATION (US) 2023-05-04 US disclosed
US-20230137582-A1 QUINOLONE DISPERSIONS SOMERSET THERAPEUTICS, LLC 2023-05-04 US disclosed
US-11638758-B2 Itraconazole compositions and dosage forms, and methods of using the same MAYNE PHARMA INTERNATIONAL PTY. LTD (AU) 2023-05-02 US disclosed
WO-2023066825-A1 FUSED BICYCLIC HETEROARYL COMPOUNDS USEFUL AS NLRP3 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2023-04-27 WO disclosed
EP-4164618-A1 3D LASER SINTERING PROCESSES FOR IMPROVED DRUG DELIVERY Board of Regents, The University of Texas System (US) 2023-04-19 EP disclosed
EP-4161627-A1 METHODS FOR DELIVERING BIOACTIVE COMPOSITIONS AND FORMULATIONS TO THE SKIN USING MICROCHANNEL DELIVERY DEVICE Aquavit Pharmaceuticals, Inc. (US) 2023-04-12 EP disclosed
CN-115955965-A Products of manufacture and methods for treating, ameliorating or preventing microbial infections 拓比利亚欧斯特有限公司 2023-04-11 CN disclosed
CN-115944654-A Methods and products for treating gastrointestinal disorders 芬奇治疗控股有限责任公司 2023-04-11 CN disclosed
US-20230095683-A1 COPROCOCCUS BACTERIA FOR USE IN THE TREATMENT OF METABOLIC SYNDROME AND INFLAMMATORY BOWEL DISEASES SORBONNE UNIVERSITE (FR) 2023-03-30 US disclosed
EP-4153745-A1 VIRAL VECTORS AND NUCLEIC ACIDS FOR REGULATED GENE THERAPY Boehringer Ingelheim International GmbH (DE) 2023-03-29 EP disclosed
EP-4153145-A1 GRANULES FOR 3D PRINTING TECHNOLOGY Board of Regents, The University of Texas System (US) 2023-03-29 EP disclosed
CN-115843565-A Method for improving plant performance 以色列农业和农村发展部农业研究组织(范卡尼中心) 2023-03-28 CN disclosed
WO-2023044316-A1 DIAGNOSIS AND TREATMENT OF HISTOPLASMOSIS THE BRIGHAM AND WOMEN’S HOSPITAL, INC. (US) 2023-03-23 WO disclosed
US-11596657-B2 Use of AhR agonist for the preventive or curative treatment of metabolic syndrome and the associated disorders INSTITUT NATIONAL DE LA RECHERCHE AGRONOMIQUE (FR) 2023-03-07 US disclosed
EP-4138832-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS Topelia Aust Limited (AU) 2023-03-01 EP disclosed
US-11590085-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-02-28 US disclosed
US-20230052945-A1 Thermally Gelling Drug Formulations UNM RAINFOREST INNOVATIONS (US) 2023-02-16 US disclosed
US-20230039551-A1 BUFFER- AND CHELATOR-FREE, STABLE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF SOMERSET THERAPEUTICS, LLC 2023-02-09 US disclosed
US-20230040283-A1 ENHANCED DELIVERY OF IMMUNOSUPPRESSIVE DRUG COMPOSITIONS FOR PULMONARY DELIVERY UNIV TEXAS (US) 2023-02-09 US disclosed
US-20230042072-A1 BUFFER-FREE, STABLE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF SOMERSET THERAPEUTICS, LLC 2023-02-09 US disclosed
WO-2023010170-A1 STABILISED COMPOSITIONS Rumin8 Pty Ltd (AU) 2023-02-09 WO disclosed
US-20230040977-A1 CHELATED, STABLE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF SOMERSET THERAPEUTICS, LLC 2023-02-09 US disclosed
US-20230040719-A1 Pharmaceutical Formulation with Improved Solubility and Bioavailability BIONANOPHARMA S.L. (ES) 2023-02-09 US disclosed
US-20230044398-A1 TREATMENT OF OPHTHALMOLOGICAL CONDITIONS USING BUFFER-FREE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE SOMERSET THERAPEUTICS, LLC 2023-02-09 US disclosed
US-20230043588-A1 BACTERIA ENGINEERED TO TREAT DISEASES THAT BENEFIT FROM REDUCED GUT INFLAMMATION AND/OR TIGHTENED GUT MUCOSAL BARRIER SYNLOGIC OPERATING COMPANY, INC. 2023-02-09 US disclosed
US-11571464-B2 C-type natriuretic peptide agent for the treatment of alopecia IGISU CO., LTD. (JP) 2023-02-07 US disclosed
CN-115684447-A Method and apparatus for quantifying target ion species 布鲁克·道尔顿有限及两合公司 2023-02-03 CN disclosed
WO-2023007514-A1 IMPROVED ORAL BIOAVAILABLE PHARMACEUTICAL COMPOSITIONS DR. REDDY'S LABORATORIES LIMITED (IN) 2023-02-02 WO disclosed
US-20230026843-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-01-26 US disclosed
US-20230028227-A1 METHOD AND DEVICE FOR THE QUANTIFICATION OF TARGET ION SPECIES BRUKER DALTONICS GMBH & CO KG (DE) 2023-01-26 US disclosed
US-20230026943-A1 BUFFER-FREE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF SOMERSET THERAPEUTICS, LLC 2023-01-26 US disclosed
EP-4114420-A1 COPROCOCCUS BACTERIA FOR USE IN THE TREATMENT OF METABOLIC SYNDROME AND INFLAMMATORY BOWEL DISEASES Institut national de recherche pour l'agriculture, l'alimentation et l'environnement (FR) 2023-01-11 EP disclosed
US-20230001396-A1 COMPOSITIONS AND METHODS FOR CONTROLLED DELIVERY AND PROTECTION OF THERAPEUTIC AGENTS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-01-05 US disclosed
US-20220401579-A1 INCLUSION COMPLEXES OF PHARMACEUTICALS AND CYCLIC OLIGOMERS DISPERSOL TECHNOLOGIES, LLC (US) 2022-12-22 US disclosed
US-20220401579-A1 INCLUSION COMPLEXES OF PHARMACEUTICALS AND CYCLIC OLIGOMERS DISPERSOL TECHNOLOGIES, LLC (US) 2022-12-22 US disclosed
EP-3325612-B1 METHODS AND COMPOSITIONS FOR STEM CELL TRANSPLANTATION ANGIOCRINE BIOSCIENCE INC (US) 2022-12-14 EP disclosed
CN-115463218-A Shh channel regulation and control of biological rhythm and related application thereof 中国人民解放军军事科学院军事医学研究院 2022-12-13 CN disclosed
US-11523987-B2 Trimcinolone and moxifloxacin methods SOMERSET THERAPEUTICS, LLC (US) 2022-12-13 US disclosed
US-20220387337-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-12-08 US disclosed
US-20220378752-A1 NOVEL THERAPEUTIC AGENT FOR PROTOTHECA DISEASE SEREN PHARMACEUTICALS INC. (JP) 2022-12-01 US disclosed
US-20220378704-A1 PROCESS FOR THE PREPARATION OF A NANOPARTICULATE ACTIVE INGREDIENT BAYER AG (DE) 2022-12-01 US disclosed
US-11510930-B2 Gatifloxacin, prednisolone, and bromfenac compositions and methods SOMERSET THERAPEUTICS, LLC (US) 2022-11-29 US disclosed
US-11510880-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-11-29 US disclosed
CN-115381776-A External spray containing itraconazole and eucalyptol and preparation method thereof 南京朗博特动物药业有限公司 2022-11-25 CN disclosed
CN-115381797-A Preparation and application of itraconazole sustained-release microspheres 江南大学 2022-11-25 CN disclosed
US-20220354778-A1 COMPOSITIONS AND METHODS OF MAKING BRITTLE-MATRIX PARTICLES THROUGH BLISTER PACK FREEZING UNIV TEXAS (US) 2022-11-10 US disclosed
CN-114996977-B Water pollution restoration simulation method and system based on hydrodynamic coupling water quality model 浙江远算科技有限公司 2022-11-04 CN disclosed
US-11484538-B2 Bromfenac, prednisolone, and moxifloxacin compositions and methods SOMERSET THERAPEUTICS, LLC (US) 2022-11-01 US disclosed
US-11485730-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-11-01 US disclosed
US-11484501-B2 Mechanochemical activated dry amorphisation by milling equilibrium between ap mesoporous silica GRACE GMBH (US) 2022-11-01 US disclosed
US-20220340551-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2022-10-27 US disclosed
US-11478424-B2 Mechanochemcial activated dry amorphisation by milling equilibrium between AP mesoporous silica GRACE GMBH (US) 2022-10-25 US disclosed
CN-115219611-A Kit for determining 7 antifungal drugs in serum by ultra-high performance liquid chromatography-tandem mass spectrometry and application thereof 上海义准生物有限公司 2022-10-21 CN disclosed
CN-115219611-A Kit for determining 7 antifungal drugs in serum by ultra-high performance liquid chromatography-tandem mass spectrometry and application thereof 上海义准生物有限公司 2022-10-21 CN disclosed
US-20220331268-A1 TREATMENT OF SKIN DISORDERS WITH TOPICAL COMBINATION COMPOSITIONS COMPRISING TAPINAROF AND AN ADDITIONAL AHR ACTIVATOR SOL-GEL TECHNOLOGIES LTD. (IL) 2022-10-20 US disclosed
WO-2022221177-A1 DIAGNOSIS AND TREATMENT OF CONGESTIVE COLON FAILURE (CCF) KHURANA VIKAS (US) 2022-10-20 WO disclosed
US-11471403-B2 Limited particle size triamcinolone and moxifloxacin compositions and associated methods of use SOMERSET THERAPEUTICS, LLC. (US) 2022-10-18 US disclosed
US-20220324849-A1 TRUNCATED ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF UNIVERSITY OF CONNECTICUT 2022-10-13 US disclosed
US-11465973-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2022-10-11 US disclosed
US-11465973-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2022-10-11 US disclosed
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US-20220313611-A1 METHODS TO PREPARE DRY POWDERS USING SUSPENSION BASED THIN FILM FREEZING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-10-06 US disclosed
WO-2022207775-A1 PROCESS FOR CONTINUOUS HOT MELT GRANULATION OF LOW SOLUBLE PHARMACEUTICALS MERCK PATENT GMBH (DE) 2022-10-06 WO disclosed
WO-2022204286-A1 COMPOSITIONS AND METHODS FOR TARGETED SYSTEMIC DELIVERY TO CELLS RECODE THERAPEUTICS, INC. (US) 2022-09-29 WO disclosed
WO-2022204043-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-09-29 WO disclosed
WO-2022204219-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS RECODE THERAPEUTICS, INC. (US) 2022-09-29 WO disclosed
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EP-4062941-A1 PROTEIN BASED EXCIPIENT FOR ACTIVE PHARMACEUTICAL INGREDIENTS Rousselot B.V. (NL) 2022-09-28 EP disclosed
CN-111588691-B Itraconazole in-situ liquid crystal gel preparation for treating vaginitis and preparation method thereof 安徽中医药大学 2022-09-23 CN disclosed
EP-4058190-A1 COMPOSITIONS AND METHODS FOR CONTROLLED DELIVERY AND PROTECTION OF THERAPEUTIC AGENTS Board of Regents, The University of Texas System (US) 2022-09-21 EP disclosed
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WO-2022192729-A1 METHODS TO PREPARE DRY POWDERS USING SUSPENSION BASED THIN FILM FREEZING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-09-15 WO disclosed
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US-11439650-B2 Thermo-kinetic mixing for pharmaceutical applications BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-09-13 US disclosed
CN-114996977-A Water pollution restoration simulation method and system based on hydrodynamic coupling water quality model 浙江远算科技有限公司 2022-09-02 CN disclosed
CN-113384570-B Application of caffeic acid methyl ester and triazole composition in preparation of antifungal products 山东省妇幼保健院 2022-08-26 CN disclosed
US-20220265833-A1 ASPARTIC PROTEASE-TRIGGERED ANTIFUNGAL HYDROGELS BROWN UNIVERSITY 2022-08-25 US disclosed
WO-2022177993-A1 SELF-ASSEMBLING NANOPARTICLES BASED ON AMPHIPHILIC PEPTIDES VACCITECH NORTH AMERICA, INC. (US) 2022-08-25 WO disclosed
US-20220257673-A1 METHODS AND PRODUCTS FOR TREATMENT OF GASTROINTESTINAL DISORDERS FINCH THERAPEUTICS HOLDINGS LLC 2022-08-18 US disclosed
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EP-4041203-A1 PROCESS FOR THE PREPARATION OF A NANOPARTICULATE ACTIVE INGREDIENT Bayer Aktiengesellschaft (DE) 2022-08-17 EP disclosed
US-20220233460-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-07-28 US disclosed
US-20220226395-A1 BACTERIA ENGINEERED TO TREAT METABOLIC DISEASES SYNLOGIC OPERATING COMPANY, INC. 2022-07-21 US disclosed
US-11390613-B2 Azole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2022-07-19 US disclosed
US-20220220079-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORAL INFECTIOUS DISEASES CELLIX BIO PRIVATE LIMITED (IN) 2022-07-14 US disclosed
US-20220220079-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORAL INFECTIOUS DISEASES CELLIX BIO PRIVATE LIMITED (IN) 2022-07-14 US disclosed
EP-3454944-B1 VOLATILE METABOLITE PROFILES FOR THE DIAGNOSIS AND TREATMENT OF MUCORALES FUNGI BRIGHAM & WOMENS HOSPITAL INC (US) 2022-07-13 EP disclosed
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US-11382899-B2 Enhanced delivery of immunosuppressive drug compositions for pulmonary delivery BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-07-12 US disclosed
US-20220213073-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2022-07-07 US disclosed
US-20220213073-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2022-07-07 US disclosed
US-20220213043-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORAL INFECTIOUS DISEASES CELLIX BIO PRIVATE LIMITED (IN) 2022-07-07 US disclosed
WO-2022147318-A1 METHODS OF TREATMENT ARENA PHARMACEUTICALS, INC. (US) 2022-07-07 WO disclosed
EP-4021416-A1 DRUG-POLYMER AMORPHOUS SOLID DISPERSIONS USING LINEAR POLY (ACRYLIC ACID) POLYMERS Lubrizol Advanced Materials, Inc. (US) 2022-07-06 EP disclosed
EP-4017524-A1 COMPOSITIONS COMPRISING HYALURONIDASE AND/OR COLLAGENASE AND/OR 4-METHYLUMBELLIFERONE (4-MU) AND METHODS OF TREATMENT USING SAME Standard of Care Corporation (US) 2022-06-29 EP disclosed
CN-114668849-A Shh channel regulation and control of biological rhythm and related application thereof 中国人民解放军军事科学院军事医学研究院 2022-06-28 CN disclosed
US-11369624-B2 Salts of prodrugs of piperazine and substituted piperidine antiviral agents VIIV HEALTHCARE UK (NO. 4) LIMITED 2022-06-28 US disclosed
CN-114660200-A Method for simultaneously measuring 4 triazole antifungal drugs in blood plasma by high performance liquid chromatography tandem mass spectrometry technology 中国人民解放军总医院 2022-06-24 CN disclosed
WO-2022128918-A1 DIAGNOSTIC METHOD FOR CANCER EVOLUTION PREDICTION, AND USES THEREOF INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2022-06-23 WO disclosed
WO-2022129661-A1 AMPHOTERICIN B FORMULATIONS FOR INHALATION BASED ON COLLAPSED MICROPARTICLES CONTAINING CARBOHYDRATES AND AMINO ACIDS UNIVERSIDAD COMPLUTENSE DE MADRID (ES) 2022-06-23 WO disclosed
US-11364197-B2 Compositions and methods of making brittle-matrix particles through blister pack freezing BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-06-21 US disclosed
WO-2022125869-A1 COMPOSITIONS AND METHODS OF MAKING COCRYSTALS USING DIELECTRIC HEATING WITH DISPERSIVE AND DISTRIBUTIVE MIXING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-06-16 WO disclosed
US-20220183967-A1 LIMITED PARTICLE SIZE TRIAMCINOLONE AND MOXIFLOXACIN COMPOSITIONS AND ASSOCIATED METHODS OF USE SOMERSET THERAPEUTICS, LLC 2022-06-16 US disclosed
US-20220183968-A1 SUSPENSION COMPONENT-SPECIFIC TRIAMCINOLONE AND MOXIFLOXACIN COMPOSITIONS AND ASSOCIATED METHODS OF USE SOMERSET THERAPEUTICS, LLC 2022-06-16 US disclosed
US-20220183966-A1 MOXIFLOXACIN AND TRIAMCINOLONE COMPOSITIONS AND ASSOCIATED METHODS SOMERSET THERAPEUTICS, LLC 2022-06-16 US disclosed
EP-4008314-A2 THERMO-KINETIC MIXING FOR PHARMACEUTICAL APPLICATIONS Board of Regents, The University of Texas System (US) 2022-06-08 EP disclosed
EP-4005600-A1 CYTOTOXIC-DRUG DELIVERING MOLECULES TARGETING HIV (CDM-HS), CYTOTOXIC ACTIVITY AGAINST THE HUMAN IMMUNODEFICIENCY VIRUS AND METHODS OF USE Yale University (US) 2022-06-01 EP disclosed
EP-3448435-B1 PROTEIN BASED EXCIPIENT FOR ACTIVE PHARMACEUTICAL INGREDIENTS ROUSSELOT B V (NL) 2022-06-01 EP disclosed
US-11339418-B2 Antimicrobial susceptibility testing and microbial identification SeLux Diagnostics, Inc. (US) 2022-05-24 US disclosed
EP-3998109-A1 NOVEL THERAPEUTIC AGENT FOR PROTOTHECA DISEASE Seren Pharmaceuticals Inc. (JP) 2022-05-18 EP disclosed
CN-114502182-A Methods and products for treating gastrointestinal disorders 芬奇治疗控股有限责任公司 2022-05-13 CN disclosed
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US-20220143143-A1 USE OF ACTIVATORS OF THE ARYL HYDROCARBON RECEPTOR FOR TREATING GLUTEN-INDUCED GASTROINTESTINAL DISEASES UNIV MCMASTER (CA) 2022-05-12 US disclosed
US-20220133638-A1 METHOD FOR PRODUCING NANOPARTICLES LEON-NANODRUGS GMBH (DE) 2022-05-05 US disclosed
WO-2022094174-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ESOPHAGEAL CONDITIONS CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-05-05 WO disclosed
WO-2022090296-A1 PHARMACEUTICAL COMPOSITION AND METHOD FOR ENHANCING SOLUBILITY OF POORLY SOLUBLE ACTIVE PHARMACEUTICAL INGREDIENTS MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
WO-2022090297-A1 METHOD FOR PRODUCING AN AMORPHOUS SOLID DISPERSION AND PHARMACEUTICAL COMPOSITION FOR STABILIZING ACTIVE PHARMACEUTICAL INGREDIENTS MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
WO-2022090295-A1 METHOD FOR PRODUCING AN AMORPHOUS SOLID DISPERSION AND PHARMACEUTICAL COMPOSITION FOR STABILIZING ACTIVE PHARMACEUTICAL INGREDIENTS MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
US-20220133637-A1 COMPOSITIONS AND METHODS FOR ORGAN SPECIFIC DELIVERY OF NUCLEIC ACIDS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-05-05 US disclosed
EP-3990679-A1 APPARATUS FOR FORMING A PLURALITY OF COATED PARTICLES, METHOD FOR FORMING A PLURALITY OF COATED PARTICLES, COATED PARTICLES Nanexa AB (SE) 2022-05-04 EP disclosed
EP-3988107-A1 BACTERIA ENGINEERED TO TREAT DISEASES THAT BENEFIT FROM REDUCED GUT INFLAMMATION AND/OR TIGHTENED GUT MUCOSAL BARRIER Synlogic Operating Company, Inc. (US) 2022-04-27 EP disclosed
US-11312707-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-04-26 US disclosed
US-11312707-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-04-26 US disclosed
US-11304911-B2 Compositions and methods for organ specific delivery of nucleic acids THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-04-19 US disclosed
EP-3980023-A1 LIPID NANOPARTICLES CONTAINING PHARMACEUTICAL AND/OR NUTRACEUTICAL AGENTS AND METHODS THEREOF Board of Regents, The University of Texas System (US) 2022-04-13 EP disclosed
US-11298315-B2 Triamcinolone and moxifloxacin compositions SOMERSET THERAPEUTICS, LLC. (US) 2022-04-12 US disclosed
CN-114302710-A Drug-polymer amorphous solid dispersions using linear poly (acrylic acid) polymers 路博润先进材料公司 2022-04-08 CN disclosed
US-20220105100-A1 SAFE BRINZOLAMIDE AND BRIMONIDINE COMPOSITIONS WITH ENHANCED BENZALKONIUM CHLORIDE CONTENT SOMERSET THERAPEUTICS, LLC 2022-04-07 US disclosed
US-20220105103-A1 SAFE USE OF BRINZOLAMIDE AND BRIMONIDINE COMPOSITIONS WITH ENHANCED BENZALKONIUM CHLORIDE CONTENT SOMERSET THERAPEUTICS, LLC 2022-04-07 US disclosed
US-20220105102-A1 METHODS OF EFFICIENTLY REDUCING INTRAOCULAR PRESSURE SOMERSET THERAPEUTICS, LLC 2022-04-07 US disclosed
US-20220106302-A1 ITRACONAZOLE ANALOGS AND USE THEREOF THE JOHNS HOPKINS UNIVERSITY 2022-04-07 US disclosed
US-20220105101-A1 EFFICIENT BRINZOLAMIDE AND BRIMONIDINE COMPOSITIONS SOMERSET THERAPEUTICS, LLC 2022-04-07 US disclosed
EP-3978499-A1 PHOTOPROTECTIVE COMPOSITIONS CONTAINING MALASSEZIA-DERIVED COMPOUNDS AND/OR CHEMICAL ANALOGS THEREOF VERSICOLOR TECHNOLOGIES, LLC (US) 2022-04-06 EP disclosed
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US-20220089579-A1 BIFUNCTIONAL MOLECULES WITH ANTIBODY-RECRUITING AND ENTRY INHIBITORY ACTIVITY AGAINST THE HUMAN IMMUNODEFICIENCY VIRUS UNIV YALE (US) 2022-03-24 US disclosed
US-20220088030-A1 METHODS FOR TREATMENT OF DISEASES BIOSSIL INC. (CA) 2022-03-24 US disclosed
US-20220088036-A1 CONCOMITANT ADMINISTRATION OF GLUCOCORTICOID RECEPTOR MODULATORS AND CYP3A INHIBITORS CORCEPT THERAPEUTICS, INC. 2022-03-24 US disclosed
US-20220088036-A1 CONCOMITANT ADMINISTRATION OF GLUCOCORTICOID RECEPTOR MODULATORS AND CYP3A INHIBITORS CORCEPT THERAPEUTICS, INC. 2022-03-24 US disclosed
US-11279936-B2 Aptamers, biosensors and detection methods for common azole-class antifungal drugs RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2022-03-22 US disclosed
US-20220072136-A1 PROTEIN BASED EXCIPIENT FOR ACTIVE PHARMACEUTICAL INGREDIENTS DISPERSOME IP APS (NL) 2022-03-10 US disclosed
US-20220062303-A1 PREDNISOLONE AND MOXIFLOXACIN COMPOSITIONS AND METHODS SOMERSET THERAPEUTICS, LLC 2022-03-03 US disclosed
US-20220062271-A1 LOTEPREDNOL AND MOXIFLOXACIN COMPOSITIONS AND METHODS SOMERSET THERAPEUTICS, LLC (US) 2022-03-03 US disclosed
US-20220062301-A1 BROMFENAC, PREDNISOLONE, AND MOXIFLOXACIN COMPOSITIONS AND METHODS SOMERSET THERAPEUTICS, LLC 2022-03-03 US disclosed
US-20220064600-A1 METHODS OF EXPANDING MYELOID CELL POPULATIONS AND USES THEREOF CELLERANT THERAPEUTICS INC (US) 2022-03-03 US disclosed
US-20220062167-A1 TRIAMCINOLONE AND MOXIFLOXACIN COMPOSITIONS SOMERSET THERAPEUTICS, LLC 2022-03-03 US disclosed
US-20220062302-A1 GATIFLOXACIN, PREDNISOLONE, AND BROMFENAC COMPOSITIONS AND METHODS SOMERSET THERAPEUTICS, LLC 2022-03-03 US disclosed
US-20220062168-A1 TRIMCINOLONE AND MOXIFLOXACIN METHODS SOMERSET THERAPEUTICS, LLC 2022-03-03 US disclosed
CN-114126609-A Novel therapeutic agent for prototheca disease 株式会社赛轮制药 2022-03-01 CN disclosed
US-20220054715-A1 Bone Morphogenetic Protein Pathway Activation, Compositions for Ossification, and Methods Related Thereto UNIV EMORY (US) 2022-02-24 US disclosed
EP-3957639-A1 PHOTOPROTECTIVE COMPOSITIONS CONTAINING MALASSEZIA-DERIVED COMPOUNDS AND/OR CHEMICAL ANALOGS THEREOF Einziger, Michael (US) 2022-02-23 EP disclosed
WO-2022036290-A1 PHARMACEUTICAL COMPOSITION CONTAINING COCRYSTALS FOR ADDITIVE MANUFACTURING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-02-17 WO disclosed
EP-3954370-A1 ANTI-FUNGAL AGENT Seren Pharmaceuticals Inc. (JP) 2022-02-16 EP disclosed
US-20220023202-A1 Medicated Hard Candy Product For Treating Esophageal Inflammation And A Method Using The Same MARTIN MICHAEL LEE (US) 2022-01-27 US disclosed
WO-2022016216-A1 BIOCOMPATIBLE POLYMER COMPOSITIONS THE UNIVERSITY OF WESTERN AUSTRALIA (AU) 2022-01-27 WO disclosed
US-11225463-B2 Compositions and methods for the treatment of oral infectious diseases CELLIX BIO PRIVATE LIMITED (IN) 2022-01-18 US disclosed
US-11220493-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-01-11 US disclosed
US-11220493-B2 Compositions and methods for the treatment of fungal infections CELLIX BIO PRIVATE LIMITED (IN) 2022-01-11 US disclosed
US-11185548-B2 Inhibitors of cytochrome P450 family 7 subfamily B member 1 (CYP7B1) for use in treating diseases HELMHOLTZ ZENTRUM MUNCHEN—DEUTSCHES FORSCHUNGSZENTRUM FÜR GESUNDHEIT UND UMWELT (GMBH) (DE) 2021-11-30 US disclosed
US-11179501-B2 Bone morphogenetic protein pathway activation, compositions for ossification, and methods related thereto EMORY UNIVERSITY (US) 2021-11-23 US disclosed
US-11028078-B2 Itraconazole analogs and use thereof THE JOHNS HOPKINS UNIVERSITY (US) 2021-06-08 US disclosed
WO-2021108022-A1 INCLUSION COMPLEXES OF PHARMACEUTICALS AND CYCLIC OLIGOMERS DISPERSOL TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
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US-20210053950-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2021-02-25 US disclosed
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US-20200361912-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2020-11-19 US disclosed
US-20200361874-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORAL INFECTIOUS DISEASES CELLIX BIO PRIVATE LIMITED (IN) 2020-11-19 US disclosed
EP-2803357-B1 Angiogenesis inhibitors UNIV JOHNS HOPKINS (US) 2020-11-18 EP disclosed
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EP-3099679-B1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF UNIV CONNECTICUT (US) 2020-05-20 EP disclosed
US-20200072711-A1 FLUORESCENT ENDOPLASMIC RETICULUM TRACKERS FOR LIVE CELL IMAGING OF PATHOGENIC YEAST RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2020-03-05 US disclosed
EP-3581566-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2019-12-18 EP disclosed
EP-3581566-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2019-12-18 EP disclosed
US-10369147-B2 Topical formulations for delivery of hedgehog inhibitor compounds and use thereof PellePharm, Inc. (US) 2019-08-06 US disclosed
US-20190224378-A1 Bone Morphogenetic Protein Pathway Activation, Compositions for Ossification, and Methods Related Thereto UNIV EMORY (US) 2019-07-25 US disclosed
US-10286113-B2 Bone morphogenetic protein pathway activation, compositions for ossification, and methods related thereto EMORY UNIVERSITY (US) 2019-05-14 US disclosed
US-20190134027-A1 TOPICAL FORMULATIONS FOR DELIVERY OF HEDGEHOG INHIBITOR COMPOUNDS AND USE THEREOF PellePharm, Inc. 2019-05-09 US disclosed
US-20190040046-A1 ITRACONAZOLE ANALOGS AND USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-02-07 US disclosed
WO-2018115319-A2 INHIBITORS OF CYTOCHROME P450 FAMILY 7 SUBFAMILY B MEMBER 1 (CYP7B1) FOR USE IN TREATING DISEASES Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (DE) 2018-06-28 WO disclosed
WO-2018096497-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF FUNGAL INFECTIONS CELLIX BIO PRIVATE LIMITED (IN) 2018-05-31 WO disclosed
WO-2018096405-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ORAL INFECTIOUS DISEASES CELLIX BIO PRIVATE LIMITED (IN) 2018-05-31 WO disclosed
US-9981956-B2 Small molecule inhibitors of fibrosis THE SCRIPPS RESEARCH INSTITUTE (US) 2018-05-29 US disclosed
US-9981956-B2 Small molecule inhibitors of fibrosis THE SCRIPPS RESEARCH INSTITUTE (US) 2018-05-29 US disclosed
US-9839636-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-12-12 US disclosed
US-9839636-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-12-12 US disclosed
US-9839636-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-12-12 US disclosed
US-20170217943-A1 SMALL MOLECULE INHIBITORS OF FIBROSIS THE SCRIPPS RESEARCH INSTITUTE 2017-08-03 US disclosed
US-20170217943-A1 SMALL MOLECULE INHIBITORS OF FIBROSIS THE SCRIPPS RESEARCH INSTITUTE 2017-08-03 US disclosed
US-20170209436-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-07-27 US disclosed
US-20170209436-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-07-27 US disclosed
US-20170209436-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-07-27 US disclosed
US-9650365-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-05-16 US disclosed
US-9650365-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-05-16 US disclosed
US-9650365-B2 Itraconazole analogues and methods of use thereof UNIVERSITY OF CONNECTICUT (US) 2017-05-16 US disclosed
US-9642865-B2 Angiogenesis inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2017-05-09 US disclosed
US-9642806-B2 Antifungal compositions with improved bioavailability JANSSEN PHARMACEUTICA NV (BE) 2017-05-09 US disclosed
US-20160361470-A1 Bone Morphogenetic Protein Pathway Activation, Compositions for Ossification, and Methods Related Thereto UNIV EMORY (US) 2016-12-15 US disclosed
US-20160354368-A1 TOPICAL FORMULATIONS FOR DELIVERY OF HEDGEHOG INHIBITOR COMPOUNDS AND USE THEREOF SOL-GEL TECHNOLOGIES LTD. (IL) 2016-12-08 US disclosed
WO-2016196928-A1 TOPICAL FORMULATIONS FOR DELIVERY OF HEDGEHOG INHIBITOR COMPOUNDS AND USE THEREOF PellePharm, Inc. (US) 2016-12-08 WO disclosed
US-20160354368-A1 TOPICAL FORMULATIONS FOR DELIVERY OF HEDGEHOG INHIBITOR COMPOUNDS AND USE THEREOF SOL-GEL TECHNOLOGIES LTD. (IL) 2016-12-08 US disclosed
US-20160340346-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-11-24 US disclosed
US-20160340346-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-11-24 US disclosed
US-20160340346-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-11-24 US disclosed
US-20160264556-A1 ITRACONAZOLE ANALOGS AND USE THEREOF UNIV JOHNS HOPKINS (US) 2016-09-15 US disclosed
US-20160264556-A1 ITRACONAZOLE ANALOGS AND USE THEREOF UNIV JOHNS HOPKINS (US) 2016-09-15 US disclosed
EP-2181330-B2 COMPOSITIONS AND MEANS FOR DIAGNOSING MICROBIAL INFECTIONS STATENS SERUMINSTITUT (DK) 2016-08-31 EP disclosed
US-20160151503-A1 COMPOSITIONS AND PREPARATION METHODS OF LOW MELTING IONIC SALTS OF POORLY-WATER SOLUBLE DRUGS MW ENCAP LIMITED (GB) 2016-06-02 US disclosed
US-20160151503-A1 COMPOSITIONS AND PREPARATION METHODS OF LOW MELTING IONIC SALTS OF POORLY-WATER SOLUBLE DRUGS MW ENCAP LIMITED (GB) 2016-06-02 US disclosed
US-9346791-B2 Itraconazole analogs and use thereof THE JOHNS HOPKINS UNIVERSITY (US) 2016-05-24 US disclosed
US-9346791-B2 Itraconazole analogs and use thereof THE JOHNS HOPKINS UNIVERSITY (US) 2016-05-24 US disclosed
EP-1912625-B1 ITRACONAZOLE COMPOSITIONS WITH IMPROVED BIOAVAILABILITY ABBVIE DEUTSCHLAND (DE) 2016-04-13 EP disclosed
WO-2015116947-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF UNIVERSITY OF CONNECTICUT (US) 2015-08-06 WO disclosed
US-9095589-B2 Chirally pure isomers of itraconazole for use as angiogenesis inhibitors JOHNS HOPKINS UNIVERSITY (US) 2015-08-04 US disclosed
US-9095589-B2 Chirally pure isomers of itraconazole for use as angiogenesis inhibitors JOHNS HOPKINS UNIVERSITY (US) 2015-08-04 US disclosed
US-8980930-B2 Angiogenesis inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2015-03-17 US disclosed
US-20150056267-A1 ANGIOGENESIS INHIBITORS UNIV JOHNS HOPKINS (US) 2015-02-26 US disclosed
EP-2803357-A2 Angiogenesis inhibitors THE JOHNS-HOPKINS UNIVERSITY (US) 2014-11-19 EP disclosed
US-20140248372-A1 BONE MORPHOGENETIC PROTEIN PATHWAY ACTIVATION, COMPOSITIONS FOR OSSIFICATION, AND METHODS RELATED THERETO EMORY UNIVERSITY (US) 2014-09-04 US disclosed
US-20140221393-A1 Itraconazole Analogs and Use Thereof THE JOHNS HOPKINS UNIVERSITY 2014-08-07 US disclosed
US-20140221393-A1 Itraconazole Analogs and Use Thereof THE JOHNS HOPKINS UNIVERSITY 2014-08-07 US disclosed
US-20140134244-A1 ANTIFUNGAL COMPOSITIONS WITH IMPROVED BIOAVAILABILITY JANSSEN PHARMACEUTICA N.V. (BE) 2014-05-15 US disclosed
US-8653083-B2 Hedgehog pathway antagonists to treat disease THE JOHNS HOPKINS UNIVERSITY (US) 2014-02-18 US disclosed
US-8591948-B2 Antifungal compositions with improved bioavailability JANSSEN PHARMACEUTICA N.V. (BE) 2013-11-26 US disclosed
EP-2181330-B1 COMPOSITIONS AND MEANS FOR DIAGNOSING MICROBIAL INFECTIONS STATENS SERUMINSTITUT (DK) 2013-11-20 EP disclosed
US-8486456-B2 Itraconazole compositions with improved bioavailability ABBOTT GMBH & CO., KG (DE) 2013-07-16 US disclosed
US-20130101657-A1 ANGIOGENESIS INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2013-04-25 US disclosed
US-20130102614-A1 CHIRALLY PURE ISOMERS OF ITRACONAZOLE FOR USE AS ANGIOGENESIS INHIBITORS JOHNS HOPKINS UNIVERSITY 2013-04-25 US disclosed
US-20130102614-A1 CHIRALLY PURE ISOMERS OF ITRACONAZOLE FOR USE AS ANGIOGENESIS INHIBITORS JOHNS HOPKINS UNIVERSITY 2013-04-25 US disclosed
US-8394813-B2 Active agent delivery systems and methods for protecting and administering active agents SHIRE LLC (US) 2013-03-12 US disclosed
EP-1919480-B1 HEDGEHOG PATHWAY ANTAGONISTS TO TREAT DISEASE UNIV JOHNS HOPKINS (US) 2013-01-16 EP disclosed
EP-2517686-A2 A kit comprising a multi-chamber container Combino Pharm, S.L. (ES) 2012-10-31 EP disclosed
EP-2431477-A1 POLYKETIDE COMPOUND Astellas Pharma Inc. (JP) 2012-03-21 EP disclosed
US-20120059038-A1 POLYKETIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2012-03-08 US disclosed
US-20120059038-A1 POLYKETIDE COMPOUND ASTELLAS PHARMA INC. (JP) 2012-03-08 US disclosed
US-20120046259-A1 COMPOSITION COMPRISING AN ANTIBIOTIC AND A CORTICOSTEROID INTERVET INC. 2012-02-23 US disclosed
EP-2404602-A1 Hedgehog pathway antagonists to treat cancer The Johns Hopkins University (US) 2012-01-11 EP disclosed
US-20110262517-A1 CHIRALLY PURE ISOMERS OF ITRACONAZOLE AND INHIBITORS OF LANOSTEROL 14A-DEMETHYLASE FOR USE AS ANGIOGENESIS INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2011-10-27 US disclosed
US-20110262517-A1 CHIRALLY PURE ISOMERS OF ITRACONAZOLE AND INHIBITORS OF LANOSTEROL 14A-DEMETHYLASE FOR USE AS ANGIOGENESIS INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2011-10-27 US disclosed
EP-2316468-A1 Delivery system and methods for protecting and administering dextroamphetamine Shire LLC (US) 2011-05-04 EP disclosed
EP-2266590-A2 Active agent delivery sytems and methods for protecting and administering active agents Shire LLC (US) 2010-12-29 EP disclosed
US-20100143455-A1 Triazole antifungal agents WU NIAN 2010-06-10 US disclosed
US-20100087409-A1 COMPOSITION COMPRISING AN ANTIBIOTIC AND A CORTICOSTEROID INTERVET INTERNATIONAL BV 2010-04-08 US disclosed
US-20100087409-A1 COMPOSITION COMPRISING AN ANTIBIOTIC AND A CORTICOSTEROID INTERVET INTERNATIONAL BV 2010-04-08 US disclosed
US-20090306228-A1 ACTIVE AGENT DELIVERY SYSTEMS AND METHODS FOR PROTECTING AND ADMINISTERING ACTIVE AGENTS SHIRE LLC (US) 2009-12-10 US disclosed
US-20090253792-A1 ACTIVE AGENT DELIVERY SYSTEMS AND METHODS FOR PROTECTING AND ADMINISTERING ACTIVE AGENTS SHIRE LLC (US) 2009-10-08 US disclosed
US-20090214656-A1 ITRACONAZOLE COMPOSITIONS WITH IMPROVED BIOAVAILABILITY ABBOTT GMBH & CO. KG (DE) 2009-08-27 US disclosed
US-20090203713-A1 Hedgehog pathway antagonists to treat disease NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2009-08-13 US disclosed
US-20090088443-A1 NOVEL CRYSTALLINE FORMS OF CONAZOLES AND METHODS OF MAKING AND USING THE SAME REMENAR JULIUS 2009-04-02 US disclosed
EP-1511490-A4 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS TRANSFORM PHARMACEUTICALS INC (US) 2009-03-11 EP disclosed
US-20080305173-A1 AMORPHOUS DRUG BEADS BOGUE BEUFORD ARLIE 2008-12-11 US disclosed
US-7459561-B2 N-substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA AG (CH) 2008-12-02 US disclosed
US-20080287299-A1 Use of Imidazole and/or Triazole Derivatives for Combating Plant Pests; as Well as Method for Controlling Diseases/Insects/Mites/Nematodes and Weeds, Particularly Foliar and/or Soil Diseases FMC QUIMICA DO BRASIL LTDA (BR) 2008-11-20 US disclosed
US-7446107-B2 Crystalline forms of conazoles and methods of making and using the same TRANSFORM PHARMACEUTICALS, INC. (US) 2008-11-04 US disclosed
US-7427600-B2 Active agent delivery systems and methods for protecting and administering active agents SHIRE LLC (US) 2008-09-23 US disclosed
US-20080193499-A1 Angiogenesis Inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2008-08-14 US disclosed
WO-2008088776-A2 AMORPHOUS DRUG BEADS CAPRICORN PHARMA INC. (US) 2008-07-24 WO disclosed
EP-1718640-A4 NOVEL CRYSTALLINE FORMS OF CONAZOLES AND METHODS OF MAKING AND USING THE SAME TRANSFORM PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed
US-20070293674-A1 Novel Saperconazole Crystalline Forms and Related Processes, Pharmaceutical Compositions and Methods TRANSFORM PHARMACEUTICALS, INC. (US) 2007-12-20 US disclosed
US-20070232529-A1 mesalamine covalently attached to carrier peptide at C-terminus, interspersed and/or side chain; releasing into bloodstream; reducing dosage NEW RIVER PHARMACEUTICALS INC. (US) 2007-10-04 US disclosed
US-20070148240-A1 Oral formulation containing itraconazole and methods for manufacturing and using the same YUNG SHIN PHARM. IND. CO., LTD. (TW) 2007-06-28 US disclosed
US-7189858-B2 N-phenyl substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA AG (CH) 2007-03-13 US disclosed
US-20070027322-A1 N-substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA INTERNATIONAL LTD. (CH) 2007-02-01 US disclosed
EP-1742941-A1 NOVEL SAPERCONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS Transform Pharmaceuticals, Inc. (US) 2007-01-17 EP disclosed
US-7163700-B2 Amorphous drug beads CAPRICORN PHARMA, INC. (US) 2007-01-16 US disclosed
US-7151182-B2 Intermediates for N-substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA AG (CH) 2006-12-19 US disclosed
US-20060263436-A1 Antifungal compositions with improved bioavailability BAERT LIEVEN E C 2006-11-23 US disclosed
EP-1718640-A1 NOVEL CRYSTALLINE FORMS OF CONAZOLES AND METHODS OF MAKING AND USING THE SAME Transform Pharmaceuticals, Inc. (US) 2006-11-08 EP disclosed
EP-1490090-A4 ACTIVE AGENT DELIVERY SYSTEMS AND METHODS FOR PROTECTING AND ADMINISTERING ACTIVE AGENTS NEW RIVER PHARMACEUTICALS INC (US) 2006-09-20 EP disclosed
US-7081255-B2 Antifungal compositions with improved bioavailability JANSSEN PHARMACEUTICA, N.V. (BE) 2006-07-25 US disclosed
US-7078526-B2 CIS-itraconazole crystalline forms and related processes, pharmaceutical compositions and methods TRANSFORM PHARMACEUTICALS, INC. (US) 2006-07-18 US disclosed
US-7060708-B2 Active agent delivery systems and methods for protecting and administering active agents NEW RIVER PHARMACEUTICALS INC. (US) 2006-06-13 US disclosed
US-20060062848-A1 Formulation comprising itraconazole NEKTAR THERAPEUTICS UK LIMITED (GB) 2006-03-23 US disclosed
WO-2005118577-A1 NOVEL SAPERCONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS TRANSFORM PHARMACEUTICALS, INC. (US) 2005-12-15 WO disclosed
US-20050226932-A1 Pharmaceutical formulations for itraconazole SAMYANG CORPORATION 2005-10-13 US disclosed
US-20050226924-A1 Composition comprising itraconazole for oral administration CHI, SANG-CHEOL (KR) 2005-10-13 US disclosed
WO-2005092884-A1 NOVEL CRYSTALLINE FORMS OF CONAZOLES AND METHODS OF MAKING AND USING THE SAME TRANSFORM PHARMACEUTICALS, INC. (US) 2005-10-06 WO disclosed
EP-1104291-B1 PELLETS HAVING A CORE COATED WITH AN ANTIFUNGAL AND A POLYMER JANSSEN PHARMACEUTICA NV (BE) 2005-09-07 EP disclosed
WO-2005060361-A2 PHARMACEUTICAL FORMULATIONS FOR ITRACONAZOLE SAMYANG CORPORATION (KR) 2005-07-07 WO disclosed
US-20050074494-A1 Itraconazole immediate release formulation ANDRX LABS, INC. 2005-04-07 US disclosed
US-20050070551-A1 Novel crystalline forms of conazoles and methods of making and using the same TRANSFORM PHARMACEUTICALS, INC. 2005-03-31 US disclosed
EP-1280795-B1 N-SUBSTITUTED CARBAMOYLOXYALKYL-AZOLIUM DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2005-03-23 EP disclosed
EP-1511490-A2 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS Transform Pharmaceuticals, Inc. (US) 2005-03-09 EP disclosed
US-20050038075-A1 Intermediates for N-substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA INTERNATIONAL LTD. (CH) 2005-02-17 US disclosed
US-20050038038-A1 N-phenyl substituted carbamoyloxyalkyl-azolium derivatives BASILEA PHARMACEUTICA INTERNATIONAL LTD. (CH) 2005-02-17 US disclosed
EP-1490090-A2 ACTIVE AGENT DELIVERY SYSTEMS AND METHODS FOR PROTECTING AND ADMINISTERING ACTIVE AGENTS New River Pharmaceuticals Inc. (US) 2004-12-29 EP disclosed
WO-2004108114-A2 ANTI-FUNGAL COMPOSITION AND A PROCESS FOR ITS MANUFACTURE PATEL DINESH SHANTILAL (IN) 2004-12-16 WO disclosed
US-6812238-B1 WATER SOLUBLE FUNGICIDES FOR SYSTEMIC MYCOSES; ORAL AND PARENTERAL ADMINISTRATION BASILEA PHARMACEUTICA AG (CH) 2004-11-02 US disclosed
US-20040115266-A1 Oral itraconazole formulations and methods of making the same STIEFEL LABORATORIES, INC. 2004-06-17 US disclosed
EP-1032263-B1 SURFACTANT-BASED ANTIMICROBIAL COMPOSITIONS AND METHODS FOR USING SAME WOODWARD LAB INC (US) 2004-06-09 EP disclosed
US-6737082-B1 Pharmaceutical oral preparation of a compound having an antifungic activity, and preparation method LICONSA LIBERACION CONTROLADA DE SUSTANCIAS ACTIVAS, S.A. (ES) 2004-05-18 US disclosed
US-20040063628-A1 Active agent delivery systems and methods for protecting and administering active agents NEW RIVER PHARMACEUTICALS INC. 2004-04-01 US disclosed
US-20040019211-A1 Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods TRANSFORM PHARMACEUTICALS, INC. (US) 2004-01-29 US disclosed
US-6673373-B2 FOR AN AZOLE ANTIFUNGAL OR ANTIBACTERIAL DRUG; CORE AND A DRUG EMULSION LAYER CONTAINING THE DRUG, AN EMULSIFIER, BINDER AND ABSORBENT AID SUCH AS CITRIC ACID; SOLUBILITY, BIOAVAILABILITY CARLSBAD TECHNOLOGY INC. 2004-01-06 US disclosed
US-6663901-B1 Itraconazole; sugar core, a coating film of a water soluble polymer, a seal coating JANSSEN PHARMACEUTICAL N.V. (BE) 2003-12-16 US disclosed
US-6663897-B2 Coating with water soluble polymer; fungicide DSM IP ASSETS B.V. (NL) 2003-12-16 US disclosed
WO-2003101392-A2 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS TRANSFORM PHARMACEUTICALS, INC. (US) 2003-12-11 WO disclosed
EP-0904060-B1 ANTIFUNGAL COMPOSITIONS WITH IMPROVED BIOAVAILABILITY JANSSEN PHARMACEUTICA NV (BE) 2003-12-10 EP disclosed
EP-1350508-A1 Antifungal formulation and the methods for manufacturing and using the same Yung Shin Pharm. Ind. Co. Ltd. (TW) 2003-10-08 EP disclosed
WO-2003079972-A2 ACTIVE AGENT DELIVERY SYSTEMS AND METHODS FOR PROTECTING AND ADMINISTERING ACTIVE AGENTS NEW RIVER PARMACEUTICALS INC. (US) 2003-10-02 WO disclosed
EP-0969821-B1 PELLETS HAVING A CORE COATED WITH AN ANTIFUNGAL AND A POLYMER JANSSEN PHARMACEUTICA NV (BE) 2003-06-04 EP disclosed
US-20030082239-A1 Antifungal compositions with improved bioavailability JANSSEN PHARMACEUTICAL, N.V. 2003-05-01 US disclosed
EP-1103252-B1 PHARMACEUTICAL ORAL PREPARATION OF A COMPOUND HAVING AN ANTIFUNGIC ACTIVITY, AND PREPARATION METHOD LICONSA LIBERACION CONTROLADA (ES) 2003-03-12 EP disclosed
US-20030026843-A1 Amorphous drug beads CAPRICORN PHARMA INC. 2003-02-06 US disclosed
EP-1280795-A2 N-SUBSTITUTED CARBAMOYLOXYALKYL-AZOLIUM DERIVATIVES Basilea Pharmaceutica AG (CH) 2003-02-05 EP disclosed
US-20020176894-A1 Antifungal formulation and the methods for manufacturing and using the same CARLSBAD TECHNOLOGY, INC. 2002-11-28 US disclosed
US-20020150620-A1 Oral itraconazole formulations and methods of making the same STIEFEL LABORATORIES, INC. 2002-10-17 US disclosed
EP-1039909-B1 METHOD OF PRODUCTION AND COMPOSITION OF AN ORAL PREPARATION OF ITRACONAZOLE CHOONGWAE PHARMA CORP (KR) 2002-10-09 EP disclosed
US-6455530-B1 FUNGICIDES SEPRACOR INC. 2002-09-24 US disclosed
EP-1143950-A3 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2002-05-15 EP disclosed
EP-0721337-B1 ORAL FORMULATIONS OF AN ANTIFUNGAL JANSSEN PHARMACEUTICA NV (BE) 2001-12-05 EP disclosed
EP-1143950-A2 TOPICAL APPLICATION PRODUCTS IPR-Institute for Pharmaceutical Research AG (CH) 2001-10-17 EP disclosed
US-20010007678-A1 ANTIFUNGAL COMPOSITIONS WITH IPMROVED BIOAVAILABILITY JANSSEN PHARMACEUTICA, N.V. (BE) 2001-07-12 US disclosed
EP-1103252-A1 PHARMACEUTICAL ORAL PREPARATION OF A COMPOUND HAVING AN ANTIFUNGIC ACTIVITY, AND PREPARATION METHOD Liconsa, Liberacion Controlada de Sustancias Activas, S.A. (ES) 2001-05-30 EP disclosed
EP-0631578-B1 ITRACONAZOLE AND SAPERCONAZOLE STEREOISOMERS JANSSEN PHARMACEUTICA NV (BE) 2001-05-23 EP disclosed
WO-2001032652-A2 N-SUBSTITUTED CARBAMOYLOXYALKYL-AZOLIUM DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed
US-6166018-A 2R, 4S, R, S- and 2S, 4R, R, S-hydroxyitraconazole SEPRACOR INC. (US) 2000-12-26 US disclosed
US-6147077-A FUNGICIDE SEPRACOR INC. (US) 2000-11-14 US disclosed
WO-2000015202-A2 TOPICAL APPLICATION PRODUCTS IPR-INSTITUTE FOR PHARMACEUTICAL RESEARCH AG (CH) 2000-03-23 WO disclosed
EP-0938487-A2 2$i(R),4$i(S),$i(R),$i(S)- AND 2$i(S),4$i(R),$i(R),$i(S)-HYDROXYITRACONAZOLE- AND HYDROXYSAPERCONAZOLE DERIVATIVES SEPRACOR, INC. (US) 1999-09-01 EP disclosed
EP-0712575-B1 Synergistic insecticidal compositions ROHM & HAAS (US) 1999-06-09 EP disclosed
EP-0759741-B1 MUCOADHESIVE EMULSIONS CONTAINING CYCLODEXTRIN JANSSEN PHARMACEUTICA NV (BE) 1998-12-23 EP disclosed
WO-1998021213-A2 2R,4S,R,S- AND 2S,4R,R,S-HYDROXYITRACONAZOLE- AND HYDROXYSAPERCONAZOLE DERIVATIVES SEPRACOR, INC. (US) 1998-05-22 WO disclosed
EP-0658103-B1 BEADS HAVING A CORE COATED WITH AN ANTIFUNGAL AND A POLYMER JANSSEN PHARMACEUTICA NV (BE) 1996-11-20 EP disclosed
US-5571829-A CYTOCHROME P450 ENZYME INHIBITOR AND AN N,N'-DIBENZOYL-N'-TERT-ALKYL-HYDRAZINE ROHM AND HAAS COMPANY (US) 1996-11-05 US disclosed
EP-0721337-A1 ORAL FORMULATIONS OF AN ANTIFUNGAL JANSSEN PHARMACEUTICA N.V. (BE) 1996-07-17 EP disclosed
EP-0712575-A1 Synergistic insecticidal compositions ROHM AND HAAS COMPANY (US) 1996-05-22 EP disclosed
US-5474997-A Administering (2R,4S)itraconazole, free of (2S,4R) stereoisomer, to reduce side effects SEPRACOR, INC. (US) 1995-12-12 US disclosed
WO-1995008993-A1 ORAL FORMULATIONS OF AN ANTIFUNGAL JANSSEN PHARMACEUTICA N.V. (BE) 1995-04-06 WO disclosed
EP-0499322-A1 (Carboxyl)alkyloxyalkyl derivatives of cyclodextrins JANSSEN PHARMACEUTICA N.V. (BE) 1992-08-19 EP disclosed
US-4916134-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACUETICA N.V. (BE) 1990-04-10 US disclosed
US-4916134-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACUETICA N.V. (BE) 1990-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (50 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240390272-A1 COMPOSITIONS AND METHODS FOR TARGETED DELIVERY TO CELLS CHMP4B, LIPA, NPC1L1 CYP3A4 4694/4885ABCG2 438/4885LMNA 350/4885
US-20050070551-A1 Novel crystalline forms of conazoles and methods of making and using the same CYP51A1, CYP3A5, ERG28 CYP3A4 10/4885ABCG2 115/4885LMNA 3498/4885
US-12097210-B2 Concomitant administration of glucocorticoid receptor modulators and CYP3A inhibitors NR3C1, NR3C2, CYP3A5 CYP3A4 21/4885ABCG2 409/4885LMNA 4861/4885
US-20230039551-A1 BUFFER- AND CHELATOR-FREE, STABLE OPHTHALMOLOGICAL COMPOSITIONS OF KETOROLAC AND PHENYLEPHRINE AND APPLICATIONS THEREOF UACA, CRYZ, MYOC CYP3A4 3871/4885ABCG2 1127/4885LMNA 1303/4885
US-20160340346-A1 ITRACONAZOLE ANALOGUES AND METHODS OF USE THEREOF GLI1, SHH, SMO CYP3A4 2373/4885ABCG2 995/4885LMNA 4777/4885
US-11648209-B2 Compositions and methods for organ specific delivery of nucleic acids POLRMT, FABP1, SNRPE CYP3A4 4622/4885ABCG2 2518/4885LMNA 185/4885
US-20070293674-A1 Novel Saperconazole Crystalline Forms and Related Processes, Pharmaceutical Compositions and Methods CYP51A1, CYP3A5, CYP3A43 CYP3A4 4/4885ABCG2 87/4885LMNA 3944/4885
US-20240293351-A1 METHODS OF ADMINISTERING SYNTHETIC TRITERPENOIDS CYP4A11, CYP3A4, CYP11B1 CYP3A4 2/4885ABCG2 131/4885LMNA 4341/4885
US-20260066250-A1 METHOD AND DEVICE FOR THE QUANTIFICATION OF TARGET ION SPECIES SRMS, IAPP, PTMS CYP3A4 4530/4885ABCG2 1800/4885LMNA 3696/4885
US-20250127887-A1 Self-Assembling Nanoparticles Based On Amphiphilic Peptides IAPP, BRCA1, ANXA11 CYP3A4 4843/4885ABCG2 4620/4885LMNA 2200/4885
US-11826373-B2 Methods for treatment of diseases SOD1, GLS, GLS2 CYP3A4 4289/4885ABCG2 4096/4885LMNA 1540/4885
US-20240269269-A1 Self-Assembling Nanoparticles UBE2B, CD4, UBE2G2 CYP3A4 4019/4885ABCG2 3818/4885LMNA 3343/4885
US-20260091097-A1 COMBINATION TREATMENT REGIMES FOR TREATING CANCER IL2, IFNG, ICOS CYP3A4 2577/4885ABCG2 4831/4885LMNA 4490/4885
US-20070027322-A1 N-substituted carbamoyloxyalkyl-azolium derivatives ERG28, CYP51A1, NAALAD2 CYP3A4 322/4885ABCG2 938/4885LMNA 4231/4885
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“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.